| Compound ID |
Compound Name |
Compound Formula |
|
CP0408834
|
2-(4-thiazol-2-ylpiperidin-1-yl)-N-(m-tolyl)acetamide
Show/Hide
|
C17H21N3OS
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0453673
|
2-[4-(2-fluorophenyl)piperidin-1-yl]-N-(m-tolyl)acetamide
Show/Hide
|
C20H23FN2O
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0036921
|
3-HYDROXYTYRAMINE HYDROCHLORIDE
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|
C8H11NO2
|
3
|
| 1 |
EC50 = 1.8 nM
|
|
|
| 2 |
EC50 = 2.2 nM
|
|
|
| 3 |
EC50 = 10 nM
|
|
|
|
CP0860027
|
(E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)propan-1-one oxime
Show/Hide
|
C19H24N4O
|
1
|
| 1 |
EC50 = 2.3 nM
|
|
|
|
CP0286510
|
6-(4-((1H-benzo[d]imidazol-2-yl)methyl)piperazin-1-yl)pyridin-3-ol
Show/Hide
|
C17H19N5O
|
2
|
| 1 |
EC50 = 2.4 nM
|
|
|
| 2 |
Ki = 17 nM
|
|
|
|
CP0006107
|
CAS_85760-74-3
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|
C13H21N3
|
3
|
| 1 |
EC50 = 2.7 nM
|
|
|
| 2 |
EC50 = 5 nM
|
|
|
| 3 |
EC50 = 83 nM
|
|
|
|
CP0502735
|
2-(5-hydroxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)-N-(m-tolyl)acetamide
Show/Hide
|
C19H23N3O2
|
1
|
| 1 |
EC50 = 3.8 nM
|
|
|
|
CP0496293
|
2-[4-(2-Nitro-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
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|
C18H19N5O2
|
1
|
| 1 |
EC50 = 3.9 nM
|
|
|
|
CP0856105
|
(E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(o-tolyl)propan-1-one oxime
Show/Hide
|
C19H24N4O
|
1
|
| 1 |
EC50 = 4.2 nM
|
|
|
|
CP0042751
|
(6aR)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol;hydrate;hydrochloride
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|
C17H17NO2
|
2
|
| 1 |
EC50 = 4.3 nM
|
|
|
| 2 |
Ki = 8.9 nM
|
|
|
|
CP0855412
|
(E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H22N4O
|
2
|
| 1 |
EC50 = 4.4 nM
|
|
|
| 2 |
Ki = 25.4 nM
|
|
|
|
CP0850200
|
(Z)-2-hydroxy-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)-propan-1-one oxime
Show/Hide
|
C19H24N4O2
|
1
|
| 1 |
EC50 = 4.9 nM
|
|
|
|
CP0200483
|
2-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
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|
C18H19ClN4
|
1
|
| 1 |
EC50 = 7.2 nM
|
|
|
|
CP0050806
|
2-[4-(4-[3H]-2-cyanophenyl)piperazinyl]-N-(2,4,6-[3H]3-3-methylphenyl)acetamide derivative
Show/Hide
|
C20H22N4O
|
1
|
| 1 |
EC50 = 7.5 nM
|
|
|
|
CP0406709
|
2-[4-(3-hydroxyphenyl)piperidin-1-yl]-N-(m-tolyl)acetamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0445989
|
2-[1-[2-(m-tolylamino)allyl]piperidin-4-yl]benzonitrile
Show/Hide
|
C21H23N3O
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0452996
|
6-Fluoro-2-(4-pyridin-2-yl-piperazin-1-ylmethyl)-1H-benzoimidazole
Show/Hide
|
C17H18FN5
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0159532
|
N-[[4-(2-cyanophenyl)piperazin-1-yl]methyl]-3-methylbenzamide
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|
C20H22N4O
|
1
|
| 1 |
EC50 = 8.3 nM
|
|
|
|
CP0881778
|
(E)-1-(2,4-difluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one oxime
Show/Hide
|
C18H20F2N4O
|
1
|
| 1 |
EC50 = 8.9 nM
|
|
|
|
CP0464229
|
3-methyl-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C19H23N3O
|
2
|
| 1 |
EC50 = 9 nM
|
|
|
| 2 |
Ki = 32 nM
|
|
|
|
CP0853251
|
(E)-1-(4-fluorophenyl)-4-(4-pyridin-2-ylpiperazin-1-yl)butan-1-one oxime
Show/Hide
|
C19H23FN4O
|
1
|
| 1 |
EC50 = 9.5 nM
|
|
|
|
CP0503097
|
3-methyl-N-(4-thiazol-2-ylpiperidin-1-ylmethyl)-benzamide
Show/Hide
|
C17H21N3OS
|
1
|
| 1 |
EC50 = 9.8 nM
|
|
|
|
CP0419364
|
1'-(1H-Benzoimidazol-2-ylmethyl)-1',2',3',6'-tetrahydro-[2,4']bipyridinyl
Show/Hide
|
C18H18N4
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0860026
|
(E)-1-(3-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H21ClN4O
|
1
|
| 1 |
EC50 = 11.9 nM
|
|
|
|
CP0376038
|
1'-(1H-Benzoimidazol-2-ylmethyl)-1',2',3',4',5',6'-hexahydro-[2,4']bipyridinyl
Show/Hide
|
C18H20N4
|
2
|
| 1 |
EC50 = 12 nM
|
|
|
| 2 |
EC50 = 14 nM
|
|
|
|
CP0031347
|
2-((4-(pyridin-2-yl)piperazin-1-yl)methyl)-1H-benzo[d]imidazole
Show/Hide
|
C17H19N5
|
1
|
| 1 |
EC50 = 12.4 nM
|
|
|
|
CP0364830
|
2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C19H22N4O
|
1
|
| 1 |
EC50 = 12.4 nM
|
|
|
|
CP0850208
|
3-[1-hydroxyimino-3-(4-pyridin-2-ylpiperazin-1-yl)propyl]-benzonitrile
Show/Hide
|
C19H21N5O
|
1
|
| 1 |
EC50 = 13.1 nM
|
|
|
|
CP0408265
|
(Z)-1-(4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23FN4O
|
2
|
| 1 |
EC50 = 13.6 nM
|
|
|
| 2 |
Ki = 53.3 nM
|
|
|
|
CP0502127
|
2-[4-(1H-Benzoimidazol-2-ylmethyl)-piperazin-1-yl]-nicotinonitrile
Show/Hide
|
C18H18N6
|
1
|
| 1 |
EC50 = 13.9 nM
|
|
|
|
CP0384374
|
2-(3',4',-5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)-N-(m-tolyl)acetamide
Show/Hide
|
C19H23N3O
|
4
|
| 1 |
EC50 = 14 nM
|
|
|
| 2 |
Ki = 3.95 nM
|
|
|
| 3 |
Ki = 8 nM
|
|
|
| 4 |
Ki = 54.2 nM
|
|
|
|
CP0439585
|
2-[4-(1H-Benzoimidazol-2-ylmethyl)-piperazin-1-yl]-benzonitrile
Show/Hide
|
C19H19N5
|
1
|
| 1 |
EC50 = 14.6 nM
|
|
|
|
CP0402831
|
2-[4-(2-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C18H19FN4
|
1
|
| 1 |
EC50 = 14.7 nM
|
|
|
|
CP0037328
|
(6aR,12bS)-10,11-Dihydroxy-5,6,6a,7,8,12b-hexahydro-benzo[a]phenanthridinium
Show/Hide
|
C17H17NO2
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0854850
|
(E)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H21FN4O
|
1
|
| 1 |
EC50 = 17.1 nM
|
|
|
|
CP0848083
|
(Z)-1-(3,5-difluorophenyl)-3-(4-(pyridin-2-yl)piperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H20F2N4O
|
1
|
| 1 |
EC50 = 17.5 nM
|
|
|
|
CP0378825
|
N-(4-fluoro-3-methylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C19H22FN3O2
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0862523
|
(E)-2-[4-(3-hydroxyimino-3-phenylpropyl)piperazin-1-yl]nicotinonitrile
Show/Hide
|
C19H21N5O
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0849239
|
(E)-1-(2-hydroxy-5-methylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C19H24N4O2
|
1
|
| 1 |
EC50 = 19.2 nM
|
|
|
|
CP0851016
|
(E)-1-(3,5-Difluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one Oxime
Show/Hide
|
C18H20F2N4O
|
1
|
| 1 |
EC50 = 19.4 nM
|
|
|
|
CP0862362
|
(Z)-2-[4-(3-hydroxyimino-3-phenylpropyl)piperazin-1-yl]nicotinonitrile
Show/Hide
|
C19H21N5O
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0846794
|
(Z)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(o-tolyl)propan-1-one oxime
Show/Hide
|
C19H24N4O
|
1
|
| 1 |
EC50 = 20.3 nM
|
|
|
|
CP0849739
|
(+/-)-trans-2,3-dihydroxy-7-propyl-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline hydrochloride
Show/Hide
|
C19H22ClNO3
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0846831
|
(Z)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H22N4O
|
1
|
| 1 |
EC50 = 21.7 nM
|
|
|
|
CP0384404
|
(Z)-1-(4-chlorophenyl)-2-hydroxy-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime
Show/Hide
|
C19H23ClN4O2
|
2
|
| 1 |
EC50 = 22.6 nM
|
|
|
| 2 |
Ki = 150 nM
|
|
|
|
CP0430324
|
2-[2-(4-Pyridin-2-yl-piperazin-1-yl)-ethyl]-1H-benzoimidazole
Show/Hide
|
C18H21N5
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0862520
|
(E)-1-(2-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H21ClN4O
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0452994
|
2-[4-(3-Fluoro-pyridin-2-yl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C17H18FN5
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0390666
|
(Z)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one Om-ethyloxime
Show/Hide
|
C19H24N4O
|
1
|
| 1 |
EC50 = 24.1 nM
|
|
|
|
CP0848082
|
(Z)-1-(2-Chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H21ClN4O
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0401628
|
2-[4-(2-Ethoxy-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C20H24N4O
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0439429
|
(E)-1-(4-fluorophenyl)-2-(4-pyridin-2-yl)ethanone O-methyloxime
Show/Hide
|
C18H21FN4O
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0161149
|
2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 = 26.8 nM
|
|
|
|
CP0393867
|
(Z)-4-[1-methoxyimino-3-(4-pyridin-2-ylpiperazin-1-yl)propyl]benzonitrile
Show/Hide
|
C20H23N5O
|
2
|
| 1 |
EC50 = 27.5 nM
|
|
|
| 2 |
Ki = 20.1 nM
|
|
|
|
CP0386031
|
(E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)propan-1-one O-methyloxime
Show/Hide
|
C20H26N4O
|
2
|
| 1 |
EC50 = 27.6 nM
|
|
|
| 2 |
Ki = 8 nM
|
|
|
|
CP0391206
|
(E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-ethyloxime
Show/Hide
|
C20H26N4O
|
2
|
| 1 |
EC50 = 28.5 nM
|
|
|
| 2 |
Ki = 38 nM
|
|
|
|
CP0268831
|
2-(4-Phenyl-piperazin-1-ylmethyl)-1H-benzoimidazole
Show/Hide
|
C18H20N4
|
1
|
| 1 |
EC50 = 30.6 nM
|
|
|
|
CP0850207
|
(E)-1-(4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H21FN4O
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0215286
|
2-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'bipyridine]-1'-yl)-N-(m-tolyl)acetamide
Show/Hide
|
C19H23N3O2
|
2
|
| 1 |
EC50 = 32 nM
|
|
|
| 2 |
Ki = 294 nM
|
|
|
|
CP0381691
|
(E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H24N4O
|
2
|
| 1 |
EC50 = 32 nM
|
|
|
| 2 |
Ki = 22.8 nM
|
|
|
|
CP0193372
|
5-Fluoro-2-(4-pyridin-2-yl-piperazin-1-ylmethyl)-1H-indole
Show/Hide
|
C18H19FN4
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0390663
|
2-[(E)-[1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propylidene]amino]oxyacetonitrile
Show/Hide
|
C20H23N5O
|
2
|
| 1 |
EC50 = 33 nM
|
|
|
| 2 |
Ki = 88 nM
|
|
|
|
CP0407226
|
1-pyridin-3-yl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C18H23N5O
|
2
|
| 1 |
EC50 = 33.3 nM
|
|
|
| 2 |
Ki = 130 nM
|
|
|
|
CP0408279
|
(Z)-1-(4-fluorophenyl)-4-(4-pyridin-2-ylpiperazin-1-yl)butan-1-one O-methyloxime
Show/Hide
|
C20H25FN4O
|
1
|
| 1 |
EC50 = 33.5 nM
|
|
|
|
CP0862370
|
(Z)-2-methoxy-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)-propan-1-one O-methyloxime
Show/Hide
|
C20H26N4O2
|
1
|
| 1 |
EC50 = 34.5 nM
|
|
|
|
CP0406707
|
2-(3-cyano-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)-N-(m-tolyl)acetamide
Show/Hide
|
C20H22N4O
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0452995
|
2-[4-(6-Methyl-pyridin-2-yl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C18H21N5
|
1
|
| 1 |
EC50 = 36.2 nM
|
|
|
|
CP0395313
|
(E)-1-(3,5-difluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C19H22F2N4O
|
2
|
| 1 |
EC50 = 37.2 nM
|
|
|
| 2 |
Ki = 110 nM
|
|
|
|
CP0376146
|
(E)-1-(4-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23ClN4O
|
2
|
| 1 |
EC50 = 37.6 nM
|
|
|
| 2 |
Ki = 38.2 nM
|
|
|
|
CP0408836
|
3,4-dimethyl-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 = 38 nM
|
|
|
|
CP0854851
|
(E)-1-phenyl-3-(4-pyrimidin-2-ylpiperazin-1-yl)propan-1-oxime
Show/Hide
|
C17H21N5O
|
1
|
| 1 |
EC50 = 39.2 nM
|
|
|
|
CP0408835
|
N-(2-methoxy-6-methylphenyl)-2-(4-pyridin-2-ylpiperidin-1-yl)acetamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0432613
|
(Z)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(o-tolyl)propan-1-one O-methyloxime
Show/Hide
|
C20H26N4O
|
1
|
| 1 |
EC50 = 40.1 nM
|
|
|
|
CP0395329
|
(E)-1-(4-fluorophenyl)-4-(4-pyridin-2-ylpiperazin-1-yl)butan-1-one O-methyloxime
Show/Hide
|
C20H25FN4O
|
1
|
| 1 |
EC50 = 41.7 nM
|
|
|
|
CP0384418
|
(E)-1-(2-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23ClN4O
|
1
|
| 1 |
EC50 = 42.3 nM
|
|
|
|
CP0424849
|
(Z)-1-(4-Fluorophenyl)-2-(4-pyridin-2-yl)ethanone O-Methyloxime
Show/Hide
|
C18H21FN4O
|
2
|
| 1 |
EC50 = 43.8 nM
|
|
|
| 2 |
Ki = 2050 nM
|
|
|
|
CP0390664
|
(E)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23FN4O
|
2
|
| 1 |
EC50 = 44.6 nM
|
|
|
| 2 |
Ki = 13.9 nM
|
|
|
|
CP0849208
|
(E)-2-hydroxy-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)-propan-1-one oxime
Show/Hide
|
C19H24N4O2
|
1
|
| 1 |
EC50 = 44.8 nM
|
|
|
|
CP0401607
|
2-(4-Pyrimidin-2-yl-piperazin-1-ylmethyl)-1H-benzoimidazole
Show/Hide
|
C16H18N6
|
1
|
| 1 |
EC50 = 44.8 nM
|
|
|
|
CP0408837
|
3,5-dichloro-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C18H19Cl2N3O2
|
1
|
| 1 |
EC50 = 45 nM
|
|
|
|
CP0395335
|
(Z)-N-ethoxy-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-imine
Show/Hide
|
C20H26N4O
|
1
|
| 1 |
EC50 = 45 nM
|
|
|
|
CP0846830
|
(E)-1-(3,5-dimethylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one oxime
Show/Hide
|
C20H26N4O
|
1
|
| 1 |
EC50 = 45.8 nM
|
|
|
|
CP0453082
|
(E)-1-(4-chlorophenyl)-2-hydroxy-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime
Show/Hide
|
C19H23ClN4O2
|
2
|
| 1 |
EC50 = 46 nM
|
|
|
| 2 |
Ki = 113 nM
|
|
|
|
CP0407232
|
(Z)-1-(4-chlorophenyl)-3-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4']bipyridinyl-1'-yl)propan-1-one O-methyl-oxime
Show/Hide
|
C20H24ClN3O2
|
1
|
| 1 |
EC50 = 46.4 nM
|
|
|
|
CP0374886
|
(Z)-1-(3,5-difluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C19H22F2N4O
|
2
|
| 1 |
EC50 = 46.7 nM
|
|
|
| 2 |
Ki = 6.3 nM
|
|
|
|
CP0395334
|
(E)-2-[4-(ethoxyimino-3-phenylpropyl)piperazin-1-yl]benzonitrile
Show/Hide
|
C22H26N4O
|
1
|
| 1 |
EC50 = 48.7 nM
|
|
|
|
CP0408376
|
(E)-1-(4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23FN4O
|
2
|
| 1 |
EC50 = 48.8 nM
|
|
|
| 2 |
Ki = 14.2 nM
|
|
|
|
CP0875445
|
(E)-1-phenyl-3-(4-thiazol-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C16H20N4OS
|
1
|
| 1 |
EC50 = 49.5 nM
|
|
|
|
CP0453675
|
3-fluoro-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C19H22FN3O2
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0420189
|
N-(3,5-dimethylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0491324
|
2-((S)-2-Methyl-4-pyridin-2-yl-piperazin-1-ylmethyl)-1H-benzoimidazole
Show/Hide
|
C18H21N5
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0453677
|
1'-(1H-benzimidazol-2-ylmethyl)-1',2',3',4',5',6'-hexahydro-[2,4'-bipyridine] 1-oxide
Show/Hide
|
C18H20N4O
|
1
|
| 1 |
EC50 = 54 nM
|
|
|
|
CP0408270
|
(Z)-1-(4-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23ClN4O
|
1
|
| 1 |
EC50 = 56.6 nM
|
|
|
|
CP0424761
|
(Z)-1-(2-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23ClN4O
|
1
|
| 1 |
EC50 = 57.2 nM
|
|
|
|
CP0861683
|
(Z)-1-(4-fluorophenyl)-4-(4-pyridin-2-ylpiperazin-1-yl)butan-1-one oxime
Show/Hide
|
C19H23FN4O
|
1
|
| 1 |
EC50 = 59.3 nM
|
|
|
|
CP0378824
|
N-(4-fluoro-2-methylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C19H22FN3O2
|
2
|
| 1 |
EC50 = 60 nM
|
|
|
| 2 |
Ki = 405 nM
|
|
|
|
CP0456872
|
N-(2-chloro-6-methylphenyl)-2-(4-pyridin-2-ylpiperidin-1-yl)acetamide
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0395340
|
(Z)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23FN4O
|
2
|
| 1 |
EC50 = 60.2 nM
|
|
|
| 2 |
Ki = 6.4 nM
|
|
|
|
CP0374846
|
(Z)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)propan-1-one O-methyloxime
Show/Hide
|
C20H26N4O
|
2
|
| 1 |
EC50 = 61 nM
|
|
|
| 2 |
Ki = 32.1 nM
|
|
|
|
CP0453676
|
N-(3-chlorophenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C18H20ClN3O2
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0453674
|
3-chloro-4-fluoro-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C18H19ClFN3O2
|
1
|
| 1 |
EC50 = 63 nM
|
|
|
|
CP0408464
|
(E)-4-[1-methoxyimino-3-(4-pyridin-2-ylpiperazin-1-yl)propyl]benzonitrile
Show/Hide
|
C20H23N5O
|
1
|
| 1 |
EC50 = 63.7 nM
|
|
|
|
CP0453357
|
2-((R)-2-Methyl-4-pyridin-2-yl-piperazin-1-ylmethyl)-1H-benzoimidazole
Show/Hide
|
C18H21N5
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0378826
|
N-(4-bromo-2-methylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C19H22BrN3O2
|
1
|
| 1 |
EC50 = 66 nM
|
|
|
|
CP0503098
|
3-ethenyl-N-[[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]methyl]benzamide
Show/Hide
|
C20H23N3O2
|
1
|
| 1 |
EC50 = 68 nM
|
|
|
|
CP0856098
|
(E)-1-phenyl-3-(4-pyrimidin-2-ylpiperazin-1-yl)propan-1-oxime
Show/Hide
|
C17H21N5O
|
1
|
| 1 |
EC50 = 69 nM
|
|
|
|
CP0445991
|
2-[4-(4-hydroxyphenyl)piperidin-1-yl]-N-(m-tolyl)acetamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0433495
|
(E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(o-tolyl)propan-1-one O-methyloxime
Show/Hide
|
C20H26N4O
|
2
|
| 1 |
EC50 = 74 nM
|
|
|
| 2 |
Ki = 11.4 nM
|
|
|
|
CP0458099
|
(Z)-1-(3,5-dimethylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C21H28N4O
|
1
|
| 1 |
EC50 = 74.7 nM
|
|
|
|
CP0378827
|
2-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)-N-(3-trifluoromethylphenyl)acetamide
