(2S,3S)-N-(2-Methoxy-5-(trifluoromethoxy)benzyl)-2-phenylpiperidin-3-amine dihydrochloride

(3S,4S)-N-[(1S)-1-[3,5-bis(trifluoromethyl)phenyl]ethyl]-3-(4-fluoro-2-methylphenyl)-N-methyl-1-oxamoylpiperidine-4-carboxamide

rac-N-{4-[cis-4-({2-Methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenylpiperidin-1-yl]-4-oxobutyl}acetamide hydrochloride

(3S,4S)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-3-(2-methylphenyl)piperidine-4-carboxamide

(3S,4S)-4-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(4-fluoro-2-methylphenyl)-4-N-methylpiperidine-1,4-dicarboxamide

rac-cis-N-Ethyl-4-({2-methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenylpiperidine-1-carboxamide hydrochloride

(3S,4S)-1-(2-acetamidoacetyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(4-fluoro-2-methylphenyl)-N-methylpiperidine-4-carboxamide

rac-cis-N-Ethyl-4-({2-(cyclopropyloxy)-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenylpiperidine-1-carboxamide hydrochloride

(3S,4S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(4-fluoro-2-methylphenyl)-1-[2-(hydroxyamino)-2-oxoacetyl]-N-methylpiperidine-4-carboxamide

(3S,4S)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(4-fluoro-2-methylphenyl)-N-methylpiperidine-4-carboxamide

(3S,4S)-4-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(4-fluoro-2-methylphenyl)-1-N,4-N-dimethylpiperidine-1,4-dicarboxamide

cis-rac-1-Acetyl-N-{2-methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}-3-phenyl-4-piperidinamine hydrochloride

(3S,4S)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(4-fluorophenyl)-N-methylpiperidine-4-carboxamide

methyl (3R,4S)-4-[[2-methoxy-5-[5-(trifluoromethyl)tetrazol-1-yl]phenyl]methylamino]-3-phenylpiperidine-1-carboxylate

rac-N-{3-[cis-4-({2-Methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenyl-1-piperidinyl]-3-oxopropyl}acetamide hydrochloride

rac-cis-N-Cyclopropyl-4-({2-methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenyl-1-piperidinecarboxamidehydrochloride

rac-cis-4-({2-Methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenyl-N-(2,2,2-trifluoroethyl)-1-piperidinecarboxamide hydrochloride

rac-cis-1-[(1-Acetyl-3-azetidinyl)carbonyl]-N-{2-methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}-3-phenyl-4-piperidinamine hydrochloride

(3S,4S)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(2-ethylphenyl)-N-methylpiperidine-4-carboxamide

(3S,4S)-4-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(4-fluoro-2-methylphenyl)-1-N-methoxy-4-N-methylpiperidine-1,4-dicarboxamide

(3R,4S)-N-[[2-methoxy-5-[5-(trifluoromethyl)tetrazol-1-yl]phenyl]methyl]-1-methylsulfonyl-3-phenylpiperidin-4-amine

rac-cis-N-Isopropyl-4-({2-methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenyl-1-piperidinecarboxamidehydrochloride

rac-N-{2-[cis-4-({2-Methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenyl-1-piperidinyl]-2-oxoethyl}-N-methylacetamide hydrochloride

rac-cis-N-Ethyl-4-({2-ethoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenylpiperidine-1-carboxamide hydrochloride

(2,5-Dimethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine

US8470816, 91

(3R,4S)-N-ethyl-3-phenyl-4-[[5-[5-(trifluoromethyl)tetrazol-1-yl]-2,3-dihydro-1-benzofuran-7-yl]methylamino]piperidine-1-carboxamide

(3R,4R)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-3-phenylpiperidine-4-carboxamide

(2S,3S)-N-(5-(1,1,1,3,3,3-hexafluoropropan-2-yl)-2-methoxybenzyl)-2-phenylpiperidin-3-amine

(2S,3S)-3-[(1R)-6-Methoxy-1-methyl-1-trifluoromethylisochroman-7-yl]methylamino-2-phenylpiperidine

R/S-(2S,3S)-N-((6-methoxy-3-(trifluoromethyl)-1,3-dihydroisobenzofuran-5-yl)methyl)-2-phenylpiperidin-3-amine

