| Compound ID |
Compound Name |
Compound Formula |
|
CP0149074
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(6-methoxypyridin-3-yl)propan-2-yl]cyclopropanecarboxamide
Show/Hide
|
C26H25FN4O3
|
3
|
| 1 |
EC50 = 1.3 nM
|
|
|
| 2 |
IC50 = 0.24 nM
|
|
|
| 3 |
IC50 = 0.4 nM
|
|
|
|
CP0476110
|
2,2-difluoro-N-[(1R,2S)-1-[1-(1-methyl-6-oxopyridin-3-yl)indazol-5-yl]oxy-1-phenylpropan-2-yl]propanamide
Show/Hide
|
C25H24F2N4O3
|
2
|
| 1 |
EC50 = 2.3 nM
|
|
|
| 2 |
IC50 = 1.6 nM
|
|
|
|
CP0063059
|
US10196374, Example 3
Show/Hide
|
C27H26F4N4O3
|
3
|
| 1 |
EC50 = 2.7 nM
|
|
|
| 2 |
IC50 = 2.2 nM
|
|
|
| 3 |
IC50 = 23 nM
|
|
|
|
CP0199185
|
US10196374, Example 5
Show/Hide
|
C27H27ClF2N4O3
|
3
|
| 1 |
EC50 = 2.9 nM
|
|
|
| 2 |
IC50 = 1.7 nM
|
|
|
| 3 |
IC50 = 324 nM
|
|
|
|
CP0320206
|
N-[(1R,2S,3S)-1-(3,5-difluorophenyl)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-3-hydroxybutan-2-yl]-5-methyl-1,3,4-oxadiazole-2-carboxamide
Show/Hide
|
C27H22F3N5O4
|
3
|
| 1 |
EC50 = 3.5 nM
|
|
|
| 2 |
IC50 = 1.6 nM
|
|
|
| 3 |
IC50 = 270 nM
|
|
|
|
CP0383864
|
2,2-difluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(6-methoxypyridin-3-yl)-3-methylbutan-2-yl]propanamide
Show/Hide
|
C27H27F3N4O3
|
3
|
| 1 |
EC50 = 3.5 nM
|
|
|
| 2 |
IC50 = 0.57 nM
|
|
|
| 3 |
IC50 = 70 nM
|
|
|
|
CP0383859
|
2,2-difluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-3-methyl-1-phenylbutan-2-yl]propanamide
Show/Hide
|
C27H26F3N3O2
|
3
|
| 1 |
EC50 = 3.9 nM
|
|
|
| 2 |
IC50 < 0.34 nM
|
|
|
| 3 |
IC50 = 13 nM
|
|
|
|
CP0125580
|
US8901310, Example 1
Show/Hide
|
C29H29F3N2O2
|
3
|
| 1 |
EC50 = 4.8 nM
|
|
|
| 2 |
IC50 = 0.69 nM
|
|
|
| 3 |
IC50 = 8.9 nM
|
|
|
|
CP0514935
|
2,2,2-trifluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-3-methyl-1-phenylbutan-2-yl]acetamide
Show/Hide
|
C26H23F4N3O2
|
3
|
| 1 |
EC50 = 5.4 nM
|
|
|
| 2 |
IC50 < 0.42 nM
|
|
|
| 3 |
IC50 = 25 nM
|
|
|
|
CP0199382
|
US10196374, Example 6
Show/Hide
|
C26H24ClF3N4O3
|
3
|
| 1 |
EC50 = 5.6 nM
|
|
|
| 2 |
IC50 = 3 nM
|
|
|
| 3 |
IC50 = 114 nM
|
|
|
|
CP0063060
|
N-[(1R,2S)-1-(2-bromo-4-cyanophenoxy)-1-(2-cyclopropylpyrimidin-5-yl)propan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C20H19BrF2N4O2
|
2
|
| 1 |
EC50 = 6.4 nM
|
|
|
| 2 |
IC50 = 1.1 nM
|
|
|
|
CP0149073
|
2,2-difluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(6-methoxypyridin-3-yl)-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C31H27F3N4O3
|
3
|
| 1 |
EC50 = 8.7 nM
|
|
|
| 2 |
IC50 = 2 nM
|
|
|
| 3 |
IC50 = 92 nM
|
|
|
|
CP0063115
|
US10196374, Example 1
Show/Hide
|
C27H28F2N4O3
|
3
|
| 1 |
EC50 = 11 nM
|
|
|
| 2 |
IC50 = 7 nM
|
|
|
| 3 |
IC50 = 160 nM
|
|
|
|
CP0429666
|
N-[(1R,2S)-1-[1-(1-ethyl-6-oxopyridin-3-yl)indazol-5-yl]oxy-1-phenylpropan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C26H26F2N4O3
|
2
|
| 1 |
EC50 = 13 nM
|
|
|
| 2 |
IC50 = 4.7 nM
|
|
|
|
CP0456226
|
