General Information of the Compound
Compound ID
CP0159376
Compound Name
2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1-[2-[2-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethoxy]ethoxy]ethyl]benzimidazole-5-carboxamide
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Structure
Formula
C40H49N5O4
Molecular Weight
663.863
Canonical SMILES
CCOc1ccc(Cc2nc3cc(ccc3n2CCOCCOCCNc2c3CCCCc3nc3ccccc23)C(=O)N(CC)CC)cc1
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InChI
InChI=1S/C40H49N5O4/c1-4-44(5-2)40(46)30-17-20-37-36(28-30)43-38(27-29-15-18-31(19-16-29)49-6-3)45(37)22-24-48-26-25-47-23-21-41-39-32-11-7-9-13-34(32)42-35-14-10-8-12-33(35)39/h7,9,11,13,15-20,28H,4-6,8,10,12,14,21-27H2,1-3H3,(H,41,42)
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InChIKey
QWAXIXJFJWHJOJ-UHFFFAOYSA-N
Physicochemical Property
logP
7.0801
Rotatable Bonds
17
Heavy Atom Count
49
Polar Areas
90.74
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
8
Complexity
49

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 155525250
ChEMBL ID
CHEMBL4456433
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00834, Cannabinoid receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 28700 nM
   TI
   LI
   LO
   TS