R/S-(2S,3S)-N-(2-methoxy-5-(2,2,2-trifluoro-1-methoxyethyl)benzyl)-2-phenylpiperidin-3-amine

R/S-(2S,3S)-N-(2-methoxy-5-(1,1,1,2-tetrafluoropropan-2-yl)benzyl)-2-phenylpiperidin-3-amine

R/S-(2S,3S)-3-(5-Methoxy-1-methyl-1-(trifluoromethyl)indane-6-yl)methylamino-2-phenylpiperidine

rac-cis-1-[(1-Acetyl-4-piperidinyl)carbonyl]-N-{2-methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}-3-phenyl-4-piperidinamine hydrochloride

N-[4-methoxy-3-[[[(2S,3S)-2-phenylpiperidin-3-yl]amino]methyl]phenyl]-N-methylmethanesulfonamide

(3S,4S)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(4-fluoro-2-methylphenyl)-N-methyl-1-[2-(methylamino)-2-oxoacetyl]piperidine-4-carboxamide

rac-cis-4-({2-Methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-N,N-dimethyl-3-phenyl-1-piperidinecarboxamide hydrochloride

(2-Ethoxy-5-trifluoromethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine

(5-Chloro-2-methoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine

(3S,4S)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-3-(3-methylphenyl)piperidine-4-carboxamide

N-[(2R)-1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-piperidin-1-ylpiperidin-1-yl)acetamide

rac-cis-1-Acetyl-N-(2-methoxy-5-(trifluoromethoxy)benzyl)-3-phenyl-4-piperidinamine hydrochloride

(+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-amine

(3R,4S)-N-ethyl-4-[[2-methoxy-5-(trifluoromethoxy)phenyl]methylamino]-3-phenylpiperidine-1-carboxamide

1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-5-phenyl-3,6-dihydro-2H-pyridine-4-carboxamide

N-[(2R)-1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-cyclohexylpiperazin-1-yl)acetamide

N-[1-[acetyl-[(2-chlorophenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-piperidin-1-ylpiperidin-1-yl)acetamide

(2-Isopropoxy-5-trifluoromethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine

(3S,4S)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-3-(4-methylphenyl)piperidine-4-carboxamide

(2-Methoxy-5-trifluoromethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine

(2S,3S)-N-(2-methoxy-5-(1,1,1-trifluoro-2-methylpropan-2-yl)benzyl)-2-phenylpiperidin-3-amine

rac-trans-N-{2-[-4-({2-Methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}amino)-3-phenyl-1-piperidinyl]-2-oxoethyl}acetamide hydrochloride

(3S,4S)-N-[(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethyl]-3-(4-fluoro-2-methylphenyl)-N-methyl-1-oxamoylpiperidine-4-carboxamide

5-(4-Fluoro-phenyl)-7-methyl-8-oxo-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide

(3S,4S)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-3-(2-propan-2-ylphenyl)piperidine-4-carboxamide

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-piperidin-1-ylpiperidin-1-yl)acetamide

7-Methyl-8-oxo-5-phenyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide

N-[3-[(3-benzhydryl-4-oxopiperidin-1-yl)methyl]-4-methoxyphenyl]methanesulfonamide

(S)-7-(3,5-Bis-trifluoromethyl-benzyl)-9-methyl-5-p-tolyl-7,8,9,10-tetrahydro-1,7,10a-triaza-cyclohepta[b]naphthalene-6,11-dione

rac-Methyl cis-4-{[2-methoxy-5-(trifluoromethoxy)benzyl]amino}-3-phenylpiperidine-1-carboxylate hydrochloride

((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-cyclohexylpiperazin-1-yl)acetamide

(2S,3S)-N-(((S)-6-methoxy-1-methyl-1-(trifluoromethyl)-3,4-dihydro-1H-isochromen-7-yl)methyl)-2-phenylpiperidin-3-amine

rac-3-(Diphenylmethyl)-1-[2-methoxy-5-(trifluoromethoxy)benzyl]piperidin-4-one hydrochloride