2,2-difluoro-N-[(1R,2S)-1-[1-(5-fluoro-1-methyl-6-oxopyridin-3-yl)indazol-5-yl]oxy-3-methyl-1-phenylbutan-2-yl]propanamide
Show/Hide
|
C27H27F3N4O3
|
3
|
| 1 |
EC50 = 18 nM
|
|
|
| 2 |
IC50 = 5.6 nM
|
|
|
| 3 |
IC50 = 301 nM
|
|
|
|
CP0456359
|
N-[(1R,2S)-1-[1-(1-cyclopropyl-6-oxopyridin-3-yl)indazol-5-yl]oxy-1-phenylpropan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C27H26F2N4O3
|
3
|
| 1 |
EC50 = 19 nM
|
|
|
| 2 |
IC50 = 3.9 nM
|
|
|
| 3 |
IC50 = 220 nM
|
|
|
|
CP0240922
|
N-[(1R,2S)-1-(2-chloro-4-cyanophenoxy)-1-(2-cyclopropylpyrimidin-5-yl)propan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C20H19ClF2N4O2
|
2
|
| 1 |
EC50 = 21 nM
|
|
|
| 2 |
IC50 = 7.8 nM
|
|
|
|
CP0179648
|
N-[(1R,2S)-1-(2-bromo-4-cyanophenoxy)-1-(2-cyclopropylpyrimidin-5-yl)propan-2-yl]-2,2,2-trifluoroacetamide
Show/Hide
|
C19H16BrF3N4O2
|
2
|
| 1 |
EC50 = 23 nM
|
|
|
| 2 |
IC50 = 2.5 nM
|
|
|
|
CP0456227
|
2,2-difluoro-N-[(1R,2S)-3-methyl-1-[1-(1-methyl-2-oxopyridin-3-yl)indazol-5-yl]oxy-1-phenylbutan-2-yl]propanamide
Show/Hide
|
C27H28F2N4O3
|
2
|
| 1 |
EC50 = 27 nM
|
|
|
| 2 |
IC50 = 11 nM
|
|
|
|
CP0477995
|
2,2-difluoro-N-[(1R,2S)-3-methyl-1-phenyl-1-[1-(1,3-thiazol-4-yl)indazol-5-yl]oxybutan-2-yl]propanamide
Show/Hide
|
C24H24F2N4O2S
|
3
|
| 1 |
EC50 = 29 nM
|
|
|
| 2 |
IC50 = 3.3 nM
|
|
|
| 3 |
IC50 = 131 nM
|
|
|
|
CP0446119
|
N-[(1R,2S)-1-(3-chloro-4-cyanophenoxy)-1-(6-methoxypyridin-3-yl)propan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C19H18ClF2N3O3
|
2
|
| 1 |
EC50 = 33 nM
|
|
|
| 2 |
IC50 = 9.3 nM
|
|
|
|
CP0446127
|
N-[(1R,2S)-1-(2-chloro-4-cyanophenoxy)-1-(6-methoxypyridin-3-yl)propan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C19H18ClF2N3O3
|
2
|
| 1 |
EC50 = 43 nM
|
|
|
| 2 |
IC50 = 16 nM
|
|
|
|
CP0383861
|
N-[(1R,2S)-1-(2-bromo-4-cyanophenoxy)-1-(2-cyclopropylpyrimidin-5-yl)butan-2-yl]-2,2,2-trifluoroacetamide
Show/Hide
|
C20H18BrF3N4O2
|
3
|
| 1 |
EC50 = 54 nM
|
|
|
| 2 |
IC50 = 9.6 nM
|
|
|
| 3 |
IC50 = 560 nM
|
|
|
|
CP0383860
|
2,2-difluoro-N-[(1R,2S)-3-methyl-1-[1-(1-methyl-2-oxopyrimidin-5-yl)indazol-5-yl]oxy-1-phenylbutan-2-yl]propanamide
Show/Hide
|
C26H27F2N5O3
|
2
|
| 1 |
EC50 = 87 nM
|
|
|
| 2 |
IC50 = 51 nM
|
|
|
|
CP0047174
|
(1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-hydroxyacetyl)-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-3,6-dien-5-one
Show/Hide
|
C21H28O5
|
2
|
| 1 |
EC50 = 110 nM
|
|
|
| 2 |
IC50 = 40 nM
|
|
|
|
CP0063057
|
N-[(1R,2S)-1-[1-(5-cyano-1-methyl-6-oxopyridin-3-yl)indazol-5-yl]oxy-3-methyl-1-phenylbutan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C28H27F2N5O3
|
2
|
| 1 |
EC50 = 110 nM
|
|
|
| 2 |
IC50 = 27 nM
|
|
|
|
CP0565693
|
2,2,2-trifluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(4-methylsulfanylphenyl)propan-2-yl]acetamide
Show/Hide
|
C25H21F4N3O2S
|
1
|
| 1 |
IC50 = 0.03 nM
|
|
|
|
CP0153948
|
2,2,2-trifluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-naphthalen-2-ylpropan-2-yl]acetamide
