| Compound ID |
Compound Name |
Compound Formula |
|
CP0016788
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 9
Show/Hide
|
C28H32FN7O2
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0025678
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 8
Show/Hide
|
C28H32FN7O2
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0510158
|
4,5-difluoro-2-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C27H30F2N8O2
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0262632
|
2-[(2-{[2-methoxy-4-(1-propyl-1,2,5,6-tetrahydropyridin-3-yl)phenyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide
Show/Hide
|
C28H31N7O2
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0020296
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 25
Show/Hide
|
C27H31FN8O2
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0299598
|
2,4-difluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C27H30F2N8O2
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0336151
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 11
Show/Hide
|
C27H31FN8O2
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0423062
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 6
Show/Hide
|
C28H30FN7O2
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0435096
|
2-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C27H32N8O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0299597
|
2,3-difluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C27H30F2N8O2
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0158666
|
2-[(2-{[2-fluoro-4-(1-propyl-1,2,5,6-tetrahydropyridin-3-yl)phenyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide
Show/Hide
|
C27H28FN7O
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0291060
|
2-[(2-{[4-(1-propyl-1,2,5,6-tetrahydropyridin-3-yl)phenyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide
Show/Hide
|
C27H29N7O
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0503001
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 12
Show/Hide
|
C24H24FN7O3
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0510157
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 10
Show/Hide
|
C27H31FN8O2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0526611
|
2-{[2-({5-chloro-2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-6-fluorobenzamide
Show/Hide
|
C27H30ClFN8O2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0037058
|
2-fluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C27H31FN8O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0386171
|
2-fluoro-6-{[2-({5-fluoro-2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C27H30F2N8O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0488073
|
2-fluoro-6-{[2-({2-methoxy-5-methyl-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C28H33FN8O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0435099
|
2-{[2-({2,5-dimethoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-6-fluorobenzamide
Show/Hide
|
C28H33FN8O3
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0463888
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 30
Show/Hide
|
C28H33FN8O2
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0531897
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 7
Show/Hide
|
C30H34FN7O2
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0070412
|
2-fluoro-6-{[2-({2-methoxy-5-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C27H31FN8O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0489779
|
2-fluoro-6-{[2-({3-fluoro-2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C27H30F2N8O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0375704
|
1-(3-(5-(4-((2-(dimethylamino)ethyl)carbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-phenoxyphenyl)urea
Show/Hide
|
C37H34N6O3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0505154
|
1-(3-(5-(3-((2-(dimethylamino)ethyl)carbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-phenoxyphenyl)urea
Show/Hide
|
C37H34N6O3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0016657
|
2-[(2-{[2-methyl-4-(1-propyl-1,2,5,6-tetrahydropyridin-3-yl)phenyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide
Show/Hide
|
C28H31N7O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0510159
|
2-fluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-N-methylbenzamide
Show/Hide
|
C28H33FN8O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0526613
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 33
Show/Hide
|
C29H35FN8O3
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0503291
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 31
Show/Hide
|
C27H31FN8O3
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0481506
|
2-fluoro-6-{[2-({2-methoxy-3-methyl-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C28H33FN8O2
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0547617
|
1-(3-(5-(4-(aminomethyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-phenoxyphenyl)urea
Show/Hide
|
C33H27N5O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0026276
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 32
Show/Hide
|
C30H37FN8O4
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0139071
|
2-fluoro-6-{[2-({2-methoxy-4-methyl-5-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C28H33FN8O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0526176
|
2-[(2-{[4-(1-propyl-1,2,5,6-tetrahydropyridin-3-yl)-2-(trifluoromethyl)phenyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide
Show/Hide
|
C28H28F3N7O
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0521169
|
1-(3-(5-(4-(aminomethyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(3-chlorophenyl)urea
Show/Hide
|
C27H22ClN5O
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0514452
|
N,N-dimethyl-3-[3-[3-[(2-phenoxyphenyl)carbamoylamino]phenyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]benzamide
Show/Hide
|
C35H29N5O3
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0435091
|
4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine, 34
Show/Hide
|
C30H37FN8O3
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0431057
|
1-(3-(5-(4-(dimethylcarbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-phenoxyphenyl)urea
Show/Hide
|
C35H29N5O3
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0514451
|
1-(3-(5-(4-((2-(dimethylamino)ethyl)carbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-fluoro-4-(trifluoromethyl)phenyl)urea
Show/Hide
|
C32H28F4N6O2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0505155
|
1-(3-(5-(3-(dimethylcarbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-(phenylamino)phenyl)urea
Show/Hide
|
C35H30N6O2
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0552080
|
2-fluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}(methyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C28H33FN8O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0295931
|
1-(3-(5-(4-(aminomethyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-fluoro-4-(trifluoromethyl)phenyl)urea
Show/Hide
|
C28H21F4N5O
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0474664
|
1-[3-[5-[3-(dimethylsulfamoyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl]phenyl]-3-(2-phenoxyphenyl)urea
Show/Hide
|
C34H29N5O4S
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0505156
|
3-{3-[3-(3-Biphenyl-2-yl-ureido)-phenyl]-1H-pyrrolo[2,3-b]pyridin-5-yl}-N,N-dimethyl-benzamide
Show/Hide
|
C35H29N5O2
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0375703
|
1-(3-(5-(3-((2-(dimethylamino)ethyl)carbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-fluoro-4-(trifluoromethyl)phenyl)urea
Show/Hide
|
C32H28F4N6O2
|
1
|
| 1 |
IC50 = 67 nM
|
|
|
|
CP0040803
|
N-(2,6-difluorophenyl)-5-[3-[2-[5-ethyl-2-methoxy-4-[4-(4-methylsulfonylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]-2-methoxybenzamide
Show/Hide
|
C44H47F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0040804
|
3-(3-(2-(4-(1,4'-bipiperidin-1'-yl)-2-methoxyphenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H40F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0042282
|
N-(2,6-difluorophenyl)-3-[3-[2-[5-ethyl-2-methoxy-4-[4-(4-methylsulfonylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H45F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0069911