(5S,9S)-4-[(2-methoxyphenyl)methyl]-9-phenyl-1,4-diazabicyclo[3.3.1]nonane

4-(4-Fluoro-phenyl)-2-methyl-1-oxo-1,2-dihydro-isoquinoline-3-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide

(2S,3S)-N-[[2-methoxy-5-(1,1,1-trifluoropropan-2-yl)phenyl]methyl]-2-phenylpiperidin-3-amine

(2-Difluoromethoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine

rac-3-(Diphenylmethyl)-1-[2-methoxy-5-(1-methylethyl)benzyl]piperidin-4-one hydrochloride

N-[(2R)-1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-[4-(hydroxymethyl)phenoxy]acetamide

(7R,9R)-7-(3,5-Bis-trifluoromethyl-benzyl)-9-methyl-5-p-tolyl-8,9,10,11-tetrahydro-7H-1,7,11a-triaza-cycloocta[b]naphthalene-6,12-dione

(2-Isopropoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine

N-[(2R)-1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-imidazol-1-ylphenoxy)acetamide

1-benzofuran-2-ylmethyl N-[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-1-[[(1S)-1-phenylethyl]amino]propan-2-yl]carbamate

(5-Dimethylamino-2-methoxy-benzyl)-((2S,3S)-2-phenyl-piperidin-3-yl)-amine

(SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2

(5S,8S)-6-[(2-methoxyphenyl)methyl]-8-phenyl-1,6-diazabicyclo[3.2.1]octane

N-[(2R)-1-[acetyl-[(2-chlorophenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-imidazol-1-ylphenoxy)acetamide

(2S,3S)-N-[[2-methoxy-5-(1,2,2,2-tetrafluoroethyl)phenyl]methyl]-2-phenylpiperidin-3-amine

N-[1-[formyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

((2S,3S)-2-Phenyl-piperidin-3-yl)-(2-trifluoromethoxy-benzyl)-amine

N-[3-(1H-indol-3-yl)-2-[[2-(4-phenylpiperazin-1-yl)acetyl]amino]propyl]-N-[(2-methoxyphenyl)methyl]propanamide

rac-3-[Bis(4-fluorophenyl)methyl]-1-[2-methoxy-5-(trifluoromethoxy)benzyl]piperidin-4-one hydrochloride

1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)carboxamidomethyl]ethyl}-2-(4-hydroxymethylphenoxy)acetamide

N-[(2R)-1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

7-(3,5-Bis-trifluoromethyl-benzyl)-5-p-tolyl-7,8,9,10-tetrahydro-1,7,10a-triaza-cyclohepta[b]naphthalene-6,11-dione

(2S,3S)-3-[2-Methoxy-5-(2,2,2-trifluoroethyl)benzylamino]-2-phenylpiperidine

(2S,3S)-N-[[2-methoxy-5-(1,1,1-trifluoro-2-methoxypropan-2-yl)phenyl]methyl]-2-phenylpiperidin-3-amine

(8S,9S)-8-benzhydryl-N-[(2-methoxyphenyl)methyl]-7-azatricyclo[4.3.1.03,7]decan-9-amine

(S)-((S)-8-Benzhydryl-7-aza-tricyclo[4.3.1.0*3,7*]dec-9-yl)-(2-methoxy-benzyl)-amine

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-benzylpiperazin-1-yl)acetamide

1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)carboxamidomethyl]ethyl}-2-[4-(1,2,3-thiadiazol-4-yl)phenoxy]acetamide

5-(4-Fluoro-phenyl)-7-methyl-8-oxo-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid 3,5-bis-trifluoromethyl-benzylamide

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

rac-3-[Bis(4-fluorophenyl)methyl]-1-(5-bromo-2-methoxybenzyl)piperidin-4-one hydrochloride

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1-benzothiophen-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

2-Methyl-1-oxo-4-phenyl-1,2-dihydro-isoquinoline-3-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide

rac-cis-N-[2-Methoxy-5-(trifluoromethoxy)benzyl]-1-(methyl sulfonyl)-3-phenyl-4-piperidin-4-amine hydrochloride