Show/Hide
|
C28H21F4N3O2
|
1
|
| 1 |
IC50 = 0.04 nM
|
|
|
|
CP0563701
|
2,2,2-trifluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-quinolin-3-ylpropan-2-yl]acetamide
Show/Hide
|
C27H20F4N4O2
|
1
|
| 1 |
IC50 = 0.04 nM
|
|
|
|
CP0532752
|
N-[(1R,2S)-1-(4-ethylphenyl)-1-[1-(4-fluorophenyl)indazol-5-yl]oxypropan-2-yl]-2,2-dimethylpropanamide
Show/Hide
|
C29H32FN3O2
|
1
|
| 1 |
IC50 = 0.05 nM
|
|
|
|
CP0504409
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-yl]-2,2-dimethylpropanamide
Show/Hide
|
C28H30FN3O3
|
1
|
| 1 |
IC50 = 0.08 nM
|
|
|
|
CP0451747
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]-5-methyl-1,3,4-oxadiazole-2-carboxamide
Show/Hide
|
C26H22FN5O3
|
1
|
| 1 |
IC50 = 0.09 nM
|
|
|
|
CP0576386
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]-5-methyl-1,2,4-oxadiazole-3-carboxamide
Show/Hide
|
C26H22FN5O3
|
1
|
| 1 |
IC50 = 0.09 nM
|
|
|
|
CP0153949
|
2,2,2-trifluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]acetamide
Show/Hide
|
C24H19F4N3O2
|
1
|
| 1 |
IC50 = 0.13 nM
|
|
|
|
CP0455011
|
N-[(1R,2S)-1-(4-ethylphenyl)-1-[1-(4-fluorophenyl)indazol-5-yl]oxypropan-2-yl]-2-hydroxyacetamide
Show/Hide
|
C26H26FN3O3
|
1
|
| 1 |
IC50 = 0.21 nM
|
|
|
|
CP0451746
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(4-methoxyphenyl)propan-2-yl]-2,2-dimethylpropanamide
Show/Hide
|
C28H30FN3O3
|
1
|
| 1 |
IC50 = 0.25 nM
|
|
|
|
CP0404495
|
(2R,3S)-3-(2-chloro-3-fluoro-4-methoxyphenyl)-2-(ethylsulfanylmethyl)-1,1,1-trifluoro-3-[(2-methylquinolin-5-yl)amino]propan-2-ol
Show/Hide
|
C23H23ClF4N2O2S
|
1
|
| 1 |
IC50 = 0.47 nM
|
|
|
|
CP0451886
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]cyclopropanecarboxamide
Show/Hide
|
C26H24FN3O2
|
1
|
| 1 |
IC50 = 0.62 nM
|
|
|
|
CP0451887
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-yl]cyclopropanesulfonamide
Show/Hide
|
C26H26FN3O4S
|
1
|
| 1 |
IC50 = 0.62 nM
|
|
|
|
CP0534627
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]-2,2-dimethylpropanamide
Show/Hide
|
C27H28FN3O2
|
1
|
| 1 |
IC50 = 0.66 nM
|
|
|
|
CP0153947
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(4-methylsulfanylphenyl)propan-2-yl]cyclopropanesulfonamide
Show/Hide
|
C26H26FN3O3S2
|
1
|
| 1 |
IC50 = 0.75 nM
|
|
|
|
CP0153950
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(4-methylsulfonylphenyl)propan-2-yl]-2-hydroxyacetamide
Show/Hide
|
C25H24FN3O5S
|
1
|
| 1 |
IC50 = 0.84 nM
|
|
|
|
CP0294288
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]cyclopropanesulfonamide
Show/Hide
|
C25H24FN3O3S
|
1
|
| 1 |
IC50 = 0.91 nM
|
|
|
|
CP0455010
|
5-[[(1S,2R,4R)-4-ethyl-6,7-difluoro-2,5-dihydroxy-2-(trifluoromethyl)-3,4-dihydro-1H-naphthalen-1-yl]amino]-1H-quinolin-2-one
Show/Hide
|
C22H19F5N2O3
|
1
|
| 1 |
IC50 = 1.15 nM
|
|
|
|
CP0322903
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(4-methylsulfonylphenyl)propan-2-yl]cyclopropanesulfonamide
Show/Hide
|
C26H26FN3O5S2
