General Information of the Compound
Compound ID
CP0173674
Compound Name
US9233968, 12
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Structure
Formula
C26H22N6O2
Molecular Weight
450.502
Canonical SMILES
Cc1cccc(NC(=O)Nc2ccc(cc2)C#Cc2ccc3nc(NC(=O)C4CC4)cn3n2)c1
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InChI
InChI=1S/C26H22N6O2/c1-17-3-2-4-22(15-17)28-26(34)27-20-10-5-18(6-11-20)7-12-21-13-14-24-29-23(16-32(24)31-21)30-25(33)19-8-9-19/h2-6,10-11,13-16,19H,8-9H2,1H3,(H,30,33)(H2,27,28,34)
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InChIKey
POLGOZRSBQTGFR-UHFFFAOYSA-N
Physicochemical Property
logP
4.43002
Rotatable Bonds
4
Heavy Atom Count
34
Polar Areas
100.42
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
5
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118638412
ChEMBL ID
CHEMBL3910382
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00844, Platelet-derived growth factor receptor beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000749 HUVEC-C Homo sapiens (Human)  1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000749 HUVEC-C Homo sapiens (Human)  1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 1308 nM