| Compound ID |
Compound Name |
Compound Formula |
|
CP0463609
|
butyl 2-[(6aR,9R,10aR)-1-hydroxy-9-(hydroxymethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C24H36O5
|
2
|
| 1 |
EC50 = 0.3 nM
|
|
|
| 2 |
Ki = 3.1 nM
|
|
|
|
CP0050487
|
(11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphthalen-1-ylcarbonyl)-9-oxa-1-azatricyclo[6.3.1.0^{4,12}]dodeca-2,4(12),5,7-tetraene
Show/Hide
|
C27H26N2O3
|
7
|
| 1 |
EC50 = 0.39 nM
|
|
|
| 2 |
EC50 = 86 nM
|
|
|
| 3 |
Ki = 1.2 nM
|
|
|
| 4 |
Ki = 2 nM
|
|
|
| 5 |
Ki = 2.1 nM
|
|
|
| 6 |
Ki = 3.7 nM
|
|
|
| 7 |
Ki = 13 nM
|
|
|
|
CP0230614
|
4-(2-{3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl}ethyl)morpholine
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|
C22H30N2O2
|
4
|
| 1 |
EC50 = 0.52 nM
|
|
|
| 2 |
EC50 = 14 nM
|
|
|
| 3 |
EC50 = 16 nM
|
|
|
| 4 |
Ki = 4.365 nM
|
|
|
|
CP0048192
|
2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl)-5-(2-methyloctan-2-yl)phenol
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|
C24H40O3
|
11
|
| 1 |
EC50 = 0.576 nM
|
|
|
| 2 |
EC50 = 2 nM
|
|
|
| 3 |
EC50 = 4.21 nM
|
|
|
| 4 |
EC50 = 5.6 nM
|
|
|
| 5 |
EC50 = 6.31 nM
|
|
|
| 6 |
EC50 = 9.8 nM
|
|
|
| 7 |
EC50 = 16.3 nM
|
|
|
| 8 |
IC50 = 8.3 nM
|
|
|
| 9 |
Ki = 0.2 nM
|
|
|
| 10 |
Ki = 0.439 nM
|
|
|
| 11 |
Ki = 0.69 nM
|
|
|
|
CP0430732
|
3-(2-(3-(2,2,3,3-Tetramethylcyclopropanecarbonyl)-1H-indol-1-yl)ethyl)oxazolidin-2-one
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|
C21H26N2O3
|
2
|
| 1 |
EC50 = 0.97 nM
|
|
|
| 2 |
EC50 = 2 nM
|
|
|
|
CP0412671
|
(6aS,10aS)-6,6,9-trimethyl-3-[(E)-C-methyl-N-(4,4,4-trifluorobutoxy)carbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C22H28F3NO3
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0402742
|
(2S,4S)-N-[(2S)-1-fluoro-3,3-dimethylbutan-2-yl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C18H22FN5O2
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0463801
|
(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-[1-(trifluoromethyl)cyclobutyl]-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C17H16F3N5O2
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0458227
|
(6aS,10aS)-6,6,9-trimethyl-3-[(E)-C-methyl-N-(3-phenylpropoxy)carbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C27H33NO3
|
2
|
| 1 |
EC50 = 1.65 nM
|
|
|
| 2 |
Ki = 2.7 nM
|
|
|
|
CP0412668
|
(6aS,10aS)-6,6,9-trimethyl-3-[(Z)-C-methyl-N-(3-phenylpropoxy)carbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C27H33NO3
|
2
|
| 1 |
EC50 = 1.7 nM
|
|
|
| 2 |
Ki = 2.9 nM
|
|
|
|
CP0490885
|
4-[(Z)-1-[(6aS,10aS)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]ethylideneamino]oxybutanenitrile
Show/Hide
|
C22H28N2O3
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
Ki = 0.4 nM
|
|
|
|
CP0439233
|
(1-(4-Hydroxybutyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
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|
C20H27NO2
|
2
|
| 1 |
EC50 = 2.1 nM
|
|
|
| 2 |
EC50 = 8 nM
|
|
|
|
CP0473684
|
(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-(1,1,1-trifluoro-2-methylpropan-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C16H16F3N5O2
|
1
|
| 1 |
EC50 = 2.3 nM
|
|
|
|
CP0403159
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
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|
C22H29NO2
|
2
|
| 1 |
EC50 = 2.7 nM
|
|
|
| 2 |
EC50 = 7 nM
|
|
|
|
CP0043110
|
(2S)-N-(5-tert-butyl-1,2-oxazol-3-yl)-1-(4-chlorophenyl)pyrrolidine-2-carboxamide
Show/Hide
|
C18H22ClN3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0403234
|
(2S,4S)-N-[(2S)-1-fluoro-3-methylbutan-2-yl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C17H20FN5O2
|
1
|
| 1 |
EC50 = 3.8 nM
|
|
|
|
CP0078200
|
[5-hydroxy-1-(oxan-4-ylmethyl)indol-3-yl]-(4-methoxyphenyl)methanone
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|
C22H23NO4
|
2
|
| 1 |
EC50 = 4.4 nM
|
|
|
| 2 |
Ki = 120.1 nM
|
|
|
|
CP0401581
|
(1-Butyl-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
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|
C20H27NO
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0294893
|
5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-3-[(E)-2-[(1S,2S,4R)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]ethenyl]pyrazole
Show/Hide
|
C30H35ClN2
|
1
|
| 1 |
EC50 = 5.32 nM
|
|
|
|
CP0469353
|
[5-hydroxy-1-(2-morpholin-4-ylethyl)indol-3-yl]-(4-methoxyphenyl)methanone
Show/Hide
|
C22H24N2O4
|
2
|
| 1 |
EC50 = 5.4 nM
|
|
|
| 2 |
Ki = 746.6 nM
|
|
|
|
CP0459091
|
(2S,4S)-N-[1-(hydroxymethyl)cyclopentyl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C18H21N5O3
|
1
|
| 1 |
EC50 = 5.6 nM
|
|
|
|
CP0460582
|
butyl 2-[(6aR,10aR)-1-hydroxy-9-(hydroxymethyl)-6,6-dimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C24H34O5
|
2
|
| 1 |
EC50 = 5.7 nM
|
|
|
| 2 |
Ki = 0.8 nM
|
|
|
|
CP0473682
|
(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-[1-(trifluoromethyl)cyclopropyl]-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C16H14F3N5O2
|
1
|
| 1 |
EC50 = 5.9 nM
|
|
|
|
CP0398538
|
(1-((Tetrahydrofuran-3-yl)methyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C21H27NO2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0405475
|
(2,2,3,3-Tetramethylcyclopropyl)(1-(4,4,4-trifluorobutyl)-1Hindol-3-yl)methanone
Show/Hide
|
C20H24F3NO
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0418693
|
6-(3-(2,2,3,3-Tetramethylcyclopropanecarbonyl)-1H-indol-1-yl)-hexan-2-one
Show/Hide
|
C22H29NO2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0204257
|
APD-371
Show/Hide
|
C18H23N5O3
|
1
|
| 1 |
EC50 = 6.2 nM
|
|
|
|
CP0373399
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-5-ol
Show/Hide
|
C22H29NO3
|
2
|
| 1 |
EC50 = 7 nM
|
|
|
| 2 |
Ki = 1.905 nM
|
|
|
|
CP0401547
|
[1-(oxan-4-ylmethyl)indol-3-yl]-(3-tricyclo[3.3.1.03,7]nonanyl)methanone
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|
C24H29NO2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0419109
|
(1-((1,3-Dioxolan-2-yl)methyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0441328
|
(2-Oxatricyclo[3.3.1.13,7]dec-1-yl)-[1-(tetrahydropyran-4-ylmethyl)-1H-indol-3-yl]methanone
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0450989
|
[5-hydroxy-1-(2-morpholin-4-ylethyl)indol-3-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C25H24N2O3
|
2
|
| 1 |
EC50 = 8.7 nM
|
|
|
| 2 |
Ki = 169 nM
|
|
|
|
CP0460583
|
butyl 2-[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C23H34O5
|
2
|
| 1 |
EC50 = 9 nM
|
|
|
| 2 |
Ki = 0.2 nM
|
|
|
|
CP0412670
|
(6aS,10aS)-3-[(E)-N-butoxy-C-methylcarbonimidoyl]-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C22H31NO3
|
2
|
| 1 |
EC50 = 9.14 nM
|
|
|
| 2 |
Ki = 16.9 nM
|
|
|
|
CP0085567
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-5-amine
Show/Hide
|
C22H30N2O2
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
Ki = 9.333 nM
|
|
|
|
CP0422343
|
6-chloro-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C22H28ClNO2
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
Ki = 2.512 nM
|
|
|
|
CP0055279
|
5-(4-chloro-3-methylphenyl)-1-phenyl-N-[(1S,2S,4R)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]pyrazole-3-carboxamide
Show/Hide
|
C27H30ClN3O
|
1
|
| 1 |
EC50 = 10.09 nM
|
|
|
|
CP0258259
|
5-tert-butyl-N-(1-hydroxy-2-methylpropan-2-yl)-1-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-3-carboxamide
Show/Hide
|
C18H23F3N4O2
|
2
|
| 1 |
EC50 = 10.7 nM
|
|
|
| 2 |
EC50 = 561.6 nM
|
|
|
|
CP0418654
|
(R)-(1-((Tetrahydrofuran-2-yl)methyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C21H27NO2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0439230
|
(1-(5-Hydroxypentyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C21H29NO2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0048193
|
5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1H-pyrazole-3-carboxylic acid (1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide
Show/Hide
|
C29H34ClN3O
|
3
|
| 1 |
EC50 = 11.5 nM
|
|
|
| 2 |
Ki = 0.6 nM
|
|
|
| 3 |
Ki = 5.4 nM
|
|
|
|
CP0445591
|
(6aS,10aS)-6,6,9-trimethyl-3-[(Z)-C-methyl-N-pentan-2-yloxycarbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C23H33NO3
|
2
|
| 1 |
EC50 = 11.5 nM
|
|
|
| 2 |
Ki = 6.1 nM
|
|
|
|
CP0334217
|
2-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-4-[(E)-2-[(1S,2S,4R)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]ethenyl]pyrrole
Show/Hide
|
C31H36ClN
|
1
|
| 1 |
EC50 = 11.56 nM
|
|
|
|
CP0445590
|
4-[(E)-1-[(6aS,10aS)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]ethylideneamino]oxybutanenitrile
Show/Hide
|
C22H28N2O3
|
2
|
| 1 |
EC50 = 12 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0102159
|
(1-(2-Methoxyethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C19H25NO2
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0297359
|
(S)-(1-((Tetrahydrofuran-2-yl)methyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C21H27NO2
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0868455
|
(R)-Spiro[2.5]octan-1-yl(1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-indol-3-yl)methanone
Show/Hide
|
C23H29NO2
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0149319
|
[5-hydroxy-1-(oxan-4-ylmethyl)indol-3-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C25H23NO3
|
2
|
| 1 |
EC50 = 14.7 nM
|
|
|
| 2 |
Ki = 275.4 nM
|
|
|
|
CP0353082
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-6-ol
Show/Hide
|
C22H29NO3
|
2
|
| 1 |
EC50 = 15 nM
|
|
|
| 2 |
Ki = 8.511 nM
|
|
|
|
CP0430960
|
(1-(2-(Tetrahydro-2H-pyran-4-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C23H31NO2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0389444
|
methyl N-[3-[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-1-adamantyl]carbamate
Show/Hide
|
C27H37NO5
|
2
|
| 1 |
EC50 = 15.8 nM
|
|
|
| 2 |
Ki = 8.4 nM
|
|
|
|
CP0401486
|
methyl 3-[3-(2,2,3,3-tetramethylcyclopropanecarbonyl)indol-1-yl]propanoate
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0227696
|
5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]pyrazole-3-carboxamide
Show/Hide
|
C29H34ClN3O
|
1
|
| 1 |
EC50 = 17.19 nM
|
|
|
|
CP0482613
|
(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-[(2S)-1,1,1-trifluoro-3-hydroxypropan-2-yl]-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C15H14F3N5O3
|
1
|
| 1 |
EC50 = 17.2 nM
|
|
|
|
CP0373396
|
5-(oxan-4-ylmethyl)-7-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-2H,5H-[1,3]dioxolo[4,5-f]indole
Show/Hide
|
C23H29NO4
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0457571
|
cyclohexyl-[5-hydroxy-1-(2-morpholin-4-ylethyl)indol-3-yl]methanone
Show/Hide
|
C21H28N2O3
|
2
|
| 1 |
EC50 = 18.6 nM
|
|
|
| 2 |
Ki = 895.3 nM
|
|
|
|
CP0139729
|
cyclopentyl-[1-(oxan-4-ylmethyl)indol-3-yl]methanone
Show/Hide
|
C20H25NO2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0405171
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole-5,6-diol
Show/Hide
|
C22H29NO4
|
2
|
| 1 |
EC50 = 21 nM
|
|
|
| 2 |
Ki = 21.38 nM
|
|
|
|
CP0412612
|
5-fluoro-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C22H28FNO2
|
2
|
| 1 |
EC50 = 22 nM
|
|
|
| 2 |
Ki = 1.585 nM
|
|
|
|
CP0439229
|
(1-(4-(Methylthio)butyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C21H29NOS
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0152977
|
5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1H-pyrazole-3-carboxylic acid ((1S,2S,4R)-1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide
Show/Hide
|
C29H34ClN3O
|
12
|
| 1 |
EC50 = 23.31 nM
|
|
|
| 2 |
IC50 = 19.95 nM
|
|
|
| 3 |
IC50 = 760 nM
|
|
|
| 4 |
IC50 = 7160 nM
|
|
|
| 5 |
Ki = 1.8 nM
|
|
|
| 6 |
Ki = 1.82 nM
|
|
|
| 7 |
Ki = 4.35 nM
|
|
|
| 8 |
Ki = 5.6 nM
|
|
|
| 9 |
Ki = 19.7 nM
|
|
|
| 10 |
Ki = 51 nM
|
|
|
| 11 |
Ki = 117 nM
|
|
|
| 12 |
Ki = 1820 nM
|
|
|
|
CP0418779
|
(1-(3-Methoxypropyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C20H27NO2
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0416863
|
(2R,4R)-N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-9-pyrazin-2-yl-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C18H23N5O2
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0419068
|
(1-(3-Hydroxypropyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C19H25NO2
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
|
CP0385957
|
[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]-(4-propylphenyl)methanone
Show/Hide
|
C22H18Cl2O3
|
1
|
| 1 |
EC50 = 28.8 nM
|
|
|
|
CP0477474
|
(1-Pentyl-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C21H29NO
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0382147
|
[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]-(4-ethylphenyl)methanone
Show/Hide
|
C21H16Cl2O3
|
1
|
| 1 |
EC50 = 29.5 nM
|
|
|
|
CP0418697
|
(1-(Pyridin-4-ylmethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C22H24N2O
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0401482
|
cycloheptyl-[1-(2-morpholin-4-ylethyl)indol-3-yl]methanone
Show/Hide
|
C22H30N2O2
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0419064
|
(1-(2-(Dimethylamino)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone p-Toluenesulfonic Acid
Show/Hide
|
C20H28N2O
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0418590
|
(1-Propyl-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C19H25NO
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0461659
|
4,5,6,7-tetrafluoro-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C22H25F4NO2
|
2
|
| 1 |
EC50 = 37 nM
|
|
|
| 2 |
Ki = 4.898 nM
|
|
|
|
CP0343767
|
9-methoxy-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[3,4-d][1,2]oxazole
Show/Hide
|
C22H31NO3
|
3
|
| 1 |
EC50 = 38.6 nM
|
|
|
| 2 |
IC50 = 4.2 nM
|
|
|
| 3 |
Ki = 12.8 nM
|
|
|
|
CP0424594
|
[3,5-dihydroxy-4-[3-(trifluoromethyl)phenyl]phenyl]-thiophen-2-ylmethanone
Show/Hide
|
C18H11F3O3S
|
1
|
| 1 |
EC50 = 38.9 nM
|
|
|
|
CP0102163
|
5-(methoxymethyl)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C24H33NO3
|
2
|
| 1 |
EC50 = 41 nM
|
|
|
| 2 |
Ki = 25.7 nM
|
|
|
|
CP0450681
|
(6aS,10aS)-6,6,9-trimethyl-3-[(E)-C-methyl-N-pentan-2-yloxycarbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C23H33NO3
|
2
|
| 1 |
EC50 = 41.3 nM
|
|
|
| 2 |
Ki = 24 nM
|
|
|
|
CP0880898
|
(R)-(1-(2-Morpholinoethyl)-1H-indol-3-yl)(spiro[2.5]octan-1-yl)-methanone
Show/Hide
|
C23H30N2O2
|
1
|
| 1 |
EC50 = 42 nM
|
|
|
|
CP0266280
|
5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S,2S,4R)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]pyrrole-3-carboxamide
Show/Hide
|
C30H35ClN2O
|
1
|
| 1 |
EC50 = 42.62 nM
|
|
|
|
CP0373389
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole-6-carbonitrile
Show/Hide
|
C23H28N2O2
|
2
|
| 1 |
EC50 = 45 nM
|
|
|
| 2 |
Ki = 5.012 nM
|
|
|
|
CP0475675
|
(2S,4S)-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C17H21N5O3
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0388239
|
(1-(2-(4-Methylthiazol-5-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C22H26N2OS
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0458225
|
(6aS,10aS)-6,6,9-trimethyl-3-[(E)-C-methyl-N-(2-phenoxyethoxy)carbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C26H31NO4
|
2
|
| 1 |
EC50 = 49.6 nM
|
|
|
| 2 |
Ki = 6.2 nM
|
|
|
|
CP0353084
|
1-[2-(morpholin-4-yl)ethyl]-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-4-amine
Show/Hide
|
C22H31N3O2
|
2
|
| 1 |
EC50 = 50 nM
|
|
|
| 2 |
Ki = 32.36 nM
|
|
|
|
CP0434538
|
4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[3,4-d][1,2]oxazol-9-ol
Show/Hide
|
C21H29NO3
|
3
|
| 1 |
EC50 = 50.2 nM
|
|
|
| 2 |
IC50 = 134 nM
|
|
|
| 3 |
Ki = 5.3 nM
|
|
|
|
CP0439231
|
(1-(2-(1H-Pyrrol-1-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C22H26N2O
|
1
|
| 1 |
EC50 = 54 nM
|
|
|
|
CP0439125
|
1-(2-(3-(2,2,3,3-Tetramethylcyclopropanecarbonyl)-1H-indol-1-yl)ethyl)pyrrolidin-2-one
Show/Hide
|
C22H28N2O2
|
1
|
| 1 |
EC50 = 55 nM
|
|
|
|
CP0418656
|
(1-(2-(Piperidin-1-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C23H32N2O
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0477572
|
(2S,4S)-N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-9-pyrazin-2-yl-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C18H23N5O2
|
1
|
| 1 |
EC50 = 59 nM
|
|
|
|
CP0225051
|
5-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C23H31NO3
|
2
|
| 1 |
EC50 = 61 nM
|
|
|
| 2 |
Ki = 4.571 nM
|
|
|
|
CP0250155
|
US9266835, 535
Show/Hide
|
C34H34Cl2F3N3O5S
|
1
|
| 1 |
EC50 = 61 nM
|
|
|
|
CP0321874
|
US9266835, 140
Show/Hide
|
C32H32Cl2F3N3O4S
|
1
|
| 1 |
EC50 = 61 nM
|
|
|
|
CP0491170
|
(1-(2-(Pyridin-3-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C23H26N2O
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0412621
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-4-ol
Show/Hide
|
C22H29NO3
|
2
|
| 1 |
EC50 = 64 nM
|
|
|
| 2 |
Ki = 3.89 nM
|
|
|
|
CP0155571
|
(2R,4R)-9-(2,4-difluorophenyl)-N-(1-hydroxy-2-methylpropan-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C18H19F2N3O2
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0048056
|
((1R,4S,5R)-4-(2,6-dimethoxy-4-(2-methyloctan-2-yl)phenyl)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl)methanol
Show/Hide
|
C27H42O3
|
1
|
| 1 |
EC50 = 64.5 nM
|
|
|
|
CP0458226
|
(6aS,10aS)-6,6,9-trimethyl-3-[(E)-C-methyl-N-(2-piperidin-1-ylethoxy)carbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C25H36N2O3
|
2
|
| 1 |
EC50 = 65.7 nM
|
|
|
| 2 |
Ki = 2.5 nM
|
|
|
|
CP0430950
|
[1-(2-morpholin-4-ylethyl)indol-3-yl]-(3-tricyclo[3.3.1.03,7]nonanyl)methanone
Show/Hide
|
C24H30N2O2
|
1
|
| 1 |
EC50 = 68 nM
|
|
|
|
CP0401544
|
(2,2,3,3-Ttetramethylcyclopropyl)(1-(2-(thiophen-3-yl)ethyl)-1H-indol-3-yl)methanone
Show/Hide
|
C22H25NOS
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0418798
|
(1-(2-(Pyrrolidin-1-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone p-Toluenesulfonic Acid
Show/Hide
|
C22H30N2O
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0401718
|
2-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-5-yl]oxyacetic acid
Show/Hide
|
C24H25NO6
|
2
|
| 1 |
EC50 = 70.2 nM
|
|
|
| 2 |
Ki = 1660 nM
|
|
|
|
CP0504771
|
Tetrahydropyranyl-methyl analogue, 48
Show/Hide
|
C23H31NO3
|
2
|
| 1 |
EC50 = 73 nM
|
|
|
| 2 |
Ki = 112.2 nM
|
|
|
|
CP0430948
|
(1-(Pyridin-3-ylmethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C22H24N2O
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
|
CP0439190
|
1-(2-(3-(2,2,3,3-Tetramethylcyclopropanecarbonyl)-1H-indol-1-yl)ethyl)pyrrolidin-2,5-dione
Show/Hide
|
C22H26N2O3
|
1
|
| 1 |
EC50 = 77 nM
|
|
|
|
CP0382099
|
4-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C23H31NO3
|
2
|
| 1 |
EC50 = 81 nM
|
|
|
| 2 |
Ki = 3.311 nM
|
|
|
|
CP0428737
|
CHEMBL3416126
Show/Hide
|
C27H35NO3
|
2
|
| 1 |
EC50 = 83.1 nM
|
|
|
| 2 |
Ki = 4.6 nM
|
|
|
|
CP0473773
|
(trans-4-Ethylcyclohexyl)(1-(2-morpholinoethyl)-1H-indol-3-yl)-methanone
Show/Hide
|
C23H32N2O2
|
1
|
| 1 |
EC50 = 85 nM
|
|
|
|
CP0439189
|
cyclohexyl-[1-(2-morpholin-4-ylethyl)indol-3-yl]methanone
Show/Hide
|
C21H28N2O2
|
1
|
| 1 |
EC50 = 86 nM
|
|
|
|
CP0382148
|
(4-chlorophenyl)-[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]methanone
Show/Hide
|
C19H11Cl3O3
|
1
|
| 1 |
EC50 = 89.7 nM
|
|
|
|
CP0411671
|
3-[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]adamantane-1-carbonitrile
Show/Hide
|
C26H33NO3
|
2
|
| 1 |
EC50 = 90.7 nM
|
|
|
| 2 |
Ki = 4.2 nM
|
|
|
|
CP0402740
|
(2S,4S)-N-(1-methylcyclopropyl)-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C16H17N5O2
|
1
|
| 1 |
EC50 = 91 nM
|
|
|
|
CP0405172
|
5-chloro-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C22H28ClNO2
|
2
|
| 1 |
EC50 = 92 nM
|
|
|
| 2 |
Ki = 3.02 nM
|
|
|
|
CP0430733
|
(1-Benzyl-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C23H25NO
|
1
|
| 1 |
EC50 = 93 nM
|
|
|
|
CP0434527
|
2-[[4,4-dimethyl-7-(2-methyloctan-2-yl)-1H-chromeno[4,3-c]pyrazol-9-yl]oxy]ethanol
Show/Hide
|
C23H34N2O3
|
3
|
| 1 |
EC50 = 95.1 nM
|
|
|
| 2 |
IC50 = 21.6 nM
|
|
|
| 3 |
Ki = 3.6 nM
|
|
|
|
CP0419110
|
(2,2,3,3-Tetramethylcyclopropyl)(1-(2-(thiophen-2-yl)ethyl)-1H-indol-3-yl)methanone
Show/Hide
|
C22H25NOS
|
1
|
| 1 |
EC50 = 96 nM
|
|
|
|
CP0412791
|
(2S,4S)-N-[(1S)-2-hydroxy-1-phenylethyl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C20H19N5O3
|
1
|
| 1 |
EC50 = 105 nM
|
|
|
|
CP0418698
|
(1-(2-(5-Chloro-1,2,4-thiadiazol-3-yl)ethyl)-1H-indol-3-yl)(2,2,3,-3-tetramethylcyclopropyl)methanone
Show/Hide
|
C20H22ClN3OS
|
1
|
| 1 |
EC50 = 109 nM
|
|
|
|
CP0385956
|
[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]-(4-methylphenyl)methanone
Show/Hide
|
C20H14Cl2O3
|
1
|
| 1 |
EC50 = 118 nM
|
|
|
|
CP0380712
|
2-(4-piperidin-1-ylphenyl)ethyl 5-chloro-3-ethyl-1H-indole-2-carboxylate
Show/Hide
|
C24H27ClN2O2
|
2
|
| 1 |
EC50 = 130 nM
|
|
|
| 2 |
IC50 = 8260 nM
|
|
|
|
CP0054364
|
6-(benzyloxy)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C29H35NO3
|
2
|
| 1 |
EC50 = 135 nM
|
|
|
| 2 |
Ki = 0.8913 nM
|
|
|
|
CP0487498
|
[4-(2,5-dichlorophenyl)-3,5-dihydroxyphenyl]-thiophen-2-ylmethanone
Show/Hide
|
C17H10Cl2O3S
|
1
|
| 1 |
EC50 = 141.25 nM
|
|
|
|
CP0382145
|
(3',5'-dichloro-2,6-dihydroxybiphenyl-4-yl)(phenyl)methanone
Show/Hide
|
C19H12Cl2O3
|
3
|
| 1 |
EC50 = 153 nM
|
|
|
| 2 |
EC50 = 154.88 nM
|
|
|
| 3 |
Ki = 2.94 nM
|
|
|
|
CP0419111
|
(1-(2-(Pyridin-4-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C23H26N2O
|
1
|
| 1 |
EC50 = 162 nM
|
|
|
|
CP0428148
|
[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]-(4-propan-2-ylphenyl)methanone
Show/Hide
|
C22H18Cl2O3
|
1
|
| 1 |
EC50 = 182 nM
|
|
|
|
CP0382098
|
1-[2-(morpholin-4-yl)ethyl]-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-6-ol
Show/Hide
|
C22H30N2O3
|
2
|
| 1 |
EC50 = 186 nM
|
|
|
| 2 |
Ki = 109.65 nM
|
|
|
|
CP0418770
|
(2,2,3,3-Tetrafluoro-1-methylcyclobutyl)(1-((tetrahydro-2Hpyran-4-yl)methyl)-1H-indol-3-yl)methanone
Show/Hide
|
C20H21F4NO2
|
1
|
| 1 |
EC50 = 197 nM
|
|
|
|
CP0507623
|
[3,5-dihydroxy-4-(3-methylphenyl)phenyl]-thiophen-2-ylmethanone
Show/Hide
|
C18H14O3S
|
1
|
| 1 |
EC50 = 199.53 nM
|
|
|
|
CP0190381
|
US9266835, 100
Show/Hide
|
C31H31Cl2F3N4O4S
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0051337
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole-5-carbonitrile
Show/Hide
|
C23H28N2O2
|
2
|
| 1 |
EC50 = 226 nM
|
|
|
| 2 |
Ki = 30.2 nM
|
|
|
|
CP0865274
|
[2-methyl-1-(2-morpholin-4-ylethyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone hydrochloride
Show/Hide
|
C23H33ClN2O2
|
1
|
| 1 |
EC50 = 227 nM
|
|
|
|
CP0507627
|
[3,5-dihydroxy-4-[3-(trifluoromethyl)phenyl]phenyl]-phenylmethanone
Show/Hide
|
C20H13F3O3
|
1
|
| 1 |
EC50 = 239.88 nM
|
|
|
|
CP0249763
|
US9266835, 122
Show/Hide
|
C34H29Cl2N3O5S
|
1
|
| 1 |
EC50 = 240 nM
|
|
|
|
CP0382150
|
(4-butylphenyl)-[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]methanone
Show/Hide
|
C23H20Cl2O3
|
1
|
| 1 |
EC50 = 254 nM
|
|
|
|
CP0424825
|
5-bromo-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C22H28BrNO2
|
2
|
| 1 |
EC50 = 280 nM
|
|
|
| 2 |
Ki = 6.607 nM
|
|
|
|
CP0416864
|
(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-[(2R)-1,1,1-trifluoro-3-hydroxypropan-2-yl]-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C15H14F3N5O3
|
1
|
| 1 |
EC50 = 280 nM
|
|
|
|
CP0401487
|
3-(3-(2,2,3,3-Tetramethylcyclopropanecarbonyl)-1H-indol-1-yl)-propanamide
Show/Hide
|
C19H24N2O2
|
1
|
| 1 |
EC50 = 294 nM
|
|
|
|
CP0537810
|
US9682955, 93
Show/Hide
|
C33H28Cl2N4O4S
|
1
|
| 1 |
EC50 = 323 nM
|
|
|
|
CP0517388
|
[4-(2,5-dichlorophenyl)-3,5-dihydroxyphenyl]-phenylmethanone
Show/Hide
|
C19H12Cl2O3
|
1
|
| 1 |
EC50 = 363.08 nM
|
|
|
|
CP0433003
|
(7E)-1-(2,4-dichlorophenyl)-5-(2-imidazol-1-ylacetyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C34H30Cl2N6O3
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0424598
|
[4-[3,5-bis(trifluoromethyl)phenyl]-3,5-dihydroxyphenyl]-phenylmethanone
Show/Hide
|
C21H12F6O3
|
1
|
| 1 |
EC50 = 371.54 nM
|
|
|
|
CP0408018
|
4-(benzyloxy)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C29H35NO3
|
2
|
| 1 |
EC50 = 383 nM
|
|
|
| 2 |
Ki = 9.333 nM
|
|
|
|
CP0419112
|
[1-(2-hydroxyethyl)indol-3-yl]-(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C18H23NO2
|
1
|
| 1 |
EC50 = 440 nM
|
|
|
|
CP0250147
|
US9266835, 108
Show/Hide
|
C32H31Cl2F3N4O5S
|
1
|
| 1 |
EC50 = 458 nM
|
|
|
|
CP0527784
|
3-[4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[3,4-d][1,2]oxazol-9-yl]oxypropan-1-ol
Show/Hide
|
C24H35NO4
|
3
|
| 1 |
EC50 = 539.6 nM
|
|
|
| 2 |
IC50 = 14 nM
|
|
|
| 3 |
Ki = 65.5 nM
|
|
|
|
CP0401484
|
(1-(2-(Pyridin-2-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C23H26N2O
|
1
|
| 1 |
EC50 = 542 nM
|
|
|
|
CP0433000
|
(8E)-8-[(5-chloropyridin-2-yl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C28H24Cl3N5O
|
1
|
| 1 |
EC50 = 560 nM
|
|
|
|
CP0416862
|
(2S,4S)-N-[(2R)-1-hydroxy-3,3-dimethylbutan-2-yl]-9-pyrazin-2-yl-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C18H23N5O2
|
1
|
| 1 |
EC50 = 560 nM
|
|
|
|
CP0405470
|
(1-((1-Methylpiperidin-2-yl)methyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C23H32N2O
|
1
|
| 1 |
EC50 = 628 nM
|
|
|
|
CP0056585
|
2-methyl-3-(naphthalen-1-ylcarbonyl)-1-propyl-1H-indole
Show/Hide
|
C23H21NO
|
1
|
| 1 |
EC50 = 634 nM
|
|
|
|
CP0385190
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-(3-sulfamoylpropanoyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H30Cl2N6O5S
|
1
|
| 1 |
EC50 = 650 nM
|
|
|
|
CP0517210
|
US9732061, Compound 36
Show/Hide
|
C24H21ClF3N5O2S2
|
1
|
| 1 |
EC50 = 665 nM
|
|
|
|
CP0533352
|
[4-[3,5-bis(trifluoromethyl)phenyl]-3,5-dihydroxyphenyl]-thiophen-2-ylmethanone
Show/Hide
|
C19H10F6O3S
|
1
|
| 1 |
EC50 = 676.08 nM
|
|
|
|
CP0430958
|
(2,2-Dichloro-1-methylcyclopropyl)(1-(2-morpholinoethyl)-1Hindol-3-yl)methanone
Show/Hide
|
C19H22Cl2N2O2
|
2
|
| 1 |
EC50 = 716 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0426521
|
3-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[6-[bis(4-chlorophenyl)methyl]-4-[[1-(trifluoromethylsulfonyl)piperidin-4-yl]amino]quinolin-8-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoic acid
Show/Hide
|
C55H76Cl2F3N3O17S
|
1
|
| 1 |
EC50 = 742 nM
|
|
|
|
CP0563716
|
(8E)-8-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H25Cl3N4O
|
1
|
| 1 |
EC50 = 743 nM
|
|
|
|
CP0401542
|
(2,2-Dichloro-1-methylcyclopropyl)(1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-indol-3-yl)methanone
Show/Hide
|
C19H21Cl2NO2
|
1
|
| 1 |
EC50 = 782 nM
|
|
|
|
CP0570537
|
US9682955, 145
Show/Hide
|
C27H23Cl2F3N4O2S
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0386505
|
(8E)-1-(3,4-dichlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-(1-pyridin-2-ylcyclopropyl)-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C30H25Cl2FN4O
|
1
|
| 1 |
EC50 = 807 nM
|
|
|
|
CP0441332
|
cyclopentyl-[1-(2-morpholin-4-ylethyl)indol-3-yl]methanone
Show/Hide
|
C20H26N2O2
|
2
|
| 1 |
EC50 = 819 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0411161
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C28H23Cl3N4O
|
1
|
| 1 |
EC50 = 854 nM
|
|
|
|
CP0418701
|
(1-(2-(Azepan-1-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C24H34N2O
|
1
|
| 1 |
EC50 = 1020 nM
|
|
|
|
CP0451950
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-[2-(tetrazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C32H28Cl2N8O3
|
1
|
| 1 |
EC50 = 1130 nM
|
|
|
|
CP0445998
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-[2-(triazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C33H29Cl2N7O3
|
1
|
| 1 |
EC50 = 1270 nM
|
|
|
|
CP0433001
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H24Cl2FN7O2
|
1
|
| 1 |
EC50 = 1310 nM
|
|
|
|
CP0419667
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-(2-sulfamoylacetyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H28Cl2N6O5S
|
1
|
| 1 |
EC50 = 1450 nM
|
|
|
|
CP0486578
|
US9682955, 41
Show/Hide
|
C37H37Cl2N5O6S
|
1
|
| 1 |
EC50 = 1470 nM
|
|
|
|
CP0418702
|
(1-(3-Morpholinopropyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C23H32N2O2
|
2
|
| 1 |
EC50 = 1524 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0400982
|
(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-(1-pyridin-2-ylcyclopropyl)-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C29H24Cl2N4O
|
1
|
| 1 |
EC50 = 1610 nM
|
|
|
|
CP0496959
|
(1-((1-Methyl-1H-imidazol-2-yl)methyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C22H27N3O
|
1
|
| 1 |
EC50 = 1619 nM
|
|
|
|
CP0562921
|
US9139546, 26
Show/Hide
|
C20H16O3
|
1
|
| 1 |
EC50 = 1659.59 nM
|
|
|
|
CP0565576
|
US9682955, 40
Show/Hide
|
C33H27Cl2F3N4O3
|
1
|
| 1 |
EC50 = 1670 nM
|
|
|
|
CP0424596
|
[4-(3,5-difluorophenyl)-3,5-dihydroxyphenyl]-phenylmethanone
Show/Hide
|
C19H12F2O3
|
1
|
| 1 |
EC50 = 1698.24 nM
|
|
|
|
CP0563751
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C32H27Cl2N7O3
|
1
|
| 1 |
EC50 = 1760 nM
|
|
|
|
CP0385182
|
3-[(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-3-[[(1R)-1-pyridin-2-ylethyl]carbamoyl]-4,6-dihydropyrazolo[4,3-c]pyridin-5-yl]-3-oxopropanoic acid
Show/Hide
|
C31H27Cl2N5O5
|
1
|
| 1 |
EC50 = 1940 nM
|
|
|
|
CP0411165
|
(8E)-1-(3,4-dichlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H25Cl2FN4O
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
|
CP0452137
|
(1-(2-(Piperazin-1-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone Trifluoroacetic Acid
Show/Hide
|
C22H31N3O
|
2
|
| 1 |
EC50 = 2200 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0257209
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[4-(2-morpholin-4-ylethoxy)phenyl]methanone
Show/Hide
|
C42H48N2O5
|
2
|
| 1 |
EC50 = 2270 nM
|
|
|
| 2 |
Ki = 580 nM
|
|
|
|
CP0263236
|
US9266835, 537
Show/Hide
|
C33H32Cl2F3N3O5S
|
1
|
| 1 |
EC50 = 2380 nM
|
|
|
|
CP0450547
|
cyclohexyl-[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]methanone
Show/Hide
|
C19H18Cl2O3
|
1
|
| 1 |
EC50 = 2540 nM
|
|
|
|
CP0334844
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[3-[2-(diethylamino)ethoxy]phenyl]methanone
Show/Hide
|
C42H50N2O4
|
2
|
| 1 |
EC50 = 2710 nM
|
|
|
| 2 |
Ki = 690 nM
|
|
|
|
CP0507626
|
[4-(furan-3-yl)-3,5-dihydroxyphenyl]-phenylmethanone
Show/Hide
|
C17H12O4
|
1
|
| 1 |
EC50 = 2754.23 nM
|
|
|
|
CP0424597
|
5-(4-benzoyl-2,6-dihydroxyphenyl)-2-fluorobenzonitrile
Show/Hide
|
C20H12FNO3
|
1
|
| 1 |
EC50 = 2818.38 nM
|
|
|
|
CP0433002
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-5-[(2S)-2,3-dihydroxypropanoyl]-N-[(1R)-1-phenylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H27Cl3N4O4
|
1
|
| 1 |
EC50 = 2910 nM
|
|
|
|
CP0451947
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-[2-(tetrazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H25Cl2FN8O2
|
1
|
| 1 |
EC50 = 3240 nM
|
|
|
|
CP0517211
|
US9732061, Compound 5
Show/Hide
|
C27H23Cl2F3N4O2S
|
1
|
| 1 |
EC50 = 3347 nM
|
|
|
|
CP0467704
|
ethyl 2-[6-[bis(4-chlorophenyl)methyl]-4-[[1-(trifluoromethylsulfonyl)piperidin-4-yl]amino]quinolin-8-yl]oxyacetate
Show/Hide
|
C32H30Cl2F3N3O5S
|
1
|
| 1 |
EC50 = 3400 nM
|
|
|
|
CP0279468
|
US9266835, 95
Show/Hide
|
C32H31Cl2N3O4
|
1
|
| 1 |
EC50 = 3650 nM
|
|
|
|
CP0433004
|
(7E)-1-(3,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-[2-(tetrazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H24Cl2FN9O2
|
1
|
| 1 |
EC50 = 3660 nM
|
|
|
|
CP0386504
|
(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C26H21Cl3N4OS
|
1
|
| 1 |
EC50 = 3820 nM
|
|
|
|
CP0388690
|
(4-tert-butylphenyl)-[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]methanone
Show/Hide
|
C23H20Cl2O3
|
1
|
| 1 |
EC50 = 3970 nM
|
|
|
|
CP0279480
|
US9266835, 57
Show/Hide
|
C31H27Cl2N5O
|
1
|
| 1 |
EC50 = 4100 nM
|
|
|
|
CP0259142
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[4-(diethylaminomethyl)phenyl]methanone
Show/Hide
|
C41H48N2O3
|
2
|
| 1 |
EC50 = 4400 nM
|
|
|
| 2 |
Ki = 1120 nM
|
|
|
|
CP0486648
|
US9682955, 54
Show/Hide
|
C34H30Cl2F3N3O4
|
1
|
| 1 |
EC50 = 4460 nM
|
|
|
|
CP0319745
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[4-[2-(diethylamino)ethoxy]phenyl]methanone
Show/Hide
|
C42H50N2O4
|
2
|
| 1 |
EC50 = 4650 nM
|
|
|
| 2 |
Ki = 1180 nM
|
|
|
|
CP0451948
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-pyrazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C33H28Cl2N6O3
|
1
|
| 1 |
EC50 = 4660 nM
|
|
|
|
CP0517384
|
[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3,5-dihydroxyphenyl]-phenylmethanone
Show/Hide
|
C21H16O5
|
1
|
| 1 |
EC50 = 4897.79 nM
|
|
|
|
CP0419665
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-5-[(2S)-2,3-dihydroxypropanoyl]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H26Cl3N5O4
|
1
|
| 1 |
EC50 = 5550 nM
|
|
|
|
CP0400984
|
(8E)-1-(2,4-dichlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C30H26Cl2FN3O
|
1
|
| 1 |
EC50 = 5590 nM
|
|
|
|
CP0486580
|
US9682955, 114
Show/Hide
|
C27H23Cl2F3N4O3S
|
1
|
| 1 |
EC50 = 5680 nM
|
|
|
|
CP0440160
|
US9815790, 2
Show/Hide
|
C43H54Cl2F3N3O10S
|
1
|
| 1 |
EC50 = 5900 nM
|
|
|
|
CP0164723
|
US9266835, 106
Show/Hide
|
C30H28Cl2N4O3
|
1
|
| 1 |
EC50 = 6500 nM
|
|
|
|
CP0563464
|
US9732061, Compound 12
Show/Hide
|
C34H30Cl2N4O2
|
1
|
| 1 |
EC50 = 6500 nM
|
|
|
|
CP0471785
|
US9266835, 532
Show/Hide
|
C30H26Cl2F3N3O5S
|
1
|
| 1 |
EC50 = 6700 nM
|
|
|
|
CP0199912
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-(4-phenylphenyl)methanone
Show/Hide
|
C42H41NO3
|
2
|
| 1 |
EC50 = 7060 nM
|
|
|
| 2 |
Ki = 1790 nM
|
|
|
|
CP0566182
|
US9815790, 1
Show/Hide
|
C37H42Cl2F3N3O7S
|
1
|
| 1 |
EC50 = 7400 nM
|
|
|
|
CP0451951
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(3,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-5-[2-(1,2,4-triazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H25Cl3N8O2
|
1
|
| 1 |
EC50 = 7850 nM
|
|
|
|
CP0411138
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-[2-(tetrazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H24Cl2FN9O2
|
1
|
| 1 |
EC50 = 8610 nM
|
|
|
|
CP0119397
|
US9266835, 538
Show/Hide
|
C33H33Cl2F3N4O4S
|
1
|
| 1 |
EC50 = 8630 nM
|
|
|
|
CP0326975
|
US9266835, 84
Show/Hide
|
C34H29Cl2N3O5S
|
1
|
| 1 |
EC50 = 8690 nM
|
|
|
|
CP0400985
|
(8E)-8-[(5-chlorothiophen-2-yl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C27H23Cl3N4OS
|
1
|
| 1 |
EC50 = 9410 nM
|
|
|
|
CP0051866
|
7-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C23H31NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 0.1259 nM
|
|
|
|
CP0051877
|
6-methyl-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C23H31NO2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 0.1479 nM
|
|
|
|
CP0054363
|
1-(oxan-4-ylmethyl)-6-phenyl-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C28H33NO2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 0.4074 nM
|
|
|
|
CP0057171
|
3-[(2-iodo-5-nitrophenyl)carbonyl]-1-[(1-methylpiperidin-2-yl)methyl]-1H-indole
Show/Hide
|
C22H22IN3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0150312
|
6-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-5-ol
Show/Hide
|
C23H31NO4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 0.6918 nM
|
|
|
|
CP0353083
|
5-(benzyloxy)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C29H35NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 1.259 nM
|
|
|
|
CP0373042
|
Tetrahydropyranyl-methyl analogue, 53
Show/Hide
|
C23H32N2O2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 61.66 nM
|
|
|
|
CP0373043
|
4-{2-[6-(benzyloxy)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl]ethyl}morpholine
Show/Hide
|
C29H36N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 2.951 nM
|
|
|
|
CP0373390
|
4-{2-[5-(benzyloxy)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl]ethyl}morpholine
Show/Hide
|
C29H36N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0373391
|
7-(benzyloxy)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C29H35NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 3.02 nM
|
|
|
|
CP0373393
|
Tetrahydropyranyl-methyl analogue, 47
Show/Hide
|
C23H32N2O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373395
|
Morpholino-ethyl analogue, 42
Show/Hide
|
C24H33N3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373398
|
6-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C23H31NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 0.5129 nM
|
|
|
|
CP0373400
|
1-(oxan-4-ylmethyl)-5-phenyl-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C28H33NO2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 58.88 nM
|
|
|
|
CP0373401
|
5-(4-bromobutoxy)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C26H36BrNO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 72.44 nM
|
|
|
|
CP0403154
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-7-ol
Show/Hide
|
C22H29NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 3.162 nM
|
|
|
|
CP0403157
|
6-bromo-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C22H28BrNO2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 0.6457 nM
|
|
|
|
CP0403161
|
4-(2-{5-methoxy-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl}ethyl)morpholine
Show/Hide
|
C23H32N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 234.42 nM
|
|
|
|
CP0405170
|
Tetrahydropyranyl-methyl analogue, 54
Show/Hide
|
C24H31NO4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 1.38 nM
|
|
|
|
CP0412610
|
6-methanesulfonyl-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C23H31NO4S
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 2.951 nM
|
|
|
|
CP0412616
|
4-{[1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-5-yl]oxy}butan-1-ol
Show/Hide
|
C26H37NO4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 263.03 nM
|
|
|
|
CP0412620
|
4-(2-{6-methoxy-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl}ethyl)morpholine
Show/Hide
|
C23H32N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 1.585 nM
|
|
|
|
CP0412624
|
Tetrahydropyranyl-methyl analogue, 50
Show/Hide
|
C24H31NO4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 239.88 nM
|
|
|
|
CP0427843
|
Morpholino-ethyl analogue, 43
Show/Hide
|
C23H33N3O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0433205
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-6-(trifluoromethyl)-1H-indole
Show/Hide
|
C23H28F3NO2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 3.467 nM
|
|
|
|
CP0436287
|
4-(2-{4-nitro-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl}ethyl)morpholine
Show/Hide
|
C22H29N3O4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 295.12 nM
|
|
|
|
CP0454165
|
5-(benzyloxy)-6-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C30H37NO4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 1.778 nM
|
|
|
|
CP0471161
|
1-[2-(morpholin-4-yl)ethyl]-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-5-ol
Show/Hide
|
C22H30N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 91.2 nM
|
|
|
|
CP0418696
|
(trans-4-Isopropylcyclohexyl)(1-(2-morpholinoethyl)-1H-indol-3-yl)methanone
Show/Hide
|
C24H34N2O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0419062
|
cyclobutyl-[1-(2-morpholin-4-ylethyl)indol-3-yl]methanone
Show/Hide
|
C19H24N2O2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0419063
|
(1-(2-Morpholinoethyl)-1H-indol-3-yl)(2,2,3,3-tetrafluoro-1-methylcyclobutyl)methanone
Show/Hide
|
C19H20F4N2O2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0431041
|
(1-(2-Aminoethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)-methanone
Show/Hide
|
C18H24N2O
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0407748
|
5-chloro-3-ethyl-N-[2-(4-pyrrolidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C23H26ClN3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0492352
|
5-chloro-3-methyl-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C23H26ClN3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0087627
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[3-(diethylaminomethyl)phenyl]methanone
Show/Hide
|
C41H48N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0120662
|
anthracen-9-yl-[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]methanone
Show/Hide
|
C44H41NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0156123
|
7-[4-(1-benzofuran-2-yl)phenoxy]-N-benzyl-N-methylheptan-1-amine
Show/Hide
|
C29H33NO2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0223129
|
(2-{4-[7-(benzylmethylamino)heptyloxy]phenyl}benzofuran-3-yl)phenylmethanone
Show/Hide
|
C36H37NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0257210
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C40H39NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0315950
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-naphthalen-2-ylmethanone
Show/Hide
|
C40H39NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0400933
|
(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C27H21Cl2F3N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0400986
|
(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-(1-pyridin-2-ylcyclopropyl)-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C28H21Cl2F3N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0400987
|
(8E)-8-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-(1-pyridin-2-ylcyclopropyl)-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H23Cl2F3N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0411162
|
(8E)-8-[(4-chlorophenyl)methylidene]-1-(3,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H25Cl3N4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0411163
|
(8E)-1-(4-chlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H26ClFN4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0411164
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C28H23Cl2FN4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0445931
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-N-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C31H28Cl3N5O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0447414
|
(7E)-1-(4-chlorophenyl)-7-[(5-chloropyridin-2-yl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C27H23Cl2N5O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0447415
|
(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C28H24Cl2N4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0451940
|
(8E)-1-(3,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-8-[[4-(trifluoromethyl)phenyl]methylidene]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C30H25Cl2F3N4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0464143
|
(8E)-8-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C28H23Cl2F3N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0509951
|
(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-(3,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C26H21Cl3N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0573762
|
(8E)-1-(2,4-dichlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-(1-pyridin-2-ylpiperidin-4-yl)-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C32H30Cl2FN5O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0386470
|
(7E)-5-(4-amino-4-oxobutanoyl)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H27Cl2FN6O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0386471