N-[1-[[(2S)-1-[benzyl(methyl)amino]-3-naphthalen-2-yl-1-oxopropan-2-yl]carbamoyl]cyclohexyl]-1H-indole-3-carboxamide

methyl 3-[[3-(1H-indol-3-yl)-2-[[2-(4-phenylpiperazin-1-yl)acetyl]amino]propyl]-[(2-methoxyphenyl)methyl]amino]-3-oxopropanoate

(2S,3S)-2-Benzhydryl-1-carbamoylmethyl-3-(2-methoxy-benzylamino)-1-azonia-bicyclo[2.2.2]octane iodide

2-Methyl-1-oxo-4-o-tolyl-1,2-dihydro-isoquinoline-3-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide

rac-cis-N-{2-Methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]benzyl}-3-phenylpiperidin-4-amine dihydrochloride

US8470816, 82

2-Dimethylamino-N-{3-(1H-indol-3-yl)-2-[2-(4-phenyl-piperazin-1-yl)-acetylamino]-propyl}-N-(2-methoxy-benzyl)-acetamide

7-(3,5-Bis-trifluoromethyl-benzyl)-5-p-tolyl-7,8,9,10,11,12-hexahydro-1,7,12a-triaza-cyclonona[b]naphthalene-6,13-dione

(S)-((S)-11-Benzhydryl-1-aza-tricyclo[5.4.0.0*3,9*]undec-10-yl)-(2-methoxy-benzyl)-amine

N-[1-[acetyl-[(2-chlorophenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

rac-cis-1-Ethyl-N-{2-Methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]}benzyl)-3-phenyl-4-piperidinamine hydrochloride

(2,4-difluorophenyl)methyl N-[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-1-[[(1S)-1-phenylethyl]amino]propan-2-yl]carbamate

(10S,11S)-11-benzhydryl-N-[(2-methoxyphenyl)methyl]-1-azatricyclo[5.4.0.03,9]undecan-10-amine

(2-fluoro-4-methylphenyl)methyl N-[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-1-[[(1S)-1-phenylethyl]amino]propan-2-yl]carbamate

(3S,6S,7S)-3-(2-Methoxy-phenyl)-7-phenyl-1,8-diaza-spiro[5.5]undecane

N-[3-(1H-indol-3-yl)-2-[[2-(4-phenylpiperazin-1-yl)acetyl]amino]propyl]-N-[(2-methoxyphenyl)methyl]benzamide

(2,5-difluorophenyl)methyl N-[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-1-[[(1S)-1-phenylethyl]amino]propan-2-yl]carbamate

((2R,3R)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine

N-[1-[acetyl(benzyl)amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

6-(3,5-Bis-trifluoromethyl-benzyl)-10-p-tolyl-7,8-dihydro-6H-1,6,8a-triaza-anthracene-5,9-dione

rac-3-[Bis(4-fluorophenyl)methyl]-1-(2,6-dimethoxybenzyl)piperidin-4-one hydrochloride

1-benzothiophen-2-ylmethyl N-[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-1-[[(1S)-1-phenylethyl]amino]propan-2-yl]carbamate

(2-Methoxy-benzyl)-((2S,3S,3aR,6aS)-2-phenyl-octahydro-cyclopenta[b]pyrrol-3-yl)-amine

(S)-((S)-9-Benzhydryl-1-aza-tricyclo[4.3.1.0*3,7*]dec-8-yl)-(2-methoxy-benzyl)-amine

2-Methyl-1-oxo-4-o-tolyl-1,2-dihydro-isoquinoline-3-carboxylic acid 3,5-bis-trifluoromethyl-benzylamide

5-(4-Fluoro-phenyl)-7-methyl-8-oxo-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (2-methoxy-benzyl)-methyl-amide

N-[1-[acetyl-[(4-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

3-benzhydryl-1-[(2-methoxy-5-nitrophenyl)methyl]piperidin-4-one

(3R,4R)-1-acetyl-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-3-phenylpiperidine-4-carboxamide

(3R,4R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-3-phenylpiperidine-4-carboxamide

(3R,4R)-1-(1-acetylpiperidine-4-carbonyl)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-phenylpiperidine-4-carboxamide

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-naphthalen-1-ylpropan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-[4-(dimethylamino)piperidin-1-yl]acetamide

