Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2,4,6-trimethyl-N-[(2S)-1-[[1-(4-methylphenyl)indazol-4-yl]amino]propan-2-yl]benzenesulfonamide
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 PubChem ID
CID: 16665286
SID: 26525334
Canonical SMILES
C[C@@H](CNc1cccc2n(ncc12)-c1ccc(C)cc1)NS(=O)(=O)c1c(C)cc(C)cc1C
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Compound Formula C26H30N4O2S
Compound Structure
Protein Name
 Protein Info 
Glucocorticoid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
>
Nuclear hormone receptor subfamily 3
>
Nuclear hormone receptor subfamily 3 group C
>
Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000464 ChaGo-K-1
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 4.5 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 3.9 nM
2 IC50 = 12 nM