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-5-[2-(methanesulfonamido)acetyl]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H27Cl3N6O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0401021
|
(7E)-5-(2-aminoacetyl)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H29Cl2N5O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0433005
|
(7E)-5-(3-amino-3-oxopropanoyl)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H25Cl2FN6O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0451949
|
(7E)-1-(4-chlorophenyl)-7-[(4-fluorophenyl)methylidene]-5-[2-(methanesulfonamido)acetyl]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H28ClFN6O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0475837
|
(7E)-1-(4-chlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H25ClFN7O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0475838
|
(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H25Cl2N7O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0545426
|
(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H24Cl2N8O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0392261
|
2-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxyacetic acid
Show/Hide
|
C24H25NO6
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki = 581.8 nM
|
|
|
|
CP0003146
|
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H21Cl3N4O
|
10
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 1.9 nM
|
|
|
| 3 |
IC50 = 1631.1 nM
|
|
|
| 4 |
IC50 = 1939.8 nM
|
|
|
| 5 |
Ki = 398.11 nM
|
|
|
| 6 |
Ki = 554 nM
|
|
|
| 7 |
Ki = 790 nM
|
|
|
| 8 |
Ki = 1640 nM
|
|
|
| 9 |
Ki > 40000 nM
|
|
|
| 10 |
Ki > 1000 nM
|
|
|
|
CP0219312
|
US9266835, 44
Show/Hide
|
C28H24Cl2F3N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0219426
|
US9266835, 541
Show/Hide
|
C28H24Cl2F3N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0219430
|
US9266835, 80
Show/Hide
|
C33H29Cl2N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0241001
|
US9266835, 117
Show/Hide
|
C29H27Cl2N3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0241006
|
US9266835, 141
Show/Hide
|
C32H34Cl2F3N5O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0243591
|
US9266835, 49
Show/Hide
|
C29H26Cl2F3N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0250148
|
US9266835, 110
Show/Hide
|
C31H30Cl2F3N3O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0266404
|
US9266835, 96
Show/Hide
|
C30H27Cl2N3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0279473
|
US9266835, 542
Show/Hide
|
C32H33Cl2F3N4O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0321871
|
US9266835, 116
Show/Hide
|
C35H29Cl2N3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0324009
|
US9266835, 127
Show/Hide
|
C35H31Cl2N3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0326974
|
US9266835, 63
Show/Hide
|
C28H27Cl2N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0346676
|
US9266835, 129
Show/Hide
|
C35H31Cl2N3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0426522
|
US9266835, 530
Show/Hide
|
C31H30Cl2F3N3O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0566181
|
2-[6-[bis(4-chlorophenyl)methyl]-4-[[1-(trifluoromethylsulfonyl)piperidin-4-yl]amino]quinolin-8-yl]oxyacetic acid
Show/Hide
|
C30H26Cl2F3N3O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0511854
|
US9682955, 107
Show/Hide
|
C27H24Cl2F3N5O2S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0472556
|
US9732061, Compound 19
Show/Hide
|
C33H28Cl2N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0472557
|
4-N-[6-[bis(4-chlorophenyl)methyl]cinnolin-4-yl]-1-N-phenylcyclohexane-1,4-diamine
Show/Hide
|
C33H30Cl2N4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0563833
|
US9732061, Compound 1
Show/Hide
|
C27H23Cl2F3N4O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0445997
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C31H28Cl2FN5O
|
1
|
| 1 |
EC50 > 11000 nM
|
|
|
|
CP0389622
|
CHEMBL3416128
Show/Hide
|
C27H35NO3S
|
2
|
| 1 |
EC50 > 400 nM
|
|
|
| 2 |
Ki = 10.3 nM
|
|
|
|
CP0382149
|
(4-chlorophenyl)-[4-(3,5-dichlorophenyl)-3-hydroxy-5-methoxyphenyl]methanone
Show/Hide
|
C20H13Cl3O3
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0385955
|
[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]-[4-(trifluoromethyl)phenyl]methanone
Show/Hide
|
C20H11Cl2F3O3
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0385958
|
[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]-(4-hydroxyphenyl)methanone
Show/Hide
|
C19H12Cl2O4
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0388694
|
(4-butylphenyl)-[4-(3,5-dichlorophenyl)-3-hydroxy-5-methoxyphenyl]methanone
Show/Hide
|
C24H22Cl2O3
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0392595
|
[4-(3,5-dichlorophenyl)-3-hydroxy-5-methoxyphenyl]-(4-methylphenyl)methanone
Show/Hide
|
C21H16Cl2O3
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0428149
|
[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]-(3-ethylphenyl)methanone
Show/Hide
|
C21H16Cl2O3
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0400705
|
N-[3-(3,3-difluoroazetidine-1-carbonyl)-5,7-dihydro-4H-thieno[2,3-c]pyran-2-yl]tricyclo[3.3.1.03,7]nonane-3-carboxamide
Show/Hide
|
C21H24F2N2O3S
|
3
|
| 1 |
IC50 = 0.1995 nM
|
|
|
| 2 |
IC50 = 5.623 nM
|
|
|
| 3 |
Ki = 5.623 nM
|
|
|
|
CP0410344
|
N-propyl-2-[(2,2,3,3-tetramethylcyclopropanecarbonyl)amino]-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
|
C19H28N2O3S
|
3
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 52.48 nM
|
|
|
| 3 |
Ki = 91.2 nM
|
|
|
|
CP0051325
|
N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H26Cl2N4O
|
2
|
| 1 |
IC50 = 1.7 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0400698
|
N-propyl-2-(tricyclo[3.3.1.03,7]nonane-3-carbonylamino)-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
|
C21H28N2O3S
|
3
|
| 1 |
IC50 = 1.95 nM
|
|
|
| 2 |
IC50 = 70.79 nM
|
|
|
| 3 |
Ki = 20.89 nM
|
|
|
|
CP0085568
|
N-cyclohexyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H22Cl2N4O
|
2
|
| 1 |
IC50 = 2.2 nM
|
|
|
| 2 |
Ki = 1.7 nM
|
|
|
|
CP0437701
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-1-(piperidin-1-yl)ethanone
Show/Hide
|
C21H18Cl4N4O
|
1
|
| 1 |
IC50 = 5.9 nM
|
|
|
|
CP0045801
|
(10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C21H30O2
|
3
|
| 1 |
IC50 = 9.5 nM
|
|
|
| 2 |
Ki = 42 nM
|
|
|
| 3 |
Ki = 71.6 nM
|
|
|
|
CP0400699
|
N-propyl-2-(tricyclo[3.3.1.03,7]nonane-3-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
Show/Hide
|
C22H30N2O2S
|
3
|
| 1 |
IC50 = 9.772 nM
|
|
|
| 2 |
IC50 = 83.18 nM
|
|
|
| 3 |
Ki = 1.95 nM
|
|
|
|
CP0230625
|
[4-[(4-fluorophenyl)methyl-methylamino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C30H24FNO3
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
Ki = 2.7 nM
|
|
|
|
CP0410345
|
2-(adamantane-1-carbonylamino)-N-propyl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
|
C22H30N2O3S
|
3
|
| 1 |
IC50 = 11.22 nM
|
|
|
| 2 |
IC50 = 42.66 nM
|
|
|
| 3 |
Ki = 33.88 nM
|
|
|
|
CP0446278
|
(6aR,9S,10aR)-6,6,9-trimethyl-3-pentyl-10,10a-dihydro-6aH-benzo[c]chromene-1,9-diol
Show/Hide
|
C21H30O3
|
4
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
IC50 = 11420 nM
|
|
|
| 3 |
Ki = 9.5 nM
|
|
|
| 4 |
Ki = 5700 nM
|
|
|
|
CP0477867
|
US9422235, 58
Show/Hide
|
C18H23F3N2O2S
|
2
|
| 1 |
IC50 = 20 nM
|
|
|
| 2 |
Ki = 12.2 nM
|
|
|
|
CP0102148
|
1-(3,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H21Cl2N5O
|
2
|
| 1 |
IC50 = 25 nM
|
|
|
| 2 |
Ki = 20 nM
|
|
|
|
CP0434540
|
15-ethyl-12,12-dimethyl-8-(2-methyloctan-2-yl)-3,11-dioxa-15,16-diazatetracyclo[8.7.0.02,7.013,17]heptadeca-1(10),2(7),8,13,16-pentaene
Show/Hide
|
C26H38N2O2
|
2
|
| 1 |
IC50 = 25.5 nM
|
|
|
| 2 |
Ki = 121.6 nM
|
|
|
|
CP0490985
|
US9422235, 3
Show/Hide
|
C17H15Cl2F3N2O2S
|
2
|
| 1 |
IC50 = 30 nM
|
|
|
| 2 |
Ki = 17 nM
|
|
|
|
CP0401720
|
(4-methoxyphenyl)-[1-(oxan-4-ylmethyl)-7-propoxyindol-3-yl]methanone
Show/Hide
|
C25H29NO4
|
2
|
| 1 |
IC50 = 30.6 nM
|
|
|
| 2 |
Ki = 5.7 nM
|
|
|
|
CP0433182
|
1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H25Cl2N5O
|
2
|
| 1 |
IC50 = 37 nM
|
|
|
| 2 |
Ki = 29 nM
|
|
|
|
CP0494872
|
US9422235, 110
Show/Hide
|
C21H29F3N2O2S
|
2
|
| 1 |
IC50 = 37.2 nM
|
|
|
| 2 |
Ki = 18.8 nM
|
|
|
|
CP0073069
|
2-(4-ethoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benzo[d]imidazole-5-carboxamide
Show/Hide
|
C26H35N3O2
|
2
|
| 1 |
IC50 = 39.81 nM
|
|
|
| 2 |
Ki = 36.7 nM
|
|
|
|
CP0396843
|
(E)-2-(benzenesulfonyl)-3-[1-(2-morpholin-4-ylethyl)indol-3-yl]prop-2-enenitrile
Show/Hide
|
C23H23N3O3S
|
1
|
| 1 |
IC50 = 40.1 nM
|
|
|
|
CP0471292
|
US9422235, 43
Show/Hide
|
C18H15ClF3N3O2S
|
2
|
| 1 |
IC50 = 50.2 nM
|
|
|
| 2 |
Ki = 29 nM
|
|
|
|
CP0225671
|
[4-[(4-fluorophenyl)methylamino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C29H22FNO3
|
2
|
| 1 |
IC50 = 70 nM
|
|
|
| 2 |
Ki = 20 nM
|
|
|
|
CP0466611
|
US9422235, 26
Show/Hide
|
C19H25F3N2O3S
|
2
|
| 1 |
IC50 = 75 nM
|
|
|
| 2 |
Ki = 36 nM
|
|
|
|
CP0372927
|
N-cyclohexyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H22Cl2N4O
|
2
|
| 1 |
IC50 = 81 nM
|
|
|
| 2 |
Ki = 64 nM
|
|
|
|
CP0045030
|
(6aR,10aR)-3-(1,1-dimethylbutyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6Hdibenzo[b,d]pyran
Show/Hide
|
C22H32O
|
6
|
| 1 |
IC50 = 81.8 nM
|
|
|
| 2 |
IC50 = 550 nM
|
|
|
| 3 |
Ki = 1.82 nM
|
|
|
| 4 |
Ki = 3 nM
|
|
|
| 5 |
Ki = 3.4 nM
|
|
|
| 6 |
Ki = 140 nM
|
|
|
|
CP0372944
|
N-cyclohexyl-1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H22F2N4O
|
2
|
| 1 |
IC50 = 83 nM
|
|
|
| 2 |
Ki = 65 nM
|
|
|
|
CP0497601
|
US9422235, 105
Show/Hide
|
C17H24F3N3O2S
|
2
|
| 1 |
IC50 = 83.4 nM
|
|
|
| 2 |
Ki = 49 nM
|
|
|
|
CP0262329
|
4-[[4-[2-(4-methoxyphenyl)-1-benzofuran-3-carbonyl]anilino]methyl]benzonitrile
Show/Hide
|
C30H22N2O3
|
2
|
| 1 |
IC50 = 90 nM
|
|
|
| 2 |
Ki = 20 nM
|
|
|
|
CP0384803
|
US9422235, 88
Show/Hide
|
C19H27F3N2O2S
|
2
|
| 1 |
IC50 = 91 nM
|
|
|
| 2 |
Ki = 56 nM
|
|
|
|
CP0512366
|
US9422235, 108
Show/Hide
|
C19H27F3N2O2S
|
2
|
| 1 |
IC50 = 95 nM
|
|
|
| 2 |
Ki = 58 nM
|
|
|
|
CP0492959
|
US9422235, 73
Show/Hide
|
C16H15ClF3N3O2S
|
2
|
| 1 |
IC50 = 95.6 nM
|
|
|
| 2 |
Ki = 43.27 nM
|
|
|
|
CP0483290
|
US9422235, 44
Show/Hide
|
C19H21F3N2O4S
|
2
|
| 1 |
IC50 = 108.9 nM
|
|
|
| 2 |
Ki = 62 nM
|
|
|
|
CP0440914
|
N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H26Cl2N4O
|
2
|
| 1 |
IC50 = 110 nM
|
|
|
| 2 |
Ki = 87 nM
|
|
|
|
CP0511966
|
US9422235, 47
Show/Hide
|
C19H19F3N2O4S
|
2
|
| 1 |
IC50 = 137.7 nM
|
|
|
| 2 |
Ki = 75.1 nM
|
|
|
|
CP0451742
|
US9422235, 94
Show/Hide
|
C16H22F3N3O2S
|
2
|
| 1 |
IC50 = 146 nM
|
|
|
| 2 |
Ki = 85 nM
|
|
|
|
CP0400473
|
US9422235, 74
Show/Hide
|
C20H27F3N2O2S
|
2
|
| 1 |
IC50 = 153 nM
|
|
|
| 2 |
Ki = 69.15 nM
|
|
|
|
CP0373861
|
1-(2,4-Dichlorophenyl)-5-(5-(hex-1-ynyl)thiophen-2-yl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C28H30Cl2N4OS
|
1
|
| 1 |
IC50 = 158 nM
|
|
|
|
CP0419646
|
US9422235, 6
Show/Hide
|
C18H19F3N2O3S
|
2
|
| 1 |
IC50 = 179 nM
|
|
|
| 2 |
Ki = 84 nM
|
|
|
|
CP0491079
|
US9422235, 32
Show/Hide
|
C19H27F3N2O3S
|
2
|
| 1 |
IC50 = 181 nM
|
|
|
| 2 |
Ki = 81 nM
|
|
|
|
CP0483272
|
US9422235, 107
Show/Hide
|
C18H26F3N3O2S
|
2
|
| 1 |
IC50 = 187 nM
|
|
|
| 2 |
Ki = 114 nM
|
|
|
|
CP0257790
|
1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H16Cl4N4O
|
2
|
| 1 |
IC50 = 190 nM
|
|
|
| 2 |
Ki = 150 nM
|
|
|
|
CP0489601
|
US9422235, 7
Show/Hide
|
C17H17F3N2O2S
|
2
|
| 1 |
IC50 = 198 nM
|
|
|
| 2 |
Ki = 90 nM
|
|
|
|
CP0073070
|
2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-(2-piperidin-1-ylethyl)benzimidazole-5-carboxamide
Show/Hide
|
C28H38N4O2
|
2
|
| 1 |
IC50 = 199.53 nM
|
|
|
| 2 |
Ki = 188 nM
|
|
|
|
CP0431778
|
1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H21Cl2N5O
|
2
|
| 1 |
IC50 = 200 nM
|
|
|
| 2 |
Ki = 1730 nM
|
|
|
|
CP0507896
|
US9422235, 35
Show/Hide
|
C19H19Cl2F3N2O3S
|
2
|
| 1 |
IC50 = 206 nM
|
|
|
| 2 |
Ki = 87 nM
|
|
|
|
CP0477868
|
US9422235, 28
Show/Hide
|
C19H22Cl2N2O5S
|
2
|
| 1 |
IC50 = 221 nM
|
|
|
| 2 |
Ki = 98 nM
|
|
|
|
CP0511965
|
US9422235, 42
Show/Hide
|
C19H21F3N2O3S
|
2
|
| 1 |
IC50 = 245 nM
|
|
|
| 2 |
Ki = 140.1 nM
|
|
|
|
CP0491076
|
US9422235, 19
Show/Hide
|
C19H22F2N2O5S
|
2
|
| 1 |
IC50 = 255 nM
|
|
|
| 2 |
Ki = 113 nM
|
|
|
|
CP0222933
|
[2-(4-methoxyphenyl)-1-benzofuran-3-yl]-[4-(pentylamino)phenyl]methanone
Show/Hide
|
C27H27NO3
|
2
|
| 1 |
IC50 = 260 nM
|
|
|
| 2 |
Ki = 70 nM
|
|
|
|
CP0460119
|
1-(2,4-Dichlorophenyl)-5-(5-(hex-1-ynyl)thiophen-2-yl)-N-hexyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C27H31Cl2N3OS
|
1
|
| 1 |
IC50 = 260.6 nM
|
|
|
|
CP0577330
|
US9422235, 106
Show/Hide
|
C19H28F3N3O2S
|
2
|
| 1 |
IC50 = 264 nM
|
|
|
| 2 |
Ki = 156 nM
|
|
|
|
CP0149320
|
[7-hydroxy-1-(oxan-4-ylmethyl)indol-3-yl]-(4-methoxyphenyl)methanone
Show/Hide
|
C22H23NO4
|
2
|
| 1 |
IC50 = 271.7 nM
|
|
|
| 2 |
Ki = 53.9 nM
|
|
|
|
CP0373859
|
N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(5-hex-1-ynylthiophen-2-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C27H29Cl2N3OS
|
1
|
| 1 |
IC50 = 278.3 nM
|
|
|
|
CP0491074
|
US9422235, 10
Show/Hide
|
C17H17Cl2F3N2O2S
|
2
|
| 1 |
IC50 = 290 nM
|
|
|
| 2 |
Ki = 168 nM
|
|
|
|
CP0446591
|
(2-tert-butylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C22H20N2O
|
2
|
| 1 |
IC50 = 300 nM
|
|
|
| 2 |
Ki = 80 nM
|
|
|
|
CP0460120
|
N-(azepan-1-yl)-1-(2,4-dichlorophenyl)-4-ethyl-5-(5-pent-1-ynylthiophen-2-yl)pyrazole-3-carboxamide
Show/Hide
|
C27H30Cl2N4OS
|
1
|
| 1 |
IC50 = 309.9 nM
|
|
|
|
CP0373860
|
1-(2,4-Dichlorophenyl)-5-(5-(hex-1-ynyl)thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4OS
|
1
|
| 1 |
IC50 = 310.5 nM
|
|
|
|
CP0458229
|
[(6aR,10aR)-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-yl] acetate
Show/Hide
|
C23H32O3
|
4
|
| 1 |
IC50 = 316 nM
|
|
|
| 2 |
IC50 = 518 nM
|
|
|
| 3 |
Ki = 158 nM
|
|
|
| 4 |
Ki = 259 nM
|
|
|
|
CP0466610
|
US9422235, 22
Show/Hide
|
C21H20F3N3O4S
|
2
|
| 1 |
IC50 = 332 nM
|
|
|
| 2 |
Ki = 146 nM
|
|
|
|
CP0489596
|
US9422235, 29
Show/Hide
|
C20H19F3N2O5S
|
2
|
| 1 |
IC50 = 344 nM
|
|
|
| 2 |
Ki = 152 nM
|
|
|
|
CP0483304
|
US9422235, 56
Show/Hide
|
C20H19ClF3N3O3S
|
2
|
| 1 |
IC50 = 359 nM
|
|
|
| 2 |
Ki = 188 nM
|
|
|
|
CP0415444
|
1-(2,4-Dichlorophenyl)-4-methyl-5-(5-(4-methylpent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4OS
|
1
|
| 1 |
IC50 = 385.9 nM
|
|
|
|
CP0516411
|
US9422235, 48
Show/Hide
|
C21H29F3N2O2S
|
2
|
| 1 |
IC50 = 398 nM
|
|
|
| 2 |
Ki = 218 nM
|
|
|
|
CP0073064
|
[2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)benzimidazol-5-yl]-piperidin-1-ylmethanone
Show/Hide
|
C27H35N3O2
|
2
|
| 1 |
IC50 = 398.11 nM
|
|
|
| 2 |
Ki = 384.5 nM
|
|
|
|
CP0356651
|
2-[(4-ethoxyphenyl)methylamino]-N,N-diethyl-1-(3-methylbutyl)benzimidazole-5-carboxamide
Show/Hide
|
C26H36N4O2
|
2
|
| 1 |
IC50 = 398.11 nM
|
|
|
| 2 |
Ki = 353.4 nM
|
|
|
|
CP0308436
|
(4-methoxyphenyl)-[2-(4-methoxyphenyl)-1-benzothiophen-3-yl]methanone
Show/Hide
|
C23H18O3S
|
2
|
| 1 |
IC50 = 400 nM
|
|
|
| 2 |
Ki = 100 nM
|
|
|
|
CP0466481
|
US9422235, 98
Show/Hide
|
C18H25F3N2O2S
|
2
|
| 1 |
IC50 = 404 nM
|
|
|
| 2 |
Ki = 235 nM
|
|
|
|
CP0327891
|
[4-(cyclopropylmethylamino)phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C26H23NO3
|
2
|
| 1 |
IC50 = 410 nM
|
|
|
| 2 |
Ki = 110 nM
|
|
|
|
CP0446280
|
[(6aR,10aR)-9-hydroperoxy-6,6,9-trimethyl-3-pentyl-10,10a-dihydro-6aH-benzo[c]chromen-1-yl] 4-methylbenzenesulfonate
Show/Hide
|
C28H36O6S
|
4
|
| 1 |
IC50 = 421 nM
|
|
|
| 2 |
IC50 = 1750 nM
|
|
|
| 3 |
Ki = 211 nM
|
|
|
| 4 |
Ki = 876 nM
|
|
|
|
CP0567673
|
US9422235, 25
Show/Hide
|
C18H25F3N2O3S
|
2
|
| 1 |
IC50 = 428 nM
|
|
|
| 2 |
Ki = 203 nM
|
|
|
|
CP0567676
|
US9422235, 75
Show/Hide
|
C21H25F3N2O4S
|
2
|
| 1 |
IC50 = 430 nM
|
|
|
| 2 |
Ki = 194.7 nM
|
|
|
|
CP0489585
|
US9422235, 109
Show/Hide
|
C19H15F6N3O2S
|
2
|
| 1 |
IC50 = 431 nM
|
|
|
| 2 |
Ki = 218 nM
|
|
|
|
CP0419674
|
US9422235, 54
Show/Hide
|
C21H25F3N2O5S
|
2
|
| 1 |
IC50 = 439 nM
|
|
|
| 2 |
Ki = 230 nM
|
|
|
|
CP0451936
|
US9422235, 66
Show/Hide
|
C19H19Cl2F3N2O2S
|
2
|
| 1 |
IC50 = 440 nM
|
|
|
| 2 |
Ki = 261 nM
|
|
|
|
CP0211385
|
[4-[3-[benzyl(methyl)amino]propoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C33H31NO4
|
2
|
| 1 |
IC50 = 440 nM
|
|
|
| 2 |
Ki = 120 nM
|
|
|
|
CP0455904
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C22H19Cl3N4O
|
1
|
| 1 |
IC50 = 486.9 nM
|
|
|
|
CP0399820
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-1,3-diaza-spiro[4.5]dec-1-en-4-one
Show/Hide
|
C25H23Cl3N4O
|
1
|
| 1 |
IC50 = 496.7 nM
|
|
|
|
CP0372932
|
1-(4-chlorophenyl)-N-(cyclohexylmethyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H25ClN4O
|
2
|
| 1 |
IC50 = 500 nM
|
|
|
| 2 |
Ki = 390 nM
|
|
|
|
CP0373045
|
N-cyclohexyl-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H25Cl3N4O
|
2
|
| 1 |
IC50 = 500 nM
|
|
|
| 2 |
Ki = 390 nM
|
|
|
|
CP0440911
|
N-[(3,4-dichlorophenyl)methyl]-1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H16Cl2F2N4O
|
2
|
| 1 |
IC50 = 500 nM
|
|
|
| 2 |
Ki = 390 nM
|
|
|
|
CP0447449
|
[2-(2-methylpropyl)benzimidazol-1-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C22H20N2O
|
2
|
| 1 |
IC50 = 500 nM
|
|
|
| 2 |
Ki = 100 nM
|
|
|
|
CP0073066
|
N,N-diethyl-1-(3-methylbutyl)-2-(4-phenoxyanilino)benzimidazole-5-carboxamide
Show/Hide
|
C29H34N4O2
|
2
|
| 1 |
IC50 = 501.19 nM
|
|
|
| 2 |
Ki = 426 nM
|
|
|
|
CP0483289
|
US9422235, 16
Show/Hide
|
C17H19F3N4O4S
|
2
|
| 1 |
IC50 = 511 nM
|
|
|
| 2 |
Ki = 220 nM
|
|
|
|
CP0466537
|
N-(azepan-1-yl)-1-(2,4-dichlorophenyl)-5-(5-hex-1-ynylthiophen-2-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C27H30Cl2N4OS
|
1
|
| 1 |
IC50 = 564 nM
|
|
|
|
CP0458228
|
9-methoxy-6,6,9-trimethyl-3-pentyl-8,10-dihydro-7H-benzo[c]chromene-1,10-diol
Show/Hide
|
C22H32O4
|
2
|
| 1 |
IC50 = 599 nM
|
|
|
| 2 |
Ki = 300 nM
|
|
|
|
CP0375064
|
N-butyl-1-(2,4-dichlorophenyl)-5-(5-hex-1-ynylthiophen-2-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H27Cl2N3OS
|
1
|
| 1 |
IC50 = 637.7 nM
|
|
|
|
CP0372929
|
1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H16Cl4N4O
|
2
|
| 1 |
IC50 = 650 nM
|
|
|
| 2 |
Ki = 510 nM
|
|
|
|
CP0176689
|
[4-(benzylamino)phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C29H23NO3
|
2
|
| 1 |
IC50 = 660 nM
|
|
|
| 2 |
Ki = 170 nM
|
|
|
|
CP0406585
|
US9422235, 103
Show/Hide
|
C15H20F3N3O3S
|
2
|
| 1 |
IC50 = 663 nM
|
|
|
| 2 |
Ki = 393 nM
|
|
|
|
CP0415446
|
N-(azepan-1-yl)-1-(2,4-dichlorophenyl)-4-methyl-5-[5-(4-methylpent-1-ynyl)thiophen-2-yl]pyrazole-3-carboxamide
Show/Hide
|
C27H30Cl2N4OS
|
1
|
| 1 |
IC50 = 687.7 nM
|
|
|
|
CP0507714
|
US9422235, 80
Show/Hide
|
C18H24F3N3O2S
|
2
|
| 1 |
IC50 = 696 nM
|
|
|
| 2 |
Ki = 373 nM
|
|
|
|
CP0458144
|
(4-methoxyphenyl)-[2-(2-methylpropyl)-1-benzothiophen-3-yl]methanone
Show/Hide
|
C20H20O2S
|
2
|
| 1 |
IC50 = 700 nM
|
|
|
| 2 |
Ki = 100 nM
|
|
|
|
CP0503126
|
N-(azepan-1-yl)-5-(5-bromothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H21BrCl2N4OS
|
1
|
| 1 |
IC50 = 704.9 nM
|
|
|
|
CP0560893
|
US9422235, 18
Show/Hide
|
C19H23FN2O5S
|
2
|
| 1 |
IC50 = 706 nM
|
|
|
| 2 |
Ki = 320 nM
|
|
|
|
CP0454268
|
N-cyclohexyl-1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H26F2N4O
|
2
|
| 1 |
IC50 = 720 nM
|
|
|
| 2 |
Ki = 570 nM
|
|
|
|
CP0419673
|
US9422235, 53
Show/Hide
|
C20H29F3N2O3S
|
2
|
| 1 |
IC50 = 743 nM
|
|
|
| 2 |
Ki = 407 nM
|
|
|
|
CP0455903
|
2-[5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C23H21BrCl2N4O
|
1
|
| 1 |
IC50 = 768.4 nM
|
|
|
|
CP0373855
|
1-(2,4-Dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-5-(5-(pent-1-ynyl)thiophen-2-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C27H28Cl2N4OS
|
1
|
| 1 |
IC50 = 785.1 nM
|
|
|
|
CP0203135
|
2-[(4-ethoxyphenyl)methyl]-N,1-bis(3-methylbutyl)benzimidazole-5-carboxamide
Show/Hide
|
C27H37N3O2
|
2
|
| 1 |
IC50 = 794.33 nM
|
|
|
| 2 |
Ki = 763.6 nM
|
|
|
|
CP0417371
|
2-[5-(4-Chloro-phenyl)-4-cyclopropyl-1-(2,4-dichloro-phenyl)-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C24H21Cl3N4O
|
1
|
| 1 |
IC50 = 822 nM
|
|
|
|
CP0477194
|
[(6aR,10R,10aR)-10-hydroperoxy-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-yl] 4-methylbenzenesulfonate
Show/Hide
|
C28H36O6S
|
2
|
| 1 |
IC50 = 851 nM
|
|
|
| 2 |
Ki = 426 nM
|
|
|
|
CP0462567
|
5-(5-bromothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H19BrCl2N4OS
|
1
|
| 1 |
IC50 = 894.6 nM
|
|
|
|
CP0441077
|
1-(heptoxymethyl)-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C26H29NO3
|
2
|
| 1 |
IC50 = 900 nM
|
|
|
| 2 |
Ki = 230 nM
|
|
|
|
CP0455906
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazole-4-thio
Show/Hide
|
C22H19Cl3N4S
|
1
|
| 1 |
IC50 = 901.4 nM
|
|
|
|
CP0460284
|
5-(5-(Cyclopentylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C29H30Cl2N4OS
|
1
|
| 1 |
IC50 = 901.7 nM
|
|
|
|
CP0375065
|
1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(pent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4OS
|
1
|
| 1 |
IC50 = 919.6 nM
|
|
|
|
CP0415442
|
5-(5-(But-1-ynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H26Cl2N4OS
|
1
|
| 1 |
IC50 = 921 nM
|
|
|
|
CP0560895
|
US9422235, 23
Show/Hide
|
C19H21F3N2O5S
|
2
|
| 1 |
IC50 = 923 nM
|
|
|
| 2 |
Ki = 407 nM
|
|
|
|
CP0519498
|
(9,9,13-trimethyl-5-pentyl-8,14-dioxatetracyclo[8.5.0.02,7.013,15]pentadeca-1(10),2(7),3,5-tetraen-3-yl) acetate
Show/Hide
|
C23H30O4
|
2
|
| 1 |
IC50 = 927 nM
|
|
|
| 2 |
Ki = 464 nM
|
|
|
|
CP0483301
|
US9422235, 17
Show/Hide
|
C19H23FN2O5S
|
2
|
| 1 |
IC50 = 953 nM
|
|
|
| 2 |
Ki = 411 nM
|
|
|
|
CP0375093
|
3-(2,4-Dichlorophenyl)-4-(5-(3-ethoxyprop-1-ynyl)thiophen-2-yl)-5-methyl-N-(piperidin-1-yl)cyclopenta-1,4-dienecarboxamide
Show/Hide
|
C25H26Cl2N4O2S
|
1
|
| 1 |
IC50 = 985.6 nM
|
|
|
|
CP0560896
|
US9422235, 79
Show/Hide
|
C18H16ClF3N2O4S
|
2
|
| 1 |
IC50 = 997 nM
|
|
|
| 2 |
Ki = 535 nM
|
|
|
|
CP0914917
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid ethanolamide
Show/Hide
|
C18H19NO3
|
2
|
| 1 |
IC50 = 1000 nM
|
|
|
| 2 |
Ki = 1030 nM
|
|
|
|
CP0181199
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-5-nitrobenzimidazole
Show/Hide
|
C21H25N3O3
|
2
|
| 1 |
IC50 = 1000 nM
|
|
|
| 2 |
Ki = 961.8 nM
|
|
|
|
CP0415440
|
N-(azepan-1-yl)-5-(5-but-1-ynylthiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H26Cl2N4OS
|
1
|
| 1 |
IC50 = 1057.8 nM
|
|
|
|
CP0455905
|
2-[1-(2,4-Dichloro-phenyl)-5-(4-methoxy-phenyl)-4-methyl-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C23H22Cl2N4O2
|
1
|
| 1 |
IC50 = 1058.5 nM
|
|
|
|
CP0527090
|
2-[5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C22H19BrCl2N4O
|
1
|
| 1 |
IC50 = 1095.5 nM
|
|
|
|
CP0458139
|
1-benzothiophen-3-yl(naphthalen-1-yl)methanone
Show/Hide
|
C19H12OS
|
2
|
| 1 |
IC50 = 1100 nM
|
|
|
| 2 |
Ki = 200 nM
|
|
|
|
CP0483263
|
US9422235, 78
Show/Hide
|
C19H18ClF3N2O4S
|
2
|
| 1 |
IC50 = 1107 nM
|
|
|
| 2 |
Ki = 560 nM
|
|
|
|
CP0451011
|
[(6aR,10S,10aR)-10-hydroxy-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-yl] 4-methylbenzenesulfonate
Show/Hide
|
C28H36O5S
|
2
|
| 1 |
IC50 = 1110 nM
|
|
|
| 2 |
Ki = 552 nM
|
|
|
|
CP0222934
|
[4-[(3,5-difluorophenyl)methylamino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C29H21F2NO3
|
2
|
| 1 |
IC50 = 1150 nM
|
|
|
| 2 |
Ki = 300 nM
|
|
|
|
CP0454981
|
1-(2,4-Dichlorophenyl)-5-(5-(3,3-dimethylbut-1-ynyl)thiophen-2-yl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C28H30Cl2N4OS
|
1
|
| 1 |
IC50 = 1158.1 nM
|
|
|
|
CP0463994
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-1-ethyl-5,5-dimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
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C23H21Cl3N4O
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1
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| 1 |
IC50 = 1173.7 nM
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CP0402743
|
US9422235, 37
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C18H13F5N2O3S
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2
|
| 1 |
IC50 = 1176 nM
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| 2 |
Ki = 471 nM
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CP0452044
|
(4-methoxyphenyl)-(2-propyl-1-benzothiophen-3-yl)methanone
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C19H18O2S
|
2
|
| 1 |
IC50 = 1200 nM
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| 2 |
Ki = 300 nM
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CP0454680
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(4-methoxyphenyl)-(2-pentyl-1-benzothiophen-3-yl)methanone
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C21H22O2S
|
2
|
| 1 |
IC50 = 1200 nM
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| 2 |
Ki = 300 nM
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CP0467679
|
1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(4-methylpent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C27H30Cl2N4OS
|
1
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| 1 |
IC50 = 1206 nM
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CP0484487
|
US9422235, 69
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C21H22F3N3O3S
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2
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| 1 |
IC50 = 1216 nM
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| 2 |
Ki = 644 nM
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CP0440912
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1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H25Cl2N5O
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2
|
| 1 |
IC50 = 1240 nM
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| 2 |
Ki = 980 nM
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CP0512349
|
US9422235, 82
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C20H20ClF3N2O4S
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2
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| 1 |
IC50 = 1253 nM
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| 2 |
Ki = 672 nM
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CP0073067
|
2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-(6-piperidin-1-ylhexyl)benzimidazole-5-carboxamide
Show/Hide
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C32H46N4O2
|
2
|
| 1 |
IC50 = 1258.93 nM
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| 2 |
Ki = 1000 nM
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CP0415438
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1-(2,4-Dichlorophenyl)-5-(5-(3-(dimethylamino)prop-1-ynyl)-thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C25H27Cl2N5OS
|
1
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| 1 |
IC50 = 1269.4 nM
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CP0373856
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5-(5-Chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H19Cl3N4OS
|
1
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| 1 |
IC50 = 1291 nM
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CP0415436
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naphthalen-1-yl-(2-pentyl-1-benzothiophen-3-yl)methanone
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C24H22OS
|
2
|
| 1 |
IC50 = 1300 nM
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| 2 |
Ki = 300 nM
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CP0463993
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-1,3-diaza-spiro[4.4]non-1-en-4-one
Show/Hide
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C24H21Cl3N4O
|
1
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| 1 |
IC50 = 1372.2 nM
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CP0466482
|
US9422235, 100
Show/Hide
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C17H18F3N3O2S
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2
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| 1 |
IC50 = 1373 nM
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| 2 |
Ki = 789 nM
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CP0446597
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[2-(4-methoxyphenyl)-1-benzothiophen-3-yl]-naphthalen-1-ylmethanone
Show/Hide
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C26H18O2S
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2
|
| 1 |
IC50 = 1400 nM
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| 2 |
Ki = 300 nM
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CP0419653
|
US9422235, 27
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C19H23ClN2O5S
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2
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| 1 |
IC50 = 1441 nM
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| 2 |
Ki = 682 nM
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CP0373854
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N-(azepan-1-yl)-1-(2,4-dichlorophenyl)-4-methyl-5-(5-pent-1-ynylthiophen-2-yl)pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4OS
|
1
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| 1 |
IC50 = 1499.2 nM
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CP0419675
|
US9422235, 55
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C21H26F3N3O3S
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2
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| 1 |
IC50 = 1520 nM
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| 2 |
Ki = 8323 nM
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CP0134010
|
[4-(heptylamino)phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
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C29H31NO3
|
2
|
| 1 |
IC50 = 1540 nM
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| 2 |
Ki = 410 nM
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CP0456628
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2-[4-Bromo-5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C21H16BrCl3N4O
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1
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| 1 |
IC50 = 1570.6 nM
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CP0489882
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5-(5-(Cyclohexylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C28H30Cl2N4OS
|
1
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| 1 |
IC50 = 1576.4 nM
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CP0516410
|
US9422235, 99
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C15H21F3N2O3S
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2
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| 1 |
IC50 = 1599 nM
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| 2 |
Ki = 919 nM
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CP0563783
|
US9422235, 15
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C18H17F5N2O3S
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2
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| 1 |
IC50 = 1638 nM
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| 2 |
Ki = 629 nM
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CP0211297
|
[4-[bis[(4-fluorophenyl)methyl]amino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C36H27F2NO3
|
2
|
| 1 |
IC50 = 1650 nM
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| 2 |
Ki = 430 nM
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CP0419754
|
(2-cyclohexylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
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C24H22N2O
|
2
|
| 1 |
IC50 = 1700 nM
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| 2 |
Ki = 400 nM
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CP0454683
|
(2-butylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
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C22H20N2O
|
2
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| 1 |
IC50 = 1700 nM
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| 2 |
Ki = 400 nM
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CP0516409
|
US9422235, 93
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C17H23F3N2O3S
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2
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| 1 |
IC50 = 1715 nM
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| 2 |
Ki = 996 nM
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CP0415434
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5-(5-(Cyclohexylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C30H32Cl2N4OS
|
1
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| 1 |
IC50 = 1725.9 nM
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CP0422466
|
1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H20Cl4N4O
|
2
|
| 1 |
IC50 = 1740 nM
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| 2 |
Ki = 1370 nM
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CP0474961
|
US9422235, 45
Show/Hide
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C22H27F3N2O4S
|
2
|
| 1 |
IC50 = 1748 nM
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| 2 |
Ki = 999 nM
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CP0373858
|
1-(2,4-Dichlorophenyl)-4-methyl-5-(5-(4-phenylbut-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C30H28Cl2N4OS
|
1
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| 1 |
IC50 = 1749.8 nM
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CP0375109
|
1-(2,4-Dichlorophenyl)-5-(5-(3-isopropoxyprop-1-ynyl)thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4O2S
|
1
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| 1 |
IC50 = 1761.1 nM
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CP0415437
|
5-(5-(Cyclopentylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C27H28Cl2N4OS
|
1
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| 1 |
IC50 = 1809.1 nM
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CP0451939
|
US9422235, 1
Show/Hide
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C19H20Cl2F3N3O3S
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2
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| 1 |
IC50 = 1837 nM
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| 2 |
Ki = 933 nM
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CP0511963
|
US9422235, 89
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C21H31F3N2O2S
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2
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| 1 |
IC50 = 1893 nM
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| 2 |
Ki = 1068 nM
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CP0386455
|
1-(2,4-Dichlorophenyl)-5-(5-(3,3-dimethylbut-1-ynyl)thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4OS
|
1
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| 1 |
IC50 = 1900.1 nM
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CP0507899
|
US9422235, 40
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C17H24N2O2S
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2
|
| 1 |
IC50 = 1940 nM
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| 2 |
Ki = 818 nM
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CP0527089
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-1-cyclopropyl-5,5-dimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C24H21Cl3N4O
|
1
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| 1 |
IC50 = 1950.4 nM
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CP0412001
|
(1-hydroxy-9-methoxy-6,6,9-trimethyl-3-pentyl-8,10-dihydro-7H-benzo[c]chromen-10-yl) acetate
Show/Hide
|
C24H34O5
|
2
|
| 1 |
IC50 = 1980 nM
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| 2 |
Ki = 990 nM
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CP0181197
|
2-(4-ethoxyanilino)-N,N-diethyl-1-(3-methylbutyl)benzimidazole-5-carboxamide
Show/Hide
|
C25H34N4O2
|
2
|
| 1 |
IC50 = 1995.26 nM
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| 2 |
Ki = 1900 nM
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CP0196094
|
2-[(4-ethoxyphenyl)methyl]-N-hexyl-1-(3-methylbutyl)benzimidazole-5-carboxamide
Show/Hide
|
C28H39N3O2
|
2
|
| 1 |
IC50 = 1995.26 nM
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| 2 |
Ki = 1900 nM
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CP0415435
|
[2-(2-methylpropyl)-1-benzothiophen-3-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C23H20OS
|
2
|
| 1 |
IC50 = 2000 nM
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| 2 |
Ki = 500 nM
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CP0412000
|
[(6aR,10aR)-8-hydroperoxy-6,6-dimethyl-9-methylidene-3-pentyl-7,8,10,10a-tetrahydro-6aH-benzo[c]chromen-1-yl] 4-methylbenzenesulfonate
Show/Hide
|
C28H36O6S
|
2
|
| 1 |
IC50 = 2060 nM
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| 2 |
Ki = 1030 nM
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CP0445204
|
US9422235, 33
Show/Hide
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C23H21F3N2O4S
|
2
|
| 1 |
IC50 = 2080 nM
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| 2 |
Ki = 880 nM
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CP0454682
|
naphthalen-1-yl-(2-propan-2-ylbenzimidazol-1-yl)methanone
Show/Hide
|
C21H18N2O
|
2
|
| 1 |
IC50 = 2100 nM
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| 2 |
Ki = 500 nM
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CP0882217
|
1-ethyl-3-(5-(naphthalen-2-ylthio)pentyl)urea
Show/Hide
|
C18H24N2OS
|
2
|
| 1 |
IC50 = 2110 nM
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| 2 |
Ki = 560 nM
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CP0507712
|
US9422235, 61
Show/Hide
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C14H17F3N2O2S
|
2
|
| 1 |
IC50 = 2133 nM
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| 2 |
Ki = 1199 nM
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CP0471293
|
US9422235, 46
Show/Hide
|
C21H24F3N3O3S
|
2
|
| 1 |
IC50 = 2150 nM
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| 2 |
Ki = 825 nM
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CP0484452
|
US9422235, 5
Show/Hide
|
C17H15Cl2FN2O
|
2
|
| 1 |
IC50 = 2150 nM
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| 2 |
Ki = 826 nM
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CP0375107
|
N-(azepan-1-yl)-5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H21Cl3N4OS
|
1
|
| 1 |
IC50 = 2156.1 nM
|
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|
CP0510719
|
(2-cyclopentylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C20H20N2O2
|
2
|
| 1 |
IC50 = 2200 nM
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| 2 |
Ki = 500 nM
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CP0386453
|
1-(2,4-Dichlorophenyl)-4-methyl-5-(5-(pent-1-ynyl)thiophen-2-1-(2,4-Dichlorophenyl)-4-methyl-5-(5-(pent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H26Cl2N4OS
|
1
|
| 1 |
IC50 = 2214 nM
|
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CP0379504
|
1-(4-chlorophenyl)-N-cyclohexyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H21ClN4O
|
2
|
| 1 |
IC50 = 2220 nM
|
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|
| 2 |
Ki = 1750 nM
|
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|
CP0471300
|
US9422235, 102
Show/Hide
|
C15H21F3N2O2S
|
2
|
| 1 |
IC50 = 2253 nM
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| 2 |
Ki = 1294 nM
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CP0474987
|
US9422235, 77
Show/Hide
|
C17H15Cl2F3N2O3S
|
2
|
| 1 |
IC50 = 2262 nM
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| 2 |
Ki = 1145 nM
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CP0451448
|
(2-tert-butylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C19H20N2O2
|
2
|
| 1 |
IC50 = 2400 nM
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| 2 |
Ki = 600 nM
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CP0483306
|
US9422235, 70
Show/Hide
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C20H18F3N3O4S
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2
|
| 1 |
IC50 = 2414 nM
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| 2 |
Ki = 1317 nM
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CP0134008
|
[4-[2-[benzyl(methyl)amino]ethoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C32H29NO4
|
2
|
| 1 |
IC50 = 2630 nM
|
|
|
| 2 |
Ki = 690 nM
|
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|
CP0517476
|
US9422235, 72
Show/Hide
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C19H22F3N3O2S
|
2
|
| 1 |
IC50 = 2655 nM
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| 2 |
Ki = 1448 nM
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CP0446595
|
2‐(4‐methoxyphenyl)‐1‐[(4‐methoxyphenyl)methyl]‐ 1,3‐benzodiazole (B14)
Show/Hide
|
C22H20N2O2
|
2
|
| 1 |
IC50 = 2700 nM
|
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|
| 2 |
Ki = 700 nM
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CP0388083
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C23H21Cl3N4O
|
1
|
| 1 |
IC50 = 2736.6 nM
|
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CP0415433
|
1-(2,4-Dichlorophenyl)-5-(5-(3-methoxyprop-1-ynyl)thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H24Cl2N4O2S
|
1
|
| 1 |
IC50 = 2737.4 nM
|
|
|
|
CP0507883
|
US9422235, 71
Show/Hide
|
C16H19F3N4O2S
|
2
|
| 1 |
IC50 = 2747 nM
|
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| 2 |
Ki = 1498 nM
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CP0422483
|
1-(4-chlorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H22ClN5O
|
2
|
| 1 |
IC50 = 2770 nM
|
|
|
| 2 |
Ki = 2180 nM
|
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|
|
CP0477866
|
US9422235, 31
Show/Hide
|
C20H21F3N2O3S
|
2
|
| 1 |
IC50 = 2778 nM
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|
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| 2 |
Ki = 1242 nM
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CP0415439
|
(2-cyclohexylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C21H22N2O2
|
2
|
| 1 |
IC50 = 2800 nM
|
|
|
| 2 |
Ki = 700 nM
|
|
|
|
CP0413640
|
US9422235, 51
Show/Hide
|
C18H19ClF3N3O3S
|
2
|
| 1 |
IC50 = 2819 nM
|
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|
| 2 |
Ki = 1851 nM
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CP0528596
|
1-Allyl-2-[5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-5,5-dimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C24H21Cl3N4O
|
1
|
| 1 |
IC50 = 2881.5 nM
|
|
|
|
CP0420581
|
(2-ethyl-1-benzothiophen-3-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C21H16OS
|
2
|
| 1 |
IC50 = 2900 nM
|
|
|
| 2 |
Ki = 700 nM
|
|
|
|
CP0420649
|
(2-cyclopentylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C23H20N2O
|
2
|
| 1 |
IC50 = 2900 nM
|
|
|
| 2 |
Ki = 700 nM
|
|
|
|
CP0372945
|
1-(2,4-difluorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H21F2N5O
|
2
|
| 1 |
IC50 = 3000 nM
|
|
|
| 2 |
Ki = 2400 nM
|
|
|
|
CP0882216
|
N-cyclopropyl-5-(naphthalen-2-yl)penta-2,4-dienamide
Show/Hide
|
C18H17NO
|
2
|
| 1 |
IC50 = 3020 nM
|
|
|