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0451748
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]benzamide
Show/Hide
|
C29H24FN3O2
|
1
|
| 1 |
IC50 = 1.41 nM
|
|
|
|
CP0113622
|
N-[(2S)-1-[[1-(4-fluorophenyl)indazol-4-yl]amino]propan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C25H27FN4O2S
|
2
|
| 1 |
IC50 = 1.47 nM
|
|
|
| 2 |
IC50 = 1.5 nM
|
|
|
|
CP0116474
|
2,4,6-trimethyl-N-[(2S)-1-[(1-phenylindazol-4-yl)amino]propan-2-yl]benzenesulfonamide
Show/Hide
|
C25H28N4O2S
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0113656
|
N-[(2S)-1-[[1-(6-fluoropyridin-3-yl)indazol-4-yl]amino]propan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C24H26FN5O2S
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0060412
|
2,4,6-trimethyl-N-[(2S)-1-[(1-pyridin-3-ylindazol-4-yl)amino]propan-2-yl]benzenesulfonamide
Show/Hide
|
C24H27N5O2S
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0432207
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]propane-2-sulfonamide
Show/Hide
|
C25H26FN3O3S
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
|
CP0551486
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]acetamide
Show/Hide
|
C24H22FN3O2
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0056982
|
N-[(2S)-1-[[1-(4-chlorophenyl)indazol-4-yl]amino]propan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C25H27ClN4O2S
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0260350
|
2,4,6-trimethyl-N-[(2S)-1-[[1-(4-methylphenyl)indazol-4-yl]amino]propan-2-yl]benzenesulfonamide
Show/Hide
|
C26H30N4O2S
|
1
|
| 1 |
IC50 = 4.5 nM
|
|
|
|
CP0455008
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]-3-methoxypropanamide
Show/Hide
|
C26H26FN3O3
|
1
|
| 1 |
IC50 = 5.09 nM
|
|
|
|
CP0260366
|
N-[(2S)-1-[[1-(3-fluorophenyl)indazol-4-yl]amino]propan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C25H27FN4O2S
|
1
|
| 1 |
IC50 = 6.1 nM
|
|
|
|
CP0060437
|
2,4,6-trimethyl-N-[(2S)-1-[[1-(3-methylphenyl)indazol-4-yl]amino]propan-2-yl]benzenesulfonamide
Show/Hide
|
C26H30N4O2S
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
|
CP0534628
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]butane-2-sulfonamide
Show/Hide
|
C26H28FN3O3S
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
|
CP0056981
|
2,4,6-trimethyl-N-[(2S)-1-[(1-pyrimidin-5-ylindazol-4-yl)amino]propan-2-yl]benzenesulfonamide
Show/Hide
|
C23H26N6O2S
|
1
|
| 1 |
IC50 = 6.9 nM
|
|
|
|
CP0429665
|
2,2-difluoro-N-[(1S,2R)-2-[1-(4-fluorophenyl)indazol-5-yl]oxy-2-(6-methoxypyridin-3-yl)-1-[(2-methylpropan-2-yl)oxy]ethyl]propanamide
Show/Hide
|
C28H29F3N4O4
|
2
|
| 1 |
IC50 = 7.1 nM
|
|
|
| 2 |
IC50 = 130 nM
|
|
|
|
CP0056980
|
1-cyclopentyl-N-[(2S)-1-[[1-(6-fluoropyridin-3-yl)indazol-4-yl]amino]propan-2-yl]-3,5-dimethylpyrazole-4-sulfonamide
Show/Hide
|
C25H30FN7O2S
|
1
|
| 1 |
IC50 = 7.2 nM
|
|
|
|
CP0577260
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]methanesulfonamide
Show/Hide