|
N-(2,6-difluorophenyl)-3-[3-[2-[2-methoxy-4-[4-(4-methylsulfonylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H41F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0177146
|
3-(3-(2-(4-(1,4'-bipiperidin-1'-yl)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C40H38F2N8O
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0380415
|
(R)-N-(2,6-difluorophenyl)-3-(3-(2-(4-(4-(3-fluoropyrrolidin-1-yl)piperidin-1-yl)-2-methoxyphenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H37F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0388757
|
N-(2,6-difluorophenyl)-3-[3-[2-[4-[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0444853
|
N-(2,6-difluorophenyl)-3-[3-[2-[2-methoxy-4-(4-morpholin-4-ylpiperidin-1-yl)anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H38F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0461635
|
N-(2,6-difluorophenyl)-3-[3-[2-[3-[2-(dimethylamino)ethoxy]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C34H29F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0461636
|
3-(3-(2-(4-(4-(4-acetylpiperazin-1-yl)piperidin-1-yl)-2-methoxyphenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H41F2N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0475298
|
N-(2,6-difluorophenyl)-3-[3-[2-[2-methoxy-4-(4-pyrrolidin-1-ylpiperidin-1-yl)anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H38F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0509038
|
N-(2,6-difluorophenyl)-3-[3-[2-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H41F2N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845764
|
3-[3-(2-{[4-(1,4'-bipiperidin-l'-yl)-2-methylphenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H40F2N8O
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845773
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(4-thiomorpholinyl)-1-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C40H38F2N8O2S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845774
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[(9aS)-hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H43F2N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845775
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[1-(2-fluoroethyl)-4-piperidinyl]-1-piperazinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845776
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(cis-4-{4-[2-(methylsulfonyl)-ethyl]-1-piperazinyl}cyclohexyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845777
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{1'-[2-(methylsulfonyl)ethyl]-4,4'-bipiperidin-1-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C45H48F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845778
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2,5-bis(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845779
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(ethyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazin-yl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H47F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845780
|
N-(2,6-difluorophenyl)-3-{3-[2-({4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)-2-[(2,2,2-trifluoroethyl)oxy]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C44H44F5N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845781
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(methyloxy)-1-piperidinyl]phenyl}-amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C37H33F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845782
|
N-(2,6-difluorophenyl)-5-[3-(2-{[2-(ethyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845783
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[2-(ethyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H43F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845802
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{1'-[2-(methylsulfonyl)ethyl]-4,4'-bipiperidin-1-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845803
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{1'-[2-(methylsulfonyl)ethyl]-1,4'-bipiperidin-4-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845804
|
N-(2,6-difluorophenyl)-3-(3-(2-((2-(methyloxy)-4-(4-(2-(methylsulfonyl)ethyl)-1,4'-bipiperidin-1'-yl)phenyl)amino)-4-pyrimidinyl)imidazo(1,2-a)pyridin-2-yl)benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845805
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-chloro-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H39ClF2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845806
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845807
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2,5-bis(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H44F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845808
|
N-(2,6-difluorophenyl)-5-{3-[2-({5-fluoro-2-(methyloxy)-4-[2-(1-piperidinyl)ethyl]phenyl}-amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
|
C39H36F3N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845809
|
3-{3-[2-({5-fluoro-2-(methyloxy)-4-[2-(1-piperidinyl)ethyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-N-(2,4,6-trifluorophenyl)benzamide
Show/Hide
|
C38H33F4N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845810
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-{3-[2-({2-(methyloxy)-4-[2-(4-methyl-1-piperazinyl)ethyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845836
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[3-(1-piperidinyl)propyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C39H37F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845845
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C43H45F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845847
|
3-[3-(2-{[4-(1,4'-bipiperidin-l'-yl)-2-(ethyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845849
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(1-piperidinylmethyl)-1-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848311
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H40F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848312
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[(3S)-3-fluoro-1-pyrrolidinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H37F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848316
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[(3R)-3-hydroxy-1-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C36H31F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848317
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H37F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848319
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C43H45F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848469
|
3-{3-[2-({4-(1,4'-bipiperidin-1'-yl)-2-[(2-methylpropyl)oxy]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C44H46F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848470
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H44F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848471
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-[4-(l-methylethyl)-1-piperazinyl]-2-(methyloxy)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C39H38F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848486
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[5-methyl-2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H43F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848489
|
N-(2,6-difluorophenyl)-3-(3-(2-(2-methyl-4-(1-methylpiperidin-4-yloxy)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C37H33F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848526
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-(4-methyl-1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848527
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-3-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(ethyloxy)benzamide
Show/Hide
|
C44H46F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848528
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848529
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H46F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848530
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-(4-hydroxy-1,4'-bipiperidin-1'-yl)-2-(methyloxy)-phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848531
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[1'-(2-fluoroethyl)-4,4'-bipiperidin-1-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H43F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848532
|
N-(2,6-difluorophenyl)-3-[3-(2-{[5-methyl-2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H39F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848534
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
|
C43H46F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848538
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-methyl-4-(4-piperidinyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C36H31F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848539
|
N-(2,3-difluorophenyl)-3-[3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C35H31F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856490
|
3-{3-[2-({4-(1,4'-bipiperidin-1'-yl)-2-[(1-methylethyl)oxy]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C43H44F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856492
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-8-methylimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856495
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[(9aS)-hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C38H34F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856496
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidin}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H41F6N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856497
|
N-(2,6-difluorophenyl)-3-(7-fluoro-3-(2-((2-(methyloxy)-4-(4-(4-(methylsulfonyl)-1-piperazinyl)-1-piperidinyl)phenyl)amino)-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H40F3N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856498
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-fluoroimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C42H41F3N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856500
|
N-(2,6-difluorophenyl)-5-{3-[2-({5-methyl-2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
|
C39H38F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856509
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-2-propylphenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C43H45F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856510
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C41H42F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856511
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-8-fluoroimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H39F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856513
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]hexahydro-1H-1,4-diazepin-1-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H44F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857311
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C40H40F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857313
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857314
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C45H49F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857317
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[3-(1-piperidinyl)propyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C40H39F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857318
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[3-(4-methyl-1-piperazinyl)propyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C39H38F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857319
|
N-(2,6-difluorophenyl)-5-{3-[2-({2-(ethyloxy)-4-[2-(4-methyl-1-piperazinyl)ethyl]-phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
|
C38H36F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857321
|
N-(2,6-difluorophenyl)-3-(3-{2-[(5-methyl-2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H39F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857322
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-[3-(2-{[2-(methyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C39H38F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857323
|
N-(2,6-difluorophenyl)-3-[8-fluoro-3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H41F4N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857326
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C44H47F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857327
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0857328
|
N-(2,6-difluorophenyl)-2-((1-methylethyl)oxy)-5-(3-(2-((2-(methyloxy)-4-(4-(4-(methylsulfonyl)-1-piperazinyl)-1-piperidinyl)phenyl)amino)-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C44H47F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0861201
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-{(3S)-3-(1-methylethyl)-4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C42H44F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0861239
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[1'-(2-fluoroethyl)-1,4'-bipiperidin-4-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H43F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0861240
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-[(9aS)-hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)-benzamide
Show/Hide
|
C39H36F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0861241
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H39F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0861242
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H40F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0863036
|
N-(2,6-difluorophenyL)-3-[8-methyl-3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H47F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0863038
|
N-(2,6-difluorophenyl)-5-{3-[2-({2-methyl-3-[(4-methyl-1-piperazinyl)methyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
|
C38H36F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0863042
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[1-(2-fluoroethyl)-4-piperidinyl]-1-piperazinyl]phenyl)amino}-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C43H44F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866109
|
N-(2,6-difluorophenyl)-5-(7-fluoro-3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C40H38F3N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866110
|
N-(2,6-difluorophenyl)-5-[3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C36H33F2N7O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866111
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C38H36F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866112
|
N-(2,6-difluorophenyl)-3-{3-[2-({5-methyl-2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C37H34F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866113
|
N-(2,6-difluorophenyl)-3-(3-(2-((5-methyl-2-(methyloxy)-4-(4-(2-(methylsulfonyl)ethyl)-1-piperidinyl)phenyl)amino)-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H39F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866114
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C37H34F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866115
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H42F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866116
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H39F5N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866958
|
N-(2,6-difluorophenyl)-3-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866959
|
N-(2,6-difluorophenyl)-3-[3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C35H31F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866960
|
3-[3-(2-{[4-(4-{bis[2-(methyloxy)ethyl]amino}-1-piperidinyl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H44F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866983
|
N-(2,6-difluorophenyl)-3-[3-(2-{[5-methyl-2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H47F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866984
|
3-[3-(2-{[4-{4-[4-(2,2-difluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(ethyloxy)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C43H43F4N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866985