| 2 |
Ki = 810 nM
|
|
|
|
CP0490939
|
US9422235, 104
Show/Hide
|
C17H18F3N3O2S
|
2
|
| 1 |
IC50 = 3167 nM
|
|
|
| 2 |
Ki = 1877 nM
|
|
|
|
CP0386648
|
6-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-5,7-diaza-spiro[3.4]oct-5-en-8-one
Show/Hide
|
C23H19Cl3N4O
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1
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| 1 |
IC50 = 3177.2 nM
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CP0454681
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(4-methoxyphenyl)-(2-propan-2-ylbenzimidazol-1-yl)methanone
Show/Hide
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C18H18N2O2
|
2
|
| 1 |
IC50 = 3200 nM
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| 2 |
Ki = 800 nM
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CP0511251
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-3,5,5-trimethyl-3,5-dihydro-imidazol-4-one
Show/Hide
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C22H19Cl3N4O
|
1
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| 1 |
IC50 = 3249.2 nM
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CP0398571
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-5,5-dimethyl-3,5-dihydro-imidazol-4-one
Show/Hide
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C21H17Cl3N4O
|
1
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| 1 |
IC50 = 3500.6 nM
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CP0446587
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(2-cyclobutylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
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C19H18N2O2
|
2
|
| 1 |
IC50 = 3600 nM
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| 2 |
Ki = 900 nM
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CP0134009
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[4-(dibenzylamino)phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
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C36H29NO3
|
2
|
| 1 |
IC50 = 3640 nM
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| 2 |
Ki = 920 nM
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CP0460128
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1-(2,4-Dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-5-(5-pentylthiophen-2-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C27H32Cl2N4OS
|
1
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| 1 |
IC50 = 3664.3 nM
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CP0491078
|
US9422235, 24
Show/Hide
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C21H26F3N3O5S
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2
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| 1 |
IC50 = 3704 nM
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| 2 |
Ki = 1633 nM
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CP0375063
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1-(2,4-Dichlorophenyl)-4-methyl-5-[((E)-5-pent-1-enyl)-thiophen-2-yl]-1H-pyrazole-3-carboxylic Acid Piperidin-1-ylamide
Show/Hide
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C25H28Cl2N4OS
|
1
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| 1 |
IC50 = 3838.3 nM
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CP0436129
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17-heptyl-1-methyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
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C26H29NO2
|
2
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| 1 |
IC50 = 3860 nM
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| 2 |
Ki = 980 nM
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CP0327836
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[2-(4-methoxyphenyl)-1-benzofuran-3-yl]-[4-[(4-methoxyphenyl)methylamino]phenyl]methanone
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C30H25NO4
|
2
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| 1 |
IC50 = 3860 nM
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| 2 |
Ki = 1020 nM
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CP0477160
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17-hexyl-1-methyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
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C25H27NO2
|
2
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| 1 |
IC50 = 3930 nM
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| 2 |
Ki = 1010 nM
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CP0477162
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1-[(heptylamino)methyl]-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
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C26H30N2O2
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2
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| 1 |
IC50 = 3930 nM
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| 2 |
Ki = 1010 nM
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CP0467612
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2-[1-(2,4-Dichloro-phenyl)-4-methyl-5-(4-trifluoromethylphenyl)-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
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C23H19Cl2F3N4O
|
1
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| 1 |
IC50 = 3968 nM
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CP0560894
|
US9422235, 20
Show/Hide
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C19H23F3N2O5S
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2
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| 1 |
IC50 = 3978 nM
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| 2 |
Ki = 1768 nM
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CP0458457
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N-[2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)benzimidazol-5-yl]benzamide
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C28H31N3O2
|
2
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| 1 |
IC50 = 3981.07 nM
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| 2 |
Ki = 4300 nM
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CP0419648
|
US9422235, 34
Show/Hide
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C21H27F3N2O6S
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2
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| 1 |
IC50 = 4000 nM
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| 2 |
Ki = 1692 nM
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CP0482647
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(6aR,9S)-9-ethoxy-6,6,9-trimethyl-3-pentyl-7,8-dihydro-6aH-benzo[c]chromene-1,4-dione
Show/Hide
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C23H32O4
|
2
|
| 1 |
IC50 = 4070 nM
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| 2 |
Ki = 2034 nM
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CP0858812
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid ethanolamide
Show/Hide
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C19H21NO3
|
2
|
| 1 |
IC50 = 4080 nM
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| 2 |
Ki = 1030 nM
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CP0419750
|
1-benzothiophen-2-yl(naphthalen-1-yl)methanone
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C19H12OS
|
2
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| 1 |
IC50 = 4100 nM
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| 2 |
Ki = 1000 nM
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CP0460118
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5-(5-(Cyclopropylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C25H24Cl2N4OS
|
1
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| 1 |
IC50 = 4234.4 nM
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CP0415470
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naphthalen-1-yl-(2-propyl-1-benzothiophen-3-yl)methanone
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C22H18OS
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2
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| 1 |
IC50 = 4300 nM
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| 2 |
Ki = 1000 nM
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CP0388082
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1Hpyrazol-3-yl]-3,5,5-trimethyl-3,5-dihydro-imidazol-4-one
Show/Hide
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C23H21Cl3N4O
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1
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| 1 |
IC50 = 4326.9 nM
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CP0460117
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5-(5-(But-1-ynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C24H24Cl2N4OS
|
1
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| 1 |
IC50 = 4328.3 nM
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CP0386647
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-thione
Show/Hide
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C23H21Cl3N4S
|
1
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| 1 |
IC50 = 4746 nM
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CP0506593
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1-Butyl-2-[5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-5,5-dimethyl-1,5-dihydro-imidazol-4one
Show/Hide
|
C25H25Cl3N4O
|
1
|
| 1 |
IC50 = 4763.3 nM
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CP0876219
|
N-(2-hydroxyethyl)-5-(naphthalen-2-yl)penta-2,4-dienamide
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|
C17H17NO2
|
2
|
| 1 |
IC50 = 4810 nM
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| 2 |
Ki = 1270 nM
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CP0445191
|
US9422235, 64
Show/Hide
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C21H25Cl2F3N2O2S
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2
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| 1 |
IC50 = 4934 nM
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| 2 |
Ki = 2774 nM
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CP0372735
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5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperidin-1-yl)-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H24Cl3N5O
|
2
|
| 1 |
IC50 = 5000 nM
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| 2 |
Ki = 3940 nM
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CP0379503
|
4-cyano-N-[(3,4-dichlorophenyl)methyl]-1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H15Cl2N5O
|
2
|
| 1 |
IC50 = 5000 nM
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| 2 |
Ki = 3940 nM
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CP0405137
|
1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H20Cl4N4O
|
2
|
| 1 |
IC50 = 5000 nM
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| 2 |
Ki = 3940 nM
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CP0440880
|
1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H25F2N5O
|
2
|
| 1 |
IC50 = 5000 nM
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| 2 |
Ki = 3940 nM
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CP0440923
|
N-[(3,4-dichlorophenyl)methyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H20Cl2F2N4O
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2
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| 1 |
IC50 = 5000 nM
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| 2 |
Ki = 3940 nM
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CP0238599
|
2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-(4-piperidin-1-ylbutyl)benzimidazole-5-carboxamide
Show/Hide
|
C30H42N4O2
|
2
|
| 1 |
IC50 = 5011.87 nM
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| 2 |
Ki = 4800 nM
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CP0389541
|
N-(1-adamantyl)-2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)benzimidazole-5-carboxamide
Show/Hide
|
C32H41N3O2
|
2
|
| 1 |
IC50 = 5011.87 nM
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| 2 |
Ki = 4700 nM
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CP0876217
|
N-(5-(naphthalen-2-ylthio)pentyl)ethanesulfonamide
Show/Hide
|
C17H23NO2S2
|
2
|
| 1 |
IC50 = 5020 nM
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| 2 |
Ki = 1320 nM
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CP0134007
|
[2-(4-methoxyphenyl)-1-benzofuran-3-yl]-[4-(pyridin-2-ylmethylamino)phenyl]methanone
Show/Hide
|
C28H22N2O3
|
2
|
| 1 |
IC50 = 5090 nM
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| 2 |
Ki = 1340 nM
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CP0522905
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1-Benzyl-2-[5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-5,5-dimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C28H23Cl3N4O
|
1
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| 1 |
IC50 = 5126.9 nM
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CP0375062
|
1-(2,4-Dichlorophenyl)-4-methyl-5-[((E)-5-pent-1-enyl)-thiophen-2-yl]-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C27H30Cl2N4OS
|
1
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| 1 |
IC50 = 5412.8 nM
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CP0396842
|
ethyl (E)-2-benzoyl-3-[1-(2-piperidin-1-ylethyl)indol-3-yl]prop-2-enoate
Show/Hide
|
C27H30N2O3
|
1
|
| 1 |
IC50 = 5480 nM
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CP0446588
|
(2-cyclobutylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
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C22H18N2O
|
2
|
| 1 |
IC50 = 5500 nM
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| 2 |
Ki = 1400 nM
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CP0463996
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-5,5-dimethyl-1-propyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C24H23Cl3N4O
|
1
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| 1 |
IC50 = 5510.1 nM
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CP0435063
|
2-[4-(dimethylamino)phenyl]ethyl 5-chloro-3-ethyl-1H-indole-2-carboxylate
Show/Hide
|
C21H23ClN2O2
|
1
|
| 1 |
IC50 = 5570 nM
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CP0386457
|
5-(5-(Cyclopropylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C27H26Cl2N4OS
|
1
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| 1 |
IC50 = 5719.5 nM
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CP0419748
|
(4-methoxyphenyl)-[2-(4-methoxyphenyl)benzimidazol-1-yl]methanone
Show/Hide
|
C22H18N2O3
|
2
|
| 1 |
IC50 = 5900 nM
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| 2 |
Ki = 1500 nM
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CP0474980
|
US9422235, 50
Show/Hide
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C20H24Cl2F3N3O2S
|
2
|
| 1 |
IC50 = 6000 nM
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| 2 |
Ki = 3939 nM
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CP0494871
|
US9422235, 30
Show/Hide
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C24H20F3N3O4S
|
2
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| 1 |
IC50 = 6000 nM
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| 2 |
Ki = 2651 nM
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CP0564898
|
US9422235, 67
Show/Hide
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C20H15Cl2F3N2O2S
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2
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| 1 |
IC50 = 6000 nM
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| 2 |
Ki = 6000 nM
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CP0435957
|
ethyl (E)-2-benzoyl-3-[1-(2-morpholin-4-ylethyl)indol-3-yl]prop-2-enoate
Show/Hide
|
C26H28N2O4
|
1
|
| 1 |
IC50 = 6220 nM
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CP0564897
|
US9422235, 65
Show/Hide
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C19H13Cl2F3N2O2S
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2
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| 1 |
IC50 = 6246 nM
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| 2 |
Ki = 3511 nM
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CP0446663
|
(2-butylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
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C19H20N2O2
|
2
|
| 1 |
IC50 = 6300 nM
|
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| 2 |
Ki = 1600 nM
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CP0489886
|
1-(2,4-Dichlorophenyl)-4-methyl-5-(5-pentylthiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H30Cl2N4OS
|
1
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| 1 |
IC50 = 6346 nM
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CP0402759
|
US9422235, 68
Show/Hide
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C18H15Cl2F3N2O4S
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2
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| 1 |
IC50 = 6404 nM
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| 2 |
Ki = 3493 nM
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CP0415487
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(2-ethyl-1-benzothiophen-3-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C18H16O2S
|
2
|
| 1 |
IC50 = 6600 nM
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| 2 |
Ki = 1600 nM
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CP0436132
|
4-chloro-17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2(7),3,5,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H26ClNO2
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2
|
| 1 |
IC50 = 6850 nM
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| 2 |
Ki = 1740 nM
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CP0410149
|
5-chloro-3-ethyl-N-[2-[4-(4-methylpiperazin-1-yl)phenyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H29ClN4O
|
1
|
| 1 |
IC50 = 6970 nM
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CP0462577
|
1-(2,4-Dichlorophenyl)-4-methyl-5-[5-(3-phenoxyprop-1-ynyl)-thiophen-2-yl]-1H-pyrazole-3-carboxylic Acid Piperidin-1-ylamide
Show/Hide
|
C29H26Cl2N4O2S
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1
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| 1 |
IC50 = 7032.2 nM
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CP0373857
|
1-(2,4-Dichlorophenyl)-5-(5-(3-(isopropylamino)prop-1-ynyl)-thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H29Cl2N5OS
|
1
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| 1 |
IC50 = 7179.1 nM
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CP0420650
|
(4-methoxyphenyl)-(2-propylbenzimidazol-1-yl)methanone
Show/Hide
|
C18H18N2O2
|
2
|
| 1 |
IC50 = 7600 nM
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| 2 |
Ki = 1900 nM
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CP0562907
|
US9422235, 83
Show/Hide
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C24H33F3N2O4S
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2
|
| 1 |
IC50 = 7663 nM
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| 2 |
Ki = 4107 nM
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CP0385256
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[2-(4-methoxyphenyl)benzimidazol-1-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C25H18N2O2
|
2
|
| 1 |
IC50 = 7700 nM
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| 2 |
Ki = 1900 nM
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CP0519327
|
17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H27NO2
|
2
|
| 1 |
IC50 = 7940 nM
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| 2 |
Ki = 2010 nM
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CP0476637
|
N,N-diethyl-2-(4-phenoxyanilino)-1-(2-piperidin-1-ylethyl)benzimidazole-5-carboxamide
Show/Hide
|
C31H37N5O2
|
2
|
| 1 |
IC50 = 7943.28 nM
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| 2 |
Ki = 8900 nM
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CP0506592
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C21H17Cl3N4O
|
1
|
| 1 |
IC50 = 7946.1 nM
|
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|
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CP0906698
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid cyclopropylamide
Show/Hide
|
C20H21NO2
|
2
|
| 1 |
IC50 = 8020 nM
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|
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| 2 |
Ki = 2040 nM
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CP0491999
|
17-hexyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C24H25NO2
|
2
|
| 1 |
IC50 = 8140 nM
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|
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| 2 |
Ki = 2060 nM
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CP0492000
|
17-octyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C26H29NO2
|
2
|
| 1 |
IC50 = 8740 nM
|
|
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| 2 |
Ki = 2220 nM
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CP0479102
|
(E)-6-Biphenyl-4-yl-4-oxohexanoic acid ethanolamide
Show/Hide
|
C20H23NO3
|
2
|
| 1 |
IC50 = 8850 nM
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|
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| 2 |
Ki = 2250 nM
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CP0380710
|
3-ethyl-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H29N3O
|
1
|
| 1 |
IC50 = 8970 nM
|
|
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CP0399752
|
5-chloro-3-ethyl-N-[2-[4-(methylamino)phenyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C20H22ClN3O
|
1
|
| 1 |
IC50 = 9130 nM
|
|
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CP0846987
|
2-ethyl-5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)penta-2,4-dienamido)acetate
Show/Hide
|
C17H19NO5
|
2
|
| 1 |
IC50 = 9690 nM
|
|
|
| 2 |
Ki = 2560 nM
|
|
|
|
CP0914916
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid glycinamide ethyl ester
Show/Hide
|
C20H21NO4
|
2
|
| 1 |
IC50 = 9820 nM
|
|
|
| 2 |
Ki = 2500 nM
|
|
|
|
CP0436133
|
1-chloro-17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H26ClNO2
|
2
|
| 1 |
IC50 = 9880 nM
|
|
|
| 2 |
Ki = 2510 nM
|
|
|
|
CP0378997
|
11-(4-hexyl-3-hydroxy-phenoxy)-undecanoic acid[2-(3,4-dihydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C31H47NO5
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0428635
|
11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid [2-(3,4-dihydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C30H45NO5
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0437123
|
12-(4-hexyl-3-hydroxy-phenoxy)-dodecanoic acid(2-hydroxy-ethyl)-amide
Show/Hide
|
C26H45NO4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0437124
|
11-(4-hexyl-3-hydroxy-phenoxy)-undecanoic acid(3-methoxy-4-hydroxy-phenyl)-amide
Show/Hide
|
C31H47NO5
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0493393
|
1-Biphenyl-4-yl-4-morpholin-4-yl-butane-1,4-dione
Show/Hide
|
C20H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858811
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid cyclopropamide
Show/Hide
|
C19H19NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858813
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid(2-hydroxy-1(R)-methylethanolamide
Show/Hide
|
C20H23NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858814
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid
Show/Hide
|
C16H14O3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858815
|
(E)-6-(3,4-Dimethoxyphenyl)-4-oxohex-5-enoic acid ethanolamide
Show/Hide
|
C16H21NO5
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858816
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic piperidinamide
Show/Hide
|
C22H25NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858817
|
(E)-6-Biphenyl-4-yl-4-oxohex-5-enoic acid ethanolamide
Show/Hide
|
C20H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0861035
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid(4-hydroxyphenyl)-amide
Show/Hide
|
C22H19NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0878641
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid(2-hydroxy-1(R)-methylethanolamide
Show/Hide
|
C19H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0878642
|
(E)-7-Naphthalen-2-yl-5-oxo-hept-6-enoic acid glycinamide ethyl ester
Show/Hide
|
C21H23NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0884366
|
(E)-N-(4-Hydroxyphenyl)-6-(4-methoxyphenyl)-4-oxohex-5-enamide
Show/Hide
|
C19H19NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0890249
|
(E)-6-(3,4-Dimethoxyphenyl)4-oxohex-5-enoic acid piperedinamide
Show/Hide
|
C19H25NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0906700
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid piperidinamide
Show/Hide
|
C21H23NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0918957
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid diethanolamide
Show/Hide
|
C20H23NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0918978
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid
Show/Hide
|
C17H16O3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0438035
|
[(Z)-3-acetyloxyprop-1-enyl] 5-methylideneoctadecanoate
Show/Hide
|
C24H42O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0461445
|
(E)-N-[(2R)-1-hydroxy-3-methoxypropan-2-yl]-N-methyloctadec-4-enamide
Show/Hide
|
C23H45NO3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0489612
|
6-methyl-N-propyl-2-(tricyclo[3.3.1.03,7]nonane-3-carbonylamino)-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide
Show/Hide
|
C22H31N3O2S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki = 91.2 nM
|
|
|
|
CP0380713
|
5-chloro-N-[2-(4-nitrophenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C17H14ClN3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0383426
|
N-[2-(4-aminophenyl)ethyl]-5-chloro-1H-indole-2-carboxamide
Show/Hide
|
C17H16ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0383427
|
5-chloro-N-[2-(4-chlorophenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C17H14Cl2N2O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0385361
|
5-chloro-3-ethyl-N-[2-(4-nitrophenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C19H18ClN3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0385362
|
5-chloro-N-[2-[4-(dimethylamino)phenyl]ethyl]-3-ethyl-1H-indole-2-carboxamide
Show/Hide
|
C21H24ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0385535
|
N-[2-(4-aminophenyl)ethyl]-5-chloro-3-ethyl-1H-indole-2-carboxamide
Show/Hide
|
C19H20ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0385536
|
5-chloro-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0387212
|
5-chloro-3-ethyl-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H28ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0389340
|
5-chloro-3-ethyl-N-[2-(4-fluorophenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C19H18ClFN2O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0395905
|
5-chloro-3-ethyl-N-[2-(4-methylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C20H21ClN2O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0395907
|
5-chloro-N-[2-(4-chlorophenyl)ethyl]-3-ethyl-1H-indole-2-carboxamide
Show/Hide
|
C19H18Cl2N2O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0400642
|
5-chloro-3-(1-hydroxyethyl)-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H28ClN3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0400643
|
5-chloro-N-[2-[4-(methylamino)phenyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C18H18ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0417341
|
5-chloro-N-[2-[4-(dimethylamino)phenyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C19H20ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0417342
|
2-(4-nitrophenyl)ethyl 5-chloro-3-ethyl-1H-indole-2-carboxylate
Show/Hide
|
C19H17ClN2O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0436061
|
3-acetyl-5-chloro-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H26ClN3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0846986
|
1-(5-(benzo[d][1,3]dioxol-5-yloxy)pentyl)urea
Show/Hide
|
C13H18N2O4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846988
|
N-(5-(naphthalen-2-yloxy)pentyl)ethanesulfonamide
Show/Hide
|
C17H23NO3S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846989
|
N-(5-(naphthalen-1-yloxy)pentyl)ethanesulfonamide
Show/Hide
|
C17H23NO3S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846990
|
1-ethyl-3-(5-(naphthalen-2-yloxy)pentyl)urea
Show/Hide
|
C18H24N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846991
|
1-(5-(benzo[d][1,3]dioxol-5-yloxy)pentyl)-3-ethylurea
Show/Hide
|
C15H22N2O4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0852446
|
2-ethyl-(6-(naphthalen-1-yloxy)hexanamido)acetate
Show/Hide
|
C20H25NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853976
|
1-ethyl-3-(5-(naphthalen-1-yloxy)pentyl)urea
Show/Hide
|
C18H24N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853977
|
2-ethyl-5-(naphthalen-2-yl)penta-2,4-dienamido)acetate
Show/Hide
|
C19H19NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853978
|
N-cyclopropyl-5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)penta-2,4-dienamide
Show/Hide
|
C16H17NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853979
|
N-(5-(benzo[d][1,3]dioxol-5-yloxy)pentyl)ethanesulfonamide
Show/Hide
|
C14H21NO5S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853980
|
5-(9H-fluoren-3-yl)-N-(2-hydroxyethyl)penta-2,4-dienamide
Show/Hide
|
C20H19NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853981
|
2-ethyl-(6-(naphthalen-2-yloxy)hexanamido)acetate
Show/Hide
|
C20H25NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858225
|
N-cyclopropyl-6-(naphthalen-2-yloxy)hexanamide
Show/Hide
|
C19H23NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858226
|
N-(2-hydroxyethyl)-6-(naphthalen-2-yloxy)hexanamide
Show/Hide
|
C18H23NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0860293
|
N-(2-hydroxyethyl)-6-(naphthalen-1-yloxy)hexanamide
Show/Hide
|
C18H23NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0860294
|
N-cyclopropyl-5-(9H-fluoren-3-yl)penta-2,4-dienamide
Show/Hide
|
C21H19NO
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0860296
|
2-ethyl-5-(9H-fluoren-3-yl)penta-2,4-dienamido)acetate
Show/Hide
|
C22H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0876218
|
N-cyclopropyl-6-(naphthalen-1-yloxy)hexanamide
Show/Hide
|
C19H23NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0876220
|
1-(5-(naphthalen-1-yloxy)pentyl)urea
Show/Hide
|
C16H20N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0401037
|
(2-methylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C19H14N2O
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0401056
|
naphthalen-1-yl-(2-propylbenzimidazol-1-yl)methanone
Show/Hide
|
C21H18N2O
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0401058
|
(4-methoxyphenyl)-(2-methylbenzimidazol-1-yl)methanone
Show/Hide
|
C16H14N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0415513
|
(4-methoxyphenyl)-[2-(2-methylpropyl)benzimidazol-1-yl]methanone
Show/Hide
|
C19H20N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0394387
|
N-[6-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxyhexyl]acetamide
Show/Hide
|
C30H38N2O5
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki = 1969 nM
|
|
|
|
CP0401724
|
methyl 5-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxypentanoate
Show/Hide
|
C28H33NO6
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki = 200.7 nM
|
|
|
|
CP0405460
|
5-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxypentanoic acid
Show/Hide
|
C27H31NO6
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki = 1307 nM
|
|
|
|
CP0436130
|
17-heptyl-1-[(heptylamino)methyl]-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C33H44N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0436131
|
17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C18H13NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0477157
|
1-bromo-17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H26BrNO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0492001
|
1-(heptoxymethyl)-17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C33H43NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0176623
|
[4-[4-[(3-fluorophenoxy)methyl]triazol-1-yl]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C31H22FN3O4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0262330
|
[4-[bis[(3,5-difluorophenyl)methyl]amino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C36H25F4NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0327835
|
[4-[4-[benzyl(methyl)amino]butoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C34H33NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0363236
|
[4-[5-[benzyl(methyl)amino]pentoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C35H35NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0467611
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-5,5-dimethyl-3,5-dihydro-imidazol-4-one
Show/Hide
|
C22H19Cl3N4O
|
1
|
| 1 |
IC50 = 10260 nM
|
|
|
|
CP0238600
|
2-(4-ethoxyanilino)-N,N-diethyl-1-(2-piperidin-1-ylethyl)benzimidazole-5-carboxamide
Show/Hide
|
C27H37N5O2
|
2
|
| 1 |
IC50 = 12589.25 nM
|
|
|
| 2 |
Ki = 10400 nM
|
|
|
|
CP0238598
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-N-phenylbenzimidazole-5-carboxamide
Show/Hide
|
C28H31N3O2
|
2
|
| 1 |
IC50 = 15848.93 nM
|
|
|
| 2 |
Ki = 14400 nM
|
|
|
|
CP0356649
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)benzimidazol-5-amine
Show/Hide
|
C21H27N3O
|
2
|
| 1 |
IC50 = 19952.62 nM
|
|
|
| 2 |
Ki = 21000 nM
|
|
|
|
CP0560888
|
US9422235, 91
Show/Hide
|
C17H25F3N2O2S
|
2
|
| 1 |
IC50 = 29390 nM
|
|
|
| 2 |
Ki = 16590 nM
|
|
|
|
CP0388772
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(2-fluorobenzyl)acetamide
Show/Hide
|
C23H15Cl4FN4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0388773
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(3-fluorobenzyl)acetamide
Show/Hide
|
C23H15Cl4FN4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0388774
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-chlorobenzyl)acetamide
Show/Hide
|
C23H15Cl5N4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0428633
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-phenylacetamide
Show/Hide
|
C22H14Cl4N4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0428634
|
2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-fluorobenzyl)acetamide
Show/Hide
|
C23H16Cl3FN4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0435287
|
N-benzyl-2-[4,5-bis(2,4-dichlorophenyl)triazol-2-yl]acetamide
Show/Hide
|
C23H16Cl4N4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0444807
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(2,5-difluorobenzyl)acetamide
Show/Hide
|
C23H14Cl4F2N4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0445458
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-cyclohexylacetamide
Show/Hide
|
C22H20Cl4N4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0455069
|
2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(2-fluorobenzyl)acetamide
Show/Hide
|
C23H16Cl3FN4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0486799
|
N-benzyl-2-[4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)triazol-2-yl]acetamide
Show/Hide
|
C23H17Cl3N4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0495914
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(2-chlorobenzyl)acetamide
Show/Hide
|
C23H15Cl5N4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0504058
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-methoxybenzyl)acetamide
Show/Hide
|
C24H18Cl4N4O2
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0521468
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-fluorobenzyl)acetamide
Show/Hide
|
C23H15Cl4FN4O
|
1
|
| 1 |
IC50 > 10 nM
|
|
|
|
CP0379501
|
4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H20Cl3N5O
|
2
|
| 1 |
IC50 > 5000 nM
|
|
|
| 2 |
Ki > 3940 nM
|
|
|
|
CP0393710
|
N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(1H-pyrrol-1-yl)-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H15Cl5N4O
|
2
|
| 1 |
IC50 > 5000 nM
|
|
|
| 2 |
Ki > 3940 nM
|
|
|
|
CP0501941
|
1-(2,4-difluorophenyl)-4-methyl-N-(morpholin-4-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C19H19F2N5O2
|
2
|
| 1 |
IC50 > 5000 nM
|
|
|
| 2 |
Ki > 3940 nM
|
|
|
|
CP0410964
|
4-oxo-1-pentyl-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C31H38N2O2S
|
1
|
| 1 |
Ki = 0.09 nM
|
|
|
|
CP0500721
|
1-butyl-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C30H36N2O2S
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0124848
|
(6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-6,6-dimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C25H38O3
|
1
|
| 1 |
Ki = 0.15 nM
|
|
|
|
CP0316457
|
(6aS,10aS)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C25H38O3
|
1
|
| 1 |
Ki = 0.15 nM
|
|
|
|
CP0516603
|
N-(1-adamantyl)-7-hydroxy-2-methyl-5-oxo-4-pentylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C23H32N4O3
|
1
|
| 1 |
Ki = 0.18 nM
|
|
|
|
CP0376757
|
N-(1-adamantyl)-2-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C25H32N2O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0513751
|
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxoquinoline-3-carboxamide
Show/Hide
|
C24H25FN2O2
|
1
|
| 1 |
Ki = 0.25 nM
|
|
|
|
CP0435697
|
7-fluoro-4-oxo-1-pentyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C25H33FN2O2
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0488979
|
US8846730, 79
Show/Hide
|
C23H30F3N3O3S
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0535627
|
US8859596, 141
Show/Hide
|
C23H31F3N4O4S
|
1
|
| 1 |
Ki = 0.32 nM
|
|
|
|
CP0453121
|
N-(1-adamantyl)-2-[5-(furan-2-yl)-1-pentylindol-3-yl]-2-oxoacetamide
Show/Hide
|
C29H34N2O3
|
1
|
| 1 |
Ki = 0.37 nM
|
|
|
|
CP0393333
|
4-oxo-7-phenylsulfanyl-1-propyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C29H34N2O2S
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0402796
|
US8846730, 40
Show/Hide
|
C25H33F3N4O4S
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0463805
|
US8859596, 193
Show/Hide
|
C23H32F3N5O2S
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0545674
|
US8859596, 198
Show/Hide
|
C25H36F3N5O2
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0458967
|
US8846730, 83
Show/Hide
|
C25H30F3N3O3S
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0573332
|
US8846730, 23
Show/Hide
|
C25H31F3N2O4S
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0476297
|
N-cyclohexyl-1-(3,4-dichlorophenyl)-4-ethyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H24Cl2N4O
|
1
|
| 1 |
Ki = 0.51 nM
|
|
|
|
CP0480579
|
N-(1-adamantyl)-8-methoxy-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C26H34N2O3
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0468403
|
US8859596, 169
Show/Hide
|
C23H31F3N4O3S
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0506904
|
US8859596, 144
Show/Hide
|
C21H29F3N4O2S
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0447476
|
5-bromopentyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C25H35BrO4
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0454191
|
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H24FN3O2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0471931
|
1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H24FN3O2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0048140
|
N-(1-adamantyl)-6-(furan-2-yl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C29H34N2O3
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0493054
|
4-Oxo-1-pentyl-6-pyrrol-1-yl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C29H35N3O2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0051827
|
8-Methyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C26H34N2O2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0375379
|
US8846730, 4
Show/Hide
|
C26H34F3N3O3S
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0429708
|
US8846730, 5
Show/Hide
|
C27H36F3N3O3S
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0390265
|
US8859596, 192
Show/Hide
|
C20H26F3N5O3S
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0545678
|
US8859596, 200
Show/Hide
|
C26H31F3N6O2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0482100
|
3-bromopropyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C23H31BrO4
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0517831
|
4-bromobutyl 1-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]cyclobutane-1-carboxylate
Show/Hide
|
C25H33BrO4
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0947552
|
S-Propyl-2-[(6aR,10aR)-6a,7,10,10a-tetrahydro-1-hydroxy-6,6,9-trimethyl-6H-dibenzo[b,d]pyran-3-yl]-2-methylpropanethioate
Show/Hide
|
C23H32O3S
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0517751
|
(6aS,10aS)-6,6,9-trimethyl-3-[(E)-C-methyl-N-(2-morpholin-4-ylethoxy)carbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C24H34N2O4
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0411351
|
US8895592, 19
Show/Hide
|
C21H27F3N2O3S
|
1
|
| 1 |
Ki = 0.73 nM
|
|
|
|
CP0449956
|
1-[(4-fluorophenyl)methyl]-4-hydroxy-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H24FN3O3
|
1
|
| 1 |
Ki = 0.75 nM
|
|
|
|
CP0529572
|
1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxoquinoline-3-carboxamide
Show/Hide
|
C24H25FN2O2
|
1
|
| 1 |
Ki = 0.75 nM
|
|
|
|
CP0436996
|
N-(1-adamantyl)-7-fluoro-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C25H31FN2O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0480040
|
1-butyl-7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C24H31FN2O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0410558
|
US8859596, 191
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0562734
|
4-bromobutyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C24H33BrO4
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0385257
|
US8895592, 32
Show/Hide
|
C23H31F3N2O3S
|
1
|
| 1 |
Ki = 0.82 nM
|
|
|
|
CP0051372
|
1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H24FN3O2
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0386407
|
N-(1-adamantyl)-7-(benzenesulfonyl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O4S
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0476372
|
5-(2-chloropyrrol-1-yl)-N-cyclohexyl-1-(3,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H21Cl3N4O
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0543942
|
US8846730, 72
Show/Hide
|
C26H33F3N2O4S
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0517832
|
4-cyanobutyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C25H33NO4
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0560405
|
N-(1-adamantyl)-7-hydroxy-1-methyl-5-oxo-4-pentyl-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C23H34N4O3
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0042459
|
(6aR,10aR)-6,6,9-Trimethyl-3-(1-methyl-1-phenyl-ethyl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C25H30O2
|
1
|
| 1 |