|
C23H22FN3O3S
|
1
|
| 1 |
IC50 = 7.4 nM
|
|
|
|
CP0451749
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-pyridin-3-ylpropan-2-yl]cyclopropanecarboxamide
Show/Hide
|
C25H23FN4O2
|
1
|
| 1 |
IC50 = 8.83 nM
|
|
|
|
CP0059291
|
1-cyclopentyl-N-[(2S)-1-[[1-(4-fluorophenyl)indazol-4-yl]amino]propan-2-yl]-3,5-dimethylpyrazole-4-sulfonamide
Show/Hide
|
C26H31FN6O2S
|
1
|
| 1 |
IC50 = 9.7 nM
|
|
|
|
CP0534626
|
N-[(3S)-1-[1-(4-fluorophenyl)indazol-4-yl]pyrrolidin-3-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C26H27FN4O2S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0059392
|
N-[(2S)-1-[[1-(4-fluorophenyl)indazol-4-yl]amino]-3-methylbutan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C27H31FN4O2S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0447689
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]propane-1-sulfonamide
Show/Hide
|
C25H26FN3O3S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0056528
|
2,4,6-trimethyl-N-[1,1,1-trifluoro-3-[1-(4-fluorophenyl)indazol-4-yl]oxypropan-2-yl]benzenesulfonamide
Show/Hide
|
C25H23F4N3O3S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0116470
|
N-[(2S)-1-[[1-(4-fluoro-3-methylphenyl)indazol-4-yl]amino]propan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C26H29FN4O2S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0035186
|
(10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]-14-hydroxy-15-methyl-14-(prop-1-yn-1-yl)tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-1,6-dien-5-one
Show/Hide
|
C29H35NO2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0056527
|
N-[(2S)-1-[[1-(4-cyanophenyl)indazol-4-yl]amino]propan-2-yl]-1-cyclopentyl-3,5-dimethylpyrazole-4-sulfonamide
Show/Hide
|
C27H31N7O2S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0148739
|
N-[(1S,2R)-2-(2-bromo-4-cyanophenoxy)-1-cyclopropyl-2-(2-cyclopropylpyrimidin-5-yl)ethyl]-2,2,2-trifluoroacetamide
Show/Hide
|
C21H18BrF3N4O2
|
2
|
| 1 |
IC50 = 21 nM
|
|
|
| 2 |
IC50 = 221 nM
|
|
|
|
CP0260348
|
N-[(2S)-4-[1-(4-fluorophenyl)indazol-4-yl]butan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C26H28FN3O2S
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0429667
|
2,2-difluoro-N-[(1R,2S)-1-[1-(6-oxo-1-propylpyridin-3-yl)indazol-5-yl]oxy-1-phenylpropan-2-yl]propanamide
Show/Hide
|
C27H28F2N4O3
|
2
|
| 1 |
IC50 = 32 nM
|
|
|
| 2 |
IC50 = 256 nM
|
|
|
|
CP0508094
|
1,1,1-trifluoro-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]methanesulfonamide
Show/Hide
|
C23H19F4N3O3S
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0514934
|
2,2-difluoro-N-[(1R,2S)-3-methyl-1-phenyl-1-[1-(1,2-thiazol-5-yl)indazol-5-yl]oxybutan-2-yl]propanamide
Show/Hide
|
C24H24F2N4O2S
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0116473
|
N-[(2S)-1-[[1-(3-methoxyphenyl)indazol-4-yl]amino]propan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C26H30N4O3S
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0056524