Show/Hide
|
C19H20F3N3O2
|
1
|
| 1 |
EC50 = 76 nM
|
|
|
|
CP0374857
|
(E)-1-phenyl-3-(4-thiazol-2-ylpiperazin-1-yl)propanon-1-one O-ethyloxime
Show/Hide
|
C18H24N4OS
|
2
|
| 1 |
EC50 = 81.8 nM
|
|
|
| 2 |
Ki = 168 nM
|
|
|
|
CP0379536
|
(Z)-1-(4-bromophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23BrN4O
|
1
|
| 1 |
EC50 = 82 nM
|
|
|
|
CP0408476
|
(E)-1-(4-chlorophenyl)-3-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4']bipyridinyl-1'-yl)propan-1-one O-methyl-oxime
Show/Hide
|
C20H24ClN3O2
|
1
|
| 1 |
EC50 = 84 nM
|
|
|
|
CP0382337
|
N-(4-fluorophenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C18H20FN3O2
|
1
|
| 1 |
EC50 = 85 nM
|
|
|
|
CP0499935
|
4-methyl-N-(1-oxy-3',4',5',6'-tetrahydro-2-H-[2,4'-bipyridine]-1'-ylmethyl)-3-trifluoromethylbenzamide
Show/Hide
|
C20H22F3N3O2
|
1
|
| 1 |
EC50 = 85 nM
|
|
|
|
CP0450413
|
2-[4-(2-Methylsulfanyl-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C19H22N4S
|
1
|
| 1 |
EC50 = 86 nM
|
|
|
|
CP0408371
|
(E)-1-(3-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23ClN4O
|
2
|
| 1 |
EC50 = 88.9 nM
|
|
|
| 2 |
Ki = 13.5 nM
|
|
|
|
CP0283744
|
ABT-670
Show/Hide
|
C19H23N3O2
|
2
|
| 1 |
EC50 = 89 nM
|
|
|
| 2 |
Ki = 1445 nM
|
|
|
|
CP0502736
|
3,5-dimethyl-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0522364
|
(Z)-1-(3,4-dimethylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C21H28N4O
|
1
|
| 1 |
EC50 = 91 nM
|
|
|
|
CP0442719
|
N-(3-ethylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 = 95 nM
|
|
|
|
CP0408420
|
(6aR,12bS)-(+)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline
Show/Hide
|
C16H15NO3
|
1
|
| 1 |
EC50 = 95 nM
|
|
|
|
CP0419605
|
(Z)-1-(3-chloro-4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H22ClFN4O
|
1
|
| 1 |
EC50 = 95 nM
|
|
|
|
CP0277559
|
N-(4-bromo-3-methylphenyl)-2-[4-(2-cyanophenyl)piperazin-1-yl]acetamide
Show/Hide
|
C20H21BrN4O
|
1
|
| 1 |
EC50 = 96 nM
|
|
|
|
CP0407233
|
(Z)-1-(4-chloro-3-methylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C20H25ClN4O
|
2
|
| 1 |
EC50 = 98 nM
|
|
|
| 2 |
Ki = 11.6 nM
|
|
|
|
CP0390665
|
(Z)-1-(4-chlorophenyl)-3-(2-methyl-4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C20H25ClN4O
|
1
|
| 1 |
EC50 = 99 nM
|
|
|
|
CP0502734
|
N-(3-methylsulfanylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C19H23N3O2S
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0485861
|
2-[4-(2-Methoxy-phenyl)-piperidin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C20H23N3O
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0378823
|
N-(2,4-difluorophenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C18H19F2N3O2
|
1
|
| 1 |
EC50 = 103 nM
|
|
|
|
CP0379538
|
(E)-1-(3,4-dimethylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C21H28N4O
|
2
|
| 1 |
EC50 = 108 nM
|
|
|
| 2 |
Ki = 27.5 nM
|
|
|
|
CP0502053
|
(E)-1-phenyl-3-(4-phenylpiperazin-1-yl)propan-1-one O-ethyloxime
Show/Hide
|
C21H27N3O
|
1
|
| 1 |
EC50 = 109 nM
|
|
|
|
CP0061859
|
(+/-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline
Show/Hide
|
C16H15NO3
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0406708
|
N-(2-ethyl-6-methylphenyl)-2-(4-pyridin-2-ylpiperidin-1-yl)acetamide
Show/Hide
|
C21H27N3O
|
1
|
| 1 |
EC50 = 111 nM
|
|
|
|
CP0379535
|
(Z)-1-(3-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23ClN4O
|
1
|
| 1 |
EC50 = 113 nM
|
|
|
|
CP0445986
|
N-[[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]methyl]naphthalene-2-carboxamide
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
EC50 = 115 nM
|
|
|
|
CP0374864
|
2-hydroxy-1-pyridin-3-yl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C18H23N5O2
|
1
|
| 1 |
EC50 = 123 nM
|
|
|
|
CP0382336
|
N-(5-chloro-2-methylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C19H22ClN3O2
|
1
|
| 1 |
EC50 = 126 nM
|
|
|
|
CP0442718
|
N-(2-methyl-5-nitrophenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C19H22N4O4
|
1
|
| 1 |
EC50 = 134 nM
|
|
|
|
CP0433042
|
2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]-N-[3-(trifluoromethoxy)phenyl]acetamide
Show/Hide
|
C19H20F3N3O3
|
1
|
| 1 |
EC50 = 135 nM
|
|
|
|
CP0428205
|
(E)-1-(4-chloro-3-methylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C20H25ClN4O
|
1
|
| 1 |
EC50 = 135 nM
|
|
|
|
CP0494784
|
2-[4-(3-Methanesulfonyl-pyridin-2-yl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C18H21N5O2S
|
1
|
| 1 |
EC50 = 136 nM
|
|
|
|
CP0403315
|
(E)-2-[4-(3-ethoxyimino-3-phenylpropyl)piperazin-1-yl]nicotinonitrile
Show/Hide
|
C21H25N5O
|
1
|
| 1 |
EC50 = 139 nM
|
|
|
|
CP0528490
|
2-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)-N-(2,4,6trichlorophenyl)acetamide
Show/Hide
|
C18H18Cl3N3O
|
1
|
| 1 |
EC50 = 145 nM
|
|
|
|
CP0374888
|
(E)-1-(3-chloro-4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H22ClFN4O
|
2
|
| 1 |
EC50 = 148 nM
|
|
|
| 2 |
Ki = 71.2 nM
|
|
|
|
CP0442716
|
3-methoxy-4-chloro-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C19H22ClN3O3
|
1
|
| 1 |
EC50 = 159 nM
|
|
|
|
CP0403493
|
N-(3,5-dichlorophenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C18H19Cl2N3O2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0526886
|
N-(3-fluorophenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C18H20FN3O2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0395338
|
(E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-isopropyloxime
Show/Hide
|
C21H28N4O
|
1
|
| 1 |
EC50 = 164 nM
|
|
|
|
CP0384369
|
2-(4-phenylpiperidin-1-yl)-N-(m-tolyl)acetamide
Show/Hide
|
C20H24N2O
|
3
|
| 1 |
EC50 = 170 nM
|
|
|
| 2 |
Ki = 1.4 nM
|
|
|
| 3 |
Ki = 25.8 nM
|
|
|
|
CP0559594
|
3-chloro-N-(1-oxy-3',4',5',6'-tetrhydro-2'H-[2,4'-bipyridine]-1'ylmethyl)-4-trifluoromethylbenzamide
Show/Hide
|
C19H19ClF3N3O3
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0374887
|
(E)-1-(3,5-dimethylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C21H28N4O
|
1
|
| 1 |
EC50 = 175 nM
|
|
|
|
CP0499928
|
N-(2,3-dichlorophenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C18H19Cl2N3O2
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
|
CP0408472
|
(E)-1-(4-bromophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C19H23BrN4O
|
1
|
| 1 |
EC50 = 183 nM
|
|
|
|
CP0395330
|
(E)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2'H-[2,4']bipyridinyl-1'-yl)propan-1-one O-methyloxime
Show/Hide
|
C20H24ClN3O
|
2
|
| 1 |
EC50 = 195 nM
|
|
|
| 2 |
Ki = 134 nM
|
|
|
|
CP0424767
|
(E)-1-(4-chlorophenyl)-2-methoxy-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime
Show/Hide
|
C20H25ClN4O2
|
1
|
| 1 |
EC50 = 195 nM
|
|
|
|
CP0437337
|
2-methoxy-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)-benzamide
Show/Hide
|
C21H26N2O2
|
2
|
| 1 |
EC50 = 206 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0394645
|
1-(4-chlorophenyl)-2-(methoxyaminomethyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime
Show/Hide
|
C21H28ClN5O2
|
2
|
| 1 |
EC50 = 206 nM
|
|
|
| 2 |
Ki = 120 nM
|
|
|
|
CP0510445
|
2-(4-Phenyl-3,6-dihydro-2H-pyridin-1-ylmethyl)-1H-benzoimidazole
Show/Hide
|
C19H19N3
|
1
|
| 1 |
EC50 = 228 nM
|
|
|
|
CP0439624
|
(6aS,12bR)-(-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline
Show/Hide
|
C16H15NO3
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0526887
|
N-(4-chloro-2,6-dimethylphenyl)-2-(4-pyridin-2-ylpiperidin-1-yl)acetamide
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
EC50 = 240 nM
|
|
|
|
CP0408474
|
(E)-1-(2,4-dichlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C19H22Cl2N4O
|
1
|
| 1 |
EC50 = 249 nM
|
|
|
|
CP0239544
|
1-(N-benzylanilino)-3-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]urea
Show/Hide
|
C28H35N5O2
|
2
|
| 1 |
EC50 = 250 nM
|
|
|
| 2 |
IC50 = 450 nM
|
|
|
|
CP0386019
|
(E)-3-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-1-phenylpropanon-1-one O-ethyloxime
Show/Hide
|
C21H28N4O
|
1
|
| 1 |
EC50 = 253 nM
|
|
|
|
CP0495961
|
N-(2-fluorophenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C18H20FN3O2
|
1
|
| 1 |
EC50 = 270 nM
|
|
|
|
CP0384421
|
(Z)-1-(4-chlorophenyl)-2-methoxy-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime
Show/Hide
|
C20H25ClN4O2
|
1
|
| 1 |
EC50 = 285 nM
|
|
|
|
CP0499936
|
N-cyclohexyl-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C18H27N3O2
|
1
|
| 1 |
EC50 = 294 nM
|
|
|
|
CP0379537
|
(Z)-1-(2,4-dichlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C19H22Cl2N4O
|
1
|
| 1 |
EC50 = 296 nM
|
|
|
|
CP0395336
|
(E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-propyloxime
Show/Hide
|
C21H28N4O
|
1
|
| 1 |
EC50 = 320 nM
|
|
|
|
CP0395004
|
3-ethoxy-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C20H25N3O3
|
1
|
| 1 |
EC50 = 324 nM
|
|
|
|
CP0394655
|
(E)-1-(4-chlorophenyl)-3-(2-methyl-4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-methyloxime
Show/Hide
|
C20H25ClN4O
|
2
|
| 1 |
EC50 = 333 nM
|
|
|
| 2 |
Ki = 67.1 nM
|
|
|
|
CP0458090
|
(E)3-[4-(2-methoxyphenyl)piperazin-1-yl]-1-phenylpropan-1-one O-ethyloxime
Show/Hide
|
C22H29N3O2
|
1
|
| 1 |
EC50 = 338 nM
|
|
|
|
CP0445984
|
N-(3-methylphenyl)-2-[4-(2-methylphenyl)piperidin-1-yl]acetamide
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
EC50 = 340 nM
|
|
|
|
CP0455560
|
N-(2-methoxy-6-methylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C20H25N3O3
|
1
|
| 1 |
EC50 = 340 nM
|
|
|
|
CP0438120
|
1-(N-benzyl-4-fluoroanilino)-3-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]urea
Show/Hide
|
C28H34FN5O2
|
2
|
| 1 |
EC50 = 340 nM
|
|
|
| 2 |
IC50 = 49 nM
|
|
|
|
CP0393866
|
(Z)-1-(3,4-dichlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C19H22Cl2N4O
|
1
|
| 1 |
EC50 = 341 nM
|
|
|
|
CP0437288
|
N-(2,6-dichloro-3-methylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C19H21Cl2N3O2
|
1
|
| 1 |
EC50 = 346 nM
|
|
|
|
CP0451711
|
N-(2,6-dimethylphenyl)-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 = 346 nM
|
|
|
|
CP0408463
|
(E)-3-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-phenylpropan-1-oneO-ethyloxime
Show/Hide
|
C23H31N3O2
|
1
|
| 1 |
EC50 = 347 nM
|
|
|
|
CP0497175
|
(E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-allyloxime
Show/Hide
|
C21H26N4O
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0445987
|
2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]-N-(3-phenylphenyl)acetamide
Show/Hide
|
C24H25N3O2
|
1
|
| 1 |
EC50 = 360 nM
|
|
|
|
CP0395337
|
(E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one O-butyloxime
Show/Hide
|
C22H30N4O
|
1
|
| 1 |
EC50 = 382 nM
|
|
|
|
CP0372267
|
4,6-Dibromo-2-(4-pyridin-2-yl-piperazin-1-ylmethyl)-1H-benzoimidazole
Show/Hide
|
C17H17Br2N5
|
1
|
| 1 |
EC50 = 416 nM
|
|
|
|
CP0403494
|
2-[4-(2-methoxyphenyl)piperidin-1-yl]-N-(m-tolyl)acetamide
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0374863
|
1-(4-chlorophenyl)-2-methyl-3-(4-pyridin-2-ylpiperazin-1-yl)-propanon-1-one O-methyloxime
Show/Hide
|
C20H25ClN4O
|
2
|
| 1 |
EC50 = 459 nM
|
|
|
| 2 |
Ki = 346 nM
|
|
|
|
CP0455559
|
N-[4-fluoro-2-(trifluoromethyl)phenyl]-2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C19H19F4N3O2
|
1
|
| 1 |
EC50 = 473 nM
|
|
|
|
CP0853248
|
(E)-1-(4-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C18H21ClN4O
|
1
|
| 1 |
EC50 = 475 nM
|
|
|
|
CP0148103
|
1-[N-[(4-fluorophenyl)methyl]anilino]-3-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]urea
Show/Hide
|
C28H34FN5O2
|
2
|
| 1 |
EC50 = 500 nM
|
|
|
| 2 |
IC50 = 620 nM
|
|
|
|
CP0445988
|
2-[4-(3-fluorophenyl)piperidin-1-yl]-N-(m-tolyl)acetamide
Show/Hide
|
C20H23FN2O
|
1
|
| 1 |
EC50 = 512 nM
|
|
|
|
CP0406710
|
N-[[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]methyl]benzamide
Show/Hide
|
C18H21N3O2
|
1
|
| 1 |
EC50 = 532 nM
|
|
|
|
CP0408475
|
(E)-1-(3,4-dichlorophenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)-propan-1-one O-methyloxime
Show/Hide
|
C19H22Cl2N4O
|
2
|
| 1 |
EC50 = 542 nM
|
|
|
| 2 |
Ki = 6.4 nM
|
|
|
|
CP0420190
|
2-[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]-N-(3-propan-2-yloxyphenyl)acetamide
Show/Hide
|
C21H27N3O3
|
1
|
| 1 |
EC50 = 555 nM
|
|
|
|
CP0891812
|
(E)-1-(4-fluorophenyl)-3-(4-(3-isopropoxyphenyl)piperazin-1-yl)propan-1-one O-methyl oxime
Show/Hide
|
C23H30FN3O2
|
1
|
| 1 |
EC50 = 594 nM
|
|
|
|
CP0862485
|
(Z)-1-(4-fluorophenyl)-3-(4-(3-isopropoxyphenyl)piperazin-1-yl)propan-1-one O-methyl oxime
Show/Hide
|
C23H30FN3O2
|
1
|
| 1 |
EC50 = 601 nM
|
|
|
|
CP0408471
|
(E)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2'H-[2,3']bipyridinyl-1'-yl)propan-1-one O-methyloxime
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
EC50 = 606 nM
|
|
|
|
CP0441840
|
(E)-1-phenyl-3-(4-pyrimidin-2-ylpiperazin-1-yl)propanon-1-one-O-ethyloxime
Show/Hide
|
C19H25N5O
|
1
|
| 1 |
EC50 = 615 nM
|
|
|
|
CP0395003
|
3-methoxy-2-methyl-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C20H25N3O3
|
1
|
| 1 |
EC50 = 685 nM
|
|
|
|
CP0382335
|
3-cyano-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C19H20N4O2
|
1
|
| 1 |
EC50 = 840 nM
|
|
|
|
CP0528491
|
6-chloro-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)nicotinamide
Show/Hide
|
C17H19ClN4O2
|
1
|
| 1 |
EC50 = 1290 nM
|
|
|
|
CP0445990
|
3-chloro-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide
Show/Hide
|
C19H22ClN3O2
|
1
|
| 1 |
EC50 = 2460 nM
|
|
|
|
CP0432611
|
(E)-3-[4-(3-methoxyphenyl)piperazin-1-yl]-1-phenylpropan-1-one O-ethyloxime
Show/Hide
|
C22H29N3O2
|
1
|
| 1 |
EC50 = 2680 nM
|
|
|
|
CP0403492
|
N-[[4-(1-oxidopyridin-1-ium-2-yl)piperidin-1-yl]methyl]pyridine-2-carboxamide
Show/Hide
|
C17H20N4O2
|
1
|
| 1 |
EC50 = 3150 nM
|
|
|
|
CP0501106
|
1-(4-chlorophenyl)-2-isopropoxymethyl-3-(4-pyridin-2-ylpiperazin-1-yl)propanon-1-one O-methyloxime
Show/Hide
|
C23H31ClN4O2
|
1
|
| 1 |
EC50 = 3210 nM
|
|
|
|
CP0845750
|
(Z)-1-(4-fluorophenyl)-2-(4-pyridin-2-yl)ethanone oxime
Show/Hide
|
C17H19FN4O
|
1
|
| 1 |
EC50 = 4290 nM
|
|
|
|
CP0379506
|
2-(4-pyridin-2-ylpiperazin-1-ylmethyl)-3,4-dihydro-2H-naphthalen-1-one O-ethyloxime
Show/Hide
|
C22H28N4O
|
1
|
| 1 |
EC50 = 4760 nM
|
|
|
|
CP0849209
|
(E)-2-methoxy-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)-propan-1-one O-methyloxime
Show/Hide
|
C20H26N4O2
|
1
|
| 1 |
EC50 = 5370 nM
|
|
|
|
CP0008601
|
4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl)
Show/Hide
|
C21H23ClFNO2
|
3
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 2.3 nM
|
|
|
| 3 |
Ki = 5 nM
|
|
|
|
CP0082340
|
2-(4-Pyridin-4-yl-piperazin-1-yl)-N-m-tolyl-acetamide
Show/Hide
|
C18H22N4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0140964
|
2-[4-(4-Bromo-2-cyano-phenyl)-piperazin-1-yl]-N-(4-bromo-3-methyl-phenyl)-acetamide
Show/Hide
|
C20H20Br2N4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0140966
|
2-[4-(4-Bromo-2-cyano-phenyl)-piperazin-1-yl]-N-(2,4,6-tribromo-3-methyl-phenyl)-acetamide
Show/Hide
|
C20H18Br4N4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0155036
|
2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide
Show/Hide
|
C19H22FN3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0276844
|
2-(4-Biphenyl-4-yl-piperazin-1-yl)-N-m-tolyl-acetamide
Show/Hide
|
C25H27N3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0277857
|
2-[4-(4-Benzyl-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide
Show/Hide
|
C26H29N3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0277858
|
2-[4-(4-Benzhydryl-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide
Show/Hide
|
C32H33N3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0302767
|
2-[4-(3-Methoxy-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0310037
|
2-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0408470
|
(Z)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2'H-[2,4']bipyridinyl-1'-yl)propan-1-one O-methyloxime
Show/Hide
|
C20H24ClN3O
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 90 nM
|
|
|
|
CP0419599
|
(E)-3-[4-(4-Methoxyphenyl)piperazin-1-yl]-1-phenylpropan-1-one O-ethyloxime
Show/Hide
|
C22H29N3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0851022
|
(E)-1-(4-fluorophenyl)-2-(4-pyridin-2-yl)ethanone oxime
Show/Hide
|
C17H19FN4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0862522
|
(E)-1-(2-benzyloxy-5-methylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one oxime
Show/Hide
|