Ki = 0.91 nM
|
|
|
|
CP0471598
|
N-(1-adamantyl)-8-nitro-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C25H31N3O4
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0443539
|
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-5-(4-methoxyphenyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C27H29FN2O3
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0390096
|
US8859596, 181
Show/Hide
|
C23H32F3N5O3S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0469773
|
US8859596, 154
Show/Hide
|
C20H25F3N4O3S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0466141
|
[2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropyl] pentanoate
Show/Hide
|
C25H36O4
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0919746
|
(4,5-bis((tetrahydro-2H-pyran-4-yl)methyl)-5H-[1,3]dioxolo[4,5-f]indol-7-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
|
C29H39NO5
|
1
|
| 1 |
Ki = 1.023 nM
|
|
|
|
CP0510098
|
3',5'-dichloro-4-(2-phenylpropan-2-yl)biphenyl-2,6-diol
Show/Hide
|
C21H18Cl2O2
|
1
|
| 1 |
Ki = 1.07 nM
|
|
|
|
CP0378066
|
1-(2-methoxyethyl)-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C29H34N2O3S
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0509469
|
US8895592, 38
Show/Hide
|
C25H28F3N5O2S
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0417828
|
US8846730, 81
Show/Hide
|
C23H29F3N2O4S
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0390100
|
US8859596, 197
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0435741
|
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxo-5-phenylpyridine-3-carboxamide
Show/Hide
|
C26H27FN2O2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0542114
|
US8846730, 75
Show/Hide
|
C22H26F3N3O4S
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0394007
|
4-cyanobutyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]acetate
Show/Hide
|
C23H29NO4
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0469875
|
N-cyclopropyl-11-(3-methoxy-5-pentylphenoxy)undecanamide
Show/Hide
|
C26H43NO3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0390569
|
N-cycloheptyl-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H24Cl2N4O
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0440242
|
N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-dichloropyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H20Cl4N4O
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0435747
|
1-[2-(dimethylamino)ethyl]-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C30H37N3O2S
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0407090
|
US8846730, 51
Show/Hide
|
C26H34F3N3O2S2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0538617
|
US8846730, 50
Show/Hide
|
C25H33F3N2O4S
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0517830
|
3-imidazol-1-ylpropyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C26H34N2O4
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0514858
|
(6aR,10aR)-3-[1-(5-Bromopentyl)cyclopentyl]-6,6a,7,8,10,10ahexahydro-1-hydroxy-6,6-dimethyl-9H-dibenzo[b,d]pyran-9-one
Show/Hide
|
C25H35BrO3
|
1
|
| 1 |
Ki = 1.32 nM
|
|
|
|
CP0460191
|
US8895592, 36
Show/Hide
|
C21H22F3N3O3S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0482099
|
3-cyanopropyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C24H31NO4
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0560406
|
N-(1-adamantyl)-4-(4-fluorobutyl)-7-hydroxy-1-methyl-5-oxo-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H31FN4O3
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0410517
|
N-(4-methylcyclohexyl)-2-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C22H30N2O2
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0414010
|
US8895592, 25
Show/Hide
|
C22H23F3N4O3S
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0406727
|
ethyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C22H30O4
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0473858
|
(R)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H26Cl2N4O
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0393334
|
N-(1-adamantyl)-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O2S
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0460111
|
US8895592, 37
Show/Hide
|
C25H28F3N5O2S
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0464067
|
US8859596, 189
Show/Hide
|
C24H32F3N5O2S
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0527324
|
(6aR,9R,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7,8,9,10,10a-hexahydro-6,6-dimethyl-6H-dibenzo[b,d]pyran-1,9 diol
Show/Hide
|
C24H35BrO3
|
1
|
| 1 |
Ki = 1.62 nM
|
|
|
|
CP0502799
|
(6aR,9S,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6a,7,8,9,10,10a-hexahydro-6,6-dimethyl-6H-dibenzo[b,d]pyran-1,9 diol
Show/Hide
|
C24H35BrO3
|
1
|
| 1 |
Ki = 1.63 nM
|
|
|
|
CP0517506
|
(3',5'-dichloro-2,6-dimethoxybiphenyl-4-yl)(phenyl)methanol
Show/Hide
|
C21H18Cl2O3
|
1
|
| 1 |
Ki = 1.66 nM
|
|
|
|
CP0456245
|
N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-ethylpyrazole-3-carboxamide
Show/Hide
|
C24H28Cl2N4O
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0467462
|
butyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C24H34O4
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0390263
|
US8859596, 190
Show/Hide
|
C23H29F3N4O2S
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0450107
|
US8859596, 147
Show/Hide
|
C24H33F3N4O3S
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0386991
|
methyl 2-(adamantane-1-carbonylamino)-5-butyl-4-methylthiophene-3-carboxylate
Show/Hide
|
C22H31NO3S
|
1
|
| 1 |
Ki = 1.72 nM
|
|
|
|
CP0513750
|
N-cycloheptyl-4-hydroxy-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H30N4O4
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0460005
|
US8846730, 73
Show/Hide
|
C23H28F3N3O4S
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0545677
|
US8859596, 164
Show/Hide
|
C22H28F6N4O2S
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0558921
|
4-cyanobutyl 1-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]cyclobutane-1-carboxylate
Show/Hide
|
C26H33NO4
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0516604
|
N-(1-adamantyl)-4-butyl-7-hydroxy-1-methyl-5-oxo-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H32N4O3
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0481084
|
N-(1-adamantyl)-5-phenyl-1-prop-2-enylindole-3-carboxamide
Show/Hide
|
C28H30N2O
|
1
|
| 1 |
Ki = 1.82 nM
|
|
|
|
CP0120450
|
N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H30N4O3
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0409164
|
N-cycloheptyl-1-(2-morpholin-4-ylethyl)-2-oxoquinoline-3-carboxamide
Show/Hide
|
C23H31N3O3
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0422475
|
US8895592, 29
Show/Hide
|
C21H22F3N3O3S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0429189
|
US8846730, 54
Show/Hide
|
C26H33F4N3O3S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0382825
|
N-(3-pentyl-1,3-benzothiazol-2-ylidene)naphthalene-1-carboxamide
Show/Hide
|
C23H22N2OS
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0671680
|
SID50107233
Show/Hide
|
C28H30N2O6S
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0525855
|
N-(1-adamantyl)-4-(4-fluorobutyl)-7-hydroxy-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H29FN4O3
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0385072
|
ethyl 2-(adamantane-1-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C22H29NO3S
|
1
|
| 1 |
Ki = 2.15 nM
|
|
|
|
CP0498832
|
N-cyclohexyl-1-[(4-fluorophenyl)methyl]-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H22FN3O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0381993
|
5-bromo-N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
|
C20H22BrFN2O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0195800
|
4-Oxo-1-pentyl-6-thiophen-2-yl-1,4-dihydro-quinoline-3-carboxylic acidadamantan-1-ylamide
Show/Hide
|
C29H34N2O2S
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0376648
|
(S)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H26Cl2N4O
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0497271
|
6-(furan-2-yl)-4-oxo-1-pentyl-N-((1R,2R,4S)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C29H36N2O3
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0426923
|
N-cyclohexyl-4-hydroxy-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C21H28N4O4
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0425247
|
methyl 2-(adamantane-1-carbonylamino)-4-ethyl-5-methylthiophene-3-carboxylate
Show/Hide
|
C20H27NO3S
|
1
|
| 1 |
Ki = 2.46 nM
|
|
|
|
CP0429455
|
N-(1-adamantyl)-5-(furan-2-yl)-1-pentylindole-3-carboxamide
Show/Hide
|
C28H34N2O2
|
1
|
| 1 |
Ki = 2.48 nM
|
|
|
|
CP0453371
|
1-(4-hydroxybutyl)-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C30H36N2O3S
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0415632
|
US8895592, 26
Show/Hide
|
C23H24F3N3O3S
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0426609
|
US8859596, 188
Show/Hide
|
C22H28F3N5O2S
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0506907
|
US8859596, 199
Show/Hide
|
C26H31F3N6O2
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0526748
|
N-(1-adamantyl)-4-butyl-7-hydroxy-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H30N4O3
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0469872
|
N-cyclopropyl-11-(3-pentyl-5-propan-2-yloxyphenoxy)undecanamide
Show/Hide
|
C28H47NO3
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0381992
|
N-cycloheptyl-5-(4-fluorophenyl)-1-[(4-fluorophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
|
C26H26F2N2O2
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0535624
|
US8859596, 165
Show/Hide
|
C23H31F3N4O2S
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0540414
|
2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methyl-N-pentylpropanamide
Show/Hide
|
C25H37NO3
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0537625
|
N-cyclohexyl-1-[(4-fluorophenyl)methyl]-2-oxoquinoline-3-carboxamide
Show/Hide
|
C23H23FN2O2
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0404948
|
7-fluoro-4-oxo-1-propyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C23H29FN2O2
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0447477
|
2-bromoethyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C22H29BrO4
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0454189
|
N-cycloheptyl-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H30N4O3
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0452614
|
butyl 1-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]cyclobutane-1-carboxylate
Show/Hide
|
C25H34O4
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0422532
|
US8846730, 53
Show/Hide
|
C26H33F4N3O3S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0519862
|
US8846730, 22
Show/Hide
|
C25H31F3N2O4S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0487732
|
(6aR,10aR)-3-[1-(6-Bromohexyl)cyclopentyl]-6,6a,7,8,10,10ahexahydro-1-hydroxy-6,6-dimethyl-9H-dibenzo[b,d]pyran-9-one
Show/Hide
|
C26H37BrO3
|
1
|
| 1 |
Ki = 3.02 nM
|
|
|
|
CP0409849
|
US8895592, 2
Show/Hide
|
C20H26ClN3O3S
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0488981
|
US8846730, 84
Show/Hide
|
C24H28F3N3O4S
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0487731
|
(6aR,10aR)-3-(1-Hexyl-cyclopent-1-yl)-6,6a,7,8,10,10a-hexahydro-1-hydroxy-6,6-dimethyl-9H-dibenzo[b,d]pyran-9-one
Show/Hide
|
C26H38O3
|
1
|
| 1 |
Ki = 3.34 nM
|
|
|
|
CP0290316
|
N-(1-adamantyl)-4-oxo-1-pentyl-6-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O2S
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0457647
|
N-(1-adamantyl)-7-(benzenesulfinyl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O3S
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0526835
|
N-cyclopropyl-11-(3-pentylphenoxy)undecanamide
Show/Hide
|
C25H41NO2
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0502931
|
N-(1-adamantyl)-1-pentyl-6-phenylindole-3-carboxamide
Show/Hide
|
C30H36N2O
|
1
|
| 1 |
Ki = 3.52 nM
|
|
|
|
CP0386405
|
N-(1-adamantyl)-6-fluoro-4-oxo-1-pentyl-7-pyrrol-1-ylquinoline-3-carboxamide
Show/Hide
|
C29H34FN3O2
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0415067
|
US8846730, 69
Show/Hide
|
C17H16Cl2N2O3
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0471615
|
butyl (2R)-2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]propanoate
Show/Hide
|
C23H32O4
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0420626
|
US8846730, 39
Show/Hide
|
C24H33F3N4O2S
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0548374
|
(6aS,10aS)-3-[(E)-N-(3-imidazol-1-ylpropoxy)-C-methylcarbonimidoyl]-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C24H31N3O3
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0195828
|
N-(1-adamantyl)-4-oxo-1-pentyl-6-phenylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0111432
|
quinolin-8-yl 4-methyl-3-piperidin-1-ylsulfonylbenzoate
Show/Hide
|
C22H22N2O4S
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0396947
|
N-cycloheptyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C24H28Cl2N4O
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0085407
|
6-(4-Hydroxy-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylicacid adamantan-1-ylamide
Show/Hide
|
C31H36N2O3
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0395647
|
1-[(4-chlorophenyl)methyl]-N-cycloheptyl-2-oxopyridine-3-carboxamide
Show/Hide
|
C20H23ClN2O2
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0415214
|
N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxoquinoline-3-carboxamide
Show/Hide
|
C23H31N3O3
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0420376
|
N-cyclopropyl-8-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]octanamide
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|
C27H45NO3
|
1
|
| 1 |
Ki = 4.2 nM
|
|
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CP0425254
|
methyl 2-(adamantane-1-carbonylamino)-5-methyl-4-propylthiophene-3-carboxylate
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|
C21H29NO3S
|
1
|
| 1 |
Ki = 4.28 nM
|
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CP0390101
|
US8859596, 151
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C22H28F3N5O2S
|
1
|
| 1 |
Ki = 4.3 nM
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CP0482473
|
(5Z,8Z,11Z,13S,14Z)-N-cyclopropyl-13-methylicosa-5,8,11,14-tetraenamide
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|
C24H39NO
|
1
|
| 1 |
Ki = 4.3 nM
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CP0054397
|
1-But-3-enyl-6-furan-2-yl-4-oxo-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
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|
C28H30N2O3
|
1
|
| 1 |
Ki = 4.4 nM
|
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CP0404949
|
1-ethyl-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C28H32N2O2S
|
1
|
| 1 |
Ki = 4.4 nM
|
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CP0409771
|
US8846730, 80
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C23H25F6N3O3S
|
1
|
| 1 |
Ki = 4.4 nM
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CP0495251
|
butyl 2-[(6aR,9S,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C23H34O5
|
1
|
| 1 |
Ki = 4.5 nM
|
|
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CP0385075
|
US8846730, 24
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C26H34F3N3O3S
|
1
|
| 1 |
Ki = 4.6 nM
|
|
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CP0401178
|
US8846730, 44
Show/Hide
|
C25H32F3N3O3S
|
1
|
| 1 |
Ki = 4.6 nM
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CP0085406
|
4-Oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C25H32N2O2
|
1
|
| 1 |
Ki = 4.7 nM
|
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CP0548834
|
N-cyclopropyl-11-(3-pentyl-5-prop-2-enoxyphenoxy)undecanamide
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|
C28H45NO3
|
1
|
| 1 |
Ki = 4.7 nM
|
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CP0398722
|
(3',5'-dichloro-2-hydroxy-6-methoxybiphenyl-4-yl)(phenyl)methanone
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|
C20H14Cl2O3
|
1
|
| 1 |
Ki = 4.77 nM
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CP0434013
|
1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
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|
C20H23FN2O2
|
1
|
| 1 |
Ki = 4.8 nM
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CP0564717
|
N-(1-adamantyl)-7-hydroxy-2-(2-hydroxyethyl)-5-oxo-4-pentylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C24H34N4O4
|
1
|
| 1 |
Ki = 4.8 nM
|
|
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CP0491211
|
US8846730, 82
Show/Hide
|
C29H40F3N3O4S
|
1
|
| 1 |
Ki = 4.9 nM
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CP0405615
|
6-bromo-4-oxo-1-pentyl-N-((1R,2R,4S)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C25H33BrN2O2
|
1
|
| 1 |
Ki = 5 nM
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CP0440547
|
US8895592, 8
Show/Hide
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C24H31F3N2O3S
|
1
|
| 1 |
Ki = 5 nM
|
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CP0420203
|
US8846730, 19
Show/Hide
|
C25H27F3N4O3S
|
1
|
| 1 |
Ki = 5 nM
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CP0394005
|
methyl 2-(adamantane-1-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
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|
C21H27NO3S
|
1
|
| 1 |
Ki = 5.08 nM
|
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CP0395641
|
5-bromo-1-butyl-N-cycloheptyl-2-oxopyridine-3-carboxamide
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|
C17H25BrN2O2
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
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CP0488394
|
US8859596, 186
Show/Hide
|
C21H28F3N5O2S
|
1
|
| 1 |
Ki = 5.1 nM
|
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CP0487733
|
(6aR,9R,10aR)-3-(1-hexylcyclobutyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
|
C25H38O3
|
1
|
| 1 |
Ki = 5.13 nM
|
|
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CP0443118
|
US8859596, 175
Show/Hide
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C22H30F3N5O2S
|
1
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| 1 |
Ki = 5.3 nM
|
|
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CP0458984
|
US8895592, 21
Show/Hide
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C22H24F3N3O3S
|
1
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| 1 |
Ki = 5.4 nM
|
|
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CP0408164
|
US8846730, 71
Show/Hide
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C26H34F3N3O4S
|
1
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| 1 |
Ki = 5.4 nM
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CP0455246
|
7-fluoro-1-(2-methoxyethyl)-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C23H29FN2O3
|
1
|
| 1 |
Ki = 5.5 nM
|
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CP0565981
|
(6aR,9R,10aR)-3-(1-adamantyl)-1-hydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-9-carbaldehyde
Show/Hide
|
C26H34O3
|
1
|
| 1 |
Ki = 5.5 nM
|
|
|
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CP0524250
|
US8846730, 38
Show/Hide
|
C24H26F3N3O3S2
|
1
|
| 1 |
Ki = 5.5 nM
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CP0506341
|
1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methyl-N-(1-phenylethyl)pyrazole-3-carboxamide
Show/Hide
|
C25H24Cl2N4O
|
1
|
| 1 |
Ki = 5.7 nM
|
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CP0380261
|
1-(2,4-Dichlorophenyl)-4-methyl-N-tert-pentyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H22Cl2N4O
|
1
|
| 1 |
Ki = 5.7 nM
|
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|
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CP0383647
|
N-(1-adamantyl)-5-(furan-2-yl)-1-prop-2-enylindole-3-carboxamide
Show/Hide
|
C26H28N2O2
|
1
|
| 1 |
Ki = 5.73 nM
|
|
|
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CP0454196
|
1-benzyl-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
Ki = 5.8 nM
|
|
|
|
CP0527323
|
(6aR,10aR)-3-[1-(5-Bromopentyl)cyclobutyl]-6,6a,7,8,10,10ahexahydro-1-hydroxy-6,6-dimethyl-9H-dibenzo[b,d]pyran-9-one
Show/Hide
|
C24H33BrO3
|
1
|
| 1 |
Ki = 5.88 nM
|
|
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CP0481802
|
methyl 2-(adamantane-1-carbonylamino)-5-ethyl-4-methylthiophene-3-carboxylate
Show/Hide
|
C20H27NO3S
|
1
|
| 1 |
Ki = 5.92 nM
|
|
|
|
CP0420476
|
US8846730, 36
Show/Hide
|
C27H29F3N2O3S
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0390095
|
US8859596, 176
Show/Hide
|
C22H28F3N5O4S
|
1
|
| 1 |
Ki = 6.1 nM
|
|
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CP0856485
|
2-Ethyl-5-methyl-1-phenyl-1H-pyrrole-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C24H30N2O
|
1
|
| 1 |
Ki = 6.15 nM
|
|
|
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CP0468042
|
US8859596, 148
Show/Hide
|
C22H30F3N5OS
|
1
|
| 1 |
Ki = 6.2 nM
|
|
|
|
CP0535625
|
US8859596, 174
Show/Hide
|
C22H30F4N4O2S
|
1
|
| 1 |
Ki = 6.2 nM
|
|
|
|
CP0531748
|
4-(4-fluorobutyl)-7-hydroxy-N-(3-hydroxy-1-adamantyl)-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H29FN4O4
|
1
|
| 1 |
Ki = 6.2 nM
|
|
|
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CP0195829
|
6-Isopropyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C28H38N2O2
|
1
|
| 1 |
Ki = 6.3 nM
|
|
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CP0433038
|
butyl (2S)-2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]propanoate
Show/Hide
|
C23H32O4
|
1
|
| 1 |
Ki = 6.3 nM
|
|
|
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CP0435085
|
N-(1-adamantyl)-1-pentyl-5-thiophen-2-ylindole-3-carboxamide
Show/Hide
|
C28H34N2OS
|
1
|
| 1 |
Ki = 6.37 nM
|
|
|
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CP0522363
|
1-benzyl-N-cycloheptyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C24H26N2O2
|
1
|
| 1 |
Ki = 6.4 nM
|
|
|
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CP0386988
|
methyl 2-(adamantane-1-carbonylamino)-5-phenylthiophene-3-carboxylate
Show/Hide
|
C23H25NO3S
|
1
|
| 1 |
Ki = 6.48 nM
|
|
|
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CP0404951
|
4-oxo-7-phenylsulfanyl-1-(4-phenylsulfanylbutyl)-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C36H40N2O2S2
|
1
|
| 1 |
Ki = 6.5 nM
|
|
|
|
CP0409765
|
US8895592, 23
Show/Hide
|
C23H32F3N3O2S
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
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CP0569467
|
N-cyclopropyl-11-(3-ethoxy-5-pentylphenoxy)undecanamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0482502
|
(5Z,8Z,11Z,13S,14Z)-N-cyclobutyl-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C25H41NO
|
1
|
| 1 |
Ki = 6.8 nM
|
|
|
|
CP0550757
|
11-(3-methoxy-5-pentylphenoxy)-N-prop-2-enylundecanamide
Show/Hide
|
C26H43NO3
|
1
|
| 1 |
Ki = 6.8 nM
|
|
|
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CP0169639
|
N-(1-adamantyl)-2-ethyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),11-tetraene-11-carboxamide
Show/Hide
|
C24H28N2O3
|
1
|
| 1 |
Ki = 6.9 nM
|
|
|
|
CP0502798
|
(6aR,10aR)-3-[1-(1,2-cis-Hexen-1-yl)-cyclopent-1-yl]-6,6a,7,8,10,10a-hexahydro-1-hydroxy-6,6-dimethyl-9H-dibenzo[b,d]pyran-9-one
Show/Hide
|
C26H36O3
|
1
|
| 1 |
Ki = 7.02 nM
|
|
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|
CP0558670
|
4-bromobutyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]acetate
Show/Hide
|
C22H29BrO4
|
1
|
| 1 |
Ki = 7.1 nM
|
|
|
|
CP0429267
|
methyl 2-(adamantane-1-carbonylamino)-5-propylthiophene-3-carboxylate
Show/Hide
|
C20H27NO3S
|
1
|
| 1 |
Ki = 7.21 nM
|
|
|
|
CP0102146
|
6-Cyclohexyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H42N2O2
|
1
|
| 1 |
Ki = 7.3 nM
|
|
|
|
CP0257260
|
1-ethyl-7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C22H27FN2O2
|
1
|
| 1 |
Ki = 7.3 nM
|
|
|
|
CP0379905
|
8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]-N-prop-2-enyloctanamide
Show/Hide
|
C26H43NO3
|
1
|
| 1 |
Ki = 7.36 nM
|
|
|
|
CP0558190
|
US8895592, 3
Show/Hide
|
C24H27F3N2O3S
|
1
|
| 1 |
Ki = 7.4 nM
|
|
|
|
CP0381716
|
US8846730, 33
Show/Hide
|
C23H30F3N3O4S
|
1
|
| 1 |
Ki = 7.4 nM
|
|
|
|
CP0546228
|
US8846730, 3
Show/Hide
|
C25H32F3N3O3S
|
1
|
| 1 |
Ki = 7.4 nM
|
|
|
|
CP0499113
|
4-hydroxy-N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H30N4O4
|
1
|
| 1 |
Ki = 7.44 nM
|
|
|
|
CP0429004
|
(7-methoxy-9-pentylcarbazol-3-yl)-piperidin-1-ylmethanone
Show/Hide
|
C24H30N2O2
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0400951
|
N-(1-adamantyl)-2,5-dimethyl-1-phenylpyrrole-3-carboxamide
Show/Hide
|
C23H28N2O
|
1
|
| 1 |
Ki = 7.59 nM
|
|
|
|
CP0536124
|
4-imidazol-1-ylbutyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C27H36N2O4
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0498834
|
1-benzyl-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
Ki = 7.8 nM
|
|
|
|
CP0395172
|
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
|
C20H23FN2O2
|
1
|
| 1 |
Ki = 7.8 nM
|
|
|
|
CP0425338
|
2-[(6aR,9S,10aR)-3-(1-adamantyl)-1-hydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-9-yl]acetaldehyde
Show/Hide
|
C27H36O3
|
1
|
| 1 |
Ki = 7.8 nM
|
|
|
|
CP0498354
|
N-cyclohexyl-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C21H28N4O3
|
1
|
| 1 |
Ki = 7.9 nM
|
|
|
|
CP0452471
|
1-[2-(dimethylamino)ethyl]-7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C24H32FN3O2
|
1
|
| 1 |
Ki = 7.9 nM
|
|
|
|
CP0458672
|
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxo-5-[(E)-2-phenylethenyl]pyridine-3-carboxamide
Show/Hide
|
C28H29FN2O2
|
1
|
| 1 |
Ki = 7.9 nM
|
|
|
|
CP0103197
|
N-(1-adamantyl)-6-imidazol-1-yl-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C28H34N4O2
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0458673
|
1-benzyl-N-cycloheptyl-2-oxopyridine-3-carboxamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0425255
|
methyl 2-(adamantane-1-carbonylamino)-5-pentyl-4-phenylthiophene-3-carboxylate
Show/Hide
|
C28H35NO3S
|
1
|
| 1 |
Ki = 8.03 nM
|
|
|
|
CP0429839
|
US8846730, 45
Show/Hide
|
C27H36F3N3O3S
|
1
|
| 1 |
Ki = 8.2 nM
|
|
|
|
CP0225272
|
6-Cyclohex-1-enyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H40N2O2
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
|
CP0395024
|
US8895592, 27
Show/Hide
|
C22H21F6N3O3S
|
1
|
| 1 |
Ki = 8.4 nM
|
|
|
|
CP0517874
|
(6aS,10aS)-6,6,9-trimethyl-3-[(E)-C-methyl-N-(2-pyrrolidin-1-ylethoxy)carbonimidoyl]-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C24H34N2O3
|
1
|
| 1 |
Ki = 8.4 nM
|
|
|
|
CP0425469
|
N-(1-adamantyl)-6-(furan-2-yl)-8-methoxy-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C30H36N2O4
|
1
|
| 1 |
Ki = 8.5 nM
|
|
|
|
CP0545676
|
US8859596, 162
Show/Hide
|
C21H31ClN4O2S
|
1
|
| 1 |
Ki = 8.5 nM
|
|
|
|
CP0429553
|
(5Z,8Z,11Z,13S,14Z)-20-azido-N-cyclopropyl-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C24H38N4O
|
1
|
| 1 |
Ki = 8.5 nM
|
|
|
|
CP0281047
|
N-(1-adamantyl)-6-ethynyl-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C27H32N2O2
|
1
|
| 1 |
Ki = 8.8 nM
|
|
|
|
CP0454190
|
1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H24FN3O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0410760
|
N-cyclohexyl-1-(2-morpholin-4-ylethyl)-2-oxoquinoline-3-carboxamide
Show/Hide
|
C22H29N3O3
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0472529
|
(6aR,9S,10aR)-3-(1-adamantyl)-1-hydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-9-carbaldehyde
Show/Hide
|
C26H34O3
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0440503
|
US8895592, 4
Show/Hide
|
C22H29ClN2O3S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0316715
|
(6aS,10aS)-3-(1,1-Dimethyl-heptyl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C25H38O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0436999
|
N-(1-adamantyl)-5,8-dimethoxy-4-oxo-1-prop-2-enylquinoline-3-carboxamide
Show/Hide
|
C25H30N2O4
|
1
|
| 1 |
Ki = 9.2 nM
|
|
|
|
CP0411384
|
US8895592, 9
Show/Hide
|
C25H34F3N3O2S
|
1
|
| 1 |
Ki = 9.2 nM
|
|
|
|
CP0425253
|
methyl 2-(adamantane-1-carbonylamino)-4,5-dimethylthiophene-3-carboxylate
Show/Hide
|
C19H25NO3S
|
1
|
| 1 |
Ki = 9.24 nM
|
|
|
|
CP0460327
|
N-(1-adamantyl)-6-bromo-4-oxo-1-pent-4-enylquinoline-3-carboxamide
Show/Hide
|
C25H29BrN2O2
|
1
|
| 1 |
Ki = 9.4 nM
|
|
|
|
CP0411670
|
(6aR,9R,10aR)-3-[3-(azidomethyl)-1-adamantyl]-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-1,9-diol
Show/Hide
|
C26H35N3O3
|
1
|
| 1 |
Ki = 9.6 nM
|
|
|
|
CP0405065
|
(6aS,10aS)-3-[(E)-N-(4-fluorobutoxy)-C-methylcarbonimidoyl]-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C22H30FNO3
|
1
|
| 1 |
Ki = 9.7 nM
|
|
|
|
CP0415721
|
US8895592, 15
Show/Hide
|
C21H27ClN2O2S
|
1
|
| 1 |
Ki = 9.9 nM
|
|
|
|
CP0563975
|
US8859596, 153
Show/Hide
|
C23H31F3N4O3S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0434997
|
N-(1-adamantyl)-2-[5-(furan-2-yl)-1-prop-2-enylindol-3-yl]-2-oxoacetamide
Show/Hide
|
C27H28N2O3
|
1
|
| 1 |
Ki = 10.3 nM
|
|
|
|
CP0527862
|
N-(cyclopropylmethyl)-11-(3-methoxy-5-pentylphenoxy)undecanamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 10.3 nM
|
|
|
|
CP0511781
|
(5Z,8Z,11Z,13S,14Z)-N-(2-chloroethyl)-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C23H38ClNO
|
1
|
| 1 |
Ki = 10.4 nM
|
|
|
|
CP0531749
|
4-butyl-7-hydroxy-N-(3-hydroxy-1-adamantyl)-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H30N4O4
|
1
|
| 1 |
Ki = 10.6 nM
|
|
|
|
CP0457644
|
(R)-7-Fluoro-4-oxo-1-pentyl-N-(1-phenylethyl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C23H25FN2O2
|
1
|
| 1 |
Ki = 10.7 nM
|
|
|
|
CP0522361
|
1-benzyl-N-cyclohexyl-7-methoxy-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H25N3O3
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0313817
|
6-(4-Chloro-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H35ClN2O2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0389373
|
US8846730, 56
Show/Hide
|
C24H27F3N4O3S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0464057
|
US8859596, 34
Show/Hide
|
C22H31F3N4O2S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0548881
|
N-cyclohexyl-2-oxo-2-(1-pentyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C27H32N2O2
|
1
|
| 1 |
Ki = 11.2 nM
|
|
|
|
CP0543794
|
2-[(6aR,9R,10aR)-3-(1-adamantyl)-1-hydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-9-yl]acetaldehyde
Show/Hide
|
C27H36O3
|
1
|
| 1 |
Ki = 11.2 nM
|
|
|
|
CP0557205
|
1-butyl-4-hydroxy-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C20H27N3O3
|
1
|
| 1 |
Ki = 11.2 nM
|
|
|
|
CP0429551
|
(5Z,8Z,11Z,13S,14Z)-13-methyl-N-prop-2-ynylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C24H37NO
|
1
|
| 1 |
Ki = 11.2 nM
|
|
|
|
CP0438382
|
AM4054
Show/Hide
|
C26H36O3
|
1
|
| 1 |
Ki = 11.3 nM
|
|
|
|
CP0379401
|
3-butyl-N-cycloheptyl-2-methoxy-5-(4-methoxyphenyl)benzamide
Show/Hide
|
C26H35NO3
|
1
|
| 1 |
Ki = 11.48 nM
|
|
|
|
CP0139727
|
N-(1-adamantyl)-4-oxo-1-pentyl-6-(trifluoromethyl)quinoline-3-carboxamide
Show/Hide
|
C26H31F3N2O2
|
1
|
| 1 |
Ki = 11.6 nM
|
|
|
|
CP0535273
|
N-(1-adamantyl)-1-pentyl-5-phenylindole-3-carboxamide
Show/Hide
|
C30H36N2O
|
1
|
| 1 |
Ki = 11.6 nM
|
|
|
|
CP0429451
|
N-(1-adamantyl)-2-(5-phenyl-1-propylindol-3-yl)acetamide
Show/Hide
|
C29H34N2O
|
1
|
| 1 |
Ki = 11.8 nM
|
|
|
|
CP0401969
|
(6aR,10aR)-3-(1-Hexyl-cyclobut-1-yl)-6,6a,7,8,10,10a-hexahydro-1-hydroxy-6,6-dimethyl-9H-dibenzo[b,d]pyran-9-one
Show/Hide
|
C25H36O3
|
1
|
| 1 |
Ki = 11.9 nM
|
|
|
|
CP0376647
|
N-(1-adamantyl)-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C27H30Cl2N4O
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0401296
|
N-cyclopentyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H24Cl2N4O
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0453835
|
N-cyclopentyl-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C20H20Cl2N4O
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0037364
|
(-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C21H30O2
|
2
|
| 1 |
Ki = 12 nM
|
|
|
| 2 |
Ki = 25 nM
|
|
|
|
CP0389343
|
US8846730, 70
Show/Hide
|
C26H34F3N3O4S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0390261
|
US8859596, 167
Show/Hide
|
C21H27F3N4O2S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0468404
|
US8859596, 194
Show/Hide
|
C23H28F6N4O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0382775
|
N-(3-pentyl-1,3-benzothiazol-2-ylidene)adamantane-1-carboxamide
Show/Hide
|
C23H30N2OS
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0436076
|
N-(1-adamantyl)-2-oxo-2-(1-pentyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C31H36N2O2
|
1
|
| 1 |
Ki = 12.7 nM
|
|
|
|
CP0248960
|
(5Z,7R,8Z,11Z,14Z)-N-[(2R)-1-hydroxypropan-2-yl]-7-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C24H41NO2
|
1
|
| 1 |
Ki = 12.8 nM
|
|
|
|
CP0432931
|
N-cyclopropyl-11-(3-hydroxy-4-pentylphenoxy)undecanamide
Show/Hide
|
C25H41NO3
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0435108
|
US8846730, 21
Show/Hide
|
C26H28F3N3O3S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0427591
|
11-(3-hydroxy-5-pentylphenoxy)undecanoic acid cyclopropylamide
Show/Hide
|
C25H41NO3
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0414615
|
(6aR,9R,10aR)-3-(3-isothiocyanato-1-adamantyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-1,9-diol
Show/Hide
|
C26H33NO3S
|
1
|
| 1 |
Ki = 13.1 nM
|
|
|
|
CP0498311
|
4-oxo-1-pentyl-7-phenylsulfanyl-N-piperidin-1-ylquinoline-3-carboxamide
Show/Hide
|
C26H31N3O2S
|
1
|
| 1 |
Ki = 13.3 nM
|
|
|
|
CP0381990
|
ethyl (E)-3-[5-(cycloheptylcarbamoyl)-1-[(4-fluorophenyl)methyl]-6-oxopyridin-3-yl]prop-2-enoate
Show/Hide
|
C25H29FN2O4
|
1
|
| 1 |
Ki = 13.7 nM
|
|
|
|
CP0449572
|
(6aR,10aR)-3-(1-adamantyl)-9-(hydroxymethyl)-6,6-dimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C26H34O3
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0470366
|
US8846730, 35
Show/Hide
|
C29H34F3N3O3S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0141726
|
N-(1-adamantyl)-6-bromo-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C25H31BrN2O2
|
1
|
| 1 |
Ki = 14.3 nM
|
|
|
|
CP0516608
|
N-(1-adamantyl)-7-hydroxy-4-(4-hydroxybutyl)-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H30N4O4
|
1
|
| 1 |
Ki = 14.3 nM
|
|
|
|
CP0472387
|
N-tert-butyl-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C19H20Cl2N4O
|
1
|
| 1 |
Ki = 14.6 nM
|
|
|
|
CP0498313
|
4-oxo-1-pentyl-7-phenylsulfanyl-N-propan-2-ylquinoline-3-carboxamide
Show/Hide
|
C24H28N2O2S
|
1
|
| 1 |
Ki = 14.8 nM
|
|
|
|
CP0477443
|
N-(1-adamantyl)-6-(furan-2-yl)-4-hydroxy-2-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C29H34N2O4
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0486536
|
US8895592, 30
Show/Hide
|
C23H28F3N3O2S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0546218
|
US8895592, 35
Show/Hide
|
C22H24F3N3O3S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0462701
|
US8846730, 2
Show/Hide
|
C24H30F3N3O3S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0426608
|
US8859596, 177
Show/Hide
|
C22H29F3N4O3S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0514857
|
(6aR,10aR)-3-[1-(1,2-cis-Hexen-1-yl)-cyclobut-1-yl]-6,6a,7,8,10,10a-hexahydro-1-hydroxy-6,6-dimethyl-9H-dibenzo[b,d]pyran-9-one
Show/Hide
|
C25H34O3
|
1
|
| 1 |
Ki = 15.1 nM
|
|
|
|
CP0393332
|
7-fluoro-1-(4-hydroxybutyl)-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C24H31FN2O3
|
1
|
| 1 |
Ki = 15.2 nM
|
|
|
|
CP0500720
|
1-ethenyl-7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C22H25FN2O2
|
1
|
| 1 |
Ki = 15.2 nM
|
|
|
|
CP0392393
|
N-cyclohexyl-1-(2,4-dichlorophenyl)-4-ethyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H24Cl2N4O
|
1
|
| 1 |
Ki = 15.8 nM
|
|
|
|
CP0102143
|
6-(2,4-Difluoro-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H34F2N2O2
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0513447
|
1-benzyl-N-cyclohexyl-2-oxoquinoline-3-carboxamide
Show/Hide
|
C23H24N2O2
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0480041
|
1-methyl-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C27H30N2O2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0397839
|
US8895592, 18
Show/Hide
|
C23H29F3N2O4S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0484505
|
US8846730, 48
Show/Hide
|
C26H34F3N3O5S2
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0443116
|
US8859596, 163
Show/Hide
|
C22H29F3N4O2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0464066
|
US8859596, 185
Show/Hide
|
C20H26F3N5O2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0546709
|
US8859596, 145
Show/Hide
|
C22H29F3N4O2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0546808
|
US8859596, 159
Show/Hide
|
C23H33F3N4O2
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0436216
|
N-(1-adamantyl)-6-(3-chloro-4-fluorophenoxy)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C31H34ClFN2O3
|
1
|
| 1 |
Ki = 16.1 nM
|
|
|
|
CP0400886
|
11-(3-hydroxy-5-pentylphenoxy)-N-prop-2-enylundecanamide
Show/Hide
|
C25H41NO3
|
1
|
| 1 |
Ki = 16.4 nM
|
|
|
|
CP0455976
|
ethyl 2-(naphthalene-1-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C22H21NO3S
|
1
|
| 1 |
Ki = 16.8 nM
|
|
|
|
CP0195802
|
N-(1-adamantyl)-6-ethyl-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C27H36N2O2
|
1
|
| 1 |
Ki = 16.9 nM
|
|
|
|
CP0429661
|
US8895592, 31
Show/Hide
|
C23H28F3N3O2S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0457643
|
(R)-4-Oxo-1-pentyl-N-(1-phenylethyl)-7-(pyrrolidin-1-yl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C27H33N3O2
|
1
|
| 1 |
Ki = 17.1 nM
|
|
|
|
CP0525854
|
4-[6-(1-adamantylcarbamoyl)-7-hydroxy-2-methyl-5-oxopyrazolo[4,3-b]pyridin-4-yl]butyl acetate
Show/Hide
|
C24H32N4O5
|
1
|
| 1 |
Ki = 17.3 nM
|
|
|
|
CP0536700
|
N-(1-adamantyl)-2-(1-but-3-enyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C30H34N2O
|
1
|
| 1 |
Ki = 17.8 nM
|
|
|
|
CP0390099
|
US8859596, 196
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0470289
|
US8859596, 180
Show/Hide
|
C22H27F3N4O3S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0395391
|
5-(2-chloropyrrol-1-yl)-N-cyclohexyl-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H21Cl3N4O
|
1
|
| 1 |
Ki = 18.3 nM
|
|
|
|
CP0423778
|
N-(1-adamantyl)-4-butyl-7-hydroxy-2-(2-hydroxyethyl)-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C23H32N4O4
|
1
|
| 1 |
Ki = 18.4 nM
|
|
|
|
CP0516606
|
4-(4-fluorobutyl)-7-hydroxy-N-(3-hydroxy-1-adamantyl)-1-methyl-5-oxo-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H31FN4O4
|
1
|
| 1 |
Ki = 18.9 nM
|
|
|
|
CP0479037
|
(6aR,9R,10aR)-6,6-Dimethyl-3-(2-oxa-tricyclo[3.3.1.1*3,7*]dec-1-yl)-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
|
C24H32O4
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0440706
|
N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(2,5-dichloropyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H20Cl4N4O
|
1
|
| 1 |
Ki = 19.1 nM
|
|
|
|
CP0453386
|
4-oxo-1-pentyl-N-phenylmethoxy-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C28H28N2O3S
|
1
|
| 1 |
Ki = 19.3 nM
|
|
|
|
CP0572166
|
4-butyl-7-hydroxy-N-(3-hydroxy-1-adamantyl)-1-methyl-5-oxo-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H32N4O4
|
1
|
| 1 |
Ki = 19.3 nM
|
|
|
|
CP0499727
|
1-butyl-N-(4-methylcyclohexyl)-2-oxoquinoline-3-carboxamide
Show/Hide
|
C21H28N2O2
|
1
|
| 1 |
Ki = 19.8 nM
|
|
|
|
CP0453373
|
N-(1-hydroxybutan-2-yl)-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C25H30N2O3S
|
1
|
| 1 |
Ki = 19.9 nM
|
|
|
|
CP0396949
|
N-(1-adamantyl)-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C25H26Cl2N4O
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0430148
|
N-cycloheptyl-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H24Cl2N4O
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0432138
|
N-cyclohexyl-1-[(4-fluorophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
|
C19H21FN2O2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0428968
|
[9-(oxan-4-ylmethyl)carbazol-3-yl]-piperidin-1-ylmethanone
Show/Hide
|
C24H28N2O2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0395560
|
N-[5-tert-butyl-3-[[(2R)-oxolan-2-yl]methyl]-1,3-thiazol-2-ylidene]-2-(pyridin-2-ylmethoxy)-5-(trifluoromethyl)benzamide
Show/Hide
|
C26H28F3N3O3S
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0395711
|
2-ethyl-5-methyl-N-naphthalen-1-yl-1-phenylpyrrole-3-carboxamide
Show/Hide
|
C24H22N2O
|
1
|
| 1 |
Ki = 20.02 nM
|
|
|
|
CP0376686
|
N-tert-butyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H24Cl2N4O
|
1
|
| 1 |
Ki = 20.2 nM
|
|
|
|
CP0434998
|
N-(1-adamantyl)-2-(1-butyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C30H36N2O
|
1
|
| 1 |
Ki = 20.5 nM
|
|
|
|
CP0195798
|
6-Iodo-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C25H31IN2O2
|
1
|
| 1 |
Ki = 20.6 nM
|
|
|
|
CP0479032
|
methyl 2-(1-adamantylcarbamoylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C21H28N2O3S
|
1
|
| 1 |
Ki = 20.97 nM
|
|
|
|
CP0491022
|
US8846730, 66
Show/Hide
|
C25H32F3N3O4S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0461549
|
US8859596, 171
Show/Hide
|
C20H27F3N4O2S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0563296
|
US8859596, 182
Show/Hide
|
C25H27F4N5O2S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0410866
|
11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]-N-[(2R)-1-hydroxypropan-2-yl]undecanamide
Show/Hide
|
C29H51NO4
|
1
|
| 1 |
Ki = 21.2 nM
|
|
|
|
CP0102145
|
6-(4-Methoxy-3,5-dimethyl-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C34H42N2O3
|
1
|
| 1 |
Ki = 21.5 nM
|
|
|
|
CP0420378
|
11-(3-butoxy-5-pentylphenoxy)-N-cyclopropylundecanamide
Show/Hide
|
C29H49NO3
|
1
|
| 1 |
Ki = 21.5 nM
|
|
|
|
CP0454192
|
1-benzyl-N-cycloheptyl-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0388921
|
3-butyl-2-methoxy-5-(4-methoxyphenyl)-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C26H35NO3
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0429838
|
US8846730, 78
Show/Hide
|
C24H32F3N3O3S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0405727
|
(5Z,8Z,11Z,13S,14Z)-N-cyclopropyl-20-isothiocyanato-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C25H38N2OS
|
1
|
| 1 |
Ki = 22.1 nM
|
|
|
|
CP0416199
|
N-(1-adamantyl)-5-(4-hydroxyphenyl)-1-prop-2-enylindole-3-carboxamide
Show/Hide
|
C28H30N2O2
|
1
|
| 1 |
Ki = 22.2 nM
|
|
|
|
CP0428319
|
N-(1-adamantyl)-6-bromo-8-methoxy-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C26H33BrN2O3
|
1
|
| 1 |
Ki = 22.9 nM
|
|
|
|
CP0527864
|
11-(3-methoxy-5-pentylphenoxy)-N-(2,2,2-trifluoroethyl)undecanamide
Show/Hide
|
C25H40F3NO3
|
1
|
| 1 |
Ki = 22.9 nM
|
|
|
|
CP0482759
|
methyl 2-(adamantane-1-carbonylamino)-5-methylthiophene-3-carboxylate
Show/Hide
|
C18H23NO3S
|
1
|
| 1 |
Ki = 23.09 nM
|
|
|
|
CP0423081
|
N-(1-adamantyl)-6-bromo-1-but-3-enyl-4-oxoquinoline-3-carboxamide
Show/Hide
|
C24H27BrN2O2
|
1
|
| 1 |
Ki = 23.8 nM
|
|
|
|
CP0543959
|
US8846730, 49
Show/Hide
|
C26H34F3N3O4S
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0464058
|
US8859596, 142
Show/Hide
|
C25H35F3N4O3
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0388546