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[4-(3,3,3-trifluoropropyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C44H44F5N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866986
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-(4-hydroxy-1-piperidinyl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C37H33F2N7O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866987
|
N-(2,6-difluorophenyl)-3-{3-[2-({5-fluoro-2-(methyloxy)-4-[2-(1-piperidinyl)ethyl]phenyl}-amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C38H34F3N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866988
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C40H40F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866989
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H42F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866990
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H38F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866991
|
N-(2,6-difluorophenyl)-3-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H38F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866992
|
N-(2,6-difluorophenyl)-3-(3-(2-((2-(ethyloxy)-4-(4-(1-methylethyl)-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H38F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866994
|
N-(2,6-difluorophenyl)-3-(8-fluoro-3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H40F3N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866995
|
N-(2,6-difluorophenyl)-3-[7-fluoro-3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H41F4N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866996
|
5-(3-{2-[(5-chloro-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C39H37ClF2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0866997
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C42H43F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0867011
|
5-(3-(2-(4-(1,4'-bipiperidin-1'-yl)-2-methoxyphenylamino)pyrimidin-4-yl)-7-methoxyimidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)-2-methoxybenzamide
Show/Hide
|
C43H44F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0867154
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H44F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0867164
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(propyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyri-din-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C43H44F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0867165
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H45F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0867166
|
3-[3-(2-{[5-chloro-4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H41ClF3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0869257
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-[3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)-ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo-[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H47F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0869420
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H42F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0870269
|
N-(2,6-difluorophenyl)-3-(3-(2-(3-(1-methyl-1H-pyrazol-4-yl)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C34H24F2N8O
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0870972
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C42H43F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0870973
|
N-(2,6-difluorophenyl)-5-(7-fluoro-3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C41H40F3N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0870974
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H41F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0870978
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[2-(methyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0870979
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0870980
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C43H45F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0870983
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C41H41F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0871077
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-fluoro-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C42H41F3N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0871078
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C40H40F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873426
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-fluoro-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H39F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873427
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[1-(2-methylpropyl)-4-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C40H39F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873428
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[(3S)-3-hydroxyl-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C36H31F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873429
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-[1-(2-fluoroethyl)-4-piperidinyl]-2-(methyloxy)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C39H36F3N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873430
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C43H45F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873431
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873432
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(2-methylpropyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C44H46F2N8O
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873433
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[4-(hexahydro-1H-azepin-1-yl)-1-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873434
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(trifluoromethyl)-1,4'-bipiperidin-1'-yl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C42H39F5N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873436
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[4-(4-ethyl-1-piperazinyl)-1-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H43F2N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873438
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873679
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C38H36F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873682
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[4-(methyloxy)-1-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C38H35F2N7O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873683
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-3-oxo-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H40F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873684
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C39H37F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0873685
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(ethyloxy)-4-[2-(4-methyl-1-piperazinyl)ethyl]-phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C37H34F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0882930
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-[3-(2-{[2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H39F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0882931
|
N-(2,6-difluorophenyl)-5-[3-(2-{[2-(ethyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C41H41F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0883050
|
5-[3-(2-{[5-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C42H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0883053
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(4-chloro-2-fluorophenyl)benzamide
Show/Hide
|
C41H40ClFN8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0883055
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[1-(2-methylpropyl)-4-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C41H41F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0883056
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[4-[4-(1-methylethyl)-1-piperazinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0883073
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoro-ethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-8-methylimidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H44F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0883074
