Brief Information of the Compound and Protein
Compound Name
2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-benzoimidazole
    Show/Hide
PubChem ID
CID: 4826074
SID: 14821537
Canonical SMILES
COc1ccccc1N1CCN(Cc2nc3ccccc3[nH]2)CC1
    Show/Hide
Compound Formula C19H22N4O
Compound Structure
Protein Name
D(4) dopamine receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Dopamine receptor
Uniprot ID
P21917
Gene Name
DRD4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 12.4 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 5.6 nM
2 Ki = 4.3 nM