|
(R)-7-Ethoxy-4-oxo-1-pentyl-N-(1-phenylethyl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C25H30N2O3
|
1
|
| 1 |
Ki = 24.2 nM
|
|
|
|
CP0104537
|
(5Z,7R,8Z,11Z,14Z)-N-(2-hydroxyethyl)-7-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C23H39NO2
|
1
|
| 1 |
Ki = 24.7 nM
|
|
|
|
CP0448313
|
(6aR,9R,10aR)-3-(3-azido-1-adamantyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-1,9-diol
Show/Hide
|
C25H33N3O3
|
1
|
| 1 |
Ki = 24.8 nM
|
|
|
|
CP0432137
|
N-cycloheptyl-2-[(4-fluorophenyl)methoxy]pyridine-3-carboxamide
Show/Hide
|
C20H23FN2O2
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0524245
|
US8846730, 63
Show/Hide
|
C29H38F3N3O5S
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0532691
|
US8846730, 34
Show/Hide
|
C27H37F3N4O3S
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0502917
|
N-(1-adamantyl)-2-oxo-2-(5-phenyl-1-prop-2-enylindol-3-yl)acetamide
Show/Hide
|
C29H30N2O2
|
1
|
| 1 |
Ki = 25.4 nM
|
|
|
|
CP0446041
|
N-(4-methylcyclohexyl)-2-oxo-1-propylquinoline-3-carboxamide
Show/Hide
|
C20H26N2O2
|
1
|
| 1 |
Ki = 25.4 nM
|
|
|
|
CP0436994
|
N-(1-adamantyl)-7-chloro-8-methyl-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C26H33ClN2O2
|
1
|
| 1 |
Ki = 25.5 nM
|
|
|
|
CP0472013
|
US8846730, 37
Show/Hide
|
C24H26F3N3O4S
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0135103
|
3-[[4,4-dimethyl-7-(2-methyloctan-2-yl)-1H-chromeno[4,3-c]pyrazol-9-yl]oxy]propan-1-ol
Show/Hide
|
C24H36N2O3
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0469873
|
N-cyclopropyl-11-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
|
C30H51NO3
|
1
|
| 1 |
Ki = 26.1 nM
|
|
|
|
CP0388957
|
N-(2,2-dimethylpropyl)-9-pentylpyrido[3,4-b]indole-3-carboxamide
Show/Hide
|
C22H29N3O
|
1
|
| 1 |
Ki = 26.5 nM
|
|
|
|
CP0470042
|
4-(2-{2-methyl-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl}ethyl)morpholine
Show/Hide
|
C23H32N2O2
|
1
|
| 1 |
Ki = 26.92 nM
|
|
|
|
CP0531130
|
US8895592, 1
Show/Hide
|
C24H34BrN3O2S
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0555631
|
US8859596, 155
Show/Hide
|
C25H35F3N4O2
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0516605
|
N-(1-adamantyl)-4-butyl-7-hydroxy-1-(2-hydroxyethyl)-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C23H32N4O4
|
1
|
| 1 |
Ki = 27.1 nM
|
|
|
|
CP0555106
|
8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]-N-(2,2,2-trifluoroethyl)octanamide
Show/Hide
|
C25H40F3NO3
|
1
|
| 1 |
Ki = 27.9 nM
|
|
|
|
CP0455045
|
N-cycloheptyl-1-(2-morpholin-4-ylethyl)-4-oxoquinoline-3-carboxamide
Show/Hide
|
C23H31N3O3
|
1
|
| 1 |
Ki = 28 nM
|
|
|
|
CP0462638
|
US8859596, 152
Show/Hide
|
C22H31F3N4O2S
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0471601
|
N-(1-adamantyl)-6-bromo-4-hydroxy-2-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C25H31BrN2O3
|
1
|
| 1 |
Ki = 29.4 nM
|
|
|
|
CP0440707
|
1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-ethyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C23H18Cl4N4O
|
1
|
| 1 |
Ki = 29.6 nM
|
|
|
|
CP0858250
|
10alpha-Hydroxy-Delta8-tetrahydrocannabinol
Show/Hide
|
C21H30O3
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0385228
|
US8895592, 24
Show/Hide
|
C23H28F3N3O2S
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0407676
|
US8846730, 6
Show/Hide
|
C26H34F3N3O3S
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0498940
|
1-benzyl-N-cyclohexyl-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0044659
|
(6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-indol-3-yl)(4-methoxyphenyl)methanone
Show/Hide
|
C23H25IN2O3
|
2
|
| 1 |
Ki = 31.2 nM
|
|
|
| 2 |
Ki = 36 nM
|
|
|
|
CP0548828
|
8-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]-N-prop-2-enyloctanamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 31.2 nM
|
|
|
|
CP0453384
|
7-fluoro-1-[(3-methylphenyl)methyl]-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C28H31FN2O2
|
1
|
| 1 |
Ki = 31.5 nM
|
|
|
|
CP0413979
|
US8895592, 7
Show/Hide
|
C25H34F3N3O2S
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0503959
|
US8859596, 183
Show/Hide
|
C23H27F3N6OS
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0473621
|
(6aR,10aR)-3-(2-Hexyl-1,3-dithiolan-2-yl)-6,6a,7,8,10,10ahexahydro-1-hydroxy-6,6-dimethyl-9H-dibenzo[b,d]pyran-9-one
Show/Hide
|
C24H34O3S2
|
1
|
| 1 |
Ki = 32.6 nM
|
|
|
|
CP0462688
|
US8846730, 7
Show/Hide
|
C27H36F3N3O3S
|
1
|
| 1 |
Ki = 33 nM
|
|
|
|
CP0527861
|
N-(2-hydroxyethyl)-11-(3-methoxy-5-pentylphenoxy)undecanamide
Show/Hide
|
C25H43NO4
|
1
|
| 1 |
Ki = 33.2 nM
|
|
|
|
CP0565979
|
(6aR,9R,10aR)-3-(1-adamantyl)-9-(2-hydroxyethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-1-ol
Show/Hide
|
C27H38O3
|
1
|
| 1 |
Ki = 33.3 nM
|
|
|
|
CP0411899
|
US8895592, 33
Show/Hide
|
C24H27F3N4O2S
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0380935
|
US8846730, 74
Show/Hide
|
C28H34F3N3O3S
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0456794
|
US8846730, 58
Show/Hide
|
C24H32F3N3O4S
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0429050
|
methyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]-2-methylpropanoate
Show/Hide
|
C21H28O4
|
1
|
| 1 |
Ki = 34.5 nM
|
|
|
|
CP0462717
|
US8895592, 20
Show/Hide
|
C23H26F3N3O3S
|
1
|
| 1 |
Ki = 35 nM
|
|
|
|
CP0425250
|
methyl 2-(adamantane-1-carbonylamino)-4-phenylthiophene-3-carboxylate
Show/Hide
|
C23H25NO3S
|
1
|
| 1 |
Ki = 35 nM
|
|
|
|
CP0429007
|
(9-pentylpyrido[3,4-b]indol-3-yl)-piperidin-1-ylmethanone
Show/Hide
|
C22H27N3O
|
1
|
| 1 |
Ki = 35.3 nM
|
|
|
|
CP0420195
|
(4-methylpiperazin-1-yl)-(9-pentylcarbazol-3-yl)methanone
Show/Hide
|
C23H29N3O
|
1
|
| 1 |
Ki = 35.4 nM
|
|
|
|
CP0499114
|
1-(3-hydroxypropyl)-N-(4-methylcyclohexyl)-2-oxoquinoline-3-carboxamide
Show/Hide
|
C20H26N2O3
|
1
|
| 1 |
Ki = 36 nM
|
|
|
|
CP0472511
|
US8846730, 55
Show/Hide
|
C26H35F3N4O2S
|
1
|
| 1 |
Ki = 36 nM
|
|
|
|
CP0415560
|
US8895592, 12
Show/Hide
|
C24H32F3N3O2S
|
1
|
| 1 |
Ki = 37 nM
|
|
|
|
CP0443573
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-[3-(trifluoromethyl)phenyl]methanone
Show/Hide
|
C23H23F3O4
|
1
|
| 1 |
Ki = 37.3 nM
|
|
|
|
CP0547736
|
2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl]benzimidazole-5-carboxamide
Show/Hide
|
C36H41N5O2
|
1
|
| 1 |
Ki = 38.5 nM
|
|
|
|
CP0427162
|
12-(3-hydroxy-5-pentyl-phenoxy)-dodecanoic acid(2-hydroxy-ethyl)-amide
Show/Hide
|
C25H43NO4
|
1
|
| 1 |
Ki = 39 nM
|
|
|
|
CP0432935
|
8-(3-hydroxy-5-pentyl-phenoxy)-octanoic acid cyclopropylamide
Show/Hide
|
C22H35NO3
|
1
|
| 1 |
Ki = 39 nM
|
|
|
|
CP0444413
|
12-(2-hexyl-5-hydroxy-phenoxy)-dodecanoic acidcyclopropylamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 39 nM
|
|
|
|
CP0546310
|
US8895592, 5
Show/Hide
|
C25H34F3N3O2S
|
1
|
| 1 |
Ki = 39 nM
|
|
|
|
CP0390258
|
US8859596, 158
Show/Hide
|
C21H29F3N4O3S
|
1
|
| 1 |
Ki = 39 nM
|
|
|
|
CP0434521
|
2-(2-hydroxyethyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
|
C23H34N2O3
|
1
|
| 1 |
Ki = 39.6 nM
|
|
|
|
CP0454197
|
1-benzyl-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
Ki = 39.8 nM
|
|
|
|
CP0552959
|
2-[2,4,4-trimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-yl]oxyethanol
Show/Hide
|
C24H36N2O3
|
1
|
| 1 |
Ki = 39.8 nM
|
|
|
|
CP0448192
|
(6aR,9R,10aR)-3-(1-adamantyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-1,9-diol
Show/Hide
|
C25H34O3
|
1
|
| 1 |
Ki = 40.5 nM
|
|
|
|
CP0054395
|
6-(4-Cyano-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C32H35N3O2
|
1
|
| 1 |
Ki = 41.9 nM
|
|
|
|
CP0526831
|
N-(2-hydroxyethyl)-8-(3-methoxy-5-pentylphenoxy)octanamide
Show/Hide
|
C22H37NO4
|
1
|
| 1 |
Ki = 41.9 nM
|
|
|
|
CP0472379
|
US8846730, 59
Show/Hide
|
C26H34N4O3S
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0390267
|
US8859596, 202
Show/Hide
|
C25H30F3N5OS
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0462788
|
US8895592, 14
Show/Hide
|
C23H30F3N3O2S
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0571106
|
US8859596, 205
Show/Hide
|
C30H37F3N6O3S
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0102144
|
6-(5-Chloro-thiophen-2-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C29H33ClN2O2S
|
1
|
| 1 |
Ki = 44.8 nM
|
|
|
|
CP0548850
|
US8846730, 41
Show/Hide
|
C23H25F3N4O3S
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0425336
|
AM4089
Show/Hide
|
C26H30O3
|
1
|
| 1 |
Ki = 46.7 nM
|
|
|
|
CP0425026
|
US8846730, 8
Show/Hide
|
C25H32F3N3O3S
|
1
|
| 1 |
Ki = 47 nM
|
|
|
|
CP0450108
|
US8859596, 201
Show/Hide
|
C19H25F3N6O2S
|
1
|
| 1 |
Ki = 47 nM
|
|
|
|
CP0516621
|
N-(cyclopropylmethyl)-11-(4-hexyl-3-methoxyphenoxy)undecanamide
Show/Hide
|
C28H47NO3
|
1
|
| 1 |
Ki = 48.8 nM
|
|
|
|
CP0454409
|
[(6aR,10aR)-3-(1-adamantyl)-1-hydroxy-6,6-dimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-9-yl]methyl 2,2-dimethylpropanoate
Show/Hide
|
C31H42O4
|
1
|
| 1 |
Ki = 49.2 nM
|
|
|
|
CP0469072
|
(9-pentylcarbazol-3-yl)-piperidin-1-ylmethanethione
Show/Hide
|
C23H28N2S
|
1
|
| 1 |
Ki = 49.6 nM
|
|
|
|
CP0051324
|
6-Bromo-4-oxo-1-prop-2-ynyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C23H23BrN2O2
|
1
|
| 1 |
Ki = 49.8 nM
|
|
|
|
CP0416198
|
N-(1-adamantyl)-2-(5-phenyl-1-prop-2-enylindol-3-yl)acetamide
Show/Hide
|
C29H32N2O
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0514780
|
N-(1-adamantyl)-2-[5-(furan-2-yl)-1-prop-2-enylindol-3-yl]acetamide
Show/Hide
|
C27H30N2O2
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0415354
|
8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]-N-[(2R)-1-hydroxypropan-2-yl]octanamide
Show/Hide
|
C26H45NO4
|
1
|
| 1 |
Ki = 50.2 nM
|
|
|
|
CP0104538
|
(5Z,8Z,11Z,13S,14Z)-N-(2-hydroxyethyl)-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C23H39NO2
|
1
|
| 1 |
Ki = 50.5 nM
|
|
|
|
CP0394003
|
methyl 2-(adamantane-1-carbonylamino)-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
Show/Hide
|
C20H25NO3S2
|
1
|
| 1 |
Ki = 50.7 nM
|
|
|
|
CP0501629
|
6-(1-Isobutyl-1H-pyrazol-4-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C32H42N4O2
|
1
|
| 1 |
Ki = 51 nM
|
|
|
|
CP0403870
|
butyl 2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]acetate
Show/Hide
|
C22H30O4
|
1
|
| 1 |
Ki = 51.5 nM
|
|
|
|
CP0547347
|
(6aS,10aS)-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C21H30O2
|
1
|
| 1 |
Ki = 51.5 nM
|
|
|
|
CP0429010
|
N,N-diethyl-9-pentylcarbazole-3-carboxamide
Show/Hide
|
C22H28N2O
|
1
|
| 1 |
Ki = 51.8 nM
|
|
|
|
CP0435424
|
(5aR,11bR)-11-hydroxy-6,6-dimethyl-9-(2-methyloctan-2-yl)-4,5,5a,11b-tetrahydro-1H-oxepino[4,3-c]chromen-3-one
Show/Hide
|
C24H36O4
|
1
|
| 1 |
Ki = 52 nM
|
|
|
|
CP0410579
|
US8859596, 168
Show/Hide
|
C24H35ClN4O3
|
1
|
| 1 |
Ki = 52 nM
|
|
|
|
CP0472586
|
US8859596, 172
Show/Hide
|
C21H24F6N4O2S
|
1
|
| 1 |
Ki = 52 nM
|
|
|
|
CP0501840
|
1-(2,4-Dichlorophenyl)-N-(3,3-dimethylbutyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H24Cl2N4O
|
1
|
| 1 |
Ki = 52.4 nM
|
|
|
|
CP0386406
|
N-(1-adamantyl)-5,8-dimethoxy-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C27H36N2O4
|
1
|
| 1 |
Ki = 52.6 nM
|
|
|
|
CP0411868
|
6-(6-Methoxy-naphthalen-2-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C36H40N2O3
|
1
|
| 1 |
Ki = 52.6 nM
|
|
|
|
CP0395646
|
1-benzyl-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
Ki = 53 nM
|
|
|
|
CP0472489
|
US8895592, 17
Show/Hide
|
C22H24F3N3O2S
|
1
|
| 1 |
Ki = 53 nM
|
|
|
|
CP0415804
|
US8846730, 17
Show/Hide
|
C25H29F3N4O3S
|
1
|
| 1 |
Ki = 53 nM
|
|
|
|
CP0542580
|
1-cyclohexyl-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
|
C27H40N2O2
|
1
|
| 1 |
Ki = 53.7 nM
|
|
|
|
CP0495980
|
5-(2-chloropyrrol-1-yl)-1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H15Cl5N4O
|
1
|
| 1 |
Ki = 53.9 nM
|
|
|
|
CP0545675
|
US8859596, 146
Show/Hide
|
C24H33F3N4O2
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0051463
|
(E)-N-(Adamant-1-yl)-6-[2-(4-methoxyphenyl)vinyl]-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C34H40N2O3
|
1
|
| 1 |
Ki = 55.9 nM
|
|
|
|
CP0392395
|
1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dimethylpyrrol-1-yl)-4-ethylpyrazole-3-carboxamide
Show/Hide
|
C25H22Cl4N4O
|
1
|
| 1 |
Ki = 56.1 nM
|
|
|
|
CP0190974
|
6-(2-Ethyl-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C33H40N2O2
|
1
|
| 1 |
Ki = 56.6 nM
|
|
|
|
CP0395708
|
2-ethyl-5-methyl-N-naphthalen-2-yl-1-phenylpyrrole-3-carboxamide
Show/Hide
|
C24H22N2O
|
1
|
| 1 |
Ki = 57 nM
|
|
|
|
CP0564718
|
7-hydroxy-N-(3-hydroxy-1-adamantyl)-2-(2-hydroxyethyl)-5-oxo-4-pentylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C24H34N4O5
|
1
|
| 1 |
Ki = 57.1 nM
|
|
|
|
CP0496490
|
2-[2-(2,4,6-Trimethyl-phenoxy)-acetylamino]-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid (1,1-dioxo-tetrahydro-1lambda*6*-thiophen-3-yl)-amide
Show/Hide
|
C24H30N2O5S2
|
1
|
| 1 |
Ki = 58 nM
|
|
|
|
CP0446046
|
2,5-dimethyl-N-naphthalen-2-yl-1-phenylpyrrole-3-carboxamide
Show/Hide
|
C23H20N2O
|
1
|
| 1 |
Ki = 58.28 nM
|
|
|
|
CP0398771
|
1-Allyl-6-furan-2-yl-4-oxo-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C27H28N2O3
|
1
|
| 1 |
Ki = 59 nM
|
|
|
|
CP0401971
|
6-(6-Methoxy-pyridin-3-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H37N3O3
|
1
|
| 1 |
Ki = 59.3 nM
|
|
|
|
CP0542582
|
2-(hydroxymethyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
|
C22H32N2O3
|
1
|
| 1 |
Ki = 59.4 nM
|
|
|
|
CP0395709
|
ethyl 2-(naphthalene-1-carbonylamino)-5-phenylthiophene-3-carboxylate
Show/Hide
|
C24H19NO3S
|
1
|
| 1 |
Ki = 59.81 nM
|
|
|
|
CP0396891
|
N-(1-adamantyl)-4-oxo-8-pentoxy-1H-quinoline-3-carboxamide
Show/Hide
|
C25H32N2O3
|
1
|
| 1 |
Ki = 60 nM
|
|
|
|
CP0379382
|
N-cycloheptyl-5-(4-fluorophenyl)-2-methoxy-3-methylbenzamide
Show/Hide
|
C22H26FNO2
|
1
|
| 1 |
Ki = 60 nM
|
|
|
|
CP0388920
|
5-(4-fluorophenyl)-2-methoxy-3-methyl-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C22H26FNO2
|
1
|
| 1 |
Ki = 60 nM
|
|
|
|
CP0429005
|
N-[3-[3-(piperidine-1-carbonyl)carbazol-9-yl]propyl]methanesulfonamide
Show/Hide
|
C22H27N3O3S
|
1
|
| 1 |
Ki = 62 nM
|
|
|
|
CP0396421
|
US8895592, 22
Show/Hide
|
C22H25F3N4O2S
|
1
|
| 1 |
Ki = 62 nM
|
|
|
|
CP0408244
|
US8846730, 43
Show/Hide
|
C26H32F3N3O4S
|
1
|
| 1 |
Ki = 62 nM
|
|
|
|
CP0516622
|
N-(cyclopropylmethyl)-11-(2-hexyl-5-methoxyphenoxy)undecanamide
Show/Hide
|
C28H47NO3
|
1
|
| 1 |
Ki = 62.6 nM
|
|
|
|
CP0484631
|
N-cycloheptyl-5-(4-fluorophenyl)-1-(2-morpholin-4-ylethyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C25H32FN3O3
|
1
|
| 1 |
Ki = 63 nM
|
|
|
|
CP0472528
|
3-(1-adamantyl)-6,6,9-trimethylbenzo[c]chromen-1-ol
Show/Hide
|
C26H30O2
|
1
|
| 1 |
Ki = 63.5 nM
|
|
|
|
CP0429266
|
methyl 5-(adamantane-1-carbonylamino)-3-methyl-1,2-oxazole-4-carboxylate
Show/Hide
|
C17H22N2O4
|
1
|
| 1 |
Ki = 64.72 nM
|
|
|
|
CP0443537
|
5-bromo-N-cycloheptyl-1-(2-morpholin-4-ylethyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C19H28BrN3O3
|
1
|
| 1 |
Ki = 65 nM
|
|
|
|
CP0506906
|
US8859596, 166
Show/Hide
|
C23H32F3N5O2S
|
1
|
| 1 |
Ki = 65 nM
|
|
|
|
CP0406215
|
(E)-N-(Adamantan-1-yl)-4-oxo-1-pentyl-6-styryl-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C33H38N2O2
|
1
|
| 1 |
Ki = 65.4 nM
|
|
|
|
CP0402075
|
N-(1-adamantyl)-6-(benzenesulfonyl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O4S
|
1
|
| 1 |
Ki = 65.9 nM
|
|
|
|
CP0434520
|
9-methoxy-2,4,4-trimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C23H34N2O2
|
1
|
| 1 |
Ki = 66.4 nM
|
|
|
|
CP0542424
|
N-(1-adamantyl)-2-(1-ethyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C28H32N2O
|
1
|
| 1 |
Ki = 67 nM
|
|
|
|
CP0488283
|
(6aR,9R,10aR)-3-(1-adamantyl)-9-[(Z)-2-methoxyethenyl]-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-1-ol
Show/Hide
|
C28H38O3
|
1
|
| 1 |
Ki = 67.2 nM
|
|
|
|
CP0464092
|
US8859596, 156
Show/Hide
|
C23H30F6N4O2
|
1
|
| 1 |
Ki = 68 nM
|
|
|
|
CP0466663
|
US8859596, 203
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
Ki = 68 nM
|
|
|
|
CP0498833
|
1-benzyl-N-[2-(4-fluorophenyl)ethyl]-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C24H20FN3O2
|
1
|
| 1 |
Ki = 69.8 nM
|
|
|
|
CP0498835
|
1-butyl-N-cyclohexyl-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C19H25N3O2
|
1
|
| 1 |
Ki = 70 nM
|
|
|
|
CP0436073
|
N-(1-adamantyl)-2-(1-pentyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C31H38N2O
|
1
|
| 1 |
Ki = 70 nM
|
|
|
|
CP0525904
|
N-(1-adamantyl)-2-(5-phenyl-1H-indol-3-yl)acetamide
Show/Hide
|
C26H28N2O
|
1
|
| 1 |
Ki = 70.8 nM
|
|
|
|
CP0493047
|
6-((E)-3,3-Dimethyl-but-1-enyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H42N2O2
|
1
|
| 1 |
Ki = 71.6 nM
|
|
|
|
CP0390454
|
1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(4,5,6,7-tetrahydroisoindol-2-yl)pyrazole-3-carboxamide
Show/Hide
|
C26H22Cl4N4O
|
1
|
| 1 |
Ki = 72.9 nM
|
|
|
|
CP0428988
|
(9-pentylcarbazol-3-yl)-piperidin-1-ylmethanone
Show/Hide
|
C23H28N2O
|
1
|
| 1 |
Ki = 73 nM
|
|
|
|
CP0462105
|
3-[3-(piperidine-1-carbonyl)carbazol-9-yl]propyl 1,1-dioxo-1,4-thiazinane-4-carboxylate
Show/Hide
|
C26H31N3O5S
|
1
|
| 1 |
Ki = 73 nM
|
|
|
|
CP0406214
|
N-(1-adamantyl)-6-(benzenesulfinyl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O3S
|
1
|
| 1 |
Ki = 73.2 nM
|
|
|
|
CP0389367
|
US8895592, 28
Show/Hide
|
C21H22F3N3O3S
|
1
|
| 1 |
Ki = 75 nM
|
|
|
|
CP0470283
|
US8859596, 149
Show/Hide
|
C24H35F3N4O2
|
1
|
| 1 |
Ki = 77 nM
|
|
|
|
CP0343766
|
9-(3-bromopropoxy)-2,4,4-trimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C25H37BrN2O2
|
1
|
| 1 |
Ki = 77.3 nM
|
|
|
|
CP0393335
|
N',N'-dimethyl-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carbohydrazide
Show/Hide
|
C23H27N3O2S
|
1
|
| 1 |
Ki = 77.5 nM
|
|
|
|
CP0536587
|
9-(2-bromoethoxy)-2-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C25H37BrN2O2
|
1
|
| 1 |
Ki = 78.7 nM
|
|
|
|
CP0454320
|
N-cyclohexyl-7-methoxy-1-(2-morpholin-4-ylethyl)-4-oxoquinoline-3-carboxamide
Show/Hide
|
C23H31N3O4
|
1
|
| 1 |
Ki = 79 nM
|
|
|
|
CP0510584
|
1-benzyl-N-cyclohexyl-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C24H26N2O3
|
1
|
| 1 |
Ki = 79 nM
|
|
|
|
CP0450454
|
1-benzyl-N-cyclohexyl-4-hydroxy-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
Ki = 79 nM
|
|
|
|
CP0432934
|
11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid cyclopropylmethyl-amide
Show/Hide
|
C26H43NO3
|
1
|
| 1 |
Ki = 80 nM
|
|
|
|
CP0376698
|
N-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C21H15Cl3N4O
|
1
|
| 1 |
Ki = 80 nM
|
|
|
|
CP0480063
|
N-cycloheptyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C24H28Cl2N4O
|
1
|
| 1 |
Ki = 80 nM
|
|
|
|
CP0388259
|
2-[(4-fluorophenyl)methoxy]-N-(4-methylcyclohexyl)pyridine-3-carboxamide
Show/Hide
|
C20H23FN2O2
|
1
|
| 1 |
Ki = 80 nM
|
|
|
|
CP0429008
|
[9-(3-methoxypropyl)carbazol-3-yl]-piperidin-1-ylmethanone
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
Ki = 83 nM
|
|
|
|
CP0455975
|
2,5-dimethyl-N-naphthalen-1-yl-1-phenylpyrrole-3-carboxamide
Show/Hide
|
C23H20N2O
|
1
|
| 1 |
Ki = 84.22 nM
|
|
|
|
CP0428977
|
morpholin-4-yl-(9-pentylcarbazol-3-yl)methanone
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
Ki = 84.5 nM
|
|
|
|
CP0512551
|
US8846730, 77
Show/Hide
|
C28H37F3N4O4S
|
1
|
| 1 |
Ki = 85 nM
|
|
|
|
CP0535626
|
US8859596, 204
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
Ki = 87 nM
|
|
|
|
CP0434530
|
9-methoxy-4,4-dimethyl-7-(2-methyloctan-2-yl)-1H-chromeno[4,3-c]pyrazole
Show/Hide
|
C22H32N2O2
|
1
|
| 1 |
Ki = 87.1 nM
|
|
|
|
CP0529927
|
9-(3-bromopropoxy)-2-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C26H39BrN2O2
|
1
|
| 1 |
Ki = 87.1 nM
|
|
|
|
CP0443757
|
[9-(3-chloropropyl)carbazol-3-yl]-piperidin-1-ylmethanone
Show/Hide
|
C21H23ClN2O
|
1
|
| 1 |
Ki = 88 nM
|
|
|
|
CP0380792
|
THC, 8 beta-OH
Show/Hide
|
C21H30O3
|
1
|
| 1 |
Ki = 88 nM
|
|
|
|
CP0952457
|
US8859596, 160
Show/Hide
|
C25H34F3N3O2
|
1
|
| 1 |
Ki = 88 nM
|
|
|
|
CP0404947
|
N-(1-azabicyclo[2.2.2]octan-3-yl)-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C28H33N3O2S
|
1
|
| 1 |
Ki = 89.1 nM
|
|
|
|
CP0379381
|
5-(4-fluorophenyl)-2-methoxy-3-methyl-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C22H26FNO2
|
1
|
| 1 |
Ki = 90 nM
|
|
|
|
CP0388919
|
2-methoxy-3-methyl-N-(4-methylcyclohexyl)-5-phenylbenzamide
Show/Hide
|
C22H27NO2
|
1
|
| 1 |
Ki = 90 nM
|
|
|
|
CP0432891
|
piperidin-1-yl-[9-(pyridin-4-ylmethyl)carbazol-3-yl]methanone
Show/Hide
|
C24H23N3O
|
1
|
| 1 |
Ki = 91 nM
|
|
|
|
CP0389942
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-[4-(cyclohexylmethylsulfonyl)piperazin-1-yl]purine
Show/Hide
|
C28H30Cl2N6O2S
|
1
|
| 1 |
Ki = 91 nM
|
|
|
|
CP0434911
|
N-[3-(morpholine-4-carbonyl)-5,7-dihydro-4H-thieno[2,3-c]pyran-2-yl]tricyclo[3.3.1.03,7]nonane-3-carboxamide
Show/Hide
|
C22H28N2O4S
|
1
|
| 1 |
Ki = 91.2 nM
|
|
|
|
CP0431465
|
US8846730, 31
Show/Hide
|
C26H34F3N3O3S
|
1
|
| 1 |
Ki = 92 nM
|
|
|
|
CP0135102
|
2-ethyl-9-methoxy-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C24H36N2O2
|
1
|
| 1 |
Ki = 92.6 nM
|
|
|
|
CP0548830
|
8-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]-N-(2,2,2-trifluoroethyl)octanamide
Show/Hide
|
C26H42F3NO3
|
1
|
| 1 |
Ki = 92.8 nM
|
|
|
|
CP0421306
|
4,4-dimethyl-7-(2-methyloctan-2-yl)-9-phenylmethoxy-1H-chromeno[4,3-c]pyrazole
Show/Hide
|
C28H36N2O2
|
1
|
| 1 |
Ki = 93.3 nM
|
|
|
|
CP0498312
|
7-fluoro-1-methyl-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C21H25FN2O2
|
1
|
| 1 |
Ki = 93.9 nM
|
|
|
|
CP0454319
|
N-cyclohexyl-7-(dimethylamino)-1-(2-morpholin-4-ylethyl)-4-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H33N5O3
|
1
|
| 1 |
Ki = 94 nM
|
|
|
|
CP0396832
|
(5aR,11bR)-11-hydroxy-6,6-dimethyl-9-(2-methyloctan-2-yl)-4,5,5a,11b-tetrahydro-1H-oxepino[4,5-c]chromen-2-one
Show/Hide
|
C24H36O4
|
1
|
| 1 |
Ki = 94 nM
|
|
|
|
CP0072767
|
(5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2-chloro-ethyl)-amide
Show/Hide
|
C22H36ClNO
|
1
|
| 1 |
Ki = 95 nM
|
|
|
|
CP0415899
|
US8895592, 11
Show/Hide
|
C26H34F3N3O3S
|
1
|
| 1 |
Ki = 95 nM
|
|
|
|
CP0414943
|
(9-hexylcarbazol-3-yl)-piperidin-1-ylmethanone
Show/Hide
|
C24H30N2O
|
1
|
| 1 |
Ki = 96 nM
|
|
|
|
CP0538165
|
US8895592, 6
Show/Hide
|
C24H29F3N4O2S
|
1
|
| 1 |
Ki = 96 nM
|
|
|
|
CP0544120
|
US8895592, 16
Show/Hide
|
C23H29N3O2S
|
1
|
| 1 |
Ki = 96 nM
|
|
|
|
CP0548584
|
11-(3-hydroxy-5-pentylphenoxy)-N-(2,2,2-trifluoroethyl)undecanamide
Show/Hide
|
C24H38F3NO3
|
1
|
| 1 |
Ki = 96.3 nM
|
|
|
|
CP0567082
|
11-(3-hydroxy-5-pentylphenoxy)-N-[(2R)-1-hydroxypropan-2-yl]undecanamide
Show/Hide
|
C25H43NO4
|
1
|
| 1 |
Ki = 97.2 nM
|
|
|
|
CP0552966
|
3-[2-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-yl]oxypropan-1-ol
Show/Hide
|
C26H40N2O3
|
1
|
| 1 |
Ki = 97.4 nM
|
|
|
|
CP0416221
|
N-(1-adamantyl)-2-(1-methyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C27H30N2O
|
1
|
| 1 |
Ki = 98 nM
|
|
|
|
CP0392392
|
5-(2-chloropyrrol-1-yl)-1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H15Cl5N4O
|
1
|
| 1 |
Ki = 98.5 nM
|
|
|
|
CP0376650
|
N-[(4-chlorophenyl)methyl]-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H17Cl3N4O
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0383135
|
N-cycloheptyl-2-methoxy-3-methyl-5-phenylbenzamide
Show/Hide
|
C22H27NO2
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0511225
|
2-[(6aR,9R,10aR)-3-(1-adamantyl)-1-hydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-9-yl]acetonitrile
Show/Hide
|
C27H35NO2
|
1
|
| 1 |
Ki = 100.3 nM
|
|
|
|
CP0429009
|
(9-pentylcarbazol-3-yl)-phenylmethanone
Show/Hide
|
C24H23NO
|
1
|
| 1 |
Ki = 101 nM
|
|
|
|
CP0407061
|
US8846730, 46
Show/Hide
|
C28H38F3N3O3S
|
1
|
| 1 |
Ki = 102 nM
|
|
|
|
CP0399232
|
(S)-4-((2',3'-dichlorobiphenyl-4-yl)methyl)-2-phenylmorpholine
Show/Hide
|
C23H21Cl2NO
|
2
|
| 1 |
Ki = 104 nM
|
|
|
| 2 |
Ki = 312 nM
|
|
|
|
CP0443540
|
1-butyl-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C17H26N2O2
|
1
|
| 1 |
Ki = 104 nM
|
|
|
|
CP0550756
|
N-(2-hydroxyethyl)-11-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
|
C29H51NO4
|
1
|
| 1 |
Ki = 104.4 nM
|
|
|
|
CP0410346
|
2-[[2-fluoro-6-(trifluoromethyl)benzoyl]amino]-N-propyl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
|
C19H18F4N2O3S
|
1
|
| 1 |
Ki = 104.71 nM
|
|
|
|
CP0453065
|
2-(bicyclo[2.2.1]heptane-2-carbonylamino)-N-propyl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
|
C19H26N2O3S
|
1
|
| 1 |
Ki = 104.71 nM
|
|
|
|
CP0382525
|
US8846730, 47
Show/Hide
|
C27H34F3N3O4S
|
1
|
| 1 |
Ki = 107 nM
|
|
|
|
CP0396951
|
N-cycloheptyl-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C24H28F2N4O
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0102214
|
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H21Cl2IN4O
|
2
|
| 1 |
Ki = 110 nM
|
|
|
| 2 |
Ki = 112 nM
|
|
|
|
CP0452193
|
2-[8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]octoxy]propane-1,3-diol
Show/Hide
|
C26H46O5
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0514781
|
N-(1-adamantyl)-2-[5-(furan-2-yl)-1-pentylindol-3-yl]acetamide
Show/Hide
|
C29H36N2O2
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0429629
|
US8895592, 13
Show/Hide
|
C24H32F3N3O2S
|
1
|
| 1 |
Ki = 111 nM
|
|
|
|
CP0400947
|
ethyl 2-(3-phenylpropanoylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C20H23NO3S
|
1
|
| 1 |
Ki = 111.87 nM
|
|
|
|
CP0508692
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-(1-benzothiophen-2-yl)methanone
Show/Hide
|
C24H24O4S
|
1
|
| 1 |
Ki = 113.1 nM
|
|
|
|
CP0489050
|
1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dimethylpyrrol-1-yl)-4-ethylpyrazole-3-carboxamide
Show/Hide
|
C25H22Cl4N4O
|
1
|
| 1 |
Ki = 113.7 nM
|
|
|
|
CP0375414
|
US8846730, 1
Show/Hide
|
C24H30F3N3O3S
|
1
|
| 1 |
Ki = 115 nM
|
|
|
|
CP0425094
|
US8846730, 67
Show/Hide
|
C25H29F3N4O3S
|
1
|
| 1 |
Ki = 115 nM
|
|
|
|
CP0409132
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-(1-benzofuran-3-yl)methanone
Show/Hide
|
C24H24O5
|
1
|
| 1 |
Ki = 118.2 nM
|
|
|
|
CP0525504
|
N-(2-morpholin-4-ylethyl)-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C27H33N3O3S
|
1
|
| 1 |
Ki = 118.7 nM
|
|
|
|
CP0410867
|
8-(3-hydroxy-5-pentylphenoxy)-N-[(2R)-1-hydroxypropan-2-yl]octanamide
Show/Hide
|
C22H37NO4
|
1
|
| 1 |
Ki = 119.3 nM
|
|
|
|
CP0405728
|
(5Z,7S,8Z,11Z,14Z)-N-[(2R)-1-hydroxypropan-2-yl]-7-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C24H41NO2
|
1
|
| 1 |
Ki = 120 nM
|
|
|
|
CP0410347
|
N-(2-methoxyethyl)-2-(tricyclo[3.3.1.03,7]nonane-3-carbonylamino)-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
|
C21H28N2O4S
|
1
|
| 1 |
Ki = 120.23 nM
|
|
|
|
CP0511224
|
(6aR,9S,10aR)-3-(1-adamantyl)-9-(hydroxymethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-1-ol
Show/Hide
|
C26H36O3
|
1
|
| 1 |
Ki = 121.2 nM
|
|
|
|
CP0465951
|
1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-tert-pentyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H26Cl2N4O
|
1
|
| 1 |
Ki = 121.5 nM
|
|
|
|
CP0429002
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-(1-benzothiophen-3-yl)methanone
Show/Hide
|
C24H24O4S
|
1
|
| 1 |
Ki = 124.8 nM
|
|
|
|
CP0418513
|
6-(3,5-Dimethyl-isoxazol-4-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C30H37N3O3
|
1
|
| 1 |
Ki = 125.7 nM
|
|
|
|
CP0443117
|
US8859596, 170
Show/Hide
|
C22H31F3N4O2S
|
1
|
| 1 |
Ki = 127 nM
|
|
|
|
CP0385040
|
11-(3-hydroxy-5-pentylphenoxy)-N-phenylundecanamide
Show/Hide
|
C28H41NO3
|
1
|
| 1 |
Ki = 127.8 nM
|
|
|
|
CP0912378
|
US8859596, 157
Show/Hide
|
C25H34F3N3O2
|
1
|
| 1 |
Ki = 128 nM
|
|
|
|
CP0876344
|
10alpha-Hydroxy-Delta9,11-hexahydrocannabinol
Show/Hide
|
C21H30O3
|
1
|
| 1 |
Ki = 129 nM
|
|
|
|
CP0385692
|
US8895592, 34
Show/Hide
|
C24H32F3N3O3S
|
1
|
| 1 |
Ki = 129 nM
|
|
|
|
CP0420377
|
N-(2-hydroxyethyl)-8-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]octanamide
Show/Hide
|
C26H45NO4
|
1
|
| 1 |
Ki = 129.4 nM
|
|
|
|
CP0409163
|
N-cyclohexyl-2-[(4-fluorophenyl)methoxy]quinoline-3-carboxamide
Show/Hide
|
C23H23FN2O2
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0443425
|
7-bromo-N-[(3,4-dichlorophenyl)methyl]-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C22H21BrCl2N2O2
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0466292
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2,2,2-trifluoroethanone
Show/Hide
|
C23H17Cl2F3N6O
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0396892
|
N-(1-adamantyl)-2-butyl-6-(furan-2-yl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C28H32N2O3
|
1
|
| 1 |
Ki = 133 nM
|
|
|
|
CP0498793
|
1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-N-(3,3-dimethylbutyl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H28Cl2N4O
|
1
|
| 1 |
Ki = 133.5 nM
|
|
|
|
CP0392391
|
1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dichloropyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H14Cl6N4O
|
1
|
| 1 |
Ki = 135.2 nM
|
|
|
|
CP0465952
|
1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(octan-2-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H32Cl2N4O
|
1
|
| 1 |
Ki = 135.5 nM
|
|
|
|
CP0248913
|
(5Z,8Z,11Z,13S,14Z)-N-cyclopentyl-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
|
C26H43NO
|
1
|
| 1 |
Ki = 139 nM
|
|
|
|
CP0404950
|
1-[(3-methylphenyl)methyl]-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C34H36N2O2S
|
1
|
| 1 |
Ki = 139.1 nM
|
|
|
|
CP0425346
|
US8846730, 30
Show/Hide
|
C26H34F3N3O3S
|
1
|
| 1 |
Ki = 141 nM
|
|
|
|
CP0413292
|
3-butyl-2-methoxy-5-(4-methoxyphenyl)-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C26H35NO3
|
1
|
| 1 |
Ki = 143 nM
|
|
|
|
CP0419213
|
2-methoxy-3-methyl-N-(4-methylcyclohexyl)-5-phenylbenzamide
Show/Hide
|
C22H27NO2
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0507345
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-(1H-indol-3-yl)methanone
Show/Hide
|
C24H25NO4
|
1
|
| 1 |
Ki = 158.6 nM
|
|
|
|
CP0532218
|
N-(1-adamantyl)-7-hydroxy-2-(2-hydroxyethyl)-5-oxo-4-propylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H30N4O4
|
1
|
| 1 |
Ki = 159 nM
|
|
|
|
CP0434519
|
1-ethyl-9-methoxy-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C24H36N2O2
|
1
|
| 1 |
Ki = 159.5 nM
|
|
|
|
CP0037555
|
(5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-tetraenamide
Show/Hide
|
C22H37NO2
|
2
|
| 1 |
Ki = 160 nM
|
|
|
| 2 |
Ki = 168 nM
|
|
|
|
CP0459063
|
1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dichloropyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H14Cl6N4O
|
1
|
| 1 |
Ki = 161.7 nM
|
|
|
|
CP0376687
|
1-(2,4-Difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-N-(3,3-dimethylbutyl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H28F2N4O
|
1
|
| 1 |
Ki = 163.4 nM
|
|
|
|
CP0400950
|
N-cyclohexyl-2,5-dimethyl-1-phenylpyrrole-3-carboxamide
Show/Hide
|
C19H24N2O
|
1
|
| 1 |
Ki = 167.81 nM
|
|
|
|
CP0430955
|
N-cyclopentyl-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C20H20Cl2N4O
|
1
|
| 1 |
Ki = 170 nM
|
|
|
|
CP0542425
|
N-(1-adamantyl)-2-(5-bromo-1-pentylindol-3-yl)acetamide
Show/Hide
|
C25H33BrN2O
|
1
|
| 1 |
Ki = 170 nM
|
|
|
|
CP0446146
|
N-cyclohexyl-2-ethyl-5-methyl-1-phenylpyrrole-3-carboxamide
Show/Hide
|
C20H26N2O
|
1
|
| 1 |
Ki = 170.81 nM
|
|
|
|
CP0420194
|
9-pentyl-N-piperidin-1-ylpyrido[3,4-b]indole-3-carboxamide
Show/Hide
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C22H28N4O
|
1
|
| 1 |
Ki = 171.1 nM
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CP0104539
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(5Z,8Z,11Z,13S,14Z)-N-[(2R)-1-hydroxypropan-2-yl]-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
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C24H41NO2
|
1
|
| 1 |
Ki = 176 nM
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CP0292304
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6-Biphenyl-4-yl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acidadamantan-1-ylamide
Show/Hide
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C37H40N2O2
|
1
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| 1 |
Ki = 181 nM
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CP0566882
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11-(3-hydroxy-5-pentylphenoxy)-N',N'-dimethylundecanehydrazide
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C24H42N2O3
|
1
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| 1 |
Ki = 182.6 nM
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CP0461548
|
US8859596, 35
Show/Hide
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C25H29F3N6OS
|
1
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| 1 |
Ki = 185 nM
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CP0420323
|
2-[6-(1-adamantylcarbamoyl)-7-hydroxy-5-oxo-4-propylpyrazolo[4,3-b]pyridin-2-yl]ethyl acetate
Show/Hide
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C24H32N4O5
|
1
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| 1 |
Ki = 186 nM
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CP0442970
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N-cycloheptyl-1-[(4-iodophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
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C20H23IN2O2
|
1
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| 1 |
Ki = 187 nM
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CP0513621
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(5Z,7S,8Z,11Z,14Z)-N-(2-hydroxyethyl)-7-methylicosa-5,8,11,14-tetraenamide
Show/Hide
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C23H39NO2
|
1
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| 1 |
Ki = 188 nM
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CP0424026
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N-(1-adamantyl)-2-(1-benzyl-5-phenylindol-3-yl)acetamide
Show/Hide
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C33H34N2O
|
1
|
| 1 |
Ki = 189 nM
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CP0398425
|
cyclopropanolamide, 14a
Show/Hide
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C23H37NO2
|
1
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| 1 |
Ki = 190 nM
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CP0419836
|
2-[6-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]hexoxy]propane-1,3-diol
Show/Hide
|
C24H42O5
|
1
|
| 1 |
Ki = 190 nM
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CP0425248
|
methyl 2-(piperidine-1-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C16H22N2O3S
|
1
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| 1 |
Ki = 195.7 nM
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CP0430952
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N-cycloheptyl-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C22H24F2N4O
|
1
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| 1 |
Ki = 200 nM
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CP0450453
|
1-benzyl-N-cyclohexyl-2-oxopyridine-3-carboxamide
Show/Hide
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C19H22N2O2
|
1
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| 1 |
Ki = 200 nM
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CP0410863
|
N-benzyl-11-(3-hydroxy-5-pentylphenoxy)undecanamide
Show/Hide
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C29H43NO3
|
1
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| 1 |
Ki = 202.3 nM
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CP0382509
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-Nheptyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H30Cl2N4O
|
1
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| 1 |
Ki = 204.8 nM
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CP0498791
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1-(2,4-Dichlorophenyl)-4-methyl-N-pentyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C20H22Cl2N4O
|
1
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| 1 |
Ki = 205.9 nM
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CP0474347
|
US8846730, 26
Show/Hide
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C26H34F3N3O3S
|
1
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| 1 |
Ki = 206 nM
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CP0429006
|
methyl 4-[3-(piperidine-1-carbonyl)carbazol-9-yl]butanoate
Show/Hide
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C23H26N2O3
|
1
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| 1 |
Ki = 208 nM
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CP0473480
|
US8846730, 12
Show/Hide
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C25H32F3N3O3S
|
1
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| 1 |
Ki = 208 nM
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CP0549308
|
2,4,4-trimethyl-7-(2-methyloctan-2-yl)-9-phenylmethoxychromeno[4,3-c]pyrazole
Show/Hide
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C29H38N2O2
|
1
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| 1 |
Ki = 208.8 nM
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CP0442880
|
US8846730, 20
Show/Hide
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C26H28F3N3O4S
|
1
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| 1 |
Ki = 209 nM
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CP0390260
|
US8859596, 161
Show/Hide
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C25H35N5O3
|
1
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| 1 |
Ki = 209 nM
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CP0507362
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-(1-benzofuran-2-yl)methanone
Show/Hide
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C24H24O5
|
1
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| 1 |
Ki = 209.4 nM
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CP0552958
|
2-[2-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-yl]oxyethanol
Show/Hide
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C25H38N2O3
|
1
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| 1 |
Ki = 210.6 nM
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CP0538058
|
2-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)-9-phenylmethoxychromeno[4,3-c]pyrazole
Show/Hide
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C30H40N2O2
|
1
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| 1 |
Ki = 212.2 nM
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CP0400702
|
N-ethyl-2-(tricyclo[3.3.1.03,7]nonane-3-carbonylamino)-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
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C20H26N2O3S
|
1
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| 1 |
Ki = 213.8 nM
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CP0508824
|
piperidin-1-yl-[9-(pyridin-2-ylmethyl)carbazol-3-yl]methanone
Show/Hide
|
C24H23N3O
|
1
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| 1 |
Ki = 215 nM
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CP0499726
|
4-hydroxy-1-(3-hydroxypropyl)-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C19H25N3O4
|
1
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| 1 |
Ki = 215 nM
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CP0506905
|
US8859596, 150
Show/Hide
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C24H33F3N4O2S
|
1
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| 1 |
Ki = 216 nM
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CP0506638
|
N-(1-adamantyl)-4-oxo-8-phenyl-1H-quinoline-3-carboxamide
Show/Hide
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C26H26N2O2
|
1
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| 1 |
Ki = 220 nM
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CP0038524
|
(5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((R)-2-hydroxy-1-methyl-ethyl)-amide
Show/Hide
|
C23H39NO2
|
1
|
| 1 |
Ki = 220 nM
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CP0447824
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[(2-fluorophenyl)methyl]urea
Show/Hide
|
C30H26Cl2FN7O
|
1
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| 1 |
Ki = 220 nM
|
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CP0375147
|
(1,1-dioxo-1,4-thiazinan-4-yl)-(9-pentylcarbazol-3-yl)methanone
Show/Hide
|
C22H26N2O3S
|
1
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| 1 |
Ki = 225 nM
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CP0453372
|
(2S)-1-(4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carbonyl)pyrrolidine-2-carboxamide
Show/Hide
|
C26H29N3O3S
|
1
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| 1 |
Ki = 230 nM
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CP0487935
|
N-(1,3-dihydroxypropan-2-yl)-11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
|
C29H51NO5
|
1
|
| 1 |
Ki = 230 nM
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CP0412798
|
1-(2,4-Dichlorophenyl)-4-methyl-N-(octan-2-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H28Cl2N4O
|
1
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| 1 |
Ki = 237.3 nM
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CP0113406
|
1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid cyclohexylamide
Show/Hide
|
C22H20Cl3N3O
|
1
|
| 1 |
Ki = 240 nM
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CP0482760
|
methyl 2-(phenoxycarbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C17H17NO4S
|
1
|
| 1 |
Ki = 244.06 nM
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CP0480943
|
US8859596, 187
Show/Hide
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C21H28F3N5OS
|
1
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| 1 |
Ki = 247 nM
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CP0529560
|
[9-[3-(1,1-dioxo-1,4-thiazinan-4-yl)propyl]carbazol-3-yl]-piperidin-1-ylmethanone
Show/Hide
|
C25H31N3O3S
|
1
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| 1 |
Ki = 249 nM
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CP0525975
|
N-cyclohexyl-2-[(4-fluorophenyl)methoxy]pyridine-3-carboxamide
Show/Hide
|
C19H21FN2O2
|
1
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| 1 |
Ki = 250 nM
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CP0384509
|
N-[11-(2-hexyl-5-hydroxyphenoxy)undecyl]cyclopropanecarboxamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 250 nM
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CP0376688
|
1-(2,4-Dichlorophenyl)-N-heptyl-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H26Cl2N4O
|
1
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| 1 |
Ki = 255.1 nM
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CP0400703
|
2-(2-oxatricyclo[3.3.1.13,7]decane-1-carbonylamino)-N-propyl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
|
C21H28N2O4S
|
1
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| 1 |
Ki = 257.04 nM
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CP0565980
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(6aR,9R,10aR)-3-(1-adamantyl)-9-(iodomethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-1-ol
Show/Hide
|
C26H35IO2
|
1
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| 1 |
Ki = 261.7 nM
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CP0395254
|
(9-butylcarbazol-3-yl)-piperidin-1-ylmethanone
Show/Hide
|
C22H26N2O
