Brief Information of the Compound and Protein
Compound Name
2,2-difluoro-N-[(1R,2S)-3-methyl-1-phenyl-1-[1-(1,2-thiazol-5-yl)indazol-5-yl]oxybutan-2-yl]propanamide
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PubChem ID
CID: 145977353
Canonical SMILES
CC(C)[C@H](NC(=O)C(C)(F)F)[C@H](Oc1ccc2n(ncc2c1)-c1ccns1)c1ccccc1
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Compound Formula C24H24F2N4O2S
Compound Structure
Protein Name
Glucocorticoid receptor
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 3
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Nuclear hormone receptor subfamily 3 group C
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Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000464 ChaGo-K-1 Homo sapiens (Human)  1
1
IC50 = 39 nM
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