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)-ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C45H49F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0883075
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-{4-[(9aS)-hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C44H45F2N9O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0888258
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H38F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0888352
|
N-(2,6-difluorophenyl)-3-[8-fluoro-3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H44F3N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0888393
|
5-(3-(2-(4-(1,4'-bipiperidin-1'-yl)-2-methoxyphenylamino)pyrimidin-4-yl)-7-methylimidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)-2-methoxybenzamide
Show/Hide
|
C43H44F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0888394
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{5-[(dimethylamino)methyl]-1,3,4-oxadiazol-2-yl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C36H29F2N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0888395
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-propylphenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C43H44F2N8O
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0894025
|
N-(2,6-difluorophenyl)-3-(8-methyl-3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0894026
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[(3S)-3-hydroxy-1,4'-bipiperidin-1'-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0895685
|
N-(2,6-difluorophenyl)-3-(3-(2-(2-methyl-4-(1-(2-(methylsulfonyl)ethyl)piperidin-4-yloxy)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H37F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0895686
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[(1S,4S)-5-(2-fluoroethyl)-2,5-diazabicyclo-[2.2.1]hept-2-yl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H42F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0895687
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1,4'-bipiperidin-1'-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C45H48F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0895688
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C43H44F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0895690
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C38H36F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0895691
|
N-(2,6-difluorophenyl)-5-[7-fluoro-3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C43H43F4N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0895693
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0895724
|
N-(2,6-difluorophenyl)-5-(3-(2-(3-(2-(dimethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-7-methylimidazo[1,2-a]pyridin-2-yl)-2-methoxybenzamide
Show/Hide
|
C36H33F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0899488
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H41F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0899576
|
N-(2,4-difluorophenyl)-3-(3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C34H29F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0899577
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[5-(1-pyrrolidinylmethyl)-1,3,4-oxadiazol-2-yl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C38H31F2N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0899726
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H39F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0899730
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C42H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0899732
|
N-(2,6-difluorophenyl)-3-(3-{2-[(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-2-propylphenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H41F2N7O3S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0901852
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H37F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0901853
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H41F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0902860
|
3-[3-(2-{[5-chloro-2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-benzamide
Show/Hide
|
C43H44ClF2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0902861
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[2-(4-methyl-1-piperazinyl)ethyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C39H38F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0904970
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(ethyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H39F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0904973
|
N-(2,6-difluorophenyl)-5-(3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)-amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C35H31F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0904974
|
3-(3-(2-(3-(2-(dimethylamino)ethoxy)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)-N-(2-fluoro-5-(trifluoromethyl)phenyl)benzamide
Show/Hide
|
C35H29F4N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0904975
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-(4-hydroxy-1-piperidinyl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C36H31F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0904977
|
3-[3-(2-{[4-(3,3-difluoro-1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H38F4N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0904979
|
N-(2,6-difluorophenyl)-3-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H38F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0904980
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C41H42F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0912085
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(trans-4-{4-[2-(methylsulfonyl)-ethyl]-1-piperazinyl}cyclohexyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0912086
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[3-(4-methyl-1-piperazinyl)propyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0912113
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-methylimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0912114
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H45F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0912115
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(4-morpholinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C35H29F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0912117
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-5-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H44F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913017
|
N-(2,6-difluorophenyl)-3-(3-(2-(2-methoxy-4-(4-(4-methyl-1,4-diazepan-1-yl)piperidin-1-yl)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913018
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[4-(dimethylamino)-1-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C38H36F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913019
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-[(3S)-3-hydroxy-1,4'-bipiperidin-1'-yl]-2-(methyloxy)-phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C42H42F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913020
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(ethyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C39H38F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913021
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl]-2-propylphenyl)amino}-4-pyrimidinyl}imidazo[1,2a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913022
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H39F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913023
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
|
C42H44F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913162
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C43H44F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913163
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-fluoroimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H39F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913164
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}-7-fluoroimidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C42H42F3N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913166
