Brief Information of the Compound and Protein
Compound Name
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-(2-sulfamoylacetyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
    Show/Hide
PubChem ID
CID: 134134129
Canonical SMILES
COc1ccc(\C=C2/CN(Cc3c(nn(c23)-c2ccc(Cl)cc2Cl)C(=O)N[C@H](C)c2ccccn2)C(=O)CS(N)(=O)=O)cc1
    Show/Hide
Compound Formula C30H28Cl2N6O5S
Compound Structure
Protein Name
Cannabinoid receptor 2
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
>
Cannabinoid receptor
Uniprot ID
P34972
Gene Name
CNR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 1450 nM
   TI
   LI
   LO
   TS