Brief Information of the Compound and Protein
Compound Name
2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-m-tolyl-acetamide
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PubChem ID
CID: 2653640
SID: 14952107
Canonical SMILES
COc1ccccc1N1CCN(CC(=O)Nc2cccc(C)c2)CC1
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Compound Formula C20H25N3O2
Compound Structure
Protein Name
D(4) dopamine receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Dopamine receptor
Uniprot ID
P21917
Gene Name
DRD4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 26.8 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 0.7 nM
2 Ki = 1.8 nM