C26H30N4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0401629
|
2-[4-(2,5-Dimethyl-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C20H24N4
|
2
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
Ki = 3.8 nM
|
|
|
|
CP0052064
|
2-[4-(3,4-Dimethyl-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
Show/Hide
|
C20H24N4
|
2
|
| 1 |
IC50 = 5 nM
|
|
|
| 2 |
Ki = 1.5 nM
|
|
|
|
CP0429805
|
5-Methyl-1-[1-(3-methyl-benzyl)-piperidin-4-yl]-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C23H27N3O
|
1
|
| 1 |
Ki = 0.33 nM
|
|
|
|
CP0099175
|
N-[1-[(4-iodophenyl)methyl]piperidin-4-yl]-N-methyl-3-propan-2-yloxypyridin-2-amine
Show/Hide
|
C21H28IN3O
|
1
|
| 1 |
Ki = 0.3311 nM
|
|
|
|
CP0375516
|
1-Benzyl-4-(3-methyl-4-phenyl-pyrazol-1-yl)-piperidine
Show/Hide
|
C22H25N3
|
1
|
| 1 |
Ki = 0.39 nM
|
|
|
|
CP0046420
|
CAS_3853
Show/Hide
|
C18H19ClN4
|
2
|
| 1 |
Ki = 0.43 nM
|
|
|
| 2 |
Ki = 2.239 nM
|
|
|
|
CP0437134
|
1-[1-(3-Chloro-benzyl)-piperidin-4-yl]-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
Ki = 0.46 nM
|
|
|
|
CP0374884
|
5-Methyl-1-(1-phenethyl-piperidin-4-yl)-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C23H27N3O
|
1
|
| 1 |
Ki = 0.56 nM
|
|
|
|
CP0467016
|
1-(1-Benzyl-piperidin-4-yl)-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H25N3O
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0375779
|
N-[4-[4-(2-methylsulfanylphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide
Show/Hide
|
C23H29N5OS
|
1
|
| 1 |
Ki = 0.63 nM
|
|
|
|
CP0377325
|
1-[1-(3-Methoxy-benzyl)-piperidin-4-yl]-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
Ki = 0.64 nM
|
|
|
|
CP0424155
|
1-(1-Benzyl-piperidin-4-yl)-4-(4-chloro-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
Ki = 0.71 nM
|
|
|
|
CP0512281
|
1-(1-Benzyl-piperidin-4-yl)-3,5-dimethyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C23H27N3O
|
1
|
| 1 |
Ki = 0.75 nM
|
|
|
|
CP0449085
|
1-(1-Benzyl-piperidin-4-yl)-3-methyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H25N3O
|
1
|
| 1 |
Ki = 0.84 nM
|
|
|
|
CP0378625
|
1-(1-Benzyl-piperidin-4-yl)-5-ethyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C23H27N3O
|
1
|
| 1 |
Ki = 0.86 nM
|
|
|
|
CP0339664
|
CHEBI:64217
Show/Hide
|
C21H26ClN3O2
|
1
|
| 1 |
Ki = 0.86 nM
|
|
|
|
CP0383198
|
3-[4-(5-Methyl-2-oxo-4-phenyl-2,3-dihydro-imidazol-1-yl)-piperidin-1-ylmethyl]-benzonitrile
Show/Hide
|
C23H24N4O
|
1
|
| 1 |
Ki = 0.96 nM
|
|
|
|
CP0232092
|
1-[3-(4-butylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C21H32N2O
|
1
|
| 1 |
Ki = 0.9772 nM
|
|
|
|
CP0420764
|
4-(1-Benzyl-piperidin-4-yl)-6-(4-chloro-phenyl)-pyrimidin-2-ylamine
Show/Hide
|
C22H23ClN4
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0378670
|
1-(1-Benzyl-piperidin-4-yl)-5-methyl-4-thiophen-2-yl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C20H23N3OS
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0455116
|
1-(1-Benzyl-piperidin-4-yl)-5-methyl-4-p-tolyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C23H27N3O
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0455407
|
1-(1-Benzyl-piperidin-4-yl)-4-(2-chloro-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0372647
|
4-[5-(4-Chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-1-phenethyl-piperidine
Show/Hide
|
C23H26ClN3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0492442
|
3-[4-(3-Methyl-4-phenyl-pyrazol-1-yl)-piperidin-1-ylmethyl]-benzonitrile
Show/Hide
|
C23H24N4
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0116478
|
1-[3-(4-benzylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C24H30N2O
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0436601
|
2-[1-(4-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole
Show/Hide
|
C19H17ClN2S
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0448500
|
1-[1-(4-Chloro-benzyl)-piperidin-4-yl]-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0036418
|
3-[4-(4-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H22N4O
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0411640
|
1-[3-(4-pentylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C22H34N2O
|
1
|
| 1 |
Ki = 1.38 nM
|
|
|
|
CP0393890
|
1-Benzyl-4-[5-(4-chloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-piperidine
Show/Hide
|
C23H26ClN3
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0394248
|
1-Benzyl-4-[5-(4-chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-piperidine
Show/Hide
|
C22H24ClN3
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0384375
|
N-(3-methylphenyl)-2-(4-naphthalen-1-ylpiperazin-1-yl)acetamide
Show/Hide
|
C23H25N3O
|
2
|
| 1 |
Ki = 1.65 nM
|
|
|
| 2 |
Ki = 28.4 nM
|
|
|
|
CP0373007
|
1-(1-Benzyl-piperidin-4-yl)-4-(4-fluoro-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H24FN3O
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0483626
|
3-(4-Phenethyl-piperidin-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C21H25N3
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0384672
|
N-(3-methylphenyl)-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide
Show/Hide
|
C18H22N4O
|
2
|
| 1 |
Ki = 1.89 nM
|
|
|
| 2 |
Ki = 212 nM
|
|
|
|
CP0489929
|
1-[3-(4-phenylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C23H28N2O
|
1
|
| 1 |
Ki = 1.95 nM
|
|
|
|
CP0049653
|
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-((R)-2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
|
C23H29N3O
|
1
|
| 1 |
Ki = 1.995 nM
|
|
|
|
CP0460142
|
1-(1-Cyclohexylmethyl-piperidin-4-yl)-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H31N3O
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0402244
|
2-(4-Phenethyl-piperidin-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C21H25N3
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0045034
|
N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide
Show/Hide
|
C23H29N5O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0404428
|
1-[1-(2-Chloro-benzyl)-piperidin-4-yl]-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0393635
|
1-[3-[4-(2-phenylethyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C25H32N2O
|
1
|
| 1 |
Ki = 2.138 nM
|
|
|
|
CP0384370
|
N-(3-ethylphenyl)-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide
Show/Hide
|
C19H24N4O
|
2
|
| 1 |
Ki = 2.23 nM
|
|
|
| 2 |
Ki = 67.9 nM
|
|
|
|
CP0427419
|
2-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)H-pyrazolo[1,5-a]pyridine
Show/Hide
|
C19H22N4O
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0081150
|
4-[3-(4-Chloro-phenyl)-4-methyl-isoxazol-5-yl]-1-phenethyl-piperidine
Show/Hide
|
C23H25ClN2O
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0375430
|
1-Benzyl-4-(5-methyl-4-phenyl-pyrazol-1-yl)-piperidine
Show/Hide
|
C22H25N3
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0133352
|
(2S)-2-[(5-chloro-2-methoxyphenoxy)methyl]-4-[(4-chlorophenyl)methyl]morpholine
Show/Hide
|
C19H21Cl2NO3
|
1
|
| 1 |
Ki = 2.818 nM
|
|
|
|
CP0232093
|
1-[3-(4-phenylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C22H27N3O
|
1
|
| 1 |
Ki = 2.884 nM
|
|
|
|
CP0393905
|
4-(4-Methyl-5-phenyl-1H-pyrazol-3-yl)-1-phenethyl-1,2,3,6-tetrahydro-pyridine
Show/Hide
|
C23H25N3
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0437126
|
1-(3-Chloro-benzyl)-4-(5-methyl-4-phenyl-pyrazol-1-yl)-piperidine
Show/Hide
|
C22H24ClN3
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0506670
|
1-(3-Chloro-benzyl)-4-(3-methyl-4-phenyl-pyrazol-1-yl)-piperidine
Show/Hide
|
C22H24ClN3
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0099174
|
4-[5-(4-Chloro-phenyl)-4-methyl-isoxazol-3-yl]-1-phenethyl-piperidine
Show/Hide
|
C23H25ClN2O
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0393889
|
1-(4-Chloro-benzyl)-4-[3-(4-chloro-phenyl)-isoxazol-5-yl]-piperidine
Show/Hide
|
C21H20Cl2N2O
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0233820
|
2-benzyl-6-(3-methoxyphenyl)-3,4-dihydro-1H-isoquinoline
Show/Hide
|
C23H23NO
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0378647
|
1-[3-[4-(5-hydroxypentyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C22H34N2O2
|
1
|
| 1 |
Ki = 4.365 nM
|
|
|
|
CP0392993
|
1-(1-Benzyl-piperidin-4-yl)-5-methyl-3,4-diphenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C28H29N3O
|
1
|
| 1 |
Ki = 4.5 nM
|
|
|
|
CP0406711
|
1-(1-Benzyl-piperidin-4-yl)-5-methyl-4-pyridin-2-yl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C21H24N4O
|
1
|
| 1 |
Ki = 4.5 nM
|
|
|
|
CP0453196
|
4-(4-Chloro-phenyl)-5-methyl-6-(1-phenethyl-piperidin-4-yl)-pyrimidin-2-ylamine
Show/Hide
|
C24H27ClN4
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
|
CP0461030
|
1-Benzyl-4-(4-methyl-5-phenyl-1H-pyrazol-3-yl)-piperidine
Show/Hide
|
C22H25N3
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
|
CP0404187
|
2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-benzothiazole
Show/Hide
|
C19H18N2S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0391270
|
N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]adamantane-1-carboxamide
Show/Hide
|
C23H32ClN3O
|
1
|
| 1 |
Ki = 5.012 nM
|
|
|
|
CP0411285
|
3-(1-octylpyrrolidin-3-yl)phenol
Show/Hide
|
C18H29NO
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0409440
|
3-[4-(5-Methyl-4-phenyl-pyrazol-1-yl)-piperidin-1-ylmethyl]-benzonitrile
Show/Hide
|
C23H24N4
|
1
|
| 1 |
Ki = 5.2 nM
|
|
|
|
CP0403521
|
1-(1-Benzyl-piperidin-4-yl)-4-(3-chloro-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
Ki = 5.2 nM
|
|
|
|
CP0393633
|
1-[3-(4-propylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C20H30N2O
|
1
|
| 1 |
Ki = 5.248 nM
|
|
|
|
CP0169831
|
4-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-1-phenethyl-piperidine
Show/Hide
|
C22H24ClN3
|
1
|
| 1 |
Ki = 5.5 nM
|
|
|
|
CP0416338
|
1-(1-Benzyl-piperidin-4-yl)-3-isoquinolin-1-yl-urea
Show/Hide
|
C22H24N4O
|
1
|
| 1 |
Ki = 5.5 nM
|
|
|
|
CP0448388
|
5-Methyl-4-phenyl-1-[1-(3-phenyl-propyl)-piperidin-4-yl]-1,3-dihydro-imidazol-2-one
Show/Hide
|
C24H29N3O
|
1
|
| 1 |
Ki = 5.5 nM
|
|
|
|
CP0384667
|
N-(3-methylphenyl)-2-(4-pyrimidin-2-ylpiperazin-1-yl)acetamide
Show/Hide
|
C17H21N5O
|
2
|
| 1 |
Ki = 5.66 nM
|
|
|
| 2 |
Ki = 318 nM
|
|
|
|
CP0393162
|
3-[2-[4-[(E)-2-phenylethenyl]-3,6-dihydro-2H-pyridin-1-yl]ethyl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C22H23N3
|
1
|
| 1 |
Ki = 6.5 nM
|
|
|
|
CP0052067
|
2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyrazolo[1,5-a]pyridine
Show/Hide
|
C18H19ClN4
|
1
|
| 1 |
Ki = 6.8 nM
|
|
|
|
CP0384376
|
N-(3-methylphenyl)-2-[4-(5-methylpyridin-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C20H25N3O
|
2
|
| 1 |
Ki = 6.87 nM
|
|
|
| 2 |
Ki = 41.7 nM
|
|
|
|
CP0453211
|
2-(1H-Pyrrolo[2,3-b]pyridin-3-ylmethyl)-1,2,3,4-tetrahydro-isoquinoline
Show/Hide
|
C17H17N3
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0091842
|
N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-2,2-dimethylbutanamide
Show/Hide
|
C18H28ClN3O
|
1
|
| 1 |
Ki = 7.943 nM
|
|
|
|
CP0391426
|
N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-1-methylcyclohexane-1-carboxamide
Show/Hide
|
C20H30ClN3O
|
1
|
| 1 |
Ki = 7.943 nM
|
|
|
|
CP0427324
|
N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-2,2-dimethylpentanamide
Show/Hide
|
C19H30ClN3O
|
1
|
| 1 |
Ki = 7.943 nM
|
|
|
|
CP0387456
|
2-[1-[(1-methylbenzimidazol-2-yl)methyl]piperidin-4-yl]-1,3-benzothiazole
Show/Hide
|
C21H22N4S
|
1
|
| 1 |
Ki = 7.943 nM
|
|
|
|
CP0436906
|
2-[1-(3-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole
Show/Hide
|
C19H17ClN2S
|
1
|
| 1 |
Ki = 8.1 nM
|
|
|
|
CP0414228
|
N-[(6,6-diphenyl-1,4-dioxan-2-yl)methyl]-2-(2-methoxyphenoxy)ethanamine
Show/Hide
|
C26H29NO4
|
1
|
| 1 |
Ki = 8.318 nM
|
|
|
|
CP0464222
|
5-Chloro-2-[1-(4-chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzooxazole
Show/Hide
|
C19H16Cl2N2O
|
1
|
| 1 |
Ki = 8.4 nM
|
|
|
|
CP0406327
|
1-Benzyl-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine
Show/Hide
|
C21H22ClN3
|
1
|
| 1 |
Ki = 9.1 nM
|
|
|
|
CP0408909
|
N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-1-methylcyclohexane-1-carboxamide
Show/Hide
|
C22H34ClN3O
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0025667
|
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
|
C18H19ClN4
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0487032
|
4-(5-Cyclohexyl-1H-pyrazol-3-yl)-1-phenethyl-piperidine
Show/Hide
|
C22H31N3
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0454722
|
5-Chloro-2-[1-(4-chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-1H-benzoimidazole
Show/Hide
|
C19H17Cl2N3
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0375428
|
1-Benzyl-4-(5-phenyl-1H-pyrazol-3-yl)-piperidine
Show/Hide
|
C21H23N3
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0405451
|
3-(1-heptylpyrrolidin-3-yl)phenol
Show/Hide
|
C17H27NO
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0853848
|
3-hydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide
Show/Hide
|
C18H22BrNO
|
1
|
| 1 |
Ki = 11.3 nM
|
|
|
|
CP0404449
|
2-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H21ClN4
|
1
|
| 1 |
Ki = 11.7 nM
|
|
|
|
CP0394250
|
(Z)-1-(1-benzylpiperidin-4-yl)-3-(4-chlorophenyl)-3-hydroxyprop-2-en-1-one
Show/Hide
|
C21H22ClNO2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0437037
|
1-(1-Benzyl-piperidin-4-yl)-4-(4-methoxy-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0375780
|
N-[3-[4-(2-methylsulfanylphenyl)piperazin-1-yl]propyl]pyrazolo[1,5-a]pyridine-3-carboxamide
Show/Hide
|
C22H27N5OS
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0416633
|
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-(3-methylphenyl)acetamide
Show/Hide
|
C18H21ClN4O
|
2
|
| 1 |
Ki = 12.5 nM
|
|
|
| 2 |
Ki = 95 nM
|
|
|
|
CP0374718
|
N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C19H30ClN3O
|
1
|
| 1 |
Ki = 12.59 nM
|
|
|
|
CP0391425
|
N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-2,2-dimethylpentanamide
Show/Hide
|
C21H34ClN3O
|
1
|
| 1 |
Ki = 12.59 nM
|
|
|
|
CP0469228
|
N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C20H33N3O2
|
1
|
| 1 |
Ki = 12.59 nM
|
|
|
|
CP0374265
|
4-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-1-cyclohexylmethyl-piperidine
Show/Hide
|
C21H28ClN3
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0518040
|
3-(1-decylpyrrolidin-3-yl)phenol
Show/Hide
|
C20H33NO
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0448976
|
1-Benzyl-4-(5-phenyl-pyrazol-1-yl)-piperidine
Show/Hide
|
C21H23N3
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0432424
|
N-[4-[4-(4-chloro-2-methoxyphenyl)piperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C20H32ClN3O2
|
1
|
| 1 |
Ki = 15.85 nM
|
|
|
|
CP0515986
|
N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-2,2-dimethylbutanamide
Show/Hide
|
C20H32ClN3O
|
1
|
| 1 |
Ki = 15.85 nM
|
|
|
|
CP0420841
|
2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-5-chloro-benzooxazole
Show/Hide
|
C19H17ClN2O
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0495061
|
1-Benzyl-4-(5-methyl-4-phenyl-[1,2,3]triazol-1-yl)-piperidine
Show/Hide
|
C21H24N4
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0432236
|
1-Benzyl-4-(4-methyl-5-phenyl-[1,2,3]triazol-1-yl)-piperidine
Show/Hide
|
C21H24N4
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0441597
|
1-(1-Benzyl-piperidin-4-yl)-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C21H23N3O
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0430826
|
1-Phenethyl-4-(5-thiophen-2-yl-1H-pyrazol-3-yl)-piperidine
Show/Hide
|
C20H23N3S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0406241
|
N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]adamantane-1-carboxamide
Show/Hide
|
C25H36ClN3O
|
1
|
| 1 |
Ki = 19.95 nM
|
|
|
|
CP0472845
|
1-[3-(4-benzylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C23H29N3O
|
1
|
| 1 |
Ki = 19.95 nM
|
|
|
|
CP0432438
|
1-(2-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine
Show/Hide
|
C21H21Cl2N3
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0430499
|
5-Chloro-2-[1-(4-chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole
Show/Hide
|
C19H16Cl2N2S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0424550
|
2-[5-(1-Phenethyl-piperidin-4-yl)-2H-pyrazol-3-yl]-pyridine
Show/Hide
|
C21H24N4
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0404174
|
