General Information of the Compound
Compound ID
CP0429666
Compound Name
N-[(1R,2S)-1-[1-(1-ethyl-6-oxopyridin-3-yl)indazol-5-yl]oxy-1-phenylpropan-2-yl]-2,2-difluoropropanamide
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Structure
Formula
C26H26F2N4O3
Molecular Weight
480.515
Canonical SMILES
CCn1cc(ccc1=O)-n1ncc2cc(O[C@@H]([C@H](C)NC(=O)C(C)(F)F)c3ccccc3)ccc12
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InChI
InChI=1S/C26H26F2N4O3/c1-4-31-16-20(10-13-23(31)33)32-22-12-11-21(14-19(22)15-29-32)35-24(18-8-6-5-7-9-18)17(2)30-25(34)26(3,27)28/h5-17,24H,4H2,1-3H3,(H,30,34)/t17-,24-/m0/s1
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InChIKey
GFAQUXPHHREEAJ-XDHUDOTRSA-N
Physicochemical Property
logP
4.4871
Rotatable Bonds
8
Heavy Atom Count
35
Polar Areas
78.15
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 145972549
ChEMBL ID
CHEMBL4215390
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00967, Glucocorticoid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000464 ChaGo-K-1 Homo sapiens (Human)  2
1
EC50 = 13 nM
   TI
   LI
   LO
   TS
2
IC50 = 4.7 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 2.5 nM