|
1
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| 1 |
Ki = 264 nM
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CP0561260
|
1-(3,4-dichlorophenyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
|
C27H32Cl2N2O2
|
1
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| 1 |
Ki = 270 nM
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CP0555377
|
US8859596, 184
Show/Hide
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C25H36F3N5O3S
|
1
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| 1 |
Ki = 279 nM
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CP0444410
|
8-(4-hexyl-3-hydroxy-phenoxy)-octanoic acidcyclopropylamide
Show/Hide
|
C23H37NO3
|
1
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| 1 |
Ki = 280 nM
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CP0429550
|
(5Z,8Z,11Z,13S,14Z)-N-[(2R)-1-hydroxypropan-2-yl]-13-methyl-18-phenoxyoctadeca-5,8,11,14-tetraenamide
Show/Hide
|
C28H41NO3
|
1
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| 1 |
Ki = 286 nM
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CP0388959
|
N-(1-adamantyl)-9-pentylcarbazole-3-carboxamide
Show/Hide
|
C28H34N2O
|
1
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| 1 |
Ki = 288.5 nM
|
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CP0472442
|
US8846730, 57
Show/Hide
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C26H34F3N3O3S
|
1
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| 1 |
Ki = 289 nM
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CP0298207
|
cyclopropanolamide, 11a
Show/Hide
|
C23H37NO2
|
1
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| 1 |
Ki = 290 nM
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CP0106737
|
N-[(2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl]-2-methyl-2-[5-(trifluoromethyl)pyridin-2-yl]oxypropanamide
Show/Hide
|
C27H25ClF3N3O2
|
1
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| 1 |
Ki = 290 nM
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CP0400884
|
N-(3,3-diphenylpropyl)-2,2-diphenylpropanamide
Show/Hide
|
C30H29NO
|
1
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| 1 |
Ki = 290 nM
|
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CP0549310
|
1-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)-9-phenylmethoxychromeno[4,3-c]pyrazole
Show/Hide
|
C30H40N2O2
|
1
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| 1 |
Ki = 295.9 nM
|
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CP0468190
|
US8895592, 10
Show/Hide
|
C24H35N3O2S
|
1
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| 1 |
Ki = 296 nM
|
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CP0526833
|
11-(3-methoxy-5-pentylphenoxy)-N-phenylundecanamide
Show/Hide
|
C29H43NO3
|
1
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| 1 |
Ki = 308.9 nM
|
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CP0428636
|
12-(3-hydroxy-5-pentyl-phenoxy)-dodecanoic acidcyclopropylamide
Show/Hide
|
C26H43NO3
|
1
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| 1 |
Ki = 310 nM
|
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CP0401267
|
N-cyclopentyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H24Cl2N4O
|
1
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| 1 |
Ki = 310 nM
|
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CP0461992
|
2,3-dihydroxypropyl 11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecanoate
Show/Hide
|
C29H50O6
|
1
|
| 1 |
Ki = 310 nM
|
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CP0469874
|
N-(cyclopropylmethyl)-11-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
|
C31H53NO3
|
1
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| 1 |
Ki = 322.3 nM
|
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CP0849493
|
9beta,10beta-Epoxyhexahydrocannabinol
Show/Hide
|
C21H30O3
|
1
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| 1 |
Ki = 335 nM
|
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CP0389443
|
3-[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]adamantane-1-carboxamide
Show/Hide
|
C26H35NO4
|
1
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| 1 |
Ki = 337 nM
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CP0385252
|
(6aR,10aR)-3-(1-adamantyl)-1-hydroxy-6,6-dimethyl-7,8,10,10a-tetrahydro-6aH-benzo[c]chromen-9-one
Show/Hide
|
C25H32O3
|
1
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| 1 |
Ki = 338 nM
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CP0488096
|
3-(1-adamantyl)-9-methoxy-6,6-dimethylbenzo[c]chromen-1-ol
Show/Hide
|
C26H30O3
|
1
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| 1 |
Ki = 338 nM
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CP0443426
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N-methoxy-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C22H24N2O3S
|
1
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| 1 |
Ki = 340 nM
|
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CP0102216
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N-(1-adamantyl)-4-oxo-1-pentyl-6-(2-phenylethynyl)quinoline-3-carboxamide
Show/Hide
|
C33H36N2O2
|
1
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| 1 |
Ki = 343 nM
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CP0563452
|
3-[2,4,4-trimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-yl]oxypropan-1-ol
Show/Hide
|
C25H38N2O3
|
1
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| 1 |
Ki = 364 nM
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CP0449575
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(6aR,9S,10aR)-3-(1-adamantyl)-9-(2-hydroxyethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-1-ol
Show/Hide
|
C27H38O3
|
1
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| 1 |
Ki = 365.3 nM
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CP0500040
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1-(2,4-Difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-Nheptyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H30F2N4O
|
1
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| 1 |
Ki = 365.5 nM
|
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CP0549309
|
1-(2-hydroxyethyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
|
C23H34N2O3
|
1
|
| 1 |
Ki = 366 nM
|
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CP0414944
|
9-pentyl-3-(piperidin-1-ylmethyl)carbazole
Show/Hide
|
C23H30N2
|
1
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| 1 |
Ki = 370 nM
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CP0879200
|
1-Butyl-2-(3,4-dichlorobenzyl)-5-trifluoromethylbenzimidazole
Show/Hide
|
C19H17Cl2F3N2
|
1
|
| 1 |
Ki = 370 nM
|
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CP0506340
|
N-[(2-bromo-3,4,5-trimethoxyphenyl)methyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C27H27BrF2N4O4
|
1
|
| 1 |
Ki = 373 nM
|
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CP0496088
|
N-cyclohexyl-1-(2,4-dichlorophenyl)-4-methyl-5-(4,5,6,7-tetrahydroisoindol-2-yl)pyrazole-3-carboxamide
Show/Hide
|
C25H28Cl2N4O
|
1
|
| 1 |
Ki = 376.4 nM
|
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CP0514782
|
N-cycloheptyl-2-[5-(furan-2-yl)-1-prop-2-enylindol-3-yl]acetamide
Show/Hide
|
C24H28N2O2
|
1
|
| 1 |
Ki = 377 nM
|
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CP0492363
|
2-[10-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]decoxy]propane-1,3-diol
Show/Hide
|
C28H50O5
|
1
|
| 1 |
Ki = 380 nM
|
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CP0500041
|
1-(2,4-Dichlorophenyl)-N-hexyl-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H24Cl2N4O
|
1
|
| 1 |
Ki = 383.3 nM
|
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CP0427500
|
8-(3-hydroxy-5-pentyl-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide
Show/Hide
|
C21H35NO4
|
1
|
| 1 |
Ki = 390 nM
|
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|
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CP0395643
|
5-bromo-2-butoxy-N-cycloheptylpyridine-3-carboxamide
Show/Hide
|
C17H25BrN2O2
|
1
|
| 1 |
Ki = 396 nM
|
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CP0388258
|
N-cycloheptyl-1-[(3-iodophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
|
C20H23IN2O2
|
1
|
| 1 |
Ki = 397 nM
|
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CP0533013
|
2-(4-methylpiperazin-1-yl)-1-(9-pentylcarbazol-3-yl)ethanone
Show/Hide
|
C24H31N3O
|
1
|
| 1 |
Ki = 398 nM
|
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|
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CP0401975
|
6-Bromo-4-oxo-1-pentyl-N-(piperidin-1-yl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C20H26BrN3O2
|
1
|
| 1 |
Ki = 400 nM
|
|
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CP0412556
|
N-cyclohexyl-2-[5-[(3-methoxyphenyl)methoxy]-1-prop-2-enylindol-3-yl]acetamide
Show/Hide
|
C27H32N2O3
|
1
|
| 1 |
Ki = 400 nM
|
|
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CP0552882
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]pentan-1-one
Show/Hide
|
C26H26Cl2N6O
|
1
|
| 1 |
Ki = 400 nM
|
|
|
|
CP0432073
|
N-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]piperidine-1-carboxamide
Show/Hide
|
C28H29Cl2N7O
|
1
|
| 1 |
Ki = 400 nM
|
|
|
|
CP0525578
|
[9-[3-(dimethylamino)propyl]carbazol-3-yl]-piperidin-1-ylmethanone
Show/Hide
|
C23H29N3O
|
1
|
| 1 |
Ki = 403 nM
|
|
|
|
CP0440708
|
N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-diethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H30Cl2N4O
|
1
|
| 1 |
Ki = 409.6 nM
|
|
|
|
CP0943932
|
1-(2-diethylaminoethyl)-2-(4-ethoxybenzyl)-5-trifluoromethylbenzimidazole
Show/Hide
|
C23H28F3N3O
|
1
|
| 1 |
Ki = 420 nM
|
|
|
|
CP0085437
|
(3-benzyl-3-methyl-2,3-dihydrobenzofuran-6-yl)(piperidin-1-yl)methanone
Show/Hide
|
C22H25NO2
|
1
|
| 1 |
Ki = 422 nM
|
|
|
|
CP0471599
|
N-(1-adamantyl)-8-methoxy-4-oxo-1-pentyl-6-phenylquinoline-3-carboxamide
Show/Hide
|
C32H38N2O3
|
1
|
| 1 |
Ki = 430 nM
|
|
|
|
CP0565261
|
butyl 2-[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]acetate
Show/Hide
|
C21H30O5
|
1
|
| 1 |
Ki = 432 nM
|
|
|
|
CP0529926
|
3-[1-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-yl]oxypropan-1-ol
Show/Hide
|
C26H40N2O3
|
1
|
| 1 |
Ki = 440 nM
|
|
|
|
CP0390455
|
1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-ethyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C23H18Cl4N4O
|
1
|
| 1 |
Ki = 454.6 nM
|
|
|
|
CP0527604
|
N-butyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H24Cl2N4O
|
1
|
| 1 |
Ki = 459.8 nM
|
|
|
|
CP0410896
|
N-[11-(3-hydroxy-5-pentylphenoxy)undecyl]cyclopropanecarboxamide
Show/Hide
|
C26H43NO3
|
1
|
| 1 |
Ki = 460 nM
|
|
|
|
CP0462464
|
N-(3-pentyl-1,3-benzothiazol-2-ylidene)-3-(trifluoromethyl)benzamide
Show/Hide
|
C20H19F3N2OS
|
1
|
| 1 |
Ki = 460 nM
|
|
|
|
CP0444415
|
11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acidcyclopropylmethyl-amide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 470 nM
|
|
|
|
CP0434010
|
N-cycloheptyl-2-phenylmethoxypyridine-3-carboxamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
Ki = 481 nM
|
|
|
|
CP0527080
|
1-(2,4-Difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-Nhexyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H28F2N4O
|
1
|
| 1 |
Ki = 487.3 nM
|
|
|
|
CP0465950
|
1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-pentyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H26Cl2N4O
|
1
|
| 1 |
Ki = 495.3 nM
|
|
|
|
CP0425251
|
methyl 4-ethyl-2-[(4-fluorobenzoyl)amino]-5-methylthiophene-3-carboxylate
Show/Hide
|
C16H16FNO3S
|
1
|
| 1 |
Ki = 495.77 nM
|
|
|
|
CP0391306
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-[4-(3,3,3-trifluoropropylsulfonyl)piperazin-1-yl]purine
Show/Hide
|
C24H21Cl2F3N6O2S
|
1
|
| 1 |
Ki = 500 nM
|
|
|
|
CP0552881
|
6-(4-butylsulfonylpiperazin-1-yl)-8-(2-chlorophenyl)-9-(4-chlorophenyl)purine
Show/Hide
|
C25H26Cl2N6O2S
|
1
|
| 1 |
Ki = 500 nM
|
|
|
|
CP0537683
|
2-(1,1-dioxo-1,4-thiazinan-4-yl)-1-(9-pentylcarbazol-3-yl)ethanone
Show/Hide
|
C23H28N2O3S
|
1
|
| 1 |
Ki = 502 nM
|
|
|
|
CP0449624
|
[9-(2-chloroethyl)carbazol-3-yl]-piperidin-1-ylmethanone
Show/Hide
|
C20H21ClN2O
|
1
|
| 1 |
Ki = 519 nM
|
|
|
|
CP0522995
|
piperidin-1-yl-(9-propylcarbazol-3-yl)methanone
Show/Hide
|
C21H24N2O
|
1
|
| 1 |
Ki = 521 nM
|
|
|
|
CP0466293
|
[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-(thian-4-yl)methanone
Show/Hide
|
C27H26Cl2N6OS
|
1
|
| 1 |
Ki = 530 nM
|
|
|
|
CP0555103
|
N-(1,3-dihydroxypropan-2-yl)-11-(3-hydroxy-5-pentylphenoxy)undecanamide
Show/Hide
|
C25H43NO5
|
1
|
| 1 |
Ki = 540 nM
|
|
|
|
CP0395713
|
2-ethyl-5-methyl-1-phenyl-N-(1-phenylethyl)pyrrole-3-carboxamide
Show/Hide
|
C22H24N2O
|
1
|
| 1 |
Ki = 540.1 nM
|
|
|
|
CP0395712
|
2,5-dimethyl-1-phenyl-N-(1-phenylethyl)pyrrole-3-carboxamide
Show/Hide
|
C21H22N2O
|
1
|
| 1 |
Ki = 546.44 nM
|
|
|
|
CP0565978
|
3-(1-adamantyl)-6,6-dimethylbenzo[c]chromene-1,9-diol
Show/Hide
|
C25H28O3
|
1
|
| 1 |
Ki = 551 nM
|
|
|
|
CP0430953
|
N-[(2-bromo-3,4,5-trimethoxyphenyl)methyl]-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C27H27BrCl2N4O4
|
1
|
| 1 |
Ki = 553 nM
|
|
|
|
CP0416055
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-phenylpropan-1-one
Show/Hide
|
C30H26Cl2N6O
|
1
|
| 1 |
Ki = 560 nM
|
|
|
|
CP0552965
|
1-(3-methoxyphenyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
|
C28H36N2O3
|
1
|
| 1 |
Ki = 562 nM
|
|
|
|
CP0561262
|
16-ethyl-12,12-dimethyl-8-(2-methyloctan-2-yl)-3,11-dioxa-15,16-diazatetracyclo[8.7.0.02,7.013,17]heptadeca-1(10),2(7),8,13(17),14-pentaene
Show/Hide
|
C26H38N2O2
|
1
|
| 1 |
Ki = 563.8 nM
|
|
|
|
CP0435742
|
N-(4-methylcyclohexyl)-2-oxo-1-propylpyridine-3-carboxamide
Show/Hide
|
C16H24N2O2
|
1
|
| 1 |
Ki = 583 nM
|
|
|
|
CP0395707
|
2,5-dimethyl-1-phenyl-N-(2-phenylethyl)pyrrole-3-carboxamide
Show/Hide
|
C21H22N2O
|
1
|
| 1 |
Ki = 584.17 nM
|
|
|
|
CP0502928
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-phenylmethanone
Show/Hide
|
C22H24O4
|
1
|
| 1 |
Ki = 587 nM
|
|
|
|
CP0395644
|
N-(4-methylcyclohexyl)-2-phenylmethoxypyridine-3-carboxamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
Ki = 594 nM
|
|
|
|
CP0553772
|
N-(1,3-dihydroxypropan-2-yl)-11-(3-methoxy-5-pentylphenoxy)undecanamide
Show/Hide
|
C26H45NO5
|
1
|
| 1 |
Ki = 597.6 nM
|
|
|
|
CP0487337
|
piperidin-1-yl-[9-(pyridin-3-ylmethyl)carbazol-3-yl]methanone
Show/Hide
|
C24H23N3O
|
1
|
| 1 |
Ki = 600 nM
|
|
|
|
CP0455587
|
3-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-1-methyl-1-(2-methylpropyl)urea
Show/Hide
|
C28H31Cl2N7O
|
1
|
| 1 |
Ki = 600 nM
|
|
|
|
CP0388378
|
N-[(2-bromo-3,4,5-trimethoxyphenyl)methyl]-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C25H23BrCl2N4O4
|
1
|
| 1 |
Ki = 609 nM
|
|
|
|
CP0466294
|
[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-(2,3-dihydro-1,4-benzodioxin-3-yl)methanone
Show/Hide
|
C30H24Cl2N6O3
|
1
|
| 1 |
Ki = 610 nM
|
|
|
|
CP0416547
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-cyclohexylpiperazine-1-carboxamide
Show/Hide
|
C28H29Cl2N7O
|
1
|
| 1 |
Ki = 620 nM
|
|
|
|
CP0386990
|
methyl 2-[(4-chlorobenzoyl)amino]-4-ethyl-5-methylthiophene-3-carboxylate
Show/Hide
|
C16H16ClNO3S
|
1
|
| 1 |
Ki = 621 nM
|
|
|
|
CP0447836
|
3-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-1-methyl-1-propylurea
Show/Hide
|
C27H29Cl2N7O
|
1
|
| 1 |
Ki = 630 nM
|
|
|
|
CP0493784
|
2-(4-Methylphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
|
C30H29NO
|
1
|
| 1 |
Ki = 650 nM
|
|
|
|
CP0400887
|
N-[11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecyl]cyclopropanecarboxamide
Show/Hide
|
C30H51NO3
|
1
|
| 1 |
Ki = 650 nM
|
|
|
|
CP0390567
|
N-[2-(2,4-dichlorophenyl)ethyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C23H18Cl2F2N4O
|
1
|
| 1 |
Ki = 667 nM
|
|
|
|
CP0511226
|
(6aR,9S,10aR)-3-(1-adamantyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-1,9-diol
Show/Hide
|
C25H34O3
|
1
|
| 1 |
Ki = 671.8 nM
|
|
|
|
CP0567079
|
11-(3-hydroxy-5-pentylphenoxy)-N-piperidin-1-ylundecanamide
Show/Hide
|
C27H46N2O3
|
1
|
| 1 |
Ki = 677.8 nM
|
|
|
|
CP0400949
|
2-ethyl-5-methyl-1-phenyl-N-(2-phenylethyl)pyrrole-3-carboxamide
Show/Hide
|
C22H24N2O
|
1
|
| 1 |
Ki = 718.2 nM
|
|
|
|
CP0439162
|
N-[2-(2,4-dichlorophenyl)ethyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H22Cl2F2N4O
|
1
|
| 1 |
Ki = 721 nM
|
|
|
|
CP0495252
|
butyl 2-[(6aR,9S,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]acetate
Show/Hide
|
C21H30O5
|
1
|
| 1 |
Ki = 733 nM
|
|
|
|
CP0390568
|
N-[(2-bromo-3,4,5-trimethoxyphenyl)methyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C25H23BrF2N4O4
|
1
|
| 1 |
Ki = 739 nM
|
|
|
|
CP0541218
|
3-[(4-methylpiperazin-1-yl)methyl]-9-pentylcarbazole
Show/Hide
|
C23H31N3
|
1
|
| 1 |
Ki = 740 nM
|
|
|
|
CP0416507
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-cyclopentylpiperazine-1-carboxamide
Show/Hide
|
C27H27Cl2N7O
|
1
|
| 1 |
Ki = 740 nM
|
|
|
|
CP0547413
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(cyclohexylmethyl)piperazine-1-carboxamide
Show/Hide
|
C29H31Cl2N7O
|
1
|
| 1 |
Ki = 740 nM
|
|
|
|
CP0482402
|
1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(cyclohexylsulfamoyl)-4-methylpiperidin-4-amine
Show/Hide
|
C29H33Cl2N7O2S
|
1
|
| 1 |
Ki = 740 nM
|
|
|
|
CP0395392
|
N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-ethylpyrazole-3-carboxamide
Show/Hide
|
C24H28Cl2N4O
|
1
|
| 1 |
Ki = 753.8 nM
|
|
|
|
CP0444362
|
5-benzyl-2-cyclohexyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one
Show/Hide
|
C23H23N3O
|
1
|
| 1 |
Ki = 790 nM
|
|
|
|
CP0376651
|
N-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C21H15Cl3N4O
|
1
|
| 1 |
Ki = 790 nM
|
|
|
|
CP0453834
|
N-[(4-chlorophenyl)methyl]-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C24H21Cl3N4O
|
1
|
| 1 |
Ki = 790 nM
|
|
|
|
CP0493783
|
2-(4-Nitrophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
|
C29H26N2O3
|
1
|
| 1 |
Ki = 790 nM
|
|
|
|
CP0524192
|
2-(4-Methoxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
|
C30H29NO2
|
1
|
| 1 |
Ki = 790 nM
|
|
|
|
CP0418900
|
1,3-dihydroxypropan-2-yl 11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecanoate
Show/Hide
|
C29H50O6
|
1
|
| 1 |
Ki = 790 nM
|
|
|
|
CP0492411
|
1,3-dihydroxypropan-2-yl 8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]octanoate
Show/Hide
|
C26H44O6
|
1
|
| 1 |
Ki = 790 nM
|
|
|
|
CP0432135
|
N-cycloheptyl-1-(2-morpholin-4-ylethyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C19H29N3O3
|
1
|
| 1 |
Ki = 790 nM
|
|
|
|
CP0465953
|
N-butyl-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C19H20Cl2N4O
|
1
|
| 1 |
Ki = 795.7 nM
|
|
|
|
CP0400439
|
1,3-dihydroxypropan-2-yl 12-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]dodecanoate
Show/Hide
|
C30H52O6
|
1
|
| 1 |
Ki = 800 nM
|
|
|
|
CP0446052
|
ethyl 2-(naphthalen-1-ylsulfonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C21H21NO4S2
|
1
|
| 1 |
Ki = 800 nM
|
|
|
|
CP0483303
|
US9422235, 39
Show/Hide
|
C16H16F2N2O2S
|
1
|
| 1 |
Ki = 800 nM
|
|
|
|
CP0533214
|
N-(1,3-dihydroxypropan-2-yl)-8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]octanamide
Show/Hide
|
C26H45NO5
|
1
|
| 1 |
Ki = 814.8 nM
|
|
|
|
CP0428969
|
(9-heptylcarbazol-3-yl)-piperidin-1-ylmethanone
Show/Hide
|
C25H32N2O
|
1
|
| 1 |
Ki = 827 nM
|
|
|
|
CP0494513
|
3-[11-(benzylamino)undecoxy]-5-pentylphenol
Show/Hide
|
C29H45NO2
|
1
|
| 1 |
Ki = 830 nM
|
|
|
|
CP0386992
|
methyl 4-(adamantane-1-carbonylamino)-1-methylpyrazole-3-carboxylate
Show/Hide
|
C17H23N3O3
|
1
|
| 1 |
Ki = 845.42 nM
|
|
|
|
CP0501760
|
1-(2-chlorophenyl)-2-(4-methoxyphenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C26H28ClN3O2
|
1
|
| 1 |
Ki = 850 nM
|
|
|
|
CP0548533
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-propylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C24H24Cl2N6O2S
|
1
|
| 1 |
Ki = 850 nM
|
|
|
|
CP0467435
|
1,3-dihydroxypropan-2-yl 11-(3-hydroxy-5-pentylphenoxy)undecanoate
Show/Hide
|
C25H42O6
|
1
|
| 1 |
Ki = 870 nM
|
|
|
|
CP0453826
|
N-cyclopentyl-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H24F2N4O
|
1
|
| 1 |
Ki = 900 nM
|
|
|
|
CP0415324
|
6-Bromo-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid cyclohexylamide
Show/Hide
|
C21H27BrN2O2
|
1
|
| 1 |
Ki = 900 nM
|
|
|
|
CP0419835
|
2-[6-(3-hydroxy-5-pentylphenoxy)hexoxy]propane-1,3-diol
Show/Hide
|
C20H34O5
|
1
|
| 1 |
Ki = 910 nM
|
|
|
|
CP0436242
|
(6aR,10aR)-9-(acetyloxymethyl)-1-hydroxy-6,6-dimethyl-3-pentyl-6a,7,8,10a-tetrahydrobenzo[c]chromene-2-carboxylic acid
Show/Hide
|
C24H32O6
|
1
|
| 1 |
Ki = 912 nM
|
|
|
|
CP0432133
|
N-cyclohexyl-2-phenylmethoxypyridine-3-carboxamide
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 916 nM
|
|
|
|
CP0453832
|
N-[(4-chlorophenyl)methyl]-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H17Cl3N4O
|
1
|
| 1 |
Ki = 940 nM
|
|
|
|
CP0859209
|
(Z)-2-(3-(2,4-Dichlorobenzyloxy)benzylidene)-6,7-dihydro-2Himidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H16Cl2N2O2S
|
1
|
| 1 |
Ki = 950 nM
|
|
|
|
CP0455325
|
7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]-1H-quinoline-3-carboxamide
Show/Hide
|
C20H23FN2O2
|
1
|
| 1 |
Ki = 957.1 nM
|
|
|
|
CP0902322
|
5-acetyl-1-(2-diethylaminoethyl)-2-(4-ethoxybenzyl)benzimidazole
Show/Hide
|
C24H31N3O2
|
1
|
| 1 |
Ki = 960 nM
|
|
|
|
CP0898591
|
(Z)-2-(3-(2-Chlorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H19ClN2O2S
|
1
|
| 1 |
Ki = 980 nM
|
|
|
|
CP0389941
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-propan-2-ylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C24H24Cl2N6O2S
|
1
|
| 1 |
Ki = 980 nM
|
|
|
|
CP0396584
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-ethylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C23H22Cl2N6O2S
|
1
|
| 1 |
Ki = 980 nM
|
|
|
|
CP0902326
|
2-[(3,4-Dichloro)benzyl]-1-[(2-dimethylamino)ethyl]-5-trifluoromethylbenzimidazole
Show/Hide
|
C19H18Cl2F3N3
|
1
|
| 1 |
Ki = 980 nM
|
|
|
|
CP0035672
|
dibenzothiazepine, 12h
Show/Hide
|
C24H20ClFN2OS
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0472488
|
US8846730, 15
Show/Hide
|
C27H36F3N3O3S
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0466477
|
5-methoxy-3-(2-methoxybenzyl)-7-methyl-2H-chromen-2-one
Show/Hide
|
C19H18O4
|
1
|
| 1 |
Ki = 1030 nM
|
|
|
|
CP0382824
|
N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-benzothiazole-2-carboxamide
Show/Hide
|
C18H16N2OS
|
1
|
| 1 |
Ki = 1060 nM
|
|
|
|
CP0431071
|
ethyl 4-[5-(2-chlorophenyl)-2-(2,4-dimethylphenyl)pyrazole-3-carbonyl]piperazine-1-carboxylate
Show/Hide
|
C25H27ClN4O3
|
1
|
| 1 |
Ki = 1069 nM
|
|
|
|
CP0482765
|
methyl 4-(adamantane-1-carbonylamino)-2-methylpyrazole-3-carboxylate
Show/Hide
|
C17H23N3O3
|
1
|
| 1 |
Ki = 1081.88 nM
|
|
|
|
CP0383283
|
N-(1-adamantyl)-2-(5-bromo-1-prop-2-enylindol-3-yl)acetamide
Show/Hide
|
C23H27BrN2O
|
1
|
| 1 |
Ki = 1090 nM
|
|
|
|
CP0388958
|
1-(9-pentylcarbazol-3-yl)-2-piperidin-1-ylethanone
Show/Hide
|
C24H30N2O
|
1
|
| 1 |
Ki = 1093 nM
|
|
|
|
CP0501759
|
1-(2-chlorophenyl)-2-(4-chlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C25H25Cl2N3O
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0486202
|
1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(2-hydroxycyclohexyl)imidazole-4-carboxamide
Show/Hide
|
C22H20Cl3N3O2
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0390566
|
N-cyclopentyl-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C20H20F2N4O
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0542696
|
2-(4-Hydroxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
|
C29H27NO2
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0484112
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-[(2-fluorophenyl)methyl]urea
Show/Hide
|
C31H28Cl2FN7O
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0849167
|
(Z)-2-(3-(Benzyloxy)benzylidene)-6,7-dihydro-2H-imidazo-[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H18N2O2S
|
1
|
| 1 |
Ki = 1110 nM
|
|
|
|
CP0400477
|
2-[6-(4-hexyl-3-hydroxyphenoxy)hexoxy]propane-1,3-diol
Show/Hide
|
C21H36O5
|
1
|
| 1 |
Ki = 1130 nM
|
|
|
|
CP0500042
|
1-(2,4-Dichlorophenyl)-N-isopropyl-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C18H18Cl2N4O
|
1
|
| 1 |
Ki = 1132.4 nM
|
|
|
|
CP0456682
|
2-[8-(3-hydroxy-5-pentylphenoxy)octoxy]propane-1,3-diol
Show/Hide
|
C22H38O5
|
1
|
| 1 |
Ki = 1160 nM
|
|
|
|
CP0498367
|
N-(1-adamantyl)-6-bromo-2-butyl-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C24H29BrN2O2
|
1
|
| 1 |
Ki = 1180 nM
|
|
|
|
CP0435620
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide
Show/Hide
|
C25H19Cl2N3O2
|
1
|
| 1 |
Ki = 1200 nM
|
|
|
|
CP0376649
|
N-[2-(4-chlorophenyl)ethyl]-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C23H19Cl3N4O
|
1
|
| 1 |
Ki = 1200 nM
|
|
|
|
CP0372348
|
2-(4-Aminophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
|
C29H28N2O
|
1
|
| 1 |
Ki = 1200 nM
|
|
|
|
CP0386993
|
methyl 2-(adamantane-1-carbonylamino)pyridine-3-carboxylate
Show/Hide
|
C18H22N2O3
|
1
|
| 1 |
Ki = 1220.19 nM
|
|
|
|
CP0372226
|
dibenzothiazepine, 12c
Show/Hide
|
C26H22ClF2N3OS
|
1
|
| 1 |
Ki = 1258.93 nM
|
|
|
|
CP0376646
|
N-[2-(3,4-dichlorophenyl)ethyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C23H18Cl2F2N4O
|
1
|
| 1 |
Ki = 1291 nM
|
|
|
|
CP0417664
|
2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C25H24Cl3N3O
|
1
|
| 1 |
Ki = 1300 nM
|
|
|
|
CP0479506
|
2-(4-bromophenyl)-N-(3,3-diphenylpropyl)acetamide
Show/Hide
|
C23H22BrNO
|
1
|
| 1 |
Ki = 1300 nM
|
|
|
|
CP0373467
|
(6aR,9S,10aR)-6,6-Dimethyl-3-(2-oxa-tricyclo[3.3.1.1*3,7*]dec-1-yl)-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
|
C24H32O4
|
1
|
| 1 |
Ki = 1300 nM
|
|
|
|
CP0466291
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-[1-(trifluoromethyl)cyclopentyl]piperazine-1-carboxamide
Show/Hide
|
C28H26Cl2F3N7O
|
1
|
| 1 |
Ki = 1300 nM
|
|
|
|
CP0466295
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(2-fluorophenyl)piperazine-1-carboxamide
Show/Hide
|
C28H22Cl2FN7O
|
1
|
| 1 |
Ki = 1300 nM
|
|
|
|
CP0533012
|
ethyl 3-[3-(piperidine-1-carbonyl)carbazol-9-yl]propanoate
Show/Hide
|
C23H26N2O3
|
1
|
| 1 |
Ki = 1313 nM
|
|
|
|
CP0425252
|
methyl 2-(adamantane-1-carbonylamino)thiophene-3-carboxylate
Show/Hide
|
C17H21NO3S
|
1
|
| 1 |
Ki = 1324.12 nM
|
|
|
|
CP0078199
|
(4-methoxyphenyl)-[1-(oxan-4-ylmethyl)-5-propoxyindol-3-yl]methanone
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 1350 nM
|
|
|
|
CP0395735
|
ethyl 9-pentylpyrido[3,4-b]indole-3-carboxylate
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
Ki = 1367 nM
|
|
|
|
CP0548838
|
N-(1,3-dihydroxypropan-2-yl)-11-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
|
C30H53NO5
|
1
|
| 1 |
Ki = 1371.2 nM
|
|
|
|
CP0428976
|
pyridin-4-ylmethyl 9-pentylcarbazole-3-carboxylate
Show/Hide
|
C24H24N2O2
|
1
|
| 1 |
Ki = 1392 nM
|
|
|
|
CP0509078
|
2-chloro-N-(3,3-diphenylpropyl)-2,2-diphenylacetamide
Show/Hide
|
C29H26ClNO
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0043807
|
1,3-dihydroxypropan-2-yl (5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoate
Show/Hide
|
C23H38O4
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0432932
|
12-(2-hexyl-5-hydroxy-phenoxy)-dodecanoic acid(2-hydroxy-ethyl)-amide
Show/Hide
|
C26H45NO4
|
1
|
| 1 |
Ki = 1420 nM
|
|
|
|
CP0563451
|
1-(2,4-dichlorophenyl)-9-methoxy-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C28H34Cl2N2O2
|
1
|
| 1 |
Ki = 1493 nM
|
|
|
|
CP0380260
|
1-(2,4-Dichlorophenyl)-4-methyl-N-propyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C18H18Cl2N4O
|
1
|
| 1 |
Ki = 1496.2 nM
|
|
|
|
CP0543211
|
3-[9-[[(2R)-1-hydroxypropan-2-yl]amino]nonoxy]-5-pentylphenol
Show/Hide
|
C23H41NO3
|
1
|
| 1 |
Ki = 1520 nM
|
|
|
|
CP0514675
|
3-(2-Chlorobenzyl)-5-methoxy-7-methyl-2H-chromen-2-one
Show/Hide
|
C18H15ClO3
|
1
|
| 1 |
Ki = 1540 nM
|
|
|
|
CP0499264
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-thiophen-3-ylmethanone
Show/Hide
|
C20H22O4S
|
1
|
| 1 |
Ki = 1551 nM
|
|
|
|
CP0868782
|
(Z)-2-(3-(4-Fluorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H19FN2O2S
|
1
|
| 1 |
Ki = 1560 nM
|
|
|
|
CP0905762
|
2-(2-benzyl-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)-N,N-diethylethanamine
Show/Hide
|
C21H24F3N3
|
1
|
| 1 |
Ki = 1580 nM
|
|
|
|
CP0428987
|
9-pentyl-N-piperidin-1-ylcarbazole-3-carboxamide
Show/Hide
|
C23H29N3O
|
1
|
| 1 |
Ki = 1609 nM
|
|
|
|
CP0919485
|
(1R,2S)-N-Oleoylcyclopropanolamide
Show/Hide
|
C19H37NO2
|
1
|
| 1 |
Ki = 1630 nM
|
|
|
|
CP0454092
|
5-benzyl-7-chloro-2-cyclohexyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one
Show/Hide
|
C23H22ClN3O
|
1
|
| 1 |
Ki = 1640 nM
|
|
|
|
CP0528608
|
11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid (3-methoxy-4-hydroxy-phenyl)-amide
Show/Hide
|
C30H45NO5
|
1
|
| 1 |
Ki = 1650 nM
|
|
|
|
CP0849218
|
(Z)-2-(3-(2,4-dichlorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H18Cl2N2O2S
|
1
|
| 1 |
Ki = 1650 nM
|
|
|
|
CP0427943
|
2-[12-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]dodecoxy]propane-1,3-diol
Show/Hide
|
C30H54O5
|
1
|
| 1 |
Ki = 1670 nM
|
|
|
|
CP0466696
|
methyl 2-(adamantane-1-carbonylamino)-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
Show/Hide
|
C20H25NO5S2
|
1
|
| 1 |
Ki = 1673.74 nM
|
|
|
|
CP0559842
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C22H20Cl2N6O2S
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0395714
|
ethyl 2-(naphthalene-2-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C22H21NO3S
|
1
|
| 1 |
Ki = 1785.22 nM
|
|
|
|
CP0527077
|
1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-Nisopropyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H22Cl2N4O
|
1
|
| 1 |
Ki = 1796.8 nM
|
|
|
|
CP0428675
|
8-(2-hexyl-5-hydroxy-phenoxy)-octanoic acidcyclopropylamide
Show/Hide
|
C23H37NO3
|
1
|
| 1 |
Ki = 1800 nM
|
|
|
|
CP0418048
|
2-(4-bromophenyl)-2-phenyl-N-(3-phenylpropyl)acetamide
Show/Hide
|
C23H22BrNO
|
1
|
| 1 |
Ki = 1800 nM
|
|
|
|
CP0479034
|
(6aR,9R,10aR)-6,6-Dimethyl-3-(2-oxa-6-aza-tricyclo[3.3.1.1*3,7*]dec-6-yl)-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
|
C23H31NO4
|
1
|
| 1 |
Ki = 1800 nM
|
|
|
|
CP0392072
|
1,3-dihydroxypropan-2-yl 8-(2-hexyl-5-hydroxyphenoxy)octanoate
Show/Hide
|
C23H38O6
|
1
|
| 1 |
Ki = 1800 nM
|
|
|
|
CP0432796
|
1,3-dihydroxypropan-2-yl 11-(2-hexyl-5-hydroxyphenoxy)undecanoate
Show/Hide
|
C26H44O6
|
1
|
| 1 |
Ki = 1800 nM
|
|
|
|
CP0900469
|
(Z)-2-(3-(Benzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H20N2O2S
|
1
|
| 1 |
Ki = 1810 nM
|
|
|
|
CP0395642
|
ethyl 4-[3-(cycloheptylcarbamoyl)-2-oxopyridin-1-yl]butanoate
Show/Hide
|
C19H28N2O4
|
1
|
| 1 |
Ki = 1832 nM
|
|
|
|
CP0410859
|
3-pentyl-5-[11-(prop-2-enylamino)undecoxy]phenol
Show/Hide
|
C25H43NO2
|
1
|
| 1 |
Ki = 1850 nM
|
|
|
|
CP0379903
|
3-[11-(cyclopropylamino)undecoxy]-5-pentylphenol
Show/Hide
|
C25H43NO2
|
1
|
| 1 |
Ki = 1890 nM
|
|
|
|
CP0522996
|
pyridin-2-ylmethyl 9-pentylcarbazole-3-carboxylate
Show/Hide
|
C24H24N2O2
|
1
|
| 1 |
Ki = 1927 nM
|
|
|
|
CP0491341
|
N-[2-(3-chloro-4-methoxyphenyl)ethyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C24H21ClF2N4O2
|
1
|
| 1 |
Ki = 1945 nM
|
|
|
|
CP0498789
|
1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-propyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H22Cl2N4O
|
1
|
| 1 |
Ki = 1953.3 nM
|
|
|
|
CP0518083
|
ethyl 2-(benzenesulfonamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C17H19NO4S2
|
1
|
| 1 |
Ki = 1993.94 nM
|
|
|
|
CP0170798
|
(S)-3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide
Show/Hide
|
C23H20Cl2N4O2S
|
2
|
| 1 |
Ki = 1995.26 nM
|
|
|
| 2 |
Ki = 7943 nM
|
|
|
|
CP0391007
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(4-fluorophenyl)piperazine-1-carboxamide
Show/Hide
|
C28H22Cl2FN7O
|
1
|
| 1 |
Ki = 2000 nM
|
|
|
|
CP0529208
|
2-(2-Methoxybenzyl)-3H-benzo[f]chromen-3-one
Show/Hide
|
C21H16O3
|
1
|
| 1 |
Ki = 2060 nM
|
|
|
|
CP0902325
|
N,N-diethyl-2-(2-(4-methoxybenzyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)ethanamine
Show/Hide
|
C22H26F3N3O
|
1
|
| 1 |
Ki = 2070 nM
|
|
|
|
CP0444412
|
11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acid(3-methoxy-4-hydroxy-phenyl)-amide
Show/Hide
|
C31H47NO5
|
1
|
| 1 |
Ki = 2100 nM
|
|
|
|
CP0394001
|
methyl 3-(adamantane-1-carbonylamino)-1H-pyrrole-2-carboxylate
Show/Hide
|
C17H22N2O3
|
1
|
| 1 |
Ki = 2141.79 nM
|
|
|
|
CP0433616
|
(6aR,9S,10S,10aR)-6,6,9-trimethyl-3-pentyl-7,8,10,10a-tetrahydro-6aH-benzo[c]chromene-1,9,10-triol
Show/Hide
|
C21H32O4
|
1
|
| 1 |
Ki = 2143 nM
|
|
|
|
CP0498065
|
5-Methoxy-7-methyl-3-(2-methylbenzyl)-2H-chromen-2-one
Show/Hide
|
C19H18O3
|
1
|
| 1 |
Ki = 2160 nM
|
|
|
|
CP0395253
|
piperidin-1-yl-[9-(3-piperidin-1-ylpropyl)carbazol-3-yl]methanone
Show/Hide
|
C26H33N3O
|
1
|
| 1 |
Ki = 2169 nM
|
|
|
|
CP0434518
|
1-(3,4-dichlorophenyl)-9-methoxy-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C28H34Cl2N2O2
|
1
|
| 1 |
Ki = 2256 nM
|
|
|
|
CP0522362
|
5-(2-morpholinoethyl)-2-phenyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
Ki = 2280 nM
|
|
|
|
CP0384969
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-1H-imidazole-4-carboxamide
Show/Hide
|
C22H21Cl2N3O
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0434259
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C24H25Cl2N3O2
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0528142
|
N-(3,3-diphenylpropyl)-2-hydroxy-2,2-diphenylacetamide
Show/Hide
|
C29H27NO2
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0416595
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-cyclopropylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C24H22Cl2N6O2S
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0508356
|
3-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-1-(2-methoxyethyl)-1-methylurea
Show/Hide
|
C27H29Cl2N7O2
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0501839
|
1-(2,4-Dichlorophenyl)-N-(5-hydroxypentyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H22Cl2N4O2
|
1
|
| 1 |
Ki = 2344.4 nM
|
|
|
|
CP0445847
|
N-(1,3-dihydroxypropan-2-yl)-11-(2-hexyl-5-hydroxyphenoxy)undecanamide
Show/Hide
|
C26H45NO5
|
1
|
| 1 |
Ki = 2370 nM
|
|
|
|
CP0432794
|
2-[10-(4-hexyl-3-hydroxyphenoxy)decoxy]propane-1,3-diol
Show/Hide
|
C25H44O5
|
1
|
| 1 |
Ki = 2390 nM
|
|
|
|
CP0427501
|
8-(4-hexyl-3-hydroxy-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide
Show/Hide
|
C22H37NO4
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0372347
|
2-(4-chlorophenyl)-N-(3,3-diphenylpropyl)acetamide
Show/Hide
|
C23H22ClNO
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0502229
|
2-(4-chlorophenyl)-2-phenyl-N-(3-phenylpropyl)acetamide
Show/Hide
|
C23H22ClNO
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0547412
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-phenylpiperazine-1-carboxamide
Show/Hide
|
C28H23Cl2N7O
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0363620
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-N-[4-(1,2,3,4-tetrahydroacridin-9-ylamino)butyl]benzimidazole-5-carboxamide
Show/Hide
|
C39H47N5O2
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0920451
|
(1S,2S)-N-Oleoylcyclopropanolamide
Show/Hide
|
C19H37NO2
|
1
|
| 1 |
Ki = 2420 nM
|
|
|
|
CP0425249
|
methyl 2-(morpholine-4-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C15H20N2O4S
|
1
|
| 1 |
Ki = 2494.08 nM
|
|
|
|
CP0159380
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-N-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl]benzimidazole-5-carboxamide
Show/Hide
|
C37H43N5O2
|
1
|
| 1 |
Ki = 2500 nM
|
|
|
|
CP0659851
|
(Z)-2-(2,4-dimethoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H16N2O3S
|
1
|
| 1 |
Ki = 2570 nM
|
|
|
|
CP0893067
|
(Z)-3-((3-oxo-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2(3H)-ylidene)methyl)phenyl 4-methylbenzoate
Show/Hide
|
C22H20N2O3S
|
1
|
| 1 |
Ki = 2580 nM
|
|
|
|
CP0398663
|
(S)-N-(2,4-dichlorophenyl)-5-((2-phenylmorpholino)methyl)pyridin-2-amine
Show/Hide
|
C22H21Cl2N3O
|
2
|
| 1 |
Ki = 2650 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0540426
|
tert-butyl N-[3-[3-(piperidine-1-carbonyl)carbazol-9-yl]propyl]carbamate
Show/Hide
|
C26H33N3O3
|
1
|
| 1 |
Ki = 2690 nM
|
|
|
|
CP0394622
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-propyl-1H-imidazole-4-carboxamide
Show/Hide
|
C25H27Cl2N3O2
|
1
|
| 1 |
Ki = 2700 nM
|
|
|
|
CP0500978
|
1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C24H25BrClN3O2
|
1
|
| 1 |
Ki = 2700 nM
|
|
|
|
CP0509567
|
(6aR,9R,10aR)-1,9-Dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-3-carboxylic acid adamantan-2-ylamide
Show/Hide
|
C26H35NO4
|
1
|
| 1 |
Ki = 2700 nM
|
|
|
|
CP0399703
|
3-(2,4-Dimethoxybenzyl)-5-methoxy-7-methyl-2Hchromen-2-one
Show/Hide
|
C20H20O5
|
1
|
| 1 |
Ki = 2780 nM
|
|
|
|
CP0517588
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-[4-(2-methylpropylsulfonyl)piperazin-1-yl]purine
Show/Hide
|
C25H26Cl2N6O2S
|
1
|
| 1 |
Ki = 2800 nM
|
|
|
|
CP0431692
|
3-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-1-propyl-1-(2,2,2-trifluoroethyl)urea
Show/Hide
|
C28H28Cl2F3N7O
|
1
|
| 1 |
Ki = 2800 nM
|
|
|
|
CP0539011
|
US10227332, No. 8
Show/Hide
|
C22H27N3O
|
1
|
| 1 |
Ki = 2833 nM
|
|
|
|
CP0390564
|
N-[2-(3-chloro-4-methoxyphenyl)ethyl]-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C24H21Cl3N4O2
|
1
|
| 1 |
Ki = 2887 nM
|
|
|
|
CP0373773
|
11-(4-hexyl-3-hydroxy-phenoxy)-undecanoic acid cyclopropylmethyl-amide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 2900 nM
|
|
|
|
CP0411062
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-[4-(oxan-4-ylmethylsulfonyl)piperazin-1-yl]purine
Show/Hide
|
C27H28Cl2N6O3S
|
1
|
| 1 |
Ki = 3000 nM
|
|
|
|
CP0416054
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-(oxolan-3-yl)ethanone
Show/Hide
|
C27H26Cl2N6O2
|
1
|
| 1 |
Ki = 3000 nM
|
|
|
|
CP0152980
|
2-[(4-ethoxyphenyl)methyl]-N-ethyl-1-(3-methylbutyl)-N-[4-(1,2,3,4-tetrahydroacridin-9-ylamino)butyl]benzimidazole-5-carboxamide
Show/Hide
|
C41H51N5O2
|
1
|
| 1 |
Ki = 3000 nM
|
|
|
|
CP0443585
|
[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-(1-methylindol-3-yl)methanone
Show/Hide
|
C25H27NO4
|
1
|
| 1 |
Ki = 3006 nM
|
|
|
|
CP0371809
|
CAS_4055807
Show/Hide
|
C26H32N2O4S
|
1
|
| 1 |
Ki = 3100 nM
|
|
|
|
CP0389946
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(2,4-difluorophenyl)piperazine-1-carboxamide
Show/Hide
|
C28H21Cl2F2N7O
|
1
|
| 1 |
Ki = 3200 nM
|
|
|
|
CP0455586
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(cyclopentylmethyl)urea
Show/Hide
|
C29H31Cl2N7O
|
1
|
| 1 |
Ki = 3200 nM
|
|
|
|
CP0379578
|
1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-N-(5-hydroxypentyl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H26Cl2N4O2
|
1
|
| 1 |
Ki = 3200.5 nM
|
|
|
|
CP0877894
|
8alpha-Hydroxy-Delta9-tetrahydrocannabinol
Show/Hide
|
C21H30O3
|
1
|
| 1 |
Ki = 3219 nM
|
|
|
|
CP0877895
|
10beta-Hydroxy-Delta8-tetrahydrocannabinol
Show/Hide
|
C21H30O3
|
1
|
| 1 |
Ki = 3274 nM
|
|
|
|
CP0514674
|
5-Methoxy-3-(3-methoxybenzyl)-7-methyl-2Hchromen-2-one
Show/Hide
|
C19H18O4
|
1
|
| 1 |
Ki = 3370 nM
|
|
|
|
CP0467012
|
ethyl 3-[3-(4-methylpiperazine-1-carbonyl)carbazol-9-yl]propanoate
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
Ki = 3376 nM
|
|
|
|
CP0509784
|
N-[(4-chlorophenyl)methyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H17ClF2N4O
|
1
|
| 1 |
Ki = 3400 nM
|
|
|
|
CP0391003
|
tert-butyl 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazine-1-carboxylate
Show/Hide
|
C26H26Cl2N6O2
|
1
|
| 1 |
Ki = 3400 nM
|
|
|
|
CP0466290
|
cyclobutyl 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazine-1-carboxylate
Show/Hide
|
C26H24Cl2N6O2
|
1
|
| 1 |
Ki = 3400 nM
|
|
|
|
CP0376756
|
N-(1-adamantyl)-8-methoxy-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C21H24N2O3
|
1
|
| 1 |
Ki = 3443 nM
|
|
|
|
CP0453830
|
N-[2-(3-chloro-4-methoxyphenyl)ethyl]-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C26H25Cl3N4O2
|
1
|
| 1 |
Ki = 3483 nM
|
|
|
|
CP0454965
|
5-Methoxy-3-(2-methoxybenzyl)-2H-chromen-2-one
Show/Hide
|
C18H16O4
|
1
|
| 1 |
Ki = 3490 nM
|
|
|
|
CP0434517
|
1-(3,4-dichlorophenyl)-9-ethoxy-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazole
Show/Hide
|
C29H36Cl2N2O2
|
1
|
| 1 |
Ki = 3545 nM
|
|
|
|
CP0556844
|
N-[2-(4-chlorophenyl)ethyl]-9-pentylcarbazole-3-carboxamide
Show/Hide
|
C26H27ClN2O
|
1
|
| 1 |
Ki = 3594 nM
|
|
|
|
CP0522936
|
5-Methoxy-3-(2-methoxybenzyl)-8-methyl-2Hchromen-2-one
Show/Hide
|
C19H18O4
|
1
|
| 1 |
Ki = 3650 nM
|
|
|
|
CP0542581
|
1-(3,4-dichlorophenyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)-9-phenylmethoxychromeno[4,3-c]pyrazole
Show/Hide
|
C34H38Cl2N2O2
|
1
|
| 1 |
Ki = 3740 nM
|
|
|
|
CP0257793
|
6-(2,4-Dichloro-benzyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C32H36Cl2N2O2
|
1
|
| 1 |
Ki = 3881 nM
|
|
|
|
CP0431070
|
1-(1-(4-chlorophenyl)-4-(3-methoxyphenyl)-5-(4-morpholinophenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethanone
Show/Hide
|
C27H27ClN4O3
|
1
|
| 1 |
Ki = 3919 nM
|
|
|
|
CP0378995
|
8-(2-hexyl-5-hydroxy-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide
Show/Hide
|
C22H37NO4
|
1
|
| 1 |
Ki = 3940 nM
|
|
|
|
CP0432937
|
12-(4-hexyl-3-hydroxy-phenoxy)-dodecanoic acidcyclopropylamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 3940 nM
|
|
|
|
CP0379559
|
CAS_22422466
Show/Hide
|
C24H27FN2O4S
|
1
|
| 1 |
Ki = 4000 nM
|
|
|
|
CP0152979
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-N-[5-(1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]benzimidazole-5-carboxamide
Show/Hide
|
C40H49N5O2
|
1
|
| 1 |
Ki = 4000 nM
|
|
|
|
CP0659892
|
(Z)-2-(3-(4-Chlorobenzyloxy)benzylidene)-6,7-dihydro-2H-imidazo-[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H17ClN2O2S
|
1
|
| 1 |
Ki = 4030 nM
|
|
|
|
CP0659893
|
(Z)-2-(3-(4-chlorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H19ClN2O2S
|
1
|
| 1 |
Ki = 4150 nM
|
|
|
|
CP0042287
|
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H19Cl2IN4O2
|
1
|
| 1 |
Ki = 4200 nM
|
|
|
|
CP0391005
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(3,4-difluorophenyl)piperazine-1-carboxamide
Show/Hide
|
C28H21Cl2F2N7O
|
1
|
| 1 |
Ki = 4200 nM
|
|
|
|
CP0375124
|
3-Benzyl-5-isopropyl-8-methylchromen-2-one
Show/Hide
|
C20H20O2
|
1
|
| 1 |
Ki = 4270 nM
|
|
|
|
CP0152986
|
2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-[6-(1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]benzimidazole-5-carboxamide
Show/Hide
|
C40H49N5O2
|
1
|
| 1 |
Ki = 4300 nM
|
|
|
|
CP0389943
|
cyclobutylmethyl 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazine-1-carboxylate
Show/Hide
|
C27H26Cl2N6O2
|
1
|
| 1 |
Ki = 4600 nM
|
|
|
|
CP0493585
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-cyclohexylurea
Show/Hide
|
C29H31Cl2N7O
|
1
|
| 1 |
Ki = 4600 nM
|
|
|
|
CP0510047
|
5-Methoxy-7-methyl-3-(4-methylbenzyl)-2H-chromen-2-one
Show/Hide
|
C19H18O3
|
1
|
| 1 |
Ki = 4760 nM
|
|
|
|
CP0528170
|
CAS_22422464
Show/Hide
|
C24H27ClN2O4S
|
1
|
| 1 |
Ki = 4800 nM
|
|
|
|
CP0461991
|