3-[5-(1-Phenethyl-piperidin-4-yl)-2H-pyrazol-3-yl]-pyridine
Show/Hide
|
C21H24N4
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0419180
|
1-Phenethyl-4-(5-phenyl-1H-pyrazol-3-yl)-piperazine
Show/Hide
|
C21H24N4
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0408943
|
N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-2,2-dimethylpropanamide
Show/Hide
|
C17H26ClN3O
|
1
|
| 1 |
Ki = 25.12 nM
|
|
|
|
CP0430505
|
2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-5-chloro-1H-benzoimidazole
Show/Hide
|
C19H18ClN3
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0421398
|
3-{2-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C20H24N4O
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0053493
|
(+)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4,9-dioxa-1-aza-phenanthren-6-ol
Show/Hide
|
C14H19NO3
|
1
|
| 1 |
Ki = 26.6 nM
|
|
|
|
CP0436445
|
1-Benzyl-4-(5-phenyl-tetrazol-2-yl)-piperidine
Show/Hide
|
C19H21N5
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0913527
|
7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C27H35N3O7
|
1
|
| 1 |
Ki = 27.2 nM
|
|
|
|
CP0451508
|
N-[2-[bis(4-fluorophenyl)methylsulfanyl]ethyl]-3-phenylpropan-1-amine
Show/Hide
|
C24H25F2NS
|
1
|
| 1 |
Ki = 28.1 nM
|
|
|
|
CP0393626
|
1-[3-[4-(2-phenylethyl)piperazin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C24H31N3O
|
1
|
| 1 |
Ki = 28.84 nM
|
|
|
|
CP0127400
|
(-)-Pramipexole
Show/Hide
|
C10H17N3S
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0392502
|
2-[2-(4-Styryl-3,6-dihydro-2H-pyridin-1-yl)-ethyl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C22H23N3
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0483245
|
N-ethyl-N-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C25H32ClFN4OS
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0913681
|
7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)quinolin-2(1H)-one oxalate
Show/Hide
|
C26H31N3O7
|
1
|
| 1 |
Ki = 30.1 nM
|
|
|
|
CP0453845
|
N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-2,2-dimethylhexanamide
Show/Hide
|
C20H32ClN3O
|
1
|
| 1 |
Ki = 31.62 nM
|
|
|
|
CP0505515
|
N-[4-[4-(4-bromophenyl)piperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C19H30BrN3O
|
1
|
| 1 |
Ki = 31.62 nM
|
|
|
|
CP0887640
|
7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)quinolin-2(1H)-one oxalate
Show/Hide
|
C27H32FN3O7
|
1
|
| 1 |
Ki = 31.9 nM
|
|
|
|
CP0492208
|
1-Benzyl-4-(4-phenyl-[1,2,3]triazol-1-yl)-piperidine
Show/Hide
|
C20H22N4
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0384372
|
N-(3-methylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propanamide
Show/Hide
|
C19H24N4O
|
2
|
| 1 |
Ki = 32.2 nM
|
|
|
| 2 |
Ki = 297 nM
|
|
|
|
CP0384371
|
N-(3-methylphenyl)-3-(4-pyrimidin-2-ylpiperazin-1-yl)propanamide
Show/Hide
|
C18H23N5O
|
2
|
| 1 |
Ki = 33 nM
|
|
|
| 2 |
Ki = 526 nM
|
|
|
|
CP0378669
|
1-Benzoyl-3-(1-benzyl-piperidin-4-yl)-urea
Show/Hide
|
C20H23N3O2
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0410033
|
3-[2-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C20H21N3
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0495774
|
3-((4-(4-chlorophenyl)-4-methoxypiperidin-1-yl)methyl)-1H-indole
Show/Hide
|
C21H23ClN2O
|
1
|
| 1 |
Ki = 34.1 nM
|
|
|
|
CP0396051
|
2-[2-[(6,6-diphenyl-1,4-dioxan-2-yl)methylamino]ethoxy]phenol
Show/Hide
|
C25H27NO4
|
1
|
| 1 |
Ki = 36.31 nM
|
|
|
|
CP0891096
|
7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C25H31N3O7
|
1
|
| 1 |
Ki = 38.5 nM
|
|
|
|
CP0429850
|
1-Benzyl-4-(4-phenyl-imidazol-1-yl)-piperidine
Show/Hide
|
C21H23N3
|
1
|
| 1 |
Ki = 40 nM
|
|
|
|
CP0860992
|
1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate
Show/Hide
|
C22H22INO6
|
1
|
| 1 |
Ki = 40.4 nM
|
|
|
|
CP0460885
|
1-(4-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-isoxazol-3-yl]-piperidine
Show/Hide
|
C21H20Cl2N2O
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0484578
|
2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-5-chloro-benzothiazole
Show/Hide
|
C19H17ClN2S
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0129619
|
N-[3-[2-[[(6S)-2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-propylamino]ethyl]-3-hydroxycyclobutyl]naphthalene-2-carboxamide
Show/Hide
|
C27H34N4O2S
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0420812
|
1-Benzyl-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-4-methyl-piperidine
Show/Hide
|
C22H24ClN3
|
1
|
| 1 |
Ki = 47 nM
|
|
|
|
CP0434427
|
2,2-dimethyl-N-[4-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]butyl]propanamide
Show/Hide
|
C20H30F3N3O
|
1
|
| 1 |
Ki = 50.12 nM
|
|
|
|
CP0389448
|
N-[(6,6-diphenyl-1,4-dioxan-2-yl)methyl]-2-[2-(methoxymethoxy)phenoxy]ethanamine
Show/Hide
|
C27H31NO5
|
1
|
| 1 |
Ki = 51.29 nM
|
|
|
|
CP0455488
|
4-[5-(1-Phenethyl-piperidin-4-yl)-2H-pyrazol-3-yl]-pyridine
Show/Hide
|
C21H24N4
|
1
|
| 1 |
Ki = 52 nM
|
|
|
|
CP0913682
|
7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)quinolin-2(1H)-one oxalate
Show/Hide
|
C25H29N3O7
|
1
|
| 1 |
Ki = 52.7 nM
|
|
|
|
CP0901061
|
1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate
Show/Hide
|
C22H23IN2O5
|
1
|
| 1 |
Ki = 53.4 nM
|
|
|
|
CP0100739
|
N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]pyrazolo[1,5-a]pyridine-3-carboxamide
Show/Hide
|
C22H27N5O2
|
1
|
| 1 |
Ki = 56 nM
|
|
|
|
CP0389575
|
4-(2-benzyl-3,4-dihydro-1H-isoquinolin-6-yl)morpholine
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 56 nM
|
|
|
|
CP0042927
|
7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}-3,4-dihydroquinolin-2(1H)-one
Show/Hide
|
C23H27Cl2N3O2
|
2
|
| 1 |
Ki = 57.1 nM
|
|
|
| 2 |
Ki = 168 nM
|
|
|
|
CP0412041
|
2-(1H-Pyrrolo[2,3-b]pyridin-2-ylmethyl)-1,2,3,4-tetrahydro-isoquinoline
Show/Hide
|
C17H17N3
|
1
|
| 1 |
Ki = 59 nM
|
|
|
|
CP0377724
|
1-(3-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine
Show/Hide
|
C21H21Cl2N3
|
1
|
| 1 |
Ki = 60 nM
|
|
|
|
CP0861004
|
4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)-piperidin-4-ol oxalate
Show/Hide
|
C23H25IN2O6
|
1
|
| 1 |
Ki = 60.4 nM
|
|
|
|
CP0183485
|
1-(4-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine
Show/Hide
|
C21H21Cl2N3
|
1
|
| 1 |
Ki = 61 nM
|
|
|
|
CP0502695
|
N-[4-(8-chloro-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-2,2-dimethylpropanamide
Show/Hide
|
C21H32ClN3O
|
1
|
| 1 |
Ki = 63.1 nM
|
|
|
|
CP0507188
|
N-[4-[4-(4-chlorophenyl)-3-methylpiperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C20H32ClN3O
|
1
|
| 1 |
Ki = 63.1 nM
|
|
|
|
CP0422138
|
2-[[4-(4-chlorophenyl)piperidin-1-yl]methyl]-1-methylbenzimidazole
Show/Hide
|
C20H22ClN3
|
1
|
| 1 |
Ki = 63.1 nM
|
|
|
|
CP0158026
|
1-butyl-4-(2-chloro-3-ethylphenyl)piperazine
Show/Hide
|
C16H25ClN2
|
1
|
| 1 |
Ki = 65.1 nM
|
|
|
|
CP0391410
|
2-[1-(4-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-1H-benzoimidazole
Show/Hide
|
C19H18ClN3
|
1
|
| 1 |
Ki = 68 nM
|
|
|
|
CP0053105
|
(S)-3-chloro-5-ethyl-N-((1-ethylpyrrolidin-2-yl)methyl)-6-hydroxy-2-methoxybenzamide
Show/Hide
|
C17H25ClN2O3
|
1
|
| 1 |
Ki = 70.4 nM
|
|
|
|
CP0404224
|
1-(1-Benzyl-piperidin-4-yl)-4-methyl-5-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C22H25N3O
|
1
|
| 1 |
Ki = 71 nM
|
|
|
|
CP0861000
|
1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1Hbenzo[d]imidazol-2-(3H)-one oxalate
Show/Hide
|
C23H23N3O5S
|
1
|
| 1 |
Ki = 72.6 nM
|
|
|
|
CP0379138
|
1-[3-[4-(3-hydroxypropyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C20H30N2O2
|
1
|
| 1 |
Ki = 74.13 nM
|
|
|
|
CP0384679
|
N-(3-methylphenyl)-3-(4-pyridin-2-ylpiperidin-1-yl)propanamide
Show/Hide
|
C20H25N3O
|
2
|
| 1 |
Ki = 76.4 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0408777
|
N-[4-[4-(2-chlorophenyl)piperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C19H30ClN3O
|
1
|
| 1 |
Ki = 79.43 nM
|
|
|
|
CP0384677
|
N-(3-ethylphenyl)-2-(4-pyridin-2-ylpiperidin-1-yl)acetamide
Show/Hide
|
C20H25N3O
|
1
|
| 1 |
Ki = 82.3 nM
|
|
|
|
CP0451957
|
N-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl]-N-methyl-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C24H30ClFN4OS
|
1
|
| 1 |
Ki = 85.1 nM
|
|
|
|
CP0350416
|
N-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-propylpropan-1-amine;hydrochloride
Show/Hide
|
C26H34ClFN4OS
|
1
|
| 1 |
Ki = 85.8 nM
|
|
|
|
CP0404235
|
2-[1-(2-Chloro-benzyl)-1,2,3,6-tetrahydro-pyridin-4-yl]-benzothiazole
Show/Hide
|
C19H17ClN2S
|
1
|
| 1 |
Ki = 87 nM
|
|
|
|
CP0224532
|
1-(2-chloro-3-ethylphenyl)-4-methylpiperazine
Show/Hide
|
C13H19ClN2
|
1
|
| 1 |
Ki = 89.9 nM
|
|
|
|
CP0367294
|
1-(2-methoxyphenyl)-4-[3-[1-(4-thiophen-3-ylphenyl)triazol-4-yl]propyl]piperazine
Show/Hide
|
C26H29N5OS
|
1
|
| 1 |
Ki = 90 nM
|
|
|
|
CP0035276
|
1-(4-fluorophenyl)-4-(4-hydroxy-5-azahexacyclo[5.4.1.02,6.03,10.04,8.09,12]dodecan-5-yl)butan-1-one
Show/Hide
|
C21H22FNO2
|
1
|
| 1 |
Ki = 93 nM
|
|
|
|
CP0391409
|
2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-benzoimidazole
Show/Hide
|
C19H19N3
|
1
|
| 1 |
Ki = 94 nM
|
|
|
|
CP0912199
|
1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate
Show/Hide
|
C22H22BrNO6
|
1
|
| 1 |
Ki = 94.5 nM
|
|
|
|
CP0455468
|
4-fluoro-N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]benzamide
Show/Hide
|
C21H25FN2O3
|
1
|
| 1 |
Ki = 95 nM
|
|
|
|
CP0436857
|
2-[2-(3-methoxyphenyl)ethyl]-1-(2-phenylethyl)-4,5-dihydroimidazole
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 95.5 nM
|
|
|
|
CP0487544
|
2-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-benzooxazole
Show/Hide
|
C19H18N2O
|
1
|
| 1 |
Ki = 97 nM
|
|
|
|
CP0509573
|
N-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C19H30ClN3O
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0441267
|
1-Methyl-2-((4-phenylpiperidin-1-yl)methyl)-1H-benzo[d]-imidazole
Show/Hide
|
C20H23N3
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0393625
|
1-[3-[4-(7-hydroxyheptyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C24H38N2O2
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0382967
|
N-[[2-(2-ethoxy-5-fluorophenyl)cyclopropyl]methyl]-N-ethyl-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C26H34ClFN4OS
|
1
|
| 1 |
Ki = 100.8 nM
|
|
|
|
CP0374292
|
3-(1-Benzyl-pyrrolidin-3-yl)-5-(4-chloro-phenyl)-1H-pyrazole
Show/Hide
|
C20H20ClN3
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0453528
|
4-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-1-(3-phenyl-propyl)-piperidine
Show/Hide
|
C23H26ClN3
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0384675
|
N-(3-methylphenyl)-2-[4-(4-methylphenyl)piperidin-1-yl]acetamide
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
Ki = 110.4 nM
|
|
|
|
CP0411284
|
3-(1-hexylpyrrolidin-3-yl)phenol
Show/Hide
|
C16H25NO
|
1
|
| 1 |
Ki = 114 nM
|
|
|
|
CP0384366
|
2-[4-(4-chlorophenyl)piperidin-1-yl]-N-(3-methylphenyl)acetamide
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
Ki = 115.2 nM
|
|
|
|
CP0383455
|
N-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-2,2-dimethylpropanamide
Show/Hide
|
C20H32ClN3O
|
1
|
| 1 |
Ki = 125.89 nM
|
|
|
|
CP0449398
|
N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-2-methylpropanamide
Show/Hide
|
C18H28ClN3O
|
1
|
| 1 |
Ki = 125.89 nM
|
|
|
|
CP0509798
|
N-[4-[4-(4-fluorophenyl)piperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C19H30FN3O
|
1
|
| 1 |
Ki = 125.89 nM
|
|
|
|
CP0422141
|
1-methyl-2-((4-(4-(trifluoromethyl)phenyl)piperidin-1-yl)methyl)-1H-benzo[d]imidazole
Show/Hide
|
C21H22F3N3
|
1
|
| 1 |
Ki = 125.89 nM
|
|
|
|
CP0446516
|
2-[[4-(4-chlorophenyl)-1-piperazinyl]methyl]-1-methylbenzimidazole
Show/Hide
|
C19H21ClN4
|
1
|
| 1 |
Ki = 125.89 nM
|
|
|
|
CP0449016
|
4-biphenyl-4-yl-1-(1H-indol-3-ylmethyl)-piperidin-4-ol
Show/Hide
|
C26H26N2O
|
1
|
| 1 |
Ki = 129 nM
|
|
|
|
CP0902372
|
4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)-piperidin-4-ol oxalate
Show/Hide
|
C23H25IN2O6
|
1
|
| 1 |
Ki = 129 nM
|
|
|
|
CP0412112
|
N-[[2-(5-chloro-2-methoxyphenyl)cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-propylpropan-1-amine;hydrochloride
Show/Hide
|
C26H34Cl2N4OS
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0355150
|
N-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C23H28ClFN4OS
|
1
|
| 1 |
Ki = 132.8 nM
|
|
|
|
CP0175178
|
11-methyl-11-aza-tricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaene
Show/Hide
|
C18H21N
|
1
|
| 1 |
Ki = 134 nM
|
|
|
|
CP0509616
|
1-Benzyl-4-(3-methyl-5-phenyl-pyrazol-1-yl)-piperidine
Show/Hide
|
C22H25N3
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0445778
|
4-chloro-N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]benzamide
Show/Hide
|
C21H25ClN2O3
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0561496
|
N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-5-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
Show/Hide
|
C23H30ClN5OS
|
1
|
| 1 |
Ki = 143 nM
|
|
|
|
CP0378380
|
1-(1-Benzyl-piperidin-4-yl)-3-pyridin-2-yl-urea
Show/Hide
|
C18H22N4O
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0412078
|
N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]-3-methoxybenzamide
Show/Hide
|
C22H28N2O4
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0372385
|
1-(benzofuran-3-ylmethyl)-4-(4-(methylthio)phenyl)piperidin-4-ol
Show/Hide
|
C21H23NO2S
|
1
|
| 1 |
Ki = 153 nM
|
|
|
|
CP0412046
|
N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]benzamide
Show/Hide
|
C21H26ClN3O
|
1
|
| 1 |
Ki = 158.49 nM
|
|
|
|
CP0440174
|
4-fluoro-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide
Show/Hide
|
C23H30FN3O2
|
1
|
| 1 |
Ki = 159 nM
|
|
|
|
CP0439296
|
1-Benzyl-4-(5-benzyl-1H-pyrazol-3-yl)-piperidine
Show/Hide
|
C22H25N3
|
1
|
| 1 |
Ki = 160 nM
|
|
|
|
CP0397772
|
N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-1H-indole-2-carboxamide
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
Ki = 161 nM
|
|
|
|
CP0869494
|
(E)-5-Methoxy-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)but-2-en-1-yl)-1H-indole-2-carboxamide oxalic acid
Show/Hide
|
C27H32N4O7
|
1
|
| 1 |
Ki = 162 nM
|
|
|
|
CP0861001
|
1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1Hbenzo[d]imidazol-2-(3H)-one oxalate
Show/Hide
|
C23H23N3O6
|
1
|
| 1 |
Ki = 163 nM
|
|
|
|
CP0093141
|
1-(2-methoxyphenyl)-4-[5-[1-(4-thiophen-3-ylphenyl)triazol-4-yl]pentyl]piperazine
Show/Hide
|
C28H33N5OS
|
1
|
| 1 |
Ki = 163 nM
|
|
|
|
CP0350418
|
N-[[2-(5-chloro-2-methoxyphenyl)cyclopropyl]methyl]-N-(cyclopropylmethyl)-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C27H34Cl2N4OS
|
1
|
| 1 |
Ki = 163 nM
|
|
|
|
CP0470669
|
3-(1-pentylpyrrolidin-3-yl)phenol
Show/Hide
|
C15H23NO
|
1
|
| 1 |
Ki = 164 nM
|
|
|
|
CP0873320
|
7-methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide
Show/Hide
|
C18H22BrNO2
|
1
|
| 1 |
Ki = 165 nM
|
|
|
|
CP0409143
|
1-(benzofuran-3-ylmethyl)-4-(3,4-dichlorophenyl)piperidin-4-ol
Show/Hide
|
C20H19Cl2NO2
|
1
|
| 1 |
Ki = 167 nM
|
|
|
|
CP0392756
|
N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]naphthalene-2-carboxamide
Show/Hide
|
C25H28N2O3
|
1
|
| 1 |
Ki = 170 nM
|
|
|
|
CP0384367
|
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-(3-ethylphenyl)acetamide
Show/Hide
|
C19H23ClN4O
|
1
|
| 1 |
Ki = 172.2 nM
|
|
|
|
CP0450101
|
N-[2-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H30N4O3
|
1
|
| 1 |
Ki = 176 nM
|
|
|
|
CP0396657
|
5-bromo-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]thiophene-2-carboxamide
Show/Hide
|
C21H28BrN3O2S
|
1
|
| 1 |
Ki = 177 nM
|
|
|
|
CP0426721
|
N-ethyl-N-[[2-[5-fluoro-2-(2-fluoroethoxy)phenyl]cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C26H33ClF2N4OS
|
1
|
| 1 |
Ki = 179.2 nM
|
|
|
|
CP0844267
|
4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)-trans-but-2-enyl)benzamides oxalic acid salt
Show/Hide
|
C29H32FN3O6S
|
1
|
| 1 |
Ki = 182 nM
|
|
|
|
CP0847131
|
7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C27H34FN3O7
|
1
|
| 1 |
Ki = 185 nM
|
|
|
|
CP0410571
|
5-[4-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]triazol-1-yl]isoquinoline
Show/Hide
|
C27H32N6O
|
1
|
| 1 |
Ki = 186 nM
|
|
|
|
CP0469462
|
N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-4-thiophen-3-ylbenzamide
Show/Hide
|
C27H33N3O2S
|
1
|
| 1 |
Ki = 187 nM
|
|
|
|
CP0477829
|
N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-5-methylthiophene-2-carboxamide