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-{3-[2-({2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C38H36F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913167
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{4-[(4-methyl-1-piperazinyl)methyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C42H43F2N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0913168
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-3-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C43H44F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0914898
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[4-(1-methylethyl)-1-piperazinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C38H36F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0919429
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C41H41F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0919430
|
N-(2,6-difluorophenyl)-5-(7-fluoro-3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C42H42F3N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0919431
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C36H32F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0920901
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-{3-[2-({2-(methyloxy)-4-[1-(2-methylpropyl)-4-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C42H43F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921732
|
N-(2,6-difluorophenyl)-3-(3-(2-(2-methyl-3-((4-methylpiperazin-1-yl)methyl)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C37H34F2N8O
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921733
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-3-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921734
|
N-(2,6-difluorophenyl)-5-{3-[2-({2-(ethyloxy)-4-[4-(1-methylethyl)-1-piperazinyl]phenyl}-amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
|
C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921735
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C41H41F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921758
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,4-difluorophenyl)benzamide
Show/Hide
|
C41H40F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921759
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-(4-hydroxy-1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C42H42F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0923164
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-{5-[(dimethylamino)methyl]-1,3,4-oxadiazol-2-yl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C37H31F2N9O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0923165
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-(4-fluoro-1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H39F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0924021
|
N-(5-chloro-2-fluorophenyl)-3-(3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C34H29ClFN7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0924036
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[2-(ethyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0926153
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2-chloro-4-fluorophenyl)benzamide
Show/Hide
|
C41H40ClFN8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0926162
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1,4'-bipiperidin-1'-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C46H50F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0926163
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-chloro-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C42H41ClF2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0926165
|
3-(3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-N-(2,4,6-trifluorophenyl)benzamide
Show/Hide
|
C34H28F3N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0926166
|
N-(2,6-difluorophenyl)-3-(3-{2-[(5-{[2-(dimethylamino)ethyl]oxy}-2-methylphenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C35H31F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0928839
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C43H44F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0928844
|
N-(2,6-difluorophenyl)-3-(3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}-2-methylphenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C35H31F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0928845
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[5-(1-pryrrolidinylmethyl)-1,3,4-oxa-diazol-2-yl]-phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C39H33F2N9O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0928846
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-ethylphenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0928847
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-[1'-(2-fluoroethyl)-4,4'-bipiperidin-1-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C44H45F3N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0929056
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(ethyloxy)-4-(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H47F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0929069
|
5-(3-{2-[(5-chloro-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)-2-(ethyloxy)benzamide
Show/Hide
|
C41H41ClF2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0944890
|
N-(2,6-difluorophenyl)-3-(3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}-7-methylimidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C35H31F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0944891
|
3-[3-(2-{[5-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H40F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0944904
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H38F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0946200
|
N-(2,6-difluorophenyl)-5-[3-(2-{[5-methyl-2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C41H41F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0946229
|
N-(2,6-difluorophenyl)-2-isopropoxy-5-{3-[2-({2-methoxy-4-[2-(4-methylpiperazin-1-yl)ethyl]phenyl}amino)pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C41H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0947312
|
N-(2,6-difluorophenyl)-5-{3-[2-({5-fluoro-2-(methyloxy)-4-[2-(4-morpholinyl)ethyl]phenyl}-amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
|
C38H34F3N7O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0952419
|
N-(2,4-difluorophenyl)-3-[3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C35H31F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0952675
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[2-(4-methyl-1-piperazinyl)ethyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C38H36F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0510553
|
1-(2-phenoxyphenyl)-3-(3-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)urea
Show/Hide
|
C32H24N4O2
|
1
|
| 1 |
IC50 = 127 nM
|
|
|
|
CP0510556
|
1-(2-(benzyloxy)phenyl)-3-(3-(5-(3-(dimethylcarbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)urea
Show/Hide
|
C36H31N5O3
|
1
|
| 1 |
IC50 = 132 nM
|
|
|
|
CP0510555
|
3-(3-(3-(3-(2-phenoxyphenyl)ureido)phenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl)benzoic acid
Show/Hide
|
C33H24N4O4
|
1
|
| 1 |
IC50 = 184 nM
|
|
|
|
CP0375702
|
1-(3-(5-(4-aminophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-fluoro-4-(trifluoromethyl)phenyl)urea
Show/Hide
|
C27H19F4N5O
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0407644
|
3-(4-(3-(3-(3-(2-phenoxyphenyl)ureido)phenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl)propanoic acid
Show/Hide
|
C35H28N4O4
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0505157
|
1-(3-(5-(3-(dimethylcarbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(3-phenoxyphenyl)urea
Show/Hide
|
C35H29N5O3
|
1
|
| 1 |
IC50 = 212 nM
|
|
|
|
CP0514454
|
1-(3-(5-(1H-pyrrol-2-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-phenoxyphenyl)urea
Show/Hide
|
C30H23N5O2
|
1
|
| 1 |
IC50 = 233 nM
|
|
|
|
CP0517509
|
1-(3-(5-(3-aminophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-fluoro-4-(trifluoromethyl)phenyl)urea
Show/Hide
|
C27H19F4N5O
|
1
|
| 1 |
IC50 = 242 nM
|
|
|
|
CP0006184
|