2,3-dihydroxypropyl 11-(2-hexyl-5-hydroxyphenoxy)undecanoate
Show/Hide
|
C26H44O6
|
1
|
| 1 |
Ki = 4820 nM
|
|
|
|
CP0371807
|
CAS_3340785
Show/Hide
|
C23H32N2O4S
|
1
|
| 1 |
Ki = 4900 nM
|
|
|
|
CP0509860
|
3-tert-butyl-1-isopropyl-1-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]quinoxalin-5(4H)-yl)-2-oxoethyl)urea
Show/Hide
|
C28H34N4O3
|
1
|
| 1 |
Ki = 4953 nM
|
|
|
|
CP0402379
|
(6aR,9S,10aR)-6,6-Dimethyl-3-(2-oxa-6-aza-tricyclo[3.3.1.1*3,7*]dec-6-ylmethyl)-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
|
C24H33NO4
|
1
|
| 1 |
Ki = 5000 nM
|
|
|
|
CP0389945
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-3,3-dimethylbutan-1-one
Show/Hide
|
C27H28Cl2N6O
|
1
|
| 1 |
Ki = 5000 nM
|
|
|
|
CP0526326
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-piperidin-1-ylethanone
Show/Hide
|
C28H29Cl2N7O
|
1
|
| 1 |
Ki = 5000 nM
|
|
|
|
CP0152985
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-N-[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]benzimidazole-5-carboxamide
Show/Hide
|
C38H45N5O2
|
1
|
| 1 |
Ki = 5000 nM
|
|
|
|
CP0456605
|
dibenzothiazepine, 12g
Show/Hide
|
C24H21ClN2OS
|
1
|
| 1 |
Ki = 5011.87 nM
|
|
|
|
CP0435608
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide
Show/Hide
|
C25H19Cl2N3O2
|
1
|
| 1 |
Ki = 5100 nM
|
|
|
|
CP0522937
|
3-(2-Hydroxybenzyl)-5-methoxy-7-methyl-2Hchromen-2-one
Show/Hide
|
C18H16O4
|
1
|
| 1 |
Ki = 5240 nM
|
|
|
|
CP0394621
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C22H21Cl2N3O2
|
1
|
| 1 |
Ki = 5300 nM
|
|
|
|
CP0859481
|
(Z)-2-(biphenyl-4-ylmethylene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C20H18N2OS
|
1
|
| 1 |
Ki = 5430 nM
|
|
|
|
CP0529207
|
5-Isopropyl-3-(2-methoxybenzyl)-7-methyl-2Hchromen-2-one
Show/Hide
|
C21H22O3
|
1
|
| 1 |
Ki = 5670 nM
|
|
|
|
CP0467642
|
5-Methoxy-3-(4-methoxybenzyl)-7-methylchromen-2-one
Show/Hide
|
C19H18O4
|
1
|
| 1 |
Ki = 5810 nM
|
|
|
|
CP0394013
|
5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-phenethylbenzofuran-2-carboxamide
Show/Hide
|
C25H30N2O4S
|
1
|
| 1 |
Ki = 6000 nM
|
|
|
|
CP0467955
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C21H19Cl2N3O2
|
1
|
| 1 |
Ki = 6300 nM
|
|
|
|
CP0465926
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] 3-formamidopropanoate
Show/Hide
|
C26H47NO5
|
1
|
| 1 |
Ki = 6400 nM
|
|
|
|
CP0489575
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(4-fluorophenyl)urea
Show/Hide
|
C29H24Cl2FN7O
|
1
|
| 1 |
Ki = 6500 nM
|
|
|
|
CP0371806
|
CAS_15991674
Show/Hide
|
C24H28N2O4S
|
1
|
| 1 |
Ki = 6600 nM
|
|
|
|
CP0398973
|
CAS_11496202
Show/Hide
|
C25H30N2O4S
|
1
|
| 1 |
Ki = 6600 nM
|
|
|
|
CP0152982
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-N-[2-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyldisulfanyl]ethyl]benzimidazole-5-carboxamide
Show/Hide
|
C39H47N5O2S2
|
1
|
| 1 |
Ki = 6800 nM
|
|
|
|
CP0416548
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-pyridin-2-ylpiperazine-1-carboxamide
Show/Hide
|
C27H22Cl2N8O
|
1
|
| 1 |
Ki = 7100 nM
|
|
|
|
CP0165128
|
2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-[5-(1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]benzimidazole-5-carboxamide
Show/Hide
|
C39H47N5O2
|
1
|
| 1 |
Ki = 7300 nM
|
|
|
|
CP0394012
|
CAS_15998702
Show/Hide
|
C22H30N2O4S
|
1
|
| 1 |
Ki = 7400 nM
|
|
|
|
CP0489860
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-1-formylpyrrolidine-2-carboxylate
Show/Hide
|
C28H49NO5
|
1
|
| 1 |
Ki = 7400 nM
|
|
|
|
CP0484113
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(4,4-difluoro-1-methylcyclohexyl)urea
Show/Hide
|
C30H31Cl2F2N7O
|
1
|
| 1 |
Ki = 7500 nM
|
|
|
|
CP0420623
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(cyclohexylmethyl)urea
Show/Hide
|
C30H33Cl2N7O
|
1
|
| 1 |
Ki = 7600 nM
|
|
|
|
CP0394718
|
1,3-dihydroxypropan-2-yl 8-(3-hydroxy-5-pentylphenoxy)octanoate
Show/Hide
|
C22H36O6
|
1
|
| 1 |
Ki = 7870 nM
|
|
|
|
CP0428008
|
1,3-dihydroxypropan-2-yl 8-(4-hexyl-3-hydroxyphenoxy)octanoate
Show/Hide
|
C23H38O6
|
1
|
| 1 |
Ki = 7870 nM
|
|
|
|
CP0440291
|
1,3-dihydroxypropan-2-yl 11-(4-hexyl-3-hydroxyphenoxy)undecanoate
Show/Hide
|
C26H44O6
|
1
|
| 1 |
Ki = 7870 nM
|
|
|
|
CP0501752
|
7-amino-1-benzyl-N-cyclohexyl-4-oxo-1,4-dihydro-1,8-naphthyridine-2-carboxamide
Show/Hide
|
C22H24N4O2
|
1
|
| 1 |
Ki = 7900 nM
|
|
|
|
CP0427498
|
11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acid[2-(3,4-dihydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C31H47NO5
|
1
|
| 1 |
Ki = 7900 nM
|
|
|
|
CP0372352
|
N-(3,3-diphenylpropyl)-2,2-diphenylacetamide
Show/Hide
|
C29H27NO
|
1
|
| 1 |
Ki = 7900 nM
|
|
|
|
CP0432136
|
N-cyclohexyl-1-(2-morpholin-4-ylethyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C18H27N3O3
|
1
|
| 1 |
Ki = 7900 nM
|
|
|
|
CP0418896
|
2,3-dihydroxypropyl 11-(3-hydroxy-5-pentylphenoxy)undecanoate
Show/Hide
|
C25H42O6
|
1
|
| 1 |
Ki = 7910 nM
|
|
|
|
CP0465176
|
2-(4-chlorophenyl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C26H25Cl3N2O
|
1
|
| 1 |
Ki = 8300 nM
|
|
|
|
CP0385440
|
(6aR,9R,10aR)-1,9-Dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C26H35NO4
|
1
|
| 1 |
Ki = 8700 nM
|
|
|
|
CP0495575
|
3-(4-Chlorobenzyl)-5-methoxy-7-methyl-2H-chromen-2-one
Show/Hide
|
C18H15ClO3
|
1
|
| 1 |
Ki = 9390 nM
|
|
|
|
CP0399367
|
CAS_4621779
Show/Hide
|
C21H30N2O4S
|
1
|
| 1 |
Ki = 9400 nM
|
|
|
|
CP0356322
|
2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-N-[6-(1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]benzimidazole-5-carboxamide
Show/Hide
|
C41H51N5O2
|
1
|
| 1 |
Ki = 9600 nM
|
|
|
|
CP0440571
|
CAS_15998061
Show/Hide
|
C26H32N2O5S
|
1
|
| 1 |
Ki = 9900 nM
|
|
|
|
CP0035557
|
(Z)-N-(2-hydroxyethyl)octadec-9-enamide
Show/Hide
|
C20H39NO2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0049976
|
(6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methylnon-6-enamide
Show/Hide
|
C18H27NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0395030
|
cyclopropanolamide, rac-10c
Show/Hide
|
C19H37NO2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0493725
|
cyclopropanolamide, rac-9c
Show/Hide
|
C19H37NO2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0058220
|
(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl (2S)-2-formamido-4-methylpentanoate
Show/Hide
|
C29H53NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0423365
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-formamido-3-methylpentanoate
Show/Hide
|
C29H53NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0423366
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] 2-acetamidoacetate
Show/Hide
|
C26H47NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0433844
|
5-oxo-L-Proline-(1S)-1-[[(2S,3S)-3-hexyl-4-oxo-2-oxetanyl]methyl]dodecyl Ester
Show/Hide
|
C27H47NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0439729
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-formamido-3-methylbutanoate
Show/Hide
|
C28H51NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0485042
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-formamidopropanoate
Show/Hide
|
C26H47NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0485066
|
(1R)-1-{[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]methyl}dodecyl N-formylglycinate
Show/Hide
|
C25H45NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0506288
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-acetamido-3-methylbutanoate
Show/Hide
|
C29H53NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0511846
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-acetamido-3-methylpentanoate
Show/Hide
|
C30H55NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0417551
|
N-benzhydryl-5-(3,5-dimethylpiperidin-1-yl)sulfonyl-2-fluorobenzamide
Show/Hide
|
C27H29FN2O3S
|
1
|
| 1 |
Ki = 10000 nM
|
|
|
|
CP0490713
|
2-(7,7-dimethyl-2-p-tolyl-7,8-dihydro-5H-pyrano[4,3-d]pyrimidin-4-ylthio)-N-(2-methoxyphenyl)propanamide
Show/Hide
|
C26H29N3O3S
|
1
|
| 1 |
Ki = 10000 nM
|
|
|
|
CP0490714
|
N-cyclopropyl-N-[2-[4-(4-methylphenyl)-4H-pyrrolo[1,2-a]quinoxalin-5-yl]-2-oxoethyl]cyclopentanecarboxamide
Show/Hide
|
C29H31N3O2
|
1
|
| 1 |
Ki = 10000 nM
|
|
|
|
CP0507878
|
4-(indolin-1-ylsulfonyl)-N-(2-phenoxyphenyl)benzamide
Show/Hide
|
C27H22N2O4S
|
1
|
| 1 |
Ki = 10000 nM
|
|
|
|
CP0092490
|
2-(2,4-dichlorophenylamino)-4-trifluoromethyl-pyrimidine-5-carboxylic acid N-(tetrahydropyran-4-ylmethyl)amide
Show/Hide
|
C18H17Cl2F3N4O2
|
2
|
| 1 |
Ki > 10000 nM
|
|
|
| 2 |
Ki > 5000 nM
|
|
|
|
CP0374924
|
3-benzyl-8-methoxychromen-2-one
Show/Hide
|
C17H14O3
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0377268
|
3-Benzyl-6-nitrochromen-2-one
Show/Hide
|
C16H11NO4
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0377269
|
6-Methoxy-3-methylchromen-2-one
Show/Hide
|
C11H10O3
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0380662
|
2-Methylbenzo[f]chromen-3-one
Show/Hide
|
C14H10O2
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0393582
|
3-Benzyl-5-methoxy-7-methylchromen-2-one
Show/Hide
|
C18H16O3
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0393608
|
7-methoxy-3-methylchromen-2-one
Show/Hide
|
C11H10O3
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0393611
|
3-Benzylchromen-2-one
Show/Hide
|
C16H12O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0393613
|
3-Benzyl-7-methoxychromen-2-one
Show/Hide
|
C17H14O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0393614
|
5-Isopropyl-3,8-dimethylchromen-2-one
Show/Hide
|
C14H16O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0395520
|
3-Benzyl-8-bromo-5-methoxychromen-2-one
Show/Hide
|
C17H13BrO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0396475
|
8-bromo-6-chloro-3-methylchromen-2-one
Show/Hide
|
C10H6BrClO2
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0396721
|
6-Iodo-3-methyl-chromen-2-one
Show/Hide
|
C10H7IO2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0399693
|
2,2-dimethyl-8-phenyl-2H-chromene-3-carbaldehyde
Show/Hide
|
C18H16O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0431359
|
3-Benzyl-6-iodochromen-2-one
Show/Hide
|
C16H11IO2
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0433057
|
3-Benzyl-6-methoxychromen-2-one
Show/Hide
|
C17H14O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0439564
|
1-(8-bromo-5-methoxy-2-methyl-2H-chromen-3-yl)ethanone
Show/Hide
|
C13H13BrO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0454966
|
8-Methoxy-3-methylchromen-2-one
Show/Hide
|
C11H10O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0454967
|
3-Benzyl-5-methoxychromen-2-one
Show/Hide
|
C17H14O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0456827
|
2-Benzylbenzo[f]chromen-3-one
Show/Hide
|
C20H14O2
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0463757
|
6-Bromo-8-methoxy-3-methylchromen-2-one
Show/Hide
|
C11H9BrO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0466479
|
1-(6-(1,3-dithiolan-2-yl)-2,2-dimethyl-2H-chromen-5-yl) 3-ethyl 2-(3-phenylallylidene)malonate
Show/Hide
|
C28H28O5S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0504198
|
2-(2-hydroxybenzylidene)-2,3,4,4a-tetrahydro-1H-xanthen-1-one
Show/Hide
|
C20H16O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0402381
|
(6aR,9R,10aR)-3-(Adamantan-1-ylaminomethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
|
C26H37NO3
|
1
|
| 1 |
Ki = 10000 nM
|
|
|
|
CP0459053
|
1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-diethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C26H24Cl4N4O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0418897
|
2-[10-(3-hydroxy-5-pentylphenoxy)decoxy]propane-1,3-diol
Show/Hide
|
C24H42O5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0418898
|
2-[12-(3-hydroxy-5-pentylphenoxy)dodecoxy]propane-1,3-diol
Show/Hide
|
C26H46O5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0438030
|
(2S)-3-hydroxy-2-[[(5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoyl]amino]propanoic acid
Show/Hide
|
C23H37NO4
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0193415
|
N-[(3,4-dichlorophenyl)methyl]-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C28H26Cl2N2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0404952
|
1-(4-chlorophenyl)-7-fluoro-4-oxo-N-piperidin-1-ylquinoline-3-carboxamide
Show/Hide
|
C21H19ClFN3O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0498310
|
N-[(3,4-dichlorophenyl)methyl]-4-oxo-1-pentyl-7-phenylquinoline-3-carboxamide
Show/Hide
|
C28H26Cl2N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0525501
|
1-(4-fluorophenyl)-4-oxo-7-phenylsulfanyl-N-piperidin-1-ylquinoline-3-carboxamide
Show/Hide
|
C27H24FN3O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0395645
|
1-(2-hydroxyethyl)-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C15H22N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0435743
|
4-[3-(cycloheptylcarbamoyl)-2-oxopyridin-1-yl]butanoic acid
Show/Hide
|
C17H24N2O4
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0481037
|
1-(3-hydroxypropyl)-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C16H24N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0125632
|
((5Z,8Z)-Icosa-5,8,11,14-tetraenoylamino)-acetic acid
Show/Hide
|
C22H35NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0659958
|
(Z)-2-(2-chlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11ClN2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0677588
|
(Z)-2-benzylidene-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H12N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0692927
|
(Z)-2-(2,3-Difluorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]thiazin-3(5H)-one
Show/Hide
|
C13H10F2N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0709769
|
(Z)-2-(3-(3-Chlorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H19ClN2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849166
|
(Z)-2-(4-bromobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11BrN2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849168
|
(Z)-2-(4-methoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C14H14N2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849169
|
(Z)-2-(2,4-Difluorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]thiazin-3(5H)-one
Show/Hide
|
C13H10F2N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849399
|
6,6-diphenyl-2,3-dihydroimidazo[2,1-b]thiazol-5(6H)-one
Show/Hide
|
C17H14N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849409
|
(Z)-2-(2-methoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C14H14N2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849467
|
(Z)-2-(3-phenoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C19H16N2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849468
|
(Z)-2-(3,4-dimethoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H16N2O3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849470
|
(Z)-2-(3-nitrobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11N3O3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849472
|
(Z)-2-(3-phenylallylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H14N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849480
|
(Z)-3-(3-phenylallylidene)-3,5,6,7-tetrahydro-2H-imidazo[2,1-b][1,3]thiazin-2-one
Show/Hide
|
C15H14N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0849481
|
1-lysophosphatidylinositol
Show/Hide
|
C29H49O12P
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0850010
|
(Z)-2-(2,6-Dichlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]thiazin-3(5H)-one
Show/Hide
|
C13H10Cl2N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0858888
|
(Z)-2-(2,3-dichlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H10Cl2N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0858889
|
(Z)-2-(4-isopropylbenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C16H18N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859207
|
(Z)-2-(4-chlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11ClN2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859208
|
(Z)-ethyl 2-(3-((3-oxo-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2(3H)-ylidene)methyl)phenoxy)acetate
Show/Hide
|
C18H20N2O4S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859210
|
2,2-diphenyl-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C19H18N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859211
|
ethyl 5-oxo-6,6-diphenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole-2-carboxylate
Show/Hide
|
C20H18N2O3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859212
|
2,2-diphenyl-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C18H16N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859457
|
(Z)-2-(3-chlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11ClN2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859466
|
(Z)-3-((3-Oxo-6,7-dihydro-3H-imidazo[2,1-b][1,3]thiazin-2(5H)-ylidene)methyl)phenyl 4-chloro-benzoate
Show/Hide
|
C20H15ClN2O3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859468
|
(Z)-2-(2,4-Dichlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]-thiazin-3(5H)-one
Show/Hide
|
C13H10Cl2N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0859491
|
3,3-diphenyl-3,5,6,7-tetrahydro-2H-imidazo[2,1-b][1,3]thiazin-2-one
Show/Hide
|
C18H16N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0866547
|
ethyl 6-oxo-5,5-diphenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole-2-carboxylate
Show/Hide
|
C20H18N2O3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0866629
|
3,3-diphenyl-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2(3H)-one
Show/Hide
|
C19H18N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0866766
|
5,5-diphenyl-2,3-dihydroimidazo[2,1-b]thiazol-6(5H)-one
Show/Hide
|
C17H14N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0866767
|
(Z)-2-(1-phenylethylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C15H16N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0867263
|
(Z)-2-(4-nitrobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11N3O3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0868197
|
(Z)-2-(3-(3,4-Dichlorobenzyloxy)benzylidene)-6,7-dihydro-2Himidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H16Cl2N2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0877023
|
(Z)-2-(3-(2-Chlorobenzyloxy)benzylidene)-6,7-dihydro-2H-imidazo-[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H17ClN2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0881784
|
(Z)-2-(3-phenoxybenzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C20H18N2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0893073
|
(Z)-3-((3-Oxo-6,7-dihydro-3H-imidazo[2,1-b][1,3]thiazin-2(5H)-ylidene)methyl)phenyl benzoate
Show/Hide
|
C20H16N2O3S
|
1
|
| 1 |
Ki >= 10000 nM
|
|
|
|
CP0905395
|
(Z)-2-(2-Fluorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11FN2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0916683
|
(Z)-2-(2,3-Dimethoxybenzylidene)-6,7-dihydro-2H-imidazo-[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H16N2O3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0381996
|
3-[12-(cyclopropylamino)dodecoxy]-5-pentylphenol
Show/Hide
|
C26H45NO2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0410861
|
N-[11-(4-hexyl-3-hydroxyphenoxy)undecyl]cyclopropanecarboxamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0411873
|
N-(1-adamantyl)-11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
|
C36H59NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0494535
|
N-(1,3-dihydroxypropan-2-yl)-11-(4-hexyl-3-hydroxyphenoxy)undecanamide
Show/Hide
|
C26H45NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0543214
|
N-(1-adamantyl)-11-(3-hydroxy-5-pentylphenoxy)undecanamide
Show/Hide
|
C32H51NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0555102
|
N-(1-adamantyl)-8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]octanamide
Show/Hide
|
C33H53NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0555105
|
N-(1-adamantyl)-11-(4-hexyl-3-hydroxyphenoxy)undecanamide
Show/Hide
|
C33H53NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0556362
|
N-(1-adamantyl)-11-(2-hexyl-3-hydroxyphenoxy)undecanamide
Show/Hide
|
C33H53NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0419212
|
N-cycloheptyl-2-methoxy-5-(4-methoxyphenyl)-3-methylbenzamide
Show/Hide
|
C23H29NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0444875
|
2-methoxy-5-(4-methoxyphenyl)-3-methyl-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C23H29NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0481742
|
2-methoxy-5-(4-methoxyphenyl)-3-methyl-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C23H29NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0163467
|
ethyl 2-amino-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C11H15NO2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0395710
|
ethyl 2-(methanesulfonamido)-5-phenylthiophene-3-carboxylate
Show/Hide
|
C14H15NO4S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0400948
|
ethyl 2-[bis(naphthalen-2-ylsulfonyl)amino]-5-phenylthiophene-3-carboxylate
Show/Hide
|
C33H25NO6S3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0400952
|
ethyl 2-(naphthalene-2-carbonylamino)-5-phenylthiophene-3-carboxylate
Show/Hide
|
C24H19NO3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0424492
|
ethyl 2-(benzenesulfonamido)-5-phenylthiophene-3-carboxylate
Show/Hide
|
C19H17NO4S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0446044
|
ethyl 2-(methanesulfonamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C12H17NO4S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0446147
|
2,5-dimethyl-1-phenylpyrrole-3-carboxylic acid
Show/Hide
|
C13H13NO2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0446148
|
ethyl 2-(naphthalen-2-ylsulfonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C21H21NO4S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0446149
|
ethyl 2-[(4-chlorophenyl)sulfonylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C17H18ClNO4S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0455958
|
ethyl 2-[(4-chlorophenyl)sulfonylamino]-5-phenylthiophene-3-carboxylate
Show/Hide
|
C19H16ClNO4S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0477627
|
2-ethyl-5-methyl-1-phenylpyrrole-3-carboxylic acid
Show/Hide
|
C14H15NO2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0514481
|
ethyl 2-(naphthalen-1-ylsulfonylamino)-5-phenylthiophene-3-carboxylate
Show/Hide
|
C23H19NO4S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0482101
|
(6aR,10aR)-3-(1-hydroxy-2-methylpropan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-ol
Show/Hide
|
C20H28O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0389944
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-ethoxyethanone
Show/Hide
|
C25H24Cl2N6O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0416545
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-cyclopentylethanone
Show/Hide
|
C28H28Cl2N6O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0548532
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-[6-(difluoromethoxy)pyridin-3-yl]piperazine-1-carboxamide
Show/Hide
|
C28H22Cl2F2N8O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0401716
|
[6-hydroxy-1-(2-morpholin-4-ylethyl)indol-3-yl]-(4-methoxyphenyl)methanone
Show/Hide
|
C22H24N2O4
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0401723
|
6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]-N-[2-[[2-[[2-[[2-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-5-yl]oxyacetyl]amino]-2-methylpropanoyl]amino]-2-methylpropanoyl]amino]ethyl]hexanamide
Show/Hide
|
C63H71BF2N8O10S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0401726
|
N-[2-[2-(2-acetamidoethoxy)ethoxy]ethyl]-5-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxypentanamide
Show/Hide
|
C35H47N3O8
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0401727
|
6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]-N-[2-[2-[2-[[2-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyacetyl]amino]ethoxy]ethoxy]ethyl]hexanamide
Show/Hide
|
C59H66BF2N7O10S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0429901
|
6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]-N-[2-[[2-methyl-2-[[2-methyl-2-[[2-[1-(2-morpholin-4-ylethyl)-3-(naphthalene-1-carbonyl)indol-5-yl]oxyacetyl]amino]propanoyl]amino]propanoyl]amino]ethyl]hexanamide
Show/Hide
|
C66H72BF2N9O9S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0429902
|
N-[2-[2-[2-[2-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-5-yl]oxyethoxy]ethoxy]ethoxy]ethyl]acetamide
Show/Hide
|
C32H42N2O8
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0458125
|
2-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyacetic acid
Show/Hide
|
C24H26N2O6
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0477175
|
N-(8-aminooctyl)-2-[1-(2-morpholin-4-ylethyl)-3-(naphthalene-1-carbonyl)indol-5-yl]oxyacetamide
Show/Hide
|
C35H44N4O4
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0477185
|
N-[2-[2-(2-acetamidoethoxy)ethoxy]ethyl]-2-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyacetamide
Show/Hide
|
C32H42N4O8
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0477186
|
N-[2-[2-(2-aminoethoxy)ethoxy]ethyl]-2-[1-(2-morpholin-4-ylethyl)-3-(naphthalene-1-carbonyl)indol-5-yl]oxyacetamide
Show/Hide
|
C33H40N4O6
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0477188
|
N-[2-[2-(2-aminoethoxy)ethoxy]ethyl]-2-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyacetamide
Show/Hide
|
C30H40N4O7
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0482638
|
N-(8-aminooctyl)-2-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyacetamide
Show/Hide
|
C32H44N4O5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0494059
|
2-[1-(2-morpholin-4-ylethyl)-3-(naphthalene-1-carbonyl)indol-5-yl]oxyacetic acid
Show/Hide
|
C27H26N2O5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0517907
|
6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]-N-[2-[2-[2-[[2-[1-(2-morpholin-4-ylethyl)-3-(naphthalene-1-carbonyl)indol-5-yl]oxyacetyl]amino]ethoxy]ethoxy]ethyl]hexanamide
Show/Hide
|
C62H66BF2N7O9S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0517908
|
6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]-N-[2-[2-[2-[5-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxypentanoylamino]ethoxy]ethoxy]ethyl]hexanamide
Show/Hide
|
C62H72BF2N7O10S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0519647
|
[5-hydroxy-1-(oxolan-3-ylmethyl)indol-3-yl]-(4-methoxyphenyl)methanone
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C21H21NO4
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1
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| 1 |
Ki > 10000 nM
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CP0536539
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N-[2-[2-[2-[6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]hexanoylamino]ethoxy]ethoxy]ethyl]-7-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyheptanamide
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C64H76BF2N7O10S
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1
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| 1 |
Ki > 10000 nM
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CP0560818
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6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]-N-[2-[[2-[[2-[[2-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyacetyl]amino]-2-methylpropanoyl]amino]-2-methylpropanoyl]amino]ethyl]hexanamide
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C63H72BF2N9O10S
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1
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| 1 |
Ki > 10000 nM
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CP0022072
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[6-(difluoromethoxy)pyridin-3-yl]urea
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C29H24Cl2F2N8O2
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1
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| 1 |
Ki > 10000 nM
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CP0420625
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-phenylurea
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C29H25Cl2N7O
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1
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| 1 |
Ki > 10000 nM
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CP0431691
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-(2,4-difluorophenyl)urea
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C30H25Cl2F2N7O
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1
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| 1 |
Ki > 10000 nM
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CP0432070
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-cyclohexylurea
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C30H33Cl2N7O
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1
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| 1 |
Ki > 10000 nM
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CP0452689
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(2,4-difluorophenyl)urea
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C29H23Cl2F2N7O
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1
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| 1 |
Ki > 10000 nM
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CP0476543
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[(4,4-difluorocyclohexyl)methyl]urea
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C30H31Cl2F2N7O
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1
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| 1 |
Ki > 10000 nM
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CP0485555
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[(4-fluorophenyl)methyl]urea
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C30H26Cl2FN7O
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1
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| 1 |
Ki > 10000 nM
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CP0485556
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[6-(trifluoromethyl)pyridin-3-yl]urea
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C29H23Cl2F3N8O
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1
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| 1 |
Ki > 10000 nM
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CP0489576
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(2-fluorophenyl)urea
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C29H24Cl2FN7O
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1
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| 1 |
Ki > 10000 nM
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CP0535473
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-[6-(difluoromethoxy)pyridin-3-yl]urea
Show/Hide
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C30H26Cl2F2N8O2
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1
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| 1 |
Ki > 10000 nM
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CP0535474
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-(2-fluorophenyl)sulfonylurea
Show/Hide
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C30H26Cl2FN7O3S
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1
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| 1 |
Ki > 10000 nM
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CP0540524
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-cyclopentylurea
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C28H29Cl2N7O
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1
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| 1 |
Ki > 10000 nM
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CP0544189
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-(4,4-difluorocyclohexyl)urea
Show/Hide
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C30H31Cl2F2N7O
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1
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| 1 |
Ki > 10000 nM
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CP0547865
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-(2-fluorophenyl)urea
Show/Hide
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C30H26Cl2FN7O
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1
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| 1 |
Ki > 10000 nM
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CP0553719
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[1-(trifluoromethyl)cyclopentyl]urea
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C29H28Cl2F3N7O
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1
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| 1 |
Ki > 10000 nM
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CP0565197
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(4,4-difluorocyclohexyl)urea
Show/Hide
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C29H29Cl2F2N7O
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1
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| 1 |
Ki > 10000 nM
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CP0382752
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N-(1,3-benzothiazol-2-yl)adamantane-1-carboxamide
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C18H20N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382754
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N-hexyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
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C17H22N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382755
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N-cyclopentyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
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C16H18N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382756
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N-benzyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
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C18H16N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382757
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N-[(2-fluorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H15FN2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382758
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N-benzyl-1,3-benzothiazole-2-carboxamide
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C15H12N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382759
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N-(1,3-benzothiazol-2-yl)-4-(trifluoromethyl)benzamide
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C15H9F3N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382776
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N-(3-pentyl-1,3-benzothiazol-2-ylidene)-4-(trifluoromethyl)benzamide
Show/Hide
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C20H19F3N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382778
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N-naphthalen-1-yl-1,3-benzothiazole-2-carboxamide
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C18H12N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382781
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N-cyclopropyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
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C14H14N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382783
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N-[(2-chlorophenyl)methyl]-1,3-benzothiazole-2-carboxamide
Show/Hide
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C15H11ClN2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382785
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(4-methyl-2-phenyl-1,3-thiazol-5-yl)-morpholin-4-ylmethanone
Show/Hide
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C15H16N2O2S
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1
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| 1 |
Ki > 10000 nM
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CP0382820
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N-(cyclohexylmethyl)-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H22N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382821
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N-(1-adamantyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
Show/Hide
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C16H22N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382822
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N-butyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C15H18N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382823
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N-[(4-fluorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H15FN2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382826
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N-(1-adamantyl)-2-tert-butyl-4-methyl-1,3-thiazole-5-carboxamide
Show/Hide
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C19H28N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382827
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N-benzyl-2,4-dimethyl-1,3-thiazole-5-carboxamide
Show/Hide
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C13H14N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0382828
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N-(cyclohexylmethyl)-1,3-benzothiazole-2-carboxamide
Show/Hide
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C15H18N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0402060
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N-(1-adamantyl)-1,3-benzothiazole-2-carboxamide
Show/Hide
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C18H20N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0427553
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N-cyclohexyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C17H20N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0427554
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N-(1-adamantyl)-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C21H24N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0427555
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N-[(2-chlorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H15ClN2OS
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1
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| 1 |
Ki > 10000 nM
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CP0427556
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N-naphthalen-2-yl-1,3-benzothiazole-2-carboxamide
Show/Hide
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C18H12N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0427561
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4-methyl-2-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-thiazole-5-carboxamide
Show/Hide
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C21H20N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0431627
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N-(1,3-benzothiazol-2-yl)-3-(trifluoromethyl)benzamide
Show/Hide
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C15H9F3N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0431630
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N-(1,3-benzothiazol-2-yl)naphthalene-1-carboxamide
Show/Hide
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C18H12N2OS
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1
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| 1 |
Ki > 10000 nM
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CP0870378
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2-(2-((1H-benzo[d][1,2,3]triazol-1-yl)methyl)-5-methyl-1H-benzo[d]imidazol-1-yl)-N,N-dimethylethanamine
Show/Hide
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C19H22N6
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1
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| 1 |
Ki > 10000 nM
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CP0877580
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1-(1-(2-(diethylamino)ethyl)-2-(4-methoxybenzyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
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C23H29N3O2
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1
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| 1 |
Ki > 10000 nM
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CP0879201
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(1S,9aR)-1-((2-(4-methoxybenzyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)methyl)octahydro-1H-quinolizine
Show/Hide
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C26H30F3N3O
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1
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| 1 |
Ki > 10000 nM
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CP0902321
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N,N-diethyl-3-(2-(4-methoxybenzyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)propan-1-amine
Show/Hide
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C23H28F3N3O
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1
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| 1 |
Ki > 10000 nM
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CP0902323
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N,N-diethyl-2-(2-(4-methoxyphenyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)ethanamine
Show/Hide
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C21H24F3N3O
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1
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| 1 |
Ki > 10000 nM
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CP0902324
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1-[2-(Diethylamino)ethyl]-2-(4-ethoxybenzyl)-5-(1-hydrazonoethyl)-1H-benzimidazole
Show/Hide
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C24H33N5O
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1
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| 1 |
Ki > 10000 nM
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CP0902327
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1-(2-((2H-benzo[d][1,2,3]triazol-2-yl)methyl)-1-(3-(diethylamino)propyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
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C23H28N6O
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1
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| 1 |
Ki > 10000 nM
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CP0905763
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(1S,9aR)-1-(2-(2-((2H-benzo[d][1,2,3]triazol-2-yl)methyl)-5-chloro-1H-benzo[d]imidazol-1-yl)ethyl)octahydro-1H-quinolizine
Show/Hide
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C25H29ClN6
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1
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| 1 |