Show/Hide
|
C22H31N3O2S
|
1
|
| 1 |
Ki = 188 nM
|
|
|
|
CP0502691
|
N-[3-[4-(4-chlorophenyl)piperazin-1-yl]propyl]-2,2-dimethylpropanamide
Show/Hide
|
C18H28ClN3O
|
1
|
| 1 |
Ki = 199.53 nM
|
|
|
|
CP0469995
|
3-[1-[(1-methylbenzimidazol-2-yl)methyl]piperidin-4-yl]-1,2-benzothiazole
Show/Hide
|
C21H22N4S
|
1
|
| 1 |
Ki = 199.53 nM
|
|
|
|
CP0362283
|
1-(2-methoxyphenyl)-4-[4-[1-(4-methylsulfanylphenyl)triazol-4-yl]butyl]piperazine
Show/Hide
|
C24H31N5OS
|
1
|
| 1 |
Ki = 200 nM
|
|
|
|
CP0920165
|
7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)quinolin-2(1H)-one oxalate
Show/Hide
|
C27H33N3O7
|
1
|
| 1 |
Ki = 201 nM
|
|
|
|
CP0847130
|
7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C26H33N3O7
|
1
|
| 1 |
Ki = 212 nM
|
|
|
|
CP0382968
|
N-[4-[propyl-[[2-[4-(trifluoromethyl)phenyl]cyclopropyl]methyl]amino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C29H34ClF3N2O
|
1
|
| 1 |
Ki = 215 nM
|
|
|
|
CP0531034
|
N-[4-[ethyl-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl]amino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
|
C26H33ClFN3O2
|
1
|
| 1 |
Ki = 220 nM
|
|
|
|
CP0389480
|
5-[1-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-4-yl]-1H-indole
Show/Hide
|
C25H30N6O
|
1
|
| 1 |
Ki = 222 nM
|
|
|
|
CP0234732
|
1-(2-methoxyphenyl)-4-[5-[1-(4-methylsulfanylphenyl)triazol-4-yl]pentyl]piperazine
Show/Hide
|
C25H33N5OS
|
1
|
| 1 |
Ki = 227 nM
|
|
|
|
CP0449146
|
1-(2-methoxyphenyl)-4-[4-(4-naphthalen-2-yltriazol-1-yl)butyl]piperazine
Show/Hide
|
C27H31N5O
|
1
|
| 1 |
Ki = 232 nM
|
|
|
|
CP0871789
|
7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C27H35N3O7
|
1
|
| 1 |
Ki = 234 nM
|
|
|
|
CP0426728
|
N-[[2-(5-chloro-2-methoxyphenyl)cyclopropyl]methyl]-N-ethyl-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C25H32Cl2N4OS
|
1
|
| 1 |
Ki = 241 nM
|
|
|
|
CP0912200
|
1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate
Show/Hide
|
C22H22INO6
|
1
|
| 1 |
Ki = 245 nM
|
|
|
|
CP0786649
|
4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt
Show/Hide
|
C29H34FN3O6S
|
1
|
| 1 |
Ki = 246 nM
|
|
|
|
CP0422137
|
2-[[4-(3-chlorophenyl)piperidin-1-yl]methyl]-1-methylbenzimidazole
Show/Hide
|
C20H22ClN3
|
1
|
| 1 |
Ki = 251.19 nM
|
|
|
|
CP0458982
|
2-[[4-(4-chloro-2-fluorophenyl)piperazin-1-yl]methyl]-1-methylbenzimidazole
Show/Hide
|
C19H20ClFN4
|
1
|
| 1 |
Ki = 251.19 nM
|
|
|
|
CP0513314
|
1-methyl-2-[[4-[3-(trifluoromethyl)phenyl]piperidin-1-yl]methyl]benzimidazole
Show/Hide
|
C21H22F3N3
|
1
|
| 1 |
Ki = 251.19 nM
|
|
|
|
CP0902371
|
1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate
Show/Hide
|
C22H22BrNO6
|
1
|
| 1 |
Ki = 254 nM
|
|
|
|
CP0393627
|
1-[3-(4-methylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C18H26N2O
|
1
|
| 1 |
Ki = 257.04 nM
|
|
|
|
CP0433591
|
6-[1-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-4-yl]quinoline
Show/Hide
|
C26H30N6O
|
1
|
| 1 |
Ki = 269 nM
|
|
|
|
CP0535381
|
N-[(3,3-diphenyl-1,4-dioxan-2-yl)methyl]-2-(2-methoxyphenoxy)ethanamine
Show/Hide
|
C26H29NO4
|
1
|
| 1 |
Ki = 275.42 nM
|
|
|
|
CP0869493
|
5-(2-fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide oxalic acid
Show/Hide
|
C28H35FN4O7
|
1
|
| 1 |
Ki = 284 nM
|
|
|
|
CP0891095
|
7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C27H35N3O8
|
1
|
| 1 |
Ki = 286 nM
|
|
|
|
CP0444479
|
N-[2-[(1R,2S)-2-[[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]methyl]cyclopropyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C25H31N5O2
|
2
|
| 1 |
Ki = 286 nM
|
|
|
| 2 |
Ki = 1520 nM
|
|
|
|
CP0470997
|
N-(cyclopropylmethyl)-N-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C27H34ClFN4OS
|
1
|
| 1 |
Ki = 291.7 nM
|
|
|
|
CP0425631
|
5-[(5S)-5-methyl-4-propylmorpholin-2-yl]pyridin-2-amine
Show/Hide
|
C13H21N3O
|
1
|
| 1 |
Ki = 292 nM
|
|
|
|
CP0381642
|
N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-1-benzothiophene-2-carboxamide
Show/Hide
|
C25H31N3O2S
|
1
|
| 1 |
Ki = 297 nM
|
|
|
|
CP0074631
|
6-methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine
Show/Hide
|
C16H19NS
|
1
|
| 1 |
Ki = 299 nM
|
|
|
|
CP0400383
|
1-(2-methoxyphenyl)-4-[4-(1-naphthalen-2-yltriazol-4-yl)butyl]piperazine
Show/Hide
|
C27H31N5O
|
1
|
| 1 |
Ki = 299 nM
|
|
|
|
CP0104676
|
Benzo[b]thiophene-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
Ki = 305 nM
|
|
|
|
CP0480201
|
N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-2-hydroxybutyl]-1H-indole-2-carboxamide
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
Ki = 305 nM
|
|
|
|
CP0382710
|
N-[2-[2-[[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]methyl]cyclopropyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C25H31N5O2
|
2
|
| 1 |
Ki = 315 nM
|
|
|
| 2 |
Ki = 6650 nM
|
|
|
|
CP0157763
|
1-(2-chloro-3-ethylphenyl)piperazine
Show/Hide
|
C12H17ClN2
|
1
|
| 1 |
Ki = 316 nM
|
|
|
|
CP0375314
|
2,2-dimethyl-N-[4-(4-phenylpiperazin-1-yl)butyl]propanamide
Show/Hide
|
C19H31N3O
|
1
|
| 1 |
Ki = 316.23 nM
|
|
|
|
CP0383454
|
N-[4-[4-(4-methoxyphenyl)piperazin-1-yl]butyl]-2,2-dimethylpropanamide
Show/Hide
|
C20H33N3O2
|
1
|
| 1 |
Ki = 316.23 nM
|
|
|
|
CP0411642
|
1-[3-(4-butylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C20H31N3O
|
1
|
| 1 |
Ki = 316.23 nM
|
|
|
|
CP0467837
|
1-((1H-indol-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol
Show/Hide
|
C21H24N2OS
|
1
|
| 1 |
Ki = 319 nM
|
|
|
|
CP0135682
|
1-butyl-4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazine
Show/Hide
|
C17H27ClN2O
|
1
|
| 1 |
Ki = 322 nM
|
|
|
|
CP0350417
|
N-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-propan-2-ylpropan-1-amine;hydrochloride
Show/Hide
|
C26H34ClFN4OS
|
1
|
| 1 |
Ki = 326.1 nM
|
|
|
|
CP0410742
|
1-[4-[1-(9H-fluoren-2-yl)triazol-4-yl]butyl]-4-(2-methoxyphenyl)piperazine
Show/Hide
|
C30H33N5O
|
1
|
| 1 |
Ki = 329 nM
|
|
|
|
CP0224535
|
N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide
Show/Hide
|
C25H31ClN4O
|
1
|
| 1 |
Ki = 334 nM
|
|
|
|
CP0197217
|
5-Iodo-benzofuran-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C24H28IN3O3
|
1
|
| 1 |
Ki = 335 nM
|
|
|
|
CP0380992
|
N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-5-phenylthiophene-2-carboxamide
Show/Hide
|
C27H33N3O2S
|
1
|
| 1 |
Ki = 342 nM
|
|
|
|
CP0902374
|
4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)-methyl)piperidin-4-ol oxalate
Show/Hide
|
C24H26BrFN2O6
|
1
|
| 1 |
Ki = 344 nM
|
|
|
|
CP0409195
|
N-[4-(4-chlorophenyl)-1-(1H-indol-3-ylmethyl)piperidin-4-yl]acetamide
Show/Hide
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C22H24ClN3O
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1
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| 1 |
Ki = 348 nM
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CP0454998
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(Z)-1-(1-benzyl-4-methylpiperidin-4-yl)-3-(4-chlorophenyl)-3-hydroxyprop-2-en-1-one
Show/Hide
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C22H24ClNO2
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1
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| 1 |
Ki = 350 nM
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CP0397169
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4-chloro-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide
Show/Hide
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C23H30ClN3O2
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1
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| 1 |
Ki = 350 nM
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CP0455469
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4-bromo-N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]benzamide
Show/Hide
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C21H25BrN2O3
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1
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| 1 |
Ki = 350 nM
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CP0912198
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8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate
Show/Hide
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C25H27N3O5S
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1
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| 1 |
Ki = 352 nM
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CP0444621
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5-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]-1H-indole
Show/Hide
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C25H30N6O
|
1
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| 1 |
Ki = 353 nM
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CP0224534
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N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide
Show/Hide
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C25H30ClN3O2
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1
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| 1 |
Ki = 356 nM
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CP0382695
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N-[4-[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]butyl]-1H-indole-2-carboxamide
Show/Hide
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C23H29N5O2
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2
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| 1 |
Ki = 357 nM
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| 2 |
Ki = 16800 nM
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CP0891097
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7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
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C26H33N3O7
|
1
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| 1 |
Ki = 359 nM
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CP0860158
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(E)-5-(2-(2-Fluoroethoxy)ethoxy)-N-(4-(4-(2-methoxyphenyl)-piperazin-1-yl)but-2-en-1-yl)-1H-indole-2-carboxamide oxalic acid
Show/Hide
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C30H37FN4O8
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1
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| 1 |
Ki = 360 nM
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CP0445424
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3-((4-(4-chlorophenyl)-4-fluoropiperidin-1-yl)methyl)-1H-indole
Show/Hide
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C20H20ClFN2
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1
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| 1 |
Ki = 365 nM
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CP0396653
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N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-4-methylsulfanylbenzamide
Show/Hide
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C24H33N3O2S
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1
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| 1 |
Ki = 372 nM
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CP0061556
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N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]-4-pyridin-2-ylbenzamide
Show/Hide
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C26H26Cl2N4O
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2
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| 1 |
Ki = 375 nM
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| 2 |
Ki = 550 nM
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CP0143978
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N-[4-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
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C27H35ClFN3O2
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1
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| 1 |
Ki = 376 nM
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CP0927947
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1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)-piperidin-4-ol oxalate
Show/Hide
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C22H23NO5S
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1
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| 1 |
Ki = 377 nM
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CP0419602
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7-ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine
Show/Hide
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C21H24N2
|
1
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| 1 |
Ki = 378.5 nM
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CP0426719
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N-[4-[ethyl-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl]amino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
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C28H34ClFN2O2
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1
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| 1 |
Ki = 384.6 nM
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CP0429530
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1-(1-Benzyl-piperidin-4-yl)-3-phenyl-urea
Show/Hide
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C19H23N3O
|
1
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| 1 |
Ki = 390 nM
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CP0093139
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1-(2-methoxyphenyl)-4-[4-[1-(4-thiophen-3-ylphenyl)triazol-4-yl]butyl]piperazine
Show/Hide
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C27H31N5OS
|
1
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| 1 |
Ki = 395 nM
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CP0452269
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1-methyl-2-[[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]methyl]benzimidazole
Show/Hide
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C20H21F3N4
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1
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| 1 |
Ki = 398.11 nM
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CP0167921
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1-(3-chloro-5-ethyl-2-methoxyphenyl)-4-methylpiperazine
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C14H21ClN2O
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1
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| 1 |
Ki = 400 nM
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CP0407660
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5-(4-fluorophenyl)-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]thiophene-2-carboxamide
Show/Hide
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C27H32FN3O2S
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1
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| 1 |
Ki = 403 nM
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CP0449024
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1-(benzofuran-3-ylmethyl)-4-(4-chlorophenyl)piperidin-4-ol
Show/Hide
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C20H20ClNO2
|
1
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| 1 |
Ki = 404 nM
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CP0508564
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1-Benzyl-3-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine
Show/Hide
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C21H22ClN3
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1
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| 1 |
Ki = 410 nM
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CP0392755
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N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]quinoline-4-carboxamide
Show/Hide
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C24H27N3O3
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1
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| 1 |
Ki = 410 nM
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CP0261925
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N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-9H-fluorene-2-carboxamide
Show/Hide
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C29H33N3O2