6,7,13,14-tetrahydroxy-2,9-dioxatetracyclo[6.6.2.0^{4,16}.0^{11,15}]hexadeca-1(14),4(16),5,7,11(15),12-hexaene-3,10-dione
Show/Hide
|
C14H6O8
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0510554
|
1-[3-[5-(furan-3-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]phenyl]-3-(2-phenoxyphenyl)urea
Show/Hide
|
C30H22N4O3
|
1
|
| 1 |
IC50 = 251 nM
|
|
|
|
CP0515946
|
1-(2-fluoro-4-(trifluoromethyl)phenyl)-3-(3-(5-(4-(piperazine-1-carbonyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)urea
Show/Hide
|
C33H28F4N6O2
|
1
|
| 1 |
IC50 = 286 nM
|
|
|
|
CP0505153
|
1-(2-fluoro-4-(trifluoromethyl)phenyl)-3-(3-(5-(3-(piperazine-1-carbonyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)urea
Show/Hide
|
C33H28F4N6O2
|
1
|
| 1 |
IC50 = 335 nM
|
|
|
|
CP0431056
|
1-(2-fluoro-4-(trifluoromethyl)phenyl)-3-(3-(5-(3-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)urea
Show/Hide
|
C27H17F5N4O
|
1
|
| 1 |
IC50 = 605 nM
|
|
|
|
CP0439847
|
1-phenyl-3-(3-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)urea
Show/Hide
|
C26H20N4O
|
1
|
| 1 |
IC50 = 749 nM
|
|
|
|
CP0845866
|
N-(2,6-difluorophenyl)-2-[(1-methylethyl)oxy]-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C43H45F2N7O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0848472
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-[(1-methylethyl)oxy]benzamide
Show/Hide
|
C43H45F2N7O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0848487
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
|
C44H47F2N7O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0857315
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
|
C43H45F2N7O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0857324
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
|
C46H51F2N9O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0870981
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C43H45F2N7O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0888354
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-[(1-methylethyl)oxy]benzamide
Show/Hide
|
C44H47F2N7O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0888370
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-[(1-methylethyl)oxy]benzamide
Show/Hide
|
C43H46F2N8O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0895692
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
|
C45H49F2N9O5S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0510552
|
1-(3-chlorophenyl)-3-(3-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)urea
Show/Hide
|
C26H19ClN4O
|
1
|
| 1 |
IC50 = 1015 nM
|
|
|
|
CP0431055
|
1-(2-fluoro-4-(trifluoromethyl)phenyl)-3-(3-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)urea
Show/Hide
|
C27H18F4N4O
|
1
|
| 1 |
IC50 = 1262 nM
|
|
|
|
CP0407643
|
1-(3-(5-(3-(dimethylcarbamoyl)phenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(4-phenoxyphenyl)urea
Show/Hide
|
C35H29N5O3
|
1
|
| 1 |
IC50 = 2039 nM
|
|
|
|
CP0506123
|
1-(3-(5-(3,4-dimethoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-3-(2-fluoro-4-(trifluoromethyl)phenyl)urea
Show/Hide
|
C29H22F4N4O3
|
1
|
| 1 |
IC50 = 2198 nM
|
|
|
|
CP0931048
|
(1S,2S)-2-((4S,7S,10S,13S)-10-benzyl-7-(2-carboxyethyl)-4-((6-chloro-1H-indol-3-yl)methyl)-14-(4-(hydroxy(phosphono)methyl)phenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C44H52ClN6O13P
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0493484
|
2-fluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide
Show/Hide
|
C28H33FN8O2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0938804
|
(1S,2S)-2-((4S,7S,10S,13S)-10-benzyl-7-(2-carboxyethyl)-4-(4-chlorobenzyl)-14-(4-(hydroxy(phosphono)methyl)phenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C42H51ClN5O13P
|
1
|
| 1 |
IC50 = 14000 nM
|
|
|
|
CP0889395
|
(4S,7S,10S,13S,16S)-4-((1H-indol-3-yl)methyl)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-13-(4-(hydroxy(phosphono)methyl)benzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C42H50N7O14P
|
1
|
| 1 |
IC50 = 15600 nM
|
|
|
|
CP0877536
|
(4S,7S,10S,13S,16S)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-4-((6-chloro-1H-indol-3-yl)methyl)-13-(4-(hydroxy(phosphono)methyl)benzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazanonadecan-19-oic acid
Show/Hide
|
C43H51ClN7O14P
|
1
|
| 1 |
IC50 = 21600 nM
|
|
|
|
CP0938805
|
(1S,2S)-2-((4R,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-14-(4-(hydroxy(phosphono)methyl)phenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C44H53N6O13P
|
1
|
| 1 |
IC50 = 22800 nM
|
|
|
|
CP0009041
|
5-propan-2-yl-7,8-dihydro-6H-indeno[1,2-b]indole-9,10-dione
Show/Hide
|
C18H17NO2
|
1
|
| 1 |
IC50 > 35000 nM
|
|
|
|
CP0938268
|
(4S,7S,10S,13S,16S)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-4-(4-chlorobenzyl)-13-(4-(hydroxy(phosphono)methyl)benzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazanonadecan-19-oic acid
Show/Hide
|
C41H50ClN6O14P
|
1
|
| 1 |
IC50 = 40500 nM
|
|
|
|
CP0877537
|
(4R,7S,10S,13S,16S)-4-((1H-indol-3-yl)methyl)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-13-(4-(hydroxy(phosphono)methyl)benzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazanonadecan-19-oic acid
Show/Hide
|
C43H52N7O14P
|
1
|
| 1 |
IC50 = 51300 nM
|
|
|
|
CP0942304
|
(4S,7S,10S,13S)-13-((R)-3-(1H-indol-3-yl)-1-(methylamino)-1-oxopropan-2-ylcarbamoyl)-10-benzyl-7-(4-(hydroxy(phosphono)methyl)benzyl)-2,5,8,11-tetraoxo-4-(pyridin-3-ylmethyl)-3,6,9,12-tetraazahexadecan-16-oic acid
Show/Hide
|
C46H53N8O12P
|
1
|
| 1 |
IC50 = 78200 nM
|
|
|
|
CP0931049
|
(4S,7S,10S,13S)-10-benzyl-13-((S)-3-(6-chloro-1H-indol-3-yl)-1-(methylamino)-1-oxopropan-2-ylcarbamoyl)-7-(4-(hydroxy(phosphono)methyl)benzyl)-2,5,8,11-tetraoxo-4-(pyridin-3-ylmethyl)-3,6,9,12-tetraazahexadecan-16-oic acid
Show/Hide
|
C46H52ClN8O12P
|
1
|
| 1 |
IC50 = 94000 nM
|
|
|
|
CP0910828
|
N-(3-chlorobenzyl)-6-nitro-9H-pyrido[2,3-b]indol-4-amine
Show/Hide
|
C18H13ClN4O2
|
1
|
| 1 |
Ki = 280 nM
|
|
|
|
CP0952563
|
N-(3-bromobenzyl)-6-nitro-9H-pyrido[2,3-b]indol-4-amine
Show/Hide
|
C18H13BrN4O2
|
1
|
| 1 |
Ki = 320 nM
|
|
|
|
CP0966032
|
N4-(3-methoxybenzyl)benzofuro[2,3-b]pyridine-4,6-diamine
Show/Hide
|
C19H17N3O2
|
1
|
| 1 |
Ki = 540 nM
|
|
|
|
CP0968343
|
N-(3-methoxybenzyl)-6-nitro-9H-pyrido[2,3-b]indol-4-amine
Show/Hide
|
C19H16N4O3
|
1
|
| 1 |
Ki = 890 nM
|
|
|
|
CP0026959
|
N-[(4-methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C19H16N2O2
|
1
|
| 1 |
Ki = 1030 nM
|
|
|
|
CP0902054
|
N4-(3-chlorobenzyl)-9H-pyrido[2,3-b]indole-4,6-diamine
Show/Hide
|
C18H15ClN4
|
1
|
| 1 |
Ki = 1920 nM
|
|
|
|
CP0853484
|
N4-(3-bromobenzyl)-9H-pyrido[2,3-b]indole-4,6-diamine
Show/Hide
|
C18H15BrN4
|
1
|
| 1 |
Ki = 2100 nM
|
|
|
|
CP0950866
|
6-nitro-N-(3-nitrobenzyl)benzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C18H12N4O5
|
1
|
| 1 |
Ki = 2390 nM
|
|
|
|
CP0883772
|
N-(3-bromobenzyl)-6-nitrobenzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C18H12BrN3O3
|
1
|
| 1 |
Ki = 2610 nM
|
|
|
|
CP0957789
|
N-(3-chlorobenzyl)-6-nitrobenzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C18H12ClN3O3
|
1
|
| 1 |
Ki = 2850 nM
|
|
|
|
CP0883773
|
N-(4-bromobenzyl)-6-nitrobenzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C18H12BrN3O3
|
1
|
| 1 |
Ki = 2870 nM
|
|
|
|
CP0941811
|
N-(4-methoxybenzyl)-6-nitrobenzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C19H15N3O4
|
1
|
| 1 |
Ki = 3400 nM
|
|
|
|
CP0853485
|
N-(4-chlorobenzyl)-6-nitrobenzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C18H12ClN3O3
|
1
|
| 1 |
Ki = 3540 nM
|
|
|
|
CP0902055
|
N4-(3-methoxybenzyl)-9H-pyrido[2,3-b]indole-4,6-diamine
Show/Hide
|
C19H18N4O
|
1
|
| 1 |
Ki = 3560 nM
|
|
|
|
CP0853483
|
N-(3-methoxybenzyl)-6-nitrobenzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C19H15N3O4
|
1
|
| 1 |
Ki = 4560 nM
|
|
|
|
CP0902051
|
N4-(3-chlorobenzyl)benzofuro[2,3-b]pyridine-4,6-diamine
Show/Hide
|
C18H14ClN3O
|
1
|
| 1 |
Ki = 4600 nM
|
|
|
|
CP0952562
|
N-(3-aminobenzyl)-6-nitrobenzofuro[2,3-b]pyridin-4-amine
Show/Hide
|
C18H14N4O3
|
1
|
| 1 |
Ki = 6180 nM
|
|
|
|
CP0853486
|
N4-(3-aminobenzyl)benzofuro[2,3-b]pyridine-4,6-diamine
Show/Hide
|
C18H16N4O
|
1
|
| 1 |
Ki = 8930 nM
|
|
|
|
CP0891047
|
(4S,7S,10S,13S,16S)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-4-((6-chloro-1H-indol-3-yl)methyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C41H46ClN7O11