N-[1-(1H-indol-3-yl)-3-[(2-methoxyphenyl)methyl-(methylcarbamoyl)amino]propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

N-[1-[acetyl-[(2-nitrophenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)acetamide

rac-3-[Bis(4-fluorophenyl)methyl]-1-(2,5-dimethoxybenzyl)piperidin-4-one hydrochloride

1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimethoxy-benzoyl)-pyrrolidin-3-yl]-ethyl}-4-phenyl-piperidine-4-carboxylic acid amide; hydrochloride

(2-fluorophenyl)methyl N-[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-1-[[(1S)-1-phenylethyl]amino]propan-2-yl]carbamate

N-[1-[acetyl-[(2-methylphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

N-[1-[acetyl-[[2-(trifluoromethyl)phenyl]methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)carboxamidomethyl]ethyl}-2-(4-hydroxyphenoxy)acetamide

(3R,4S)-1-acetyl-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-N-methyl-3-phenylpiperidine-4-carboxamide

(S)-((S)-3-Benzhydryl-octahydro-2,5-methano-isoquinolin-4-yl)-(2-methoxy-benzyl)-amine

1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)carboxamidomethyl]ethyl}-4-(4-methoxyphenyl)-4-oxobutanamide

7-Methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (3,5-dichloro-benzyl)-methyl-amide

6-Chloro-2-methyl-1-oxo-4-phenyl-1,2-dihydro-isoquinoline-3-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide

1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)carboxamidomethyl]ethyl}-2-(4-acetylphenoxy)acetamide

(3R,4R)-N-ethyl-4-[[2-methoxy-5-(trifluoromethoxy)phenyl]methylamino]-3-phenylpiperidine-1-carboxamide

N-[1-(1H-indol-3-yl)-3-[(2-methoxyphenyl)methyl-methylsulfonylamino]propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

rac-3-[Bis(4-fluorophenyl)methyl]-1-(5-fluoro-2-methoxybenzyl)piperidin-4-one hydrochloride

(S)-((S)-9-Benzhydryl-8-aza-tricyclo[5.3.1.0*3,8*]undec-10-yl)-(2-methoxy-benzyl)-amine

1-(2-Chloro-benzyl)-1-methyl-3-(2,6,7-trimethyl-1-oxo-4-phenyl-1,2-dihydro-isoquinolin-3-yl)-urea

7-Methyl-8-oxo-5-p-tolyl-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (3,5-dimethyl-benzyl)-methyl-amide

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperidin-1-yl)acetamide

N-[1-[acetyl-[(3-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-phenylpiperazin-1-yl)acetamide

rac-cis-1-Ethyl-N-[2-methoxy-5-(trifluoromethoxy)benzyl]-3-phenyl-4-piperidinamine hydrochloride

rac-3-[Bis(4-fluorophenyl)methyl]-1-[2-(trifluoromethyl)benzyl]piperidin-4-one hydrochloride

N-[(1S,2R)-2-[[(1R)-1-[methyl-(2-phenylacetyl)amino]-2-naphthalen-2-ylethyl]carbamoyl]cyclohexyl]-1H-indole-3-carboxamide

5-(4-Fluoro-phenyl)-7-methyl-8-oxo-7,8-dihydro-[1,7]naphthyridine-6-carboxylic acid (3,5-dimethyl-benzyl)-methyl-amide

N-[1-[acetyl-[(2-methoxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propan-2-yl]-2-(4-methylpiperazin-1-yl)acetamide

ethyl N-[3-(1H-indol-3-yl)-2-[[2-(4-phenylpiperazin-1-yl)acetyl]amino]propyl]-N-[(2-methoxyphenyl)methyl]carbamate

cis-(3RS,4SR)-N-[3,5-Bis(trifluoromethyl)benzyl]-N-methyl-3-phenylpiperidine-4-carboxamide hydrochloride

rac-1-(5-Amino-2-methoxybenzyl)-3-(diphenylmethyl)piperidin-4-one dihydrochloride

1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)carboxamidomethyl]ethyl}-4-(4-fluorophenyl)-4-oxobutanamide

rac-2-({3-[Bis(4-fluorophenyl)methyl]-4-oxopiperidin-1-yl}methyl)benzonitrile hydrochloride