Ki > 10000 nM
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CP0905764
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1-(2-((1H-benzo[d][1,2,3]triazol-1-yl)methyl)-1-(2-(diethylamino)ethyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
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C22H26N6O
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1
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| 1 |
Ki > 10000 nM
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CP0929327
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1-(2-(4-methoxybenzyl)-1-(((1S,9aR)-octahydro-1H-quinolizin-1-yl)methyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
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C27H33N3O2
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1
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| 1 |
Ki > 10000 nM
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CP0929328
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2-(3,4-Dichlorobenzyl)-1-[(2-methoxy)ethyl]-5-trifluoromethylbenzimidazole
Show/Hide
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C18H15Cl2F3N2O
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1
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| 1 |
Ki = 10000 nM
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CP0942687
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1-(2-(4-chlorobenzyl)-1-(2-(diethylamino)ethyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
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C22H26ClN3O
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1
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| 1 |
Ki > 10000 nM
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CP0418899
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2,3-dihydroxypropyl 11-(4-hexyl-3-hydroxyphenoxy)undecanoate
Show/Hide
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C26H44O6
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1
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| 1 |
Ki = 10440 nM
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CP0509565
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(6aR,9S,10aR)-6,6-Dimethyl-3-(2-oxa-6-aza-tricyclo[3.3.1.1*3,7*]dec-6-yl)-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
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C23H31NO4
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1
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| 1 |
Ki = 14900 nM
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CP0473176
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(6aR,9S,10aR)-1,9-Dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-3-carboxylic acid adamantan-2-ylamide
Show/Hide
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C26H35NO4
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1
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| 1 |
Ki = 15000 nM
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CP0479035
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(6aR,9R,10aR)-6,6-Dimethyl-3-(2-oxa-6-aza-tricyclo[3.3.1.1*3,7*]dec-6-ylmethyl)-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
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C24H33NO4
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1
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| 1 |
Ki = 15000 nM
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CP0868783
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(Z)-2-(4-(dimethylamino)benzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
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C15H17N3OS
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1
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| 1 |
Ki = 16600 nM
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CP0371808
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CAS_3379236
Show/Hide
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C23H32N2O4S
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1
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| 1 |
Ki = 17400 nM
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CP0152981
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2-[(4-ethoxyphenyl)methyl]-1-(3-methylbutyl)-N-[2-[2-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethoxy]ethoxy]ethyl]benzimidazole-5-carboxamide
Show/Hide
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C41H51N5O4
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1
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| 1 |
Ki = 17400 nM
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CP0528073
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5-(3,5-dimethyl-piperidine-1-sulfonyl)-3-methyl-benzofuran-2-carboxylic acid 4-methyl-benzylamide
Show/Hide
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C25H30N2O4S
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1
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| 1 |
Ki = 19100 nM
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CP0373465
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(6aR,9R,10aR)-3-(Adamantan-2-ylaminomethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
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C26H37NO3
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1
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| 1 |
Ki = 20000 nM
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CP0385439
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((6aR,9R,10aR)-1,9-Dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromen-3-yl)-(2-oxa-6-aza-tricyclo[3.3.1.1*3,7*]dec-6-yl)-methanone
Show/Hide
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C24H31NO5
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1
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| 1 |
Ki = 20000 nM
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CP0371805
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CAS_15998383
Show/Hide
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C25H30N2O5S
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1
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| 1 |
Ki = 22800 nM
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CP0379561
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5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzofuran-2-carboxamide
Show/Hide
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C27H32N2O4S
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1
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| 1 |
Ki = 22800 nM
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CP0373464
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(6aR,9S,10aR)-3-(Adamantan-1-ylaminomethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
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C26H37NO3
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1
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| 1 |
Ki = 25000 nM
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CP0479036
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(6aR,9S,10aR)-3-(Adamantan-2-ylaminomethyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-1,9-diol
Show/Hide
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C26H37NO3
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1
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| 1 |
Ki = 25000 nM
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CP0509566
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((6aR,9S,10aR)-1,9-Dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromen-3-yl)-(2-oxa-6-aza-tricyclo[3.3.1.1*3,7*]dec-6-yl)-methanone
Show/Hide
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C24H31NO5
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1
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| 1 |
Ki = 25000 nM
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CP0152984
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2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-[4-(1,2,3,4-tetrahydroacridin-9-ylamino)butyl]benzimidazole-5-carboxamide
Show/Hide
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C38H45N5O2
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1
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| 1 |
Ki = 26900 nM
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CP0159376
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2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-[2-[2-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethoxy]ethoxy]ethyl]benzimidazole-5-carboxamide
Show/Hide
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C40H49N5O4
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1
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| 1 |
Ki = 28700 nM
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CP0431579
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2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]benzimidazole-5-carboxamide
Show/Hide
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C37H43N5O2
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1
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| 1 |
Ki = 30700 nM
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CP0402380
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(6aR,9S,10aR)-1,9-Dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene-3-carboxylic acid adamantan-1-ylamide
Show/Hide
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C26H35NO4
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1
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| 1 |
Ki = 35000 nM
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CP0434522
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2-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
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C23H34N2O2
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1
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| 1 |
Ki > 40000 nM
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CP0434524
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4,4-dimethyl-7-(2-methyloctan-2-yl)-1H-chromeno[4,3-c]pyrazol-9-ol
Show/Hide
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C21H30N2O2
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1
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| 1 |
Ki > 40000 nM
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CP0434526
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3-[1-(3,4-dichlorophenyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-yl]oxypropan-1-ol
Show/Hide
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C30H38Cl2N2O3
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1
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| 1 |
Ki > 40000 nM
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CP0434528
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1-ethyl-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
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C23H34N2O2
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1
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| 1 |
Ki > 40000 nM
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CP0434529
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1-(3,5-difluorophenyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
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C27H32F2N2O2
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1
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| 1 |
Ki > 40000 nM
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CP0549312
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2,4,4-trimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
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C22H32N2O2
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1
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| 1 |
Ki > 40000 nM
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CP0556764
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1-(2,4-dichlorophenyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)-9-phenylmethoxychromeno[4,3-c]pyrazole
Show/Hide
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C34H38Cl2N2O2
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1
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| 1 |
Ki > 40000 nM
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CP0561261
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3-[1-(2,4-dichlorophenyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-yl]oxypropan-1-ol
Show/Hide
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C30H38Cl2N2O3
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1
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| 1 |
Ki > 40000 nM
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CP0574985
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1-(2,4-dichlorophenyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
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C27H32Cl2N2O2
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1
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| 1 |
Ki > 40000 nM
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CP0483265
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US9422235, 97
Show/Hide
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C14H17F3N2O2S
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1
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| 1 |
Ki = 86980 nM
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CP0486261
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1-(4-chlorophenyl)-N-cyclohexyl-2-o-tolyl-1H-imidazole-4-carboxamide
Show/Hide
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C23H24ClN3O
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1
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| 1 |
Ki > 1000 nM
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CP0405468
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3-(3-(2,2,3,3-Tetramethylcyclopropanecarbonyl)-1H-indol-1-yl)propanoic Acid
Show/Hide
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C19H23NO3
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1
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| 1 |
Ki > 1000 nM
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CP0418655
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(1-(2-(1-methylpiperidin-4-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
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C24H34N2O
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1
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| 1 |
Ki > 1000 nM
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CP0430771
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(1-(2-(4-Methylpiperazin-1-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
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C23H33N3O
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1
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| 1 |
Ki > 1000 nM
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CP0430957
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2-(Tetrahydro-2H-pyran-4-yl)-1-(3-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1H-indol-1-yl)ethanone
Show/Hide
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C23H29NO3
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1
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| 1 |
Ki > 1000 nM
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CP0491470
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(1-(2-(Piperidin-4-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
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C23H32N2O
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1
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| 1 |
Ki > 1000 nM
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CP0496258
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(1-(2-(1-Methylpyrrolidin-2-yl)ethyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
Show/Hide
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C23H32N2O
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1
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| 1 |
Ki > 1000 nM
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CP0434919
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N-propyl-2-(tricyclo[3.3.1.03,7]nonane-3-carbonylamino)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-3-carboxamide
Show/Hide
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C21H29N3O2S
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1
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| 1 |
Ki > 1000 nM
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CP0429003
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[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-pyridin-3-ylmethanone
Show/Hide
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C21H23NO4
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1
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| 1 |
Ki > 1000 nM
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CP0481436
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[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-pyridin-4-ylmethanone
Show/Hide
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C21H23NO4
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1
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| 1 |
Ki > 1000 nM
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CP0507347
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[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-(1,3-thiazol-4-yl)methanone
Show/Hide
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C19H21NO4S
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1
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| 1 |
Ki > 1000 nM
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CP0524968
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[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]-pyridin-2-ylmethanone
Show/Hide
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C21H23NO4
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1
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| 1 |
Ki > 1000 nM
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CP0445554
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[1-[(cyclohexylideneamino)oxycarbonylamino]-3-methoxypropan-2-yl] (Z)-octadec-9-enoate
Show/Hide
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C29H52N2O5
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1
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| 1 |
Ki > 1000 nM
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CP0445555
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[1-methoxy-3-[4-(4-phenylphenyl)butanoylamino]propan-2-yl] 4-(4-phenylphenyl)butanoate
Show/Hide
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C36H39NO4
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1
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| 1 |
Ki > 1000 nM
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CP0449775
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[1-methoxy-3-(octanoylamino)propan-2-yl] octanoate
Show/Hide
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C20H39NO4
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1
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| 1 |
Ki > 1000 nM
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CP0453559
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[1-[(cyclohexylideneamino)oxycarbonylamino]-3-methoxypropan-2-yl] octanoate
Show/Hide
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C19H34N2O5
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1
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| 1 |
Ki > 1000 nM
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CP0482396
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[1-methoxy-3-(octoxycarbonylamino)propan-2-yl] octanoate
Show/Hide
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C21H41NO5
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1
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| 1 |
Ki > 1000 nM
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CP0482398
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[1-methoxy-3-(octylcarbamoyloxy)propan-2-yl] octanoate
Show/Hide
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C21H41NO5
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1
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| 1 |
Ki > 1000 nM
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CP0482399
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[1-methoxy-3-(octanoylamino)propan-2-yl] (Z)-octadec-9-enoate
Show/Hide
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C30H57NO4
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1
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| 1 |
Ki > 1000 nM
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CP0497836
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[1-methoxy-3-(octoxycarbonylamino)propan-2-yl] (Z)-octadec-9-enoate
Show/Hide
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C31H59NO5
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1
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| 1 |
Ki > 1000 nM
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CP0497837
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[1-[(cyclohexylideneamino)oxycarbonylamino]-3-methoxypropan-2-yl] 4-(4-phenylphenyl)butanoate
Show/Hide
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C27H34N2O5
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1
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| 1 |
Ki > 1000 nM
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CP0497838
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[2-[tert-butyl(diphenyl)silyl]oxy-2-methoxyethyl] N-octylcarbamate
Show/Hide
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C28H43NO4Si
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1
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| 1 |
Ki > 1000 nM
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CP0507761
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[1-methoxy-3-(octylcarbamoyloxy)propan-2-yl] (Z)-octadec-9-enoate
Show/Hide
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C31H59NO5
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1
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| 1 |
Ki > 1000 nM
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CP0507763
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(cyclohexylideneamino) N-(2-hydroxy-3-methoxypropyl)carbamate
Show/Hide
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C11H20N2O4
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1
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| 1 |
Ki > 1000 nM
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CP0507765
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(3-methoxy-2-octanoyloxypropyl) octanoate
Show/Hide
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C20H38O5
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1
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| 1 |
Ki > 1000 nM
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CP0534221
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[3-methoxy-2-(octylcarbamoyloxy)propyl] N-octylcarbamate
Show/Hide
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C22H44N2O5
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1
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| 1 |
Ki > 1000 nM
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CP0534531
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[1-methoxy-3-(octylcarbamoyloxy)propan-2-yl] (5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoate
Show/Hide
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C33H57NO5
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1
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| 1 |
Ki > 1000 nM
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CP0565516
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[3-methoxy-2-[4-(4-phenylphenyl)butanoyloxy]propyl] 4-(4-phenylphenyl)butanoate
Show/Hide
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C36H38O5
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1
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| 1 |
Ki > 1000 nM
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CP0435367
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2-[(3R,4R)-5-hydroxy-3-(2-hydroxyethyl)-2,2-dimethyl-7-(2-methyloctan-2-yl)-3,4-dihydrochromen-4-yl]acetic acid
Show/Hide
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C24H38O5
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1
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| 1 |
Ki > 1000 nM
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CP0481412
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3-[(3R,4R)-5-hydroxy-4-(hydroxymethyl)-2,2-dimethyl-7-(2-methyloctan-2-yl)-3,4-dihydrochromen-3-yl]propanoic acid
Show/Hide
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C24H38O5
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1
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| 1 |
Ki > 1000 nM
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CP0089105
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(Z)-7-[(1R,2R,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-5-phenylpent-1-enyl]-5-oxocyclopentyl]-N-[(2S)-1-hydroxypropan-2-yl]hept-5-enamide
Show/Hide
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C26H37NO5
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1
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| 1 |
Ki > 1000 nM
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CP0089197
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(Z)-7-[(1R,2R,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-5-phenylpent-1-enyl]-5-oxocyclopentyl]-N-(3-hydroxypropyl)hept-5-enamide
Show/Hide
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C26H37NO5
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1
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| 1 |
Ki > 1000 nM
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CP0116592
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(Z)-N-(2-hydroxyethyl)-7-[(1R,2R,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-5-(4-iodophenyl)pent-1-enyl]-5-oxocyclopentyl]hept-5-enamide
Show/Hide
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C25H34INO5
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1
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| 1 |
Ki > 1000 nM
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CP0116593
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(Z)-7-[(1R,2R,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-5-phenylpent-1-enyl]-5-oxocyclopentyl]-N-[(2R)-1-hydroxypropan-2-yl]hept-5-enamide
Show/Hide
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C26H37NO5
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1
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| 1 |
Ki > 1000 nM
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CP0147320
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(Z)-N-(2-hydroxyethyl)-7-[(1R,2R,3R)-3-hydroxy-2-[(E,3R)-3-hydroxy-5-phenylpent-1-enyl]-5-oxocyclopentyl]hept-5-enamide
Show/Hide
|
C25H35NO5
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1
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| 1 |
Ki > 1000 nM
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CP0147321
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(Z)-N-(2-hydroxyethyl)-7-[(1R,2R,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-5-phenylpent-1-enyl]-5-oxocyclopentyl]hept-5-enamide
Show/Hide
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C25H35NO5
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1
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| 1 |
Ki > 1000 nM
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CP0409943
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(6aR,9R,10aR)-3-[3-(aminomethyl)-1-adamantyl]-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-1,9-diol
Show/Hide
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C26H37NO3
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1
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| 1 |
Ki > 1000 nM
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CP0414203
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3-[(6aR,9R,10aR)-1,9-dihydroxy-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromen-3-yl]adamantane-1-carboxylic acid
Show/Hide
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C26H34O5
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1
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| 1 |
Ki > 1000 nM
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CP0428792
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(6aR,9R,10aR)-3-(3-amino-1-adamantyl)-6,6-dimethyl-6a,7,8,9,10,10a-hexahydrobenzo[c]chromene-1,9-diol
Show/Hide
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C25H35NO3
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1
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| 1 |
Ki > 1000 nM
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CP0424188
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US8859596, 178
Show/Hide
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C24H28F6N4O3
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1
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| 1 |
Ki > 1000 nM
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CP0443119
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US8859596, 179
Show/Hide
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C23H26F6N4O2
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1
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| 1 |
Ki > 1000 nM
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CP0405726
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(5Z,8Z,11Z,13R,14Z)-N-[(2R)-1-hydroxypropan-2-yl]-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
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C24H41NO2
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1
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| 1 |
Ki > 1000 nM
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CP0429549
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(5Z,8Z,10R,11Z,14Z)-N-(2-hydroxyethyl)-10-methylicosa-5,8,11,14-tetraenamide
Show/Hide
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C23H39NO2
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1
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| 1 |
Ki > 1000 nM
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CP0482472
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(5Z,8Z,10S,11Z,14Z)-N-(2-hydroxyethyl)-10-methylicosa-5,8,11,14-tetraenamide
Show/Hide
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C23H39NO2
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1
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| 1 |
Ki > 1000 nM
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CP0543345
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(5Z,8Z,11Z,13R,14Z)-N-(2-hydroxyethyl)-13-methylicosa-5,8,11,14-tetraenamide
Show/Hide
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C23H39NO2
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1
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| 1 |
Ki > 1000 nM
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CP0158863
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2-[((11Z,14Z)-Icosa-5,8,11,14-tetraenyl)oxy]-propane-1,3-diol
Show/Hide
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C23H40O3
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1
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| 1 |
Ki > 3000 nM
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CP0372933
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1-(4-chlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-3-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-4-carboxamide
Show/Hide
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C22H17Cl3N4O
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1
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| 1 |
Ki > 3940 nM
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CP0372969
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1-(4-chlorophenyl)-3-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-4-carboxamide
Show/Hide
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C20H22ClN5O
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1
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| 1 |
Ki > 3940 nM
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CP0384279
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4-cyano-1-phenyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C20H20N6O
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1
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| 1 |
Ki > 3940 nM
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CP0431799
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1-(4-chlorophenyl)-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C19H20ClN5O
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1
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| 1 |
Ki > 3940 nM
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CP0431800
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1-(4-chlorophenyl)-4-cyano-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C20H19ClN6O
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1
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| 1 |
Ki > 3940 nM
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CP0431801
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1-phenyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C19H21N5O
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1
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| 1 |
Ki > 3940 nM
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CP0458171
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4-methyl-1-phenyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C20H23N5O
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1
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| 1 |
Ki > 3940 nM
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CP0376645
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N-[2-(4-chlorophenyl)ethyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H23ClF2N4O
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1
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| 1 |
Ki > 3940 nM
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CP0376652
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1-(2,4-dichlorophenyl)-N-[2-(2,4-dichlorophenyl)ethyl]-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H22Cl4N4O
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1
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| 1 |
Ki > 3940 nM
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CP0376697
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N-[2-(4-chlorophenyl)ethyl]-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H19Cl3N4O
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1
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| 1 |
Ki > 3940 nM
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CP0390565
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N-[(4-chlorophenyl)methyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C24H21ClF2N4O
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1
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| 1 |
Ki > 3940 nM
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CP0396948
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N-[2-(4-chlorophenyl)ethyl]-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H23Cl3N4O
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1
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| 1 |
Ki > 3940 nM
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CP0396952
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N-(4-chlorophenyl)-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C23H19ClF2N4O
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1
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| 1 |
Ki > 3940 nM
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CP0396953
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N-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C23H19Cl3N4O
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1
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| 1 |
Ki > 3940 nM
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CP0439166
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N-[2-(4-chlorophenyl)ethyl]-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H23Cl3N4O
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1
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| 1 |
Ki > 3940 nM
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CP0439167
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N-[(4-chlorophenyl)methyl]-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C24H21Cl3N4O
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1
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| 1 |
Ki > 3940 nM
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CP0450845
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1-(2,4-dichlorophenyl)-N-[2-(3,4-dichlorophenyl)ethyl]-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H18Cl4N4O
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1
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| 1 |
Ki > 3940 nM
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CP0453827
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N-[2-(3-chloro-4-methoxyphenyl)ethyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C26H25ClF2N4O2
|
1
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| 1 |
Ki > 3940 nM
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CP0453828
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N-[2-(3,4-dichlorophenyl)ethyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H22Cl2F2N4O
|
1
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| 1 |
Ki > 3940 nM
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CP0453829
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N-(4-chlorophenyl)-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C21H15ClF2N4O
|
1
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| 1 |
Ki > 3940 nM
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CP0453831
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1-(2,4-dichlorophenyl)-N-[2-(3,4-dichlorophenyl)ethyl]-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
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C25H22Cl4N4O
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1
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| 1 |
Ki > 3940 nM
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CP0453833
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N-[2-(4-chlorophenyl)ethyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
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C23H19ClF2N4O
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1
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| 1 |
Ki > 3940 nM
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CP0494321
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N-[(4-chlorophenyl)-phenylmethyl]-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
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C30H25Cl3N4O
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1
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| 1 |
Ki > 3940 nM
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CP0496213
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N-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C23H19Cl3N4O
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1
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| 1 |
Ki > 3940 nM
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CP0506396
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1-(2,4-dichlorophenyl)-N-[2-(2,4-dichlorophenyl)ethyl]-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
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C23H18Cl4N4O
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1
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| 1 |
Ki > 3940 nM
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CP0098948
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Impulsin
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C18H37NO2
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1
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| 1 |
Ki > 5000 nM
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CP0461224
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2-cyclohexyl-5-(2-morpholinoethyl)-2H-pyrazolo[4,3-c]quinolin-3(5H)-one
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C22H28N4O2
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1
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| 1 |
Ki > 7900 nM
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CP0372349
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2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
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C29H26ClNO
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1
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| 1 |
Ki > 7900 nM
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CP0372351
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2,2-diphenyl-N-(3-phenylpropyl)acetamide
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C23H23NO
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1
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| 1 |
Ki > 7900 nM
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CP0372609
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2-(4-Bromophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
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C29H26BrNO
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1
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| 1 |
Ki > 7900 nM
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CP0496637
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N-(3,3-diphenylpropyl)-2-phenylacetamide
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C23H23NO
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1
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| 1 |
Ki > 7900 nM
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