|
1
|
| 1 |
Km = 5100 nM
|
|
|
|
CP0849344
|
(1S,2S)-2-((4S,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C43H50N6O10
|
1
|
| 1 |
Km = 8600 nM
|
|
|
|
CP0920986
|
(1R,2R)-2-((4S,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclopentanecarboxylic acid
Show/Hide
|
C42H48N6O10
|
1
|
| 1 |
Km = 15100 nM
|
|
|
|
CP0938265
|
(1S,2S)-2-((4S,7S,10S,13S)-10-benzyl-7-(2-carboxyethyl)-4-(4-chlorobenzyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C41H48ClN5O10
|
1
|
| 1 |
Km = 15400 nM
|
|
|
|
CP0886391
|
(4S,7S,10S,13S,16S)-4-((1H-indol-3-yl)methyl)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C41H47N7O11
|
1
|
| 1 |
Km = 16000 nM
|
|
|
|
CP0845821
|
(S)-5-((S)-3-(1H-indol-3-yl)-1-(methylamino)-1-oxopropan-2-ylamino)-4-((S)-2-((S)-3-(4-hydroxyphenyl)-2-(2-nitrobenzamido)propanamido)-3-phenylpropanamido)-5-oxopentanoic acid
Show/Hide
|
C42H43N7O10
|
1
|
| 1 |
Km = 19100 nM
|
|
|
|
CP0912795
|
(4S,10S,13S,16S)-16-acetamido-10-benzyl-4-((6-chloro-1H-indol-3-yl)methyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C38H42ClN7O9
|
1
|
| 1 |
Km = 19300 nM
|
|
|
|
CP0912759
|
(4S,7S,10S,13S,16S)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-4-(4-chlorobenzyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C39H45ClN6O11
|
1
|
| 1 |
Km = 19700 nM
|
|
|
|
CP0866644
|
(4S,7S,10S,13S,16S)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-13-(4-hydroxybenzyl)-4-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C43H48N6O11
|
1
|
| 1 |
Km = 19900 nM
|
|
|
|
CP0866633
|
(4S,7S,10S,13S,16S)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-4-((6-chloro-1H-indol-3-yl)methyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazanonadecan-19-oic acid
Show/Hide
|
C42H48ClN7O11
|
1
|
| 1 |
Km = 23500 nM
|
|
|
|
CP0845879
|
(4S,7S,10S,13S,16S)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-4-(3,4-dichlorobenzyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C39H44Cl2N6O11
|
1
|
| 1 |
Km = 25700 nM
|
|
|
|
CP0912755
|
(S)-4-((S)-2-((S)-3-(4-hydroxyphenyl)-2-(2-nitrobenzamido)propanamido)-3-phenylpropanamido)-5-((S)-1-(methylamino)-1-oxo-3-phenylpropan-2-ylamino)-5-oxopentanoic acid
Show/Hide
|
C40H42N6O10
|
1
|
| 1 |
Km = 28700 nM
|
|
|
|
CP0938264
|
(1S,2R)-2-((4S,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C43H50N6O10
|
1
|
| 1 |
Km = 28700 nM
|
|
|
|
CP0938267
|
(4S,7S,10S,13S)-10-benzyl-13-((S)-3-(6-chloro-1H-indol-3-yl)-1-(methylamino)-1-oxopropan-2-ylcarbamoyl)-7-(4-hydroxybenzyl)-2,5,8,11-tetraoxo-4-(pyridin-3-ylmethyl)-3,6,9,12-tetraazahexadecan-16-oic acid
Show/Hide
|
C45H49ClN8O9
|
1
|
| 1 |
Km = 35300 nM
|
|
|
|
CP0889392
|
(1R,2R)-2-((4S,7S,10S,13S)-4,10-dibenzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclopentanecarboxylic acid
Show/Hide
|
C40H47N5O10
|
1
|
| 1 |
Km = 36300 nM
|
|
|
|
CP0912794
|
2-((4S,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclobutanecarboxylic acid
Show/Hide
|
C41H46N6O10
|
1
|
| 1 |
Km = 36900 nM
|
|
|
|
CP0849350
|
(1S,2S)-2-((4S,7S,10S,13S)-4,10-dibenzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C41H49N5O10
|
1
|
| 1 |
Km = 43100 nM
|
|
|
|
CP0849346
|
(4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-4-amino-4-oxo-butanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenyl-propanoyl]amino]-5-[[(1S)-1-(1H-indol-3-ylmethyl)-2-(methylamino)-2-oxo-ethyl]amino]-5-oxo-pentanoic acid
Show/Hide
|
C41H48N8O10
|
1
|
| 1 |
Km = 48000 nM
|
|
|
|
CP0889394
|
(4S,10S,13S,16S)-4-((1H-indol-3-yl)methyl)-16-acetamido-10-benzyl-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C38H43N7O9
|
1
|
| 1 |
Km = 70300 nM
|
|
|
|
CP0860222
|
2-((4S,7S,10S,13S)-4,10-dibenzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclobutanecarboxylic acid
Show/Hide
|
C39H45N5O10
|
1
|
| 1 |
Km = 73600 nM
|
|
|
|
CP0877534
|
(4S,7S,10S,13S,16S)-16-acetamido-4,10-dibenzyl-7-(2-carboxyethyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C39H46N6O11
|
1
|
| 1 |
Km = 82300 nM
|
|
|
|
CP0888598
|
(1S,2R)-2-((4S,7S,10S,13S)-4,10-dibenzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C41H49N5O10
|
1
|
| 1 |
Km = 103000 nM
|
|
|
|
CP0915950
|
(4S,10S,13S,16S)-16-acetamido-10-benzyl-4-(3,4-dichlorobenzyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C36H40Cl2N6O9
|
1
|
| 1 |
Km = 106000 nM
|
|
|
|
CP0905990
|
(4S,7S,10S,13S,16S)-4-((1H-indol-3-yl)methyl)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazanonadecan-19-oic acid
Show/Hide
|
C42H49N7O11
|
1
|
| 1 |
Km = 114000 nM
|
|
|
|
CP0866643
|
(4S,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C39H44N6O10
|
1
|
| 1 |
Km = 144000 nM
|
|
|
|
CP0866632
|
(4S,10S,13S,16S)-16-acetamido-10-benzyl-4-(4-chlorobenzyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C36H41ClN6O9
|
1
|
| 1 |
Km = 156000 nM
|
|
|
|
CP0845877
|
(4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-4-amino-4-oxo-butanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenyl-propanoyl]amino]-5-[[(1S)-1-benzyl-2-(methylamino)-2-oxo-ethyl]amino]-5-oxo-pentanoic acid
Show/Hide
|
C39H47N7O10
|
1
|
| 1 |
Km = 167000 nM
|
|
|
|
CP0861750
|
(1S,2S)-2-((4R,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C43H50N6O10
|
1
|
| 1 |
Km = 188000 nM
|
|
|
|
CP0915949
|
(1R,2R)-2-((4S,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C43H50N6O10
|
1
|
| 1 |
Km = 204000 nM
|
|
|
|
CP0912793
|
(1S,2S)-2-((4S,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-10-benzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclopentanecarboxylic acid
Show/Hide
|
C42H48N6O10
|
1
|
| 1 |
Km = 230000 nM
|
|
|
|
CP0861751
|
(4S,7S,10S,13S,16S)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-4-(4-chlorobenzyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazanonadecan-19-oic acid
Show/Hide
|
C40H47ClN6O11
|
1
|
| 1 |
Km = 278000 nM
|
|
|
|
CP0877554
|
(1S,2S)-2-((4S,7S,10S,13S)-4,10-dibenzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclopentanecarboxylic acid
Show/Hide
|
C40H47N5O10
|
1
|
| 1 |
Km = 397000 nM
|
|
|
|
CP0909413
|
(4S,10S,13S,16S)-16-acetamido-10-benzyl-13-(4-hydroxybenzyl)-4-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C40H44N6O9
|
1
|
| 1 |
Km = 473000 nM
|
|
|
|
CP0860223
|
(4R,7S,10S,13S,16S)-4-((1H-indol-3-yl)methyl)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C41H47N7O11
|
1
|
| 1 |
Km = 514000 nM
|
|
|
|
CP0845878
|
(1R,2R)-2-((4S,7S,10S,13S)-4,10-dibenzyl-7-(2-carboxyethyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C41H49N5O10
|
1
|
| 1 |
Km = 587000 nM
|
|
|
|
CP0942305
|
(4R,10S,13S,16S)-4-((1H-indol-3-yl)methyl)-16-acetamido-10-benzyl-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C38H43N7O9
|
1
|
| 1 |
Km = 907000 nM
|
|
|
|
CP0908550
|
(4S,7S,10S,13S)-4,10-dibenzyl-7-(2-carboxyethyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazaoctadecan-18-oic acid
Show/Hide
|
C37H43N5O10
|
1
|
| 1 |
Km = 947000 nM
|
|
|
|
CP0845820
|
(4S,7S,10S,13S)-10-benzyl-13-((S)-3-(4-chlorophenyl)-1-(methylamino)-1-oxopropan-2-ylcarbamoyl)-7-(4-hydroxybenzyl)-2,5,8,11-tetraoxo-4-(pyridin-3-ylmethyl)-3,6,9,12-tetraazahexadecan-16-oic acid
Show/Hide
|
C43H48ClN7O9
|
1
|
| 1 |
Km > 1000000 nM
|
|
|
|
CP0856483
|
(4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(3-pyridyl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenyl-propanoyl]amino]-5-[[(1S)-1-(1H-indol-3-ylmethyl)-2-(methylamino)-2-oxo-ethyl]amino]-5-oxo-pentanoic acid
Show/Hide
|
C45H50N8O9
|
1
|
| 1 |
Km > 1000000 nM
|
|
|
|
CP0877535
|
(4S,7S,10S,13S)-13-((R)-3-(1H-indol-3-yl)-1-(methylamino)-1-oxopropan-2-ylcarbamoyl)-10-benzyl-7-(4-hydroxybenzyl)-2,5,8,11-tetraoxo-4-(pyridin-3-ylmethyl)-3,6,9,12-tetraazahexadecan-16-oic acid
Show/Hide
|
C45H50N8O9
|
1
|
| 1 |
Km > 1000000 nM
|
|
|
|
CP0938266
|
(4R,7S,10S,13S,16S)-4-((1H-indol-3-yl)methyl)-16-acetamido-10-benzyl-7-(2-carboxyethyl)-13-(4-hydroxybenzyl)-3,6,9,12,15-pentaoxo-2,5,8,11,14-pentaazanonadecan-19-oic acid
Show/Hide
|
C42H49N7O11
|
1
|
| 1 |
Km > 1000000 nM
|
|
|
|
CP0912796
|
(1S,2S)-2-((4S,7S,10S,13S)-10-benzyl-7-(2-carboxyethyl)-4-((6-chloro-1H-indol-3-yl)methyl)-14-(4-hydroxyphenyl)-3,6,9,12-tetraoxo-2,5,8,11-tetraazatetradecan-13-ylcarbamoyl)cyclohexanecarboxylic acid
Show/Hide
|
C43H49ClN6O10
|
1
|
| 1 |
Km < 5000 nM
|
|
|
