Brief Information of the Compound and Protein
Compound Name
2-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
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PubChem ID
CID: 9945233
SID: 14919672
Canonical SMILES
Clc1ccccc1N1CCN(Cc2nc3ccccc3[nH]2)CC1
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Compound Formula C18H19ClN4
Compound Structure
Protein Name
D(4) dopamine receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Dopamine receptor
Uniprot ID
P21917
Gene Name
DRD4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 7.2 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 1 nM
2 Ki = 8.5 nM