|
1-cyclopentyl-3,5-dimethyl-N-[(2S)-1-[(1-pyrimidin-5-ylindazol-4-yl)amino]propan-2-yl]pyrazole-4-sulfonamide
Show/Hide
|
C24H30N8O2S
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0458739
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]-2-methylpropane-1-sulfonamide
Show/Hide
|
C26H28FN3O3S
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0056983
|
N-[(2S)-1-[1-(4-fluorophenyl)indazol-4-yl]oxypropan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C25H26FN3O3S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0179647
|
N-[(1R,2S)-1-(4-cyanophenoxy)-1-(6-methoxypyridin-3-yl)propan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C19H19F2N3O3
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0478000
|
2,2-difluoro-N-[(1R,2S)-1-[1-[1-(1-hydroxyethyl)-6-oxopyridin-3-yl]indazol-5-yl]oxy-1-phenylpropan-2-yl]propanamide
Show/Hide
|
C26H26F2N4O4
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0029908
|
2-[(4R)-4-[(5-ethylsulfonyl-1H-pyrrolo[2,3-c]pyridin-2-yl)methyl]-5,5,5-trifluoro-4-hydroxy-2-methylpentan-2-yl]-5-fluorobenzamide
Show/Hide
|
C23H25F4N3O4S
|
1
|
| 1 |
IC50 = 84 nM
|
|
|
|
CP0504408
|
N-[(2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxypropan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C25H26FN3O3S
|
1
|
| 1 |
IC50 = 98 nM
|
|
|
|
CP0446132
|
N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-yl]pentane-1-sulfonamide
Show/Hide
|
C27H30FN3O3S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0240918
|
N-[(1R,2S)-1-[1-[1-(cyclopropylmethyl)-6-oxopyridin-3-yl]indazol-5-yl]oxy-1-phenylpropan-2-yl]-2,2-difluoropropanamide
Show/Hide
|
C28H28F2N4O3
|
2
|
| 1 |
IC50 = 226 nM
|
|
|
| 2 |
IC50 = 449 nM
|
|
|
|
CP0063061
|
N-[(1R,2S)-1-(2-bromo-4-cyanophenoxy)-1-(2-cyclopropylpyrimidin-5-yl)-3-[(2-methylpropan-2-yl)oxy]propan-2-yl]-2,2,2-trifluoroacetamide
Show/Hide
|
C23H24BrF3N4O3
|
1
|
| 1 |
IC50 = 516 nM
|
|
|
|
CP0411644
|
N-[(2S)-1-(1H-indazol-4-ylamino)propan-2-yl]-2,4,6-trimethylbenzenesulfonamide
Show/Hide
|
C19H24N4O2S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0247159
|
2,4,6-trimethyl-N-[(2S)-1-quinolin-5-yloxypropan-2-yl]benzenesulfonamide
Show/Hide
|
C21H24N2O3S
|
1
|
| 1 |
IC50 = 960 nM
|
|
|
|
CP0113623
|
2,4,6-trimethyl-N-[(2S)-1-[(8-methylquinolin-5-yl)amino]propan-2-yl]benzenesulfonamide
Show/Hide
|
C22H27N3O2S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0380944
|
2,4,6-trimethyl-N-[(2S)-1-(quinolin-5-ylamino)propan-2-yl]benzenesulfonamide
Show/Hide
|
C21H25N3O2S
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0060414
|
2,4,6-trimethyl-N-[(2S)-1-[(2-methylquinolin-5-yl)amino]propan-2-yl]benzenesulfonamide
Show/Hide
|
C22H27N3O2S
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0495197
|
2,4,6-trichloro-N-[(2S)-1-quinolin-5-yloxypropan-2-yl]benzenesulfonamide
Show/Hide
|
C18H15Cl3N2O3S
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