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1
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| 1 |
Ki = 425 nM
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CP0452963
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1-(2-methoxyphenyl)-4-[4-[4-(4-phenylphenyl)triazol-1-yl]butyl]piperazine
Show/Hide
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C29H33N5O
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1
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| 1 |
Ki = 425 nM
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CP0375438
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N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-1-benzofuran-2-carboxamide
Show/Hide
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C25H31N3O3
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1
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| 1 |
Ki = 429 nM
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CP0396656
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2,3-dimethoxy-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide
Show/Hide
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C25H35N3O4
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1
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| 1 |
Ki = 441 nM
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CP0850773
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5-Hydroxy-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide oxalic acid
Show/Hide
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C26H32N4O7
|
1
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| 1 |
Ki = 444 nM
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CP0041232
|
1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-ol
Show/Hide
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C20H21ClN2O
|
2
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| 1 |
Ki = 449 nM
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| 2 |
Ki = 1520 nM
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CP0327018
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N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-5-iodo-1H-indole-2-carboxamide
Show/Hide
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C24H29IN4O3
|
1
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| 1 |
Ki = 455 nM
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CP0441507
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1-Benzyl-4-(5-methyl-1H-pyrazol-3-yl)-piperidine
Show/Hide
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C16H21N3
|
1
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| 1 |
Ki = 470 nM
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CP0314424
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1H-Indole-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
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C24H30N4O2
|
1
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| 1 |
Ki = 476 nM
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CP0266687
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1-(2-methoxyphenyl)-4-[4-(4-phenyltriazol-1-yl)butyl]piperazine
Show/Hide
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C23H29N5O
|
1
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| 1 |
Ki = 480 nM
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CP0367693
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13-methyl-4-thia-6,13-diazapentacyclo[10.7.1.02,10.03,7.016,20]icosa-1(19),2(10),3(7),5,8,16(20),17-heptaen-5-amine
Show/Hide
|
C18H17N3S
|
1
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| 1 |
Ki = 481 nM
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CP0410743
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1-(2-methoxyphenyl)-4-[4-(1-phenyltriazol-4-yl)butyl]piperazine
Show/Hide
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C23H29N5O
|
1
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| 1 |
Ki = 486 nM
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CP0919567
|
8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate
Show/Hide
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C25H27N3O6
|
1
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| 1 |
Ki = 492 nM
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CP0421285
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N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-5-ethyl-1H-imidazole-2-carboxamide
Show/Hide
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C22H32ClN5O
|
1
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| 1 |
Ki = 500 nM
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CP0228691
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N-[[2-(2-ethoxy-5-fluorophenyl)cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C24H30ClFN4OS
|
1
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| 1 |
Ki = 501.2 nM
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CP0424341
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N-[(E)-4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]but-2-enyl]-5-methyl-1H-imidazole-2-carboxamide
Show/Hide
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C21H28ClN5O
|
1
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| 1 |
Ki = 503 nM
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CP0400385
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5-[4-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]triazol-1-yl]-1H-indole
Show/Hide
|
C24H26Cl2N6
|
1
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| 1 |
Ki = 510 nM
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CP0426726
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N-[4-[[2-(4-chlorophenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
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C26H33Cl2N3O
|
1
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| 1 |
Ki = 510 nM
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CP0375440
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4-(2-fluoroethyl)-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide
Show/Hide
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C25H34FN3O2
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1
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| 1 |
Ki = 522 nM
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CP0488182
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N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-5-methyl-1H-imidazole-2-carboxamide
Show/Hide
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C21H30ClN5O
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1
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| 1 |
Ki = 529 nM
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CP0426722
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N-[4-[[2-(5-chloro-2-methoxyphenyl)cyclopropyl]methyl-ethylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
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C28H34Cl2N2O2
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1
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| 1 |
Ki = 553 nM
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CP0481782
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N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]-4-methoxybenzamide
Show/Hide
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C22H28N2O4
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1
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| 1 |
Ki = 560 nM
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CP0898479
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5-(2-(2-(2-Fluoroethoxy)ethoxy)ethoxy)-N-(4-(4-(2-methoxy-phenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide oxalic acid
Show/Hide
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C32H43FN4O9
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1
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| 1 |
Ki = 565 nM
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CP0409144
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1-((5-methoxy-1H-indol-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol
Show/Hide
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C22H26N2O2S
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1
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| 1 |
Ki = 567 nM
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CP0412254
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N-[4-[[2-(5-chloro-2-methoxyphenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
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C27H35Cl2N3O2
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1
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| 1 |
Ki = 575 nM
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CP0533678
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N-[4-[[(1R,2R)-2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
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C30H37ClFN3O2
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1
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| 1 |
Ki = 575 nM
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CP0139957
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3-[Bis-(4-fluoro-phenyl)-methoxy]-8-butyl-8-aza-bicyclo[3.2.1]octane
Show/Hide
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C24H29F2NO
|
1
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| 1 |
Ki = 583 nM
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CP0410746
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1-[4-[4-(9H-fluoren-2-yl)triazol-1-yl]butyl]-4-(2-methoxyphenyl)piperazine
Show/Hide
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C30H33N5O
|
1
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| 1 |
Ki = 588 nM
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CP0381617
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4-(dimethylamino)-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide
Show/Hide
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C25H36N4O2
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1
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| 1 |
Ki = 608 nM
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CP0919397
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1-((1H-Pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate
Show/Hide
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C21H22BrN3O5
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1
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| 1 |
Ki = 620 nM
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CP0234177
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2-[[4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]methyl]-1-methylbenzimidazole
Show/Hide
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C19H19ClF3N5
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1
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| 1 |
Ki = 630.96 nM
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CP0473888
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1-methyl-2-[[4-[2-(trifluoromethyl)phenyl]piperazin-1-yl]methyl]benzimidazole
Show/Hide
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C20H21F3N4
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1
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| 1 |
Ki = 630.96 nM
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CP0861002
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1-((1H-Pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate
Show/Hide
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C21H22IN3O5
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1
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| 1 |
Ki = 634 nM
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CP0772206
|
SID56463240
Show/Hide
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C26H32ClN3O2
|
1
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| 1 |
Ki = 634 nM
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CP0288362
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N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]-1H-indole-2-carboxamide
Show/Hide
|
C23H24Cl2N4O
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1
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| 1 |
Ki = 640 nM
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CP0381618
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6-chloro-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
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C22H29ClN4O2
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1
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| 1 |
Ki = 641 nM
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CP0406019
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1-((1H-indol-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol
Show/Hide
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C20H21BrN2O
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1
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| 1 |
Ki = 652 nM
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CP0397771
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N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-9-oxofluorene-4-carboxamide
Show/Hide
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C30H33N3O3
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1
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| 1 |
Ki = 657 nM
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CP0412077
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4-hydroxy-N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]benzamide
Show/Hide
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C21H26N2O4
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1
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| 1 |
Ki = 660 nM
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CP0904688
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4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)-methyl)piperidin-4-ol oxalate
Show/Hide
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C24H26BrFN2O6
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1
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| 1 |
Ki = 668 nM
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CP0426729
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N-[4-[[2-(3-fluorophenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
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C26H33ClFN3O
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1
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| 1 |
Ki = 671 nM
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CP0348222
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N-[4-[[(1R,2R)-2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C29H34Cl3N3O
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1
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| 1 |
Ki = 676 nM
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CP0426727
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N-[4-[[(1S,2S)-2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
|
C26H32Cl3N3O
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1
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| 1 |
Ki = 676 nM
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CP0449018
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1-((1H-indazol-3-yl)methyl)-4-(3,4-dichlorophenyl)piperidin-4-ol
Show/Hide
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C19H19Cl2N3O
|
1
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| 1 |
Ki = 677 nM
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CP0449017
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1-((1H-indol-3-yl)methyl)-4-(4-methoxyphenyl)piperidin-4-ol
Show/Hide
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C21H24N2O2
|
1
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| 1 |
Ki = 679 nM
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CP0506201
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4-(4-bromophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol
Show/Hide
