General Information of the Compound
Compound ID
CP0400987
Compound Name
(8E)-8-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-(1-pyridin-2-ylcyclopropyl)-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
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Structure
Formula
C29H23Cl2F3N4OS
Molecular Weight
603.497
Canonical SMILES
FC(F)(F)c1ccc(c(Cl)c1)-n1nc(C(=O)NC2(CC2)c2ccccn2)c2CCCC\C(=C/c3ccc(Cl)s3)c12
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InChI
InChI=1S/C29H23Cl2F3N4OS/c30-21-16-18(29(32,33)34)8-10-22(21)38-26-17(15-19-9-11-24(31)40-19)5-1-2-6-20(26)25(37-38)27(39)36-28(12-13-28)23-7-3-4-14-35-23/h3-4,7-11,14-16H,1-2,5-6,12-13H2,(H,36,39)/b17-15+
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InChIKey
VPTHGWFPZPEPCX-BMRADRMJSA-N
Physicochemical Property
logP
8.3405
Rotatable Bonds
5
Heavy Atom Count
40
Polar Areas
59.81
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
40

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 134145283
ChEMBL ID
CHEMBL3941829
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01298, Cannabinoid receptor 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 8 nM
   TI
   LI
   LO
   TS
Protein ID: PT00834, Cannabinoid receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS