Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-(2-{3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl}ethyl)morpholine
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 PubChem ID
CID: 11584525
SID: 17155420
Canonical SMILES
CC1(C)C(C(=O)c2cn(CCN3CCOCC3)c3ccccc23)C1(C)C
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Compound Formula C22H30N2O2
Compound Structure
Protein Name
 Protein Info 
Cannabinoid receptor 2
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
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Cannabinoid receptor
Uniprot ID
P34972
Gene Name
CNR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  4
1
EC50 = 0.52 nM
   TI
   LI
   LO
   TS
2
EC50 = 14 nM
   TI
   LI
   LO
   TS
3
EC50 = 16 nM
   TI
   LI
   LO
   TS
4
Ki = 4.365 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 0.77 nM
2 Ki = 4.4 nM