|
C21H23BrN2O2
|
1
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| 1 |
Ki = 700 nM
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CP0397770
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N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-4-(methylamino)benzamide
Show/Hide
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C24H34N4O2
|
1
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| 1 |
Ki = 706 nM
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CP0224533
|
N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide
Show/Hide
|
C26H32ClN3O3
|
1
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| 1 |
Ki = 714 nM
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CP0538565
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N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]-4-phenylbenzamide
Show/Hide
|
C27H30N2O3
|
1
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| 1 |
Ki = 720 nM
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CP0001212
|
1-(2-methoxyphenyl)-4-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]piperazine
Show/Hide
|
C23H29N5OS
|
1
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| 1 |
Ki = 721 nM
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CP0397773
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4-ethenyl-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide
Show/Hide
|
C25H33N3O2
|
1
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| 1 |
Ki = 728 nM
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CP0375439
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4-(2-hydroxyethyl)-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide
Show/Hide
|
C25H35N3O3
|
1
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| 1 |
Ki = 748 nM
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CP0234731
|
4-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]-N,N-dimethylaniline
Show/Hide
|
C25H34N6O
|
1
|
| 1 |
Ki = 758 nM
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CP0143982
|
N-[4-[[(1S,2S)-2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C28H33Cl3N2O
|
1
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| 1 |
Ki = 776 nM
|
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CP0452272
|
2-[4-[(1-methylbenzimidazol-2-yl)methyl]piperazin-1-yl]-1,3-benzothiazole
Show/Hide
|
C20H21N5S
|
1
|
| 1 |
Ki = 794.33 nM
|
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CP0231075
|
4-(2-fluoroethyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide
Show/Hide
|
C24H32FN3O2
|
1
|
| 1 |
Ki = 804 nM
|
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CP0159265
|
N-[4-[4-(3-cyanophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide
Show/Hide
|
C26H28N4OS
|
1
|
| 1 |
Ki = 806 nM
|
|
|
|
CP0267566
|
N-[4-[[(1R,2R)-2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C28H33Cl3N2O
|
1
|
| 1 |
Ki = 813 nM
|
|
|
|
CP0424340
|
N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide
Show/Hide
|
C24H30ClN5O
|
1
|
| 1 |
Ki = 819 nM
|
|
|
|
CP0465278
|
6-bromo-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C22H29BrN4O2
|
1
|
| 1 |
Ki = 830 nM
|
|
|
|
CP0377177
|
4-(4-bromophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol
Show/Hide
|
C21H23BrN2O2
|
1
|
| 1 |
Ki = 840 nM
|
|
|
|
CP0528465
|
N-[4-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C29H36ClFN2O2
|
1
|
| 1 |
Ki = 844 nM
|
|
|
|
CP0348221
|
N-[4-[[(1S,2S)-2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C30H37ClFN3O2
|
1
|
| 1 |
Ki = 851 nM
|
|
|
|
CP0887642
|
7-(4-(3-Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate
Show/Hide
|
C29H36N4O7
|
1
|
| 1 |
Ki = 865 nM
|
|
|
|
CP0362281
|
5-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]isoquinoline
Show/Hide
|
C26H30N6O
|
1
|
| 1 |
Ki = 875 nM
|
|
|
|
CP0543970
|
N-[4-[[2-(3-chlorophenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
|
C26H33Cl2N3O
|
1
|
| 1 |
Ki = 878 nM
|
|
|
|
CP0653272
|
4-(Dimethylamino)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt
Show/Hide
|
C27H37FN4O6
|
1
|
| 1 |
Ki = 890 nM
|
|
|
|
CP0722004
|
4-(2-Fluoroethyl)-N-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt
Show/Hide
|
C27H33F2N3O6
|
1
|
| 1 |
Ki = 890 nM
|
|
|
|
CP0181036
|
4-(dimethylamino)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide
Show/Hide
|
C24H34N4O2
|
1
|
| 1 |
Ki = 896 nM
|
|
|
|
CP0248165
|
2-benzyl-5-(3-methoxyphenyl)-1,3-dihydroisoindole
Show/Hide
|
C22H21NO
|
1
|
| 1 |
Ki = 904 nM
|
|
|
|
CP0384469
|
N-[4-[[(1S,2S)-2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C29H34Cl3N3O
|
1
|
| 1 |
Ki = 912 nM
|
|
|
|
CP0380731
|
1'-phenethyl-3-phenylspiro[2,4,5,6-tetrahydrocyclopenta[c]pyrazole-6,4'-(hexahydropyridine)]
Show/Hide
|
C24H27N3
|
1
|
| 1 |
Ki = 930 nM
|
|
|
|
CP0919407
|
1-((1H-Pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate
Show/Hide
|
C22H25N3O5S
|
1
|
| 1 |
Ki = 937 nM
|
|
|
|
CP0860998
|
8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate
Show/Hide
|
C26H28FN3O6
|
1
|
| 1 |
Ki = 945 nM
|
|
|
|
CP0143979
|
N-[4-[[2-(5-chloro-2-methoxyphenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C29H36Cl2N2O2
|
1
|
| 1 |
Ki = 945 nM
|
|
|
|
CP0451956
|
N-[[2-[5-fluoro-2-(2-fluoroethoxy)phenyl]cyclopropyl]methyl]-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C24H29ClF2N4OS
|
1
|
| 1 |
Ki = 962.3 nM
|
|
|
|
CP0096655
|
5-fluoro-N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H29FN4O3
|
1
|
| 1 |
Ki = 967 nM
|
|
|
|
CP0447274
|
N-[[2-[5-fluoro-2-(2-fluoroethoxy)phenyl]cyclopropyl]methyl]-N-methyl-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C25H31ClF2N4OS
|
1
|
| 1 |
Ki = 977.2 nM
|
|
|
|
CP0902370
|
8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate
Show/Hide
|
C29H31FN6O6
|
1
|
| 1 |
Ki = 978 nM
|
|
|
|
CP0228692
|
N-[[2-(2-ethoxy-5-fluorophenyl)cyclopropyl]methyl]-N-methyl-3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propan-1-amine;hydrochloride
Show/Hide
|
C25H32ClFN4OS
|
1
|
| 1 |
Ki = 988.6 nM
|
|
|
|
CP0785530
|
4-(2-Fluoroethoxy)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt
Show/Hide
|
C27H35F2N3O7
|
1
|
| 1 |
Ki = 990 nM
|
|
|
|
CP0387459
|
1-methyl-2-[[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]methyl]benzimidazole
Show/Hide
|
C19H20F3N5
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0065124
|
9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
Show/Hide
|
C28H27Cl2N3O
|
1
|
| 1 |
Ki = 1020 nM
|
|
|
|
CP0887641
|
7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C27H32N4O7
|
1
|
| 1 |
Ki = 1029 nM
|
|
|
|
CP0096659
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-2-hydroxybutyl]-1H-indole-2-carboxamide
Show/Hide
|
C23H26Cl2N4O2
|
1
|
| 1 |
Ki = 1040 nM
|
|
|
|
CP0382966
|
N-[4-[[(1R,2R)-2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
|
C26H32Cl3N3O
|
1
|
| 1 |
Ki = 1047 nM
|
|
|
|
CP0135680
|
N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide
Show/Hide
|
C26H33ClN4O2
|
1
|
| 1 |
Ki = 1050 nM
|
|
|
|
CP0044765
|
Benzofuran-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
Show/Hide
|
C23H23Cl2N3O2
|
1
|
| 1 |
Ki = 1070 nM
|
|
|
|
CP0421766
|
1-((1H-indol-3-yl)methyl)-4-(3,4-dichlorophenyl)piperidin-4-ol
Show/Hide
|
C20H20Cl2N2O
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0350421
|
N-[4-[[2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
|
C26H32Cl3N3O
|
1
|
| 1 |
Ki = 1131 nM
|
|
|
|
CP0343822
|
N-[4-[[2-(5-fluoro-2-methoxyphenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C30H37ClFN3O2
|
1
|
| 1 |
Ki = 1142 nM
|
|
|
|
CP0405450
|
3-(1-butylpyrrolidin-3-yl)phenol
Show/Hide
|
C14H21NO
|
1
|
| 1 |
Ki = 1174 nM
|
|
|
|
CP0449025
|
3-((4-(allyloxy)-4-(4-chlorophenyl)piperidin-1-yl)methyl)-1H-indole
Show/Hide
|
C23H25ClN2O
|
1
|
| 1 |
Ki = 1190 nM
|
|
|
|
CP0487134
|
4-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-1-methyl-piperidine
Show/Hide
|
C15H18ClN3
|
1
|
| 1 |
Ki = 1200 nM
|
|
|
|
CP0460824
|
1-Benzyl-4-(5-phenyl-tetrazol-1-yl)-piperidine
Show/Hide
|
C19H21N5
|
1
|
| 1 |
Ki = 1200 nM
|
|
|
|
CP0041389
|
Benzofuran-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C23H25Cl2N3O2
|
1
|
| 1 |
Ki = 1220 nM
|
|
|
|
CP0377890
|
US8748608, 19
Show/Hide
|
C29H33N3O3
|
1
|
| 1 |
Ki = 1230 nM
|
|
|
|
CP0502409
|
N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]acetamide
Show/Hide
|
C16H24ClN3O
|
1
|
| 1 |
Ki = 1258.93 nM
|
|
|
|
CP0288361
|
N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-5-iodo-1-benzofuran-2-carboxamide
Show/Hide
|
C24H28IN3O4
|
1
|
| 1 |
Ki = 1290 nM
|
|
|
|
CP0426723
|
N-[4-[[2-(3-fluorophenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C28H34ClFN2O
|
1
|
| 1 |
Ki = 1298 nM
|
|
|
|
CP0891093
|
7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C26H31ClN2O7
|
1
|
| 1 |
Ki = 1311 nM
|
|
|
|
CP0426724
|
N-[4-[[2-(3-chlorophenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C28H34Cl2N2O
|
1
|
| 1 |
Ki = 1318 nM
|
|
|
|
CP0447271
|
N-[4-[[2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C28H33Cl3N2O
|
1
|
| 1 |
Ki = 1339 nM
|
|
|
|
CP0891094
|
7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate
Show/Hide
|
C27H31ClN4O7
|
1
|
| 1 |
Ki = 1352 nM
|
|
|
|
CP0464320
|
1-((1H-indol-3-yl)methyl)-4-(4-hydroxyphenyl)piperidin-4-ol
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
Ki = 1360 nM
|
|
|
|
CP0043442
|
Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C23H25Cl2N3OS
|
1
|
| 1 |
Ki = 1370 nM
|
|
|
|
CP0421822
|
1-[(6,6-diphenyl-1,4-dioxan-2-yl)methyl]-4-(2-methoxyphenyl)piperazine
Show/Hide
|
C28H32N2O3
|
1
|
| 1 |
Ki = 1380.38 nM
|
|
|
|
CP0861003
|
1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate
Show/Hide
|
C24H26N4O6
|
1
|
| 1 |
Ki = 1390 nM
|
|
|
|
CP0786650
|
4-(2-Fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)-piperazin-1-yl)-butyl)benzamide oxalic acid salt
Show/Hide
|
C26H34FN3O7
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0450713
|
N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]pyridine-4-carboxamide
Show/Hide
|
C20H25N3O3
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0228693
|
N-[4-[[2-(4-chlorophenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C29H35Cl2N3O
|
1
|
| 1 |
Ki = 1413 nM
|
|
|
|
CP0277135
|
N-[[(1S,2R)-2-[[4-(2,3-dichlorophenyl)piperazin-1-yl]methyl]cyclopropyl]methyl]-4-pyridin-2-ylbenzamide
Show/Hide
|
C27H28Cl2N4O
|
1
|
| 1 |
Ki = 1460 nM
|
|
|
|
CP0449021
|
1-((1H-indol-3-yl)methyl)-4-(4-(hexyloxy)phenyl)piperidin-4-ol
Show/Hide
|
C26H34N2O2
|
1
|
| 1 |
Ki = 1490 nM
|
|
|
|
CP0277136
|
US8748608, 18
Show/Hide
|
C27H32N4O3
|
1
|
| 1 |
Ki = 1490 nM
|
|
|
|
CP0190971
|
N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H29FN4O2
|
1
|
| 1 |
Ki = 1490 nM
|
|
|
|
CP0455471
|
N-[4-(7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]-4-iodobenzamide
Show/Hide
|
C21H25IN2O3
|
1
|
| 1 |
Ki = 1500 nM
|
|
|
|
CP0369518
|
N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-5-methoxy-1H-indole-2-carboxamide
Show/Hide
|
C25H32N4O4
|
1
|
| 1 |
Ki = 1530 nM
|
|
|
|
CP0409196
|
1-((1H-indol-3-yl)methyl)-4-(2,3-dichlorophenyl)piperidin-4-ol
Show/Hide
|
C20H20Cl2N2O
|
1
|
| 1 |
Ki = 1550 nM
|
|
|
|
CP0426725
|
N-[4-[[2-(4-chlorophenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C28H34Cl2N2O
|
1
|
| 1 |
Ki = 1585 nM
|
|
|
|
CP0318039
|
3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic acid ethyl ester
Show/Hide
|
C15H20N2O2
|
1
|
| 1 |
Ki = 1600 nM
|
|
|
|
CP0143981
|
N-[4-[[2-(4-fluorophenyl)cyclopropyl]methyl-propylamino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
|
C26H33ClFN3O
|
1
|
| 1 |
Ki = 1609 nM
|
|
|
|
CP0392147
|
3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-pyrrolo[2,3-f][3]benzazecine
Show/Hide
|
C17H22N2
|
1
|
| 1 |
Ki = 1647 nM
|
|
|
|
CP0253779
|
5-Iodo-benzofuran-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C23H24Cl2IN3O2
|
1
|
| 1 |
Ki = 1720 nM
|
|
|
|
CP0385310
|
US10913711, Compound 10j
Show/Hide
|
C28H32F2N2O2S
|
1
|
| 1 |
Ki = 1750 nM
|
|
|
|
CP0047599
|
Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
Show/Hide
|
C23H23Cl2N3OS
|
1
|
| 1 |
Ki = 1770 nM
|
|
|
|
CP0355151
|
N-[4-[[2-(5-chloro-2-methoxyphenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C30H37Cl2N3O2
|
1
|
| 1 |
Ki = 1833 nM
|
|
|
|
CP0293888
|
N-[(3S)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide
Show/Hide
|
C23H26Cl2N4O2
|
2
|
| 1 |
Ki = 1900 nM
|
|
|
| 2 |
Ki > 5000 nM
|
|
|
|
CP0288363
|
N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H30N4O3
|
1
|
| 1 |
Ki = 1920 nM
|
|
|
|
CP0449019
|
(1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-yl)methanol
Show/Hide
|
C21H23ClN2O
|
1
|
| 1 |
Ki = 1940 nM
|
|
|
|
CP0480200
|
N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-5-methyl-1H-imidazole-2-carboxamide
Show/Hide
|
C21H30ClN5O2
|
1
|
| 1 |
Ki = 1960 nM
|
|
|
|
CP0350422
|
N-[4-[[2-(2,3-dichlorophenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C29H34Cl3N3O
|
1
|
| 1 |
Ki = 2011 nM
|
|
|
|
CP0197218
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-5-methoxy-1H-indole-2-carboxamide
Show/Hide
|
C24H28Cl2N4O3
|
2
|
| 1 |
Ki = 2040 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0463737
|
N-[4-[propyl-[[2-[4-(trifluoromethyl)phenyl]cyclopropyl]methyl]amino]butyl]-1H-indole-2-carboxamide;hydrochloride
Show/Hide
|
C27H33ClF3N3O
|
1
|
| 1 |
Ki = 2073 nM
|
|
|
|
CP0771814
|
4-(2-(2-(2-Fluoroethoxy)ethoxy)ethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-l)butyl)benzamide oxalic acid salt
Show/Hide
|
C30H42FN3O9
|
1
|
| 1 |
Ki = 2100 nM
|
|
|
|
CP0369519
|
N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide
Show/Hide
|
C24H29N3O4
|
1
|
| 1 |
Ki = 2140 nM
|
|
|
|
CP0467820
|
1-((1H-indazol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-ol
Show/Hide
|
C19H20ClN3O
|
1
|
| 1 |
Ki = 2146 nM
|
|
|
|
CP0470998
|
N-[4-[propyl-[[2-[4-(trifluoromethyl)phenyl]cyclopropyl]methyl]amino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C30H35ClF3N3O
|
1
|
| 1 |
Ki = 2171 nM
|
|
|
|
CP0549074
|
N-[4-[[2-(4-fluorophenyl)cyclopropyl]methyl-propylamino]butyl]naphthalene-2-carboxamide;hydrochloride
Show/Hide
|
C28H34ClFN2O
|
1
|
| 1 |
Ki = 2171 nM
|
|
|
|
CP0470995
|
N-[4-[[2-(3-fluorophenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C29H35ClFN3O
|
1
|
| 1 |
Ki = 2222 nM
|
|
|
|
CP0919398
|
1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate
Show/Hide
|
C24H26N4O6
|
1
|
| 1 |
Ki = 2230 nM
|
|
|
|
CP0421765
|
1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidine-4-carbonitrile
Show/Hide
|
C21H20ClN3
|
1
|
| 1 |
Ki = 2270 nM
|
|
|
|
CP0427783
|
1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-amine
Show/Hide
|
C20H22ClN3
|
1
|
| 1 |
Ki = 2293 nM
|
|
|
|
CP0135681
|
1-(3-chloro-5-ethyl-2-methoxyphenyl)piperazine
Show/Hide
|
C13H19ClN2O
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0143980
|
N-[4-[[2-(3-chlorophenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C29H35Cl2N3O
|
1
|
| 1 |
Ki = 2326 nM
|
|
|
|
CP0156136
|
N-[4-[4-(2-chloro-5-methylphenyl)piperazin-1-yl]butyl]-2-oxo-3H-1,3-benzoxazole-5-carboxamide
Show/Hide
|
C23H27ClN4O3
|
1
|
| 1 |
Ki = 2370 nM
|
|
|
|
CP0250704
|
N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-1-benzofuran-2-carboxamide
Show/Hide
|
C25H30ClN3O3
|
1
|
| 1 |
Ki = 2380 nM
|
|
|
|
CP0372387
|
1-((1H-indol-3-yl)methyl)-3-(4-chlorophenyl)piperidin-3-ol
Show/Hide
|
C20H21ClN2O
|
1
|
| 1 |
Ki = 2440 nM
|
|
|
|
CP0136531
|
2-[[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl]-1-methylbenzimidazole
Show/Hide
|
C17H19ClN6
|
1
|
| 1 |
Ki = 2511.89 nM
|
|
|
|
CP0439090
|
2-[[4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]piperidin-1-yl]methyl]-1-methylbenzimidazole
Show/Hide
|
C20H20ClF3N4
|
1
|
| 1 |
Ki = 2511.89 nM
|
|
|
|
CP0392149
|
2,3-dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine
Show/Hide
|
C20H25NO2
|
1
|
| 1 |
Ki = 2514 nM
|
|
|
|
CP0057840
|
US8748608, 34
Show/Hide
|
C23H26Cl2N4O2
|
2
|
| 1 |
Ki = 2600 nM
|
|
|
| 2 |
Ki = 4900 nM
|
|
|
|
CP0414849
|
1-Benzyl-3-(1-benzyl-piperidin-4-yl)-urea
Show/Hide
|
C20H25N3O
|
1
|
| 1 |
Ki = 2700 nM
|
|
|
|
CP0445423
|
3-((4-(4-chlorophenyl)-4-methylpiperidin-1-yl)methyl)-1H-indole
Show/Hide
|
C21H23ClN2
|
1
|
| 1 |
Ki = 2750 nM
|
|
|
|
CP0449014
|
1-((1H-indol-3-yl)methyl)-4-(2-chlorophenyl)piperidin-4-ol
Show/Hide
|
C20H21ClN2O
|
1
|
| 1 |
Ki = 2820 nM
|
|
|
|
CP0431105
|
N-[4-[[2-(4-fluorophenyl)cyclopropyl]methyl-propylamino]butyl]-4-pyridin-2-ylbenzamide;hydrochloride
Show/Hide
|
C29H35ClFN3O
|
1
|
| 1 |
Ki = 2884 nM
|
|
|
|
CP0438521
|
N-[2-[(1S,2R)-2-[[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]methyl]cyclopropyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C25H31N5O2
|
2
|
| 1 |
Ki = 2930 nM
|
|
|
| 2 |
Ki = 62700 nM
|
|
|
|
CP0427930
|
4-(4-chlorophenyl)-1-((2-methyl-1H-indol-3-yl)methyl)piperidin-4-ol
Show/Hide
|
C21H23ClN2O
|
1
|
| 1 |
Ki = 2990 nM
|
|
|
|
CP0190972
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-4-pyridin-2-ylbenzamide
Show/Hide
|
C26H27Cl2FN4O
|
1
|
| 1 |
Ki = 3090 nM
|
|
|
|
CP0294037
|
N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-9H-fluorene-2-carboxamide
Show/Hide
|
C29H32FN3O2
|
1
|
| 1 |
Ki = 3180 nM
|
|
|
|
CP0382713
|
7-[4-[(5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
|
C23H30N4O3
|
1
|
| 1 |
Ki = 3220 nM
|
|
|
|
CP0258057
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1H-indole-2-carboxamide
Show/Hide
|
C23H25Cl2FN4O
|
1
|
| 1 |
Ki = 3360 nM
|
|
|
|
CP0122857
|
(R)-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-3-hydroxybutyl)-1H-indole-2-carboxamide
Show/Hide
|
C23H26Cl2N4O2
|
2
|
| 1 |
Ki = 3430 nM
|
|
|
| 2 |
Ki = 4000 nM
|
|
|
|
CP0409198
|
ethyl 4-(4-chlorophenyl)-1-(1H-indol-3-ylmethyl)piperidine-4-carboxylate
Show/Hide
|
C23H25ClN2O2
|
1
|
| 1 |
Ki = 3520 nM
|
|
|
|
CP0435244
|
1-((1H-indol-3-yl)methyl)-4-(3-chlorophenyl)piperidin-4-ol
Show/Hide
|
C20H21ClN2O
|
1
|
| 1 |
Ki = 3540 nM
|
|
|
|
CP0381742
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-9H-fluorene-3-carboxamide
Show/Hide
|
C28H29Cl2N3O2
|
1
|
| 1 |
Ki = 3670 nM
|
|
|
|
CP0079495
|
9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C28H29Cl2N3O
|
1
|
| 1 |
Ki = 3670 nM
|
|
|
|
CP0501761
|
1-((1H-indol-3-yl)methyl)-4-(3-(trifluoromethyl)phenyl)piperidin-4-ol
Show/Hide
|
C21H21F3N2O
|
1
|
| 1 |
Ki = 3750 nM
|
|
|
|
CP0464096
|
US10913711, Compound 10d
Show/Hide
|
C22H28F2N2O2S
|
1
|
| 1 |
Ki = 3820 nM
|
|
|
|
CP0467819
|
1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)azepan-4-ol
Show/Hide
|
C21H23ClN2O
|
1
|
| 1 |
Ki = 3870 nM
|
|
|
|
CP0372344
|
1-((1H-indol-3-yl)methyl)-4-(4-chlorobenzyl)piperidin-4-ol
Show/Hide
|
C21H23ClN2O
|
1
|
| 1 |
Ki = 3930 nM
|
|
|
|
CP0467821
|
methyl 4-(4-chlorophenyl)-1-(1H-indol-3-ylmethyl)piperidine-4-carboxylate
Show/Hide
|
C22H23ClN2O2
|
1
|
| 1 |
Ki = 3930 nM
|
|
|
|
CP0449020
|
N-[[4-(4-chlorophenyl)-1-(1H-indol-3-ylmethyl)piperidin-4-yl]methyl]acetamide
Show/Hide
|
C23H26ClN3O
|
1
|
| 1 |
Ki = 4450 nM
|
|
|
|
CP0433590
|
1-(2,3-dichlorophenyl)-4-[4-[1-(9H-fluoren-2-yl)triazol-4-yl]butyl]piperazine
Show/Hide
|
C29H29Cl2N5
|
1
|
| 1 |
Ki = 4450 nM
|
|
|
|
CP0064183
|
4-[3-methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy]furo[3,2-c]pyridine
Show/Hide
|
C21H16N4O2
|
1
|
| 1 |
Ki = 4500 nM
|
|
|
|
CP0041034
|
US8748608, 16
Show/Hide
|
C26H28Cl2N4O2
|
1
|
| 1 |
Ki = 4620 nM
|
|
|
|
CP0449653
|
1-Benzyl-2-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine
Show/Hide
|
C21H22ClN3
|
1
|
| 1 |
Ki = 4800 nM
|
|
|
|
CP0244206
|
7-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]thieno[2,3-c]pyridine
Show/Hide
|
C21H12F3N3OS
|
1
|
| 1 |
Ki = 4900 nM
|
|
|
|
CP0421988
|
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-pyridin-3-ylacetamide
Show/Hide
|
C16H18ClN5O
|
1
|
| 1 |
Ki = 5000 nM
|
|
|
|
CP0449015
|
4-(4-chlorophenyl)-1-((1-methyl-1H-indol-3-yl)methyl)piperidin-4-ol
Show/Hide
|
C21H23ClN2O
|
1
|
| 1 |
Ki = 5140 nM
|
|
|
|
CP0443872
|
N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-hydroxybutyl]-1-benzofuran-2-carboxamide
Show/Hide
|
C26H32ClN3O4
|
1
|
| 1 |
Ki = 5290 nM
|
|
|
|
CP0243806
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzofuran-2-carboxamide
Show/Hide
|
C23H24Cl2FN3O2
|
1
|
| 1 |
Ki = 5340 nM
|
|
|
|
CP0157764
|
N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
Ki = 5520 nM
|
|
|
|
CP0449026
|
1-((1H-indol-3-yl)methyl)-4-(4-fluorophenyl)piperidin-4-ol
Show/Hide
|
C20H21FN2O
|
1
|
| 1 |
Ki = 6090 nM
|
|
|
|
CP0451512
|
1-[4-[2-[bis(4-fluorophenyl)methylsulfanyl]ethyl]piperazin-1-yl]propan-2-ol
Show/Hide
|
C22H28F2N2OS
|
1
|
| 1 |
Ki = 6300 nM
|
|
|
|
CP0384381
|
N-pyridin-3-yl-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide
Show/Hide
|
C16H19N5O
|
1
|
| 1 |
Ki = 6407 nM
|
|
|
|
CP0064188
|
4-[4-(6-methylimidazo[1,2-a]pyrazin-5-yl)-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
Show/Hide
|
C21H13F3N4O2
|
1
|
| 1 |
Ki = 6900 nM
|
|
|
|
CP0369306
|
4-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
Show/Hide
|
C21H12F3N3O2
|
1
|
| 1 |
Ki = 6900 nM
|
|
|
|
CP0372388
|
4-(4-chlorophenyl)-1-((1-hexyl-1H-indol-3-yl)methyl)piperidin-4-ol
Show/Hide
|
C26H33ClN2O
|
1
|
| 1 |
Ki = 8890 nM
|
|
|
|
CP0426667
|
1-[[(2R)-3,3-diphenyl-1,4-dioxan-2-yl]methyl]-4-(2-methoxyphenyl)piperazine
Show/Hide
|
C28H32N2O3
|
1
|
| 1 |
Ki = 9772.37 nM
|
|
|
|
CP0091917
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-5-iodo-1H-indole-2-carboxamide
Show/Hide
|
C23H25Cl2IN4O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0197219
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-1-benzofuran-2-carboxamide
Show/Hide
|
C23H25Cl2N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0288360
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-5-iodo-1-benzofuran-2-carboxamide
Show/Hide
|
C23H24Cl2IN3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0919396
|
1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate
Show/Hide
|
C23H26N2O6
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0002070
|
1-(1H-Indol-3-yl)-2-propanamine
Show/Hide
|
C11H14N2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0002071
|
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-N-prop-2-enylprop-2-en-1-amine
Show/Hide
|
C17H22N2O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0864137
|
1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-butyl)-4-(2,3-dichlorophenyl)piperazine
Show/Hide
|
C28H29Cl2N5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0075581
|
N-[4-[4-(3,5-dichlorophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide
Show/Hide
|
C25H27Cl2N3OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0434495
|
N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]imidazo[1,2-a]pyridine-2-carboxamide
Show/Hide
|
C24H30ClN5O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0157762
|
N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide
Show/Hide
|
C26H33ClN4O3
|
1
|
| 1 |
Ki = 13900 nM
|
|
|
|
CP0414817
|
N-[(3S)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzofuran-2-carboxamide
Show/Hide
|
C23H24Cl2FN3O2
|
1
|
| 1 |
Ki > 14000 nM
|
|
|
|
CP0372386
|
(1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-yl)methanamine
Show/Hide
|
C21H24ClN3
|
1
|
| 1 |
Ki > 20000 nM
|
|
|
|
CP0501799
|
1-((1H-indol-2-yl)methyl)-4-(4-chlorophenyl)piperidin-4-ol
Show/Hide
|
C20H21ClN2O
|
1
|
| 1 |
Ki > 20000 nM
|
|
|
|
CP0389182
|
1-(2,3-dichlorophenyl)-4-[4-[4-(9H-fluoren-2-yl)triazol-1-yl]butyl]piperazine
Show/Hide
|
C29H29Cl2N5
|
1
|
| 1 |
Ki > 20000 nM
|
|
|
|
CP0397790
|
1-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-(4-naphthalen-2-yltriazol-1-yl)butan-2-ol
Show/Hide
|
C26H27Cl2N5O
|
1
|
| 1 |
Ki > 20000 nM
|
|
|
|
CP0456678
|
5-[5-[3-[(1S,5R)-1-[2-fluoro-4-(trifluoromethyl)phenyl]-3-azabicyclo[3.1.0]hexan-3-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
Show/Hide
|
C22H23F4N5OS
|
1
|
| 1 |
Ki = 35600 nM
|
|
|
|
CP0384383
|
2-(4-pyridin-2-ylpiperazin-1-yl)-N-pyrimidin-5-ylacetamide
Show/Hide
|
C15H18N6O
|
1
|
| 1 |
Ki = 39290 nM
|
|
|
|
CP0384678
|
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-pyrimidin-5-ylacetamide
Show/Hide
|
C15H17ClN6O
|
1
|
| 1 |
Ki > 50000 nM
|
|
|
|
CP0390315
|
(R)-Modafinil
Show/Hide
|
C15H15NO2S
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
|
CP0467854
|
5-[(5S)-5-methyl-4-propylmorpholin-2-yl]-N,N-dipropylpyridin-2-amine
Show/Hide
|
C19H33N3O
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
|
CP0410750
|
6-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]isoquinoline
Show/Hide
|
C26H30N6O
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0410751
|
4-[4-(9H-fluoren-2-yl)triazol-1-yl]-1-[4-(2-methoxyphenyl)piperazin-1-yl]butan-2-ol
Show/Hide
|
C30H33N5O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0547198
|
1-(2,3-dichlorophenyl)-4-[4-(4-naphthalen-2-yltriazol-1-yl)butyl]piperazine
Show/Hide
|
C26H27Cl2N5
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0909483
|
6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline
Show/Hide
|
C25H26Cl2N6
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0504457
|
4-(4-chlorophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol
Show/Hide
|
C21H23ClN2O2
|
1
|
| 1 |
Ki > 2000 nM
|
|
|
|
CP0389180
|
1-(2,3-dichlorophenyl)-4-[4-(1-naphthalen-2-yltriazol-4-yl)butyl]piperazine
Show/Hide
|
C26H27Cl2N5
|
1
|
| 1 |
Ki > 2000 nM
|
|
|
|
CP0410753
|
1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-(4-naphthalen-2-yltriazol-1-yl)butan-2-ol
Show/Hide
|
C27H31N5O2
|
1
|
| 1 |
Ki > 2000 nM
|
|
|
|
CP0433565
|
1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-[4-(4-phenylphenyl)triazol-1-yl]butan-2-ol
Show/Hide
|
C29H33N5O2
|
1
|
| 1 |
Ki > 2000 nM
|
|
|
|
CP0443217
|
5-[1-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]triazol-4-yl]-1H-indole
Show/Hide
|
C24H26Cl2N6
|
1
|
| 1 |
Ki > 2000 nM
|
|
|
|
CP0380824
|
5-Methyl-1-(1-methyl-piperidin-4-yl)-4-phenyl-1,3-dihydro-imidazol-2-one
Show/Hide
|
C16H21N3O
|
1
|
| 1 |
Ki > 2500 nM
|
|
|
|
CP0410131
|
N-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-fluorobutyl]-1-benzofuran-2-carboxamide
Show/Hide
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C23H24Cl2FN3O2
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1
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| 1 |
Ki > 3000 nM
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CP0381741
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1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-(4-phenyltriazol-1-yl)butan-2-ol
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C23H29N5O2
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1
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| 1 |
Ki > 3000 nM
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CP0381747
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1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-(4-quinolin-6-yltriazol-1-yl)butan-2-ol
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C26H30N6O2
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1
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| 1 |
Ki > 3000 nM
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CP0443218
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1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-[4-(2-methoxyphenyl)triazol-1-yl]butan-2-ol
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C24H31N5O3
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1
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| 1 |
Ki > 3000 nM
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CP0045069
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2-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-N,N-dimethylethanamine
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C19H22N2O3S
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1
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| 1 |
Ki > 3200 nM
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CP0186950
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(4S,5S)-4-Dimethylamino-1-(toluene-4-sulfonyl)-1,3,4,5-tetrahydro-benzo[cd]indol-5-ol
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C20H22N2O3S
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1
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| 1 |
Ki > 3200 nM
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CP0255950
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2-[1-(benzenesulfonyl)indol-3-yl]-N,N-dimethylethanamine
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C18H20N2O2S
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1
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| 1 |
Ki > 3200 nM
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CP0330654
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2-[1-(benzenesulfonyl)indol-4-yl]-N,N-dimethylethanamine
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C18H20N2O2S
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1
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| 1 |
Ki > 3200 nM
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CP0379189
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2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine
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C16H16N2O2S
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1
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| 1 |
Ki > 3200 nM
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CP0418991
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[1-(benzenesulfonyl)-4-[2-(dimethylamino)ethyl]indol-2-yl]-phenylmethanone
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C25H24N2O3S
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1
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| 1 |
Ki > 3200 nM
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CP0442957
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4-[3-(4-CHLOROPHENYL)-1H-PYRAZOL-5-YL]PIPERIDINE
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C14H16ClN3
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1
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| 1 |
Ki > 3300 nM
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CP0504160
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4-(4-chlorophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol
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C21H23ClN2O2
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1
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| 1 |
Ki > 3500 nM
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CP0409092
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[3-[2-(dimethylamino)ethyl]-5-hydroxyindol-1-yl]-phenylmethanone
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C19H20N2O2
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1
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| 1 |
Ki > 3900 nM
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CP0392142
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7-cyclopropylmethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine
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C23H26N2
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1
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| 1 |
Ki > 5000 nM
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CP0156829
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N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-5-fluoro-1H-indole-2-carboxamide
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C23H25Cl2FN4O2
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1
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| 1 |
Ki > 5000 nM
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CP0389447
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1-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-[4-(4-phenylphenyl)triazol-1-yl]butan-2-ol
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C28H29Cl2N5O
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1
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| 1 |
Ki > 7000 nM
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CP0410937
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N-[(3R)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzofuran-2-carboxamide
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C23H24Cl2FN3O2
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1
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| 1 |
Ki > 9000 nM
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