| Compound ID |
Compound Name |
Compound Formula |
|
CP0955941
|
(S)-6-(cyclopropylmethyl)-N-((S)-1-(5-(7-methoxyquinolin-6-yl)-1H-imidazol-2-yl)-7-oxononyl)-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C34H45N5O3
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0568215
|
(2S)-6-(cyclopropylmethyl)-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C35H47N5O3
|
1
|
| 1 |
IC50 < 0.3 nM
|
|
|
|
CP0571293
|
(2S)-6-cyclobutyl-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C35H47N5O3
|
1
|
| 1 |
IC50 < 0.3 nM
|
|
|
|
CP0577445
|
(2S)-6-(cyclopropylmethyl)-N-[(1S)-1-[5-(2-ethyl-7-methoxyquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C36H49N5O3
|
1
|
| 1 |
IC50 < 0.3 nM
|
|
|
|
CP0579552
|
(2S)-N-[(1S)-1-[5-(2-cyclopropyl-7-methoxyquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-(cyclopropylmethyl)-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C37H49N5O3
|
1
|
| 1 |
IC50 < 0.3 nM
|
|
|
|
CP0008777
|
JNJ-26481585
Show/Hide
|
C21H26N6O2
|
2
|
| 1 |
IC50 = 0.33 nM
|
|
|
| 2 |
IC50 = 2.16 nM
|
|
|
|
CP0577441
|
(2S)-6-ethyl-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H45N5O3
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0636220
|
(S)-N-(1-(5-(2-fluorophenyl)-1H-imidazol-2-yl)-7-(isoxazol-3-yl)-7-oxoheptyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C24H28FN5O3
|
1
|
| 1 |
IC50 = 0.47 nM
|
|
|
|
CP0570249
|
(2S)-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-propan-2-yl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C34H47N5O3
|
1
|
| 1 |
IC50 = 0.59 nM
|
|
|
|
CP0577693
|
(2S)-N-[(1S)-1-[5-(2-cyclopropyl-7-methoxyquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C34H45N5O3
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0138710
|
(2S)-6-(cyclopropylmethyl)-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C35H46N4O4
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0577129
|
(2S)-6-ethyl-N-[(1S)-1-[5-(7-methoxy-1-methyl-2-oxoquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H45N5O4
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0577442
|
(2S)-N-[(1S)-1-[5-(2,7-dimethylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H43N5O2
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0638656
|
(S)-N-(1-(5-(2-fluorophenyl)-1H-imidazol-2-yl)-7-(5-methylisoxazol-3-yl)-7-oxoheptyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C25H30FN5O3
|
1
|
| 1 |
IC50 = 0.76 nM
|
|
|
|
CP0015199
|
N-[(1S)-1-[5-(2-fluorophenyl)-1,3-oxazol-2-yl]-7-(1,2-oxazol-3-yl)-7-oxoheptyl]-1-methylazetidine-3-carboxamide
Show/Hide
|
C24H27FN4O4
|
1
|
| 1 |
IC50 = 0.82 nM
|
|
|
|
CP0543661
|
(2S)-6-ethyl-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H44N4O4
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0570394
|
(2S)-N-[(1S)-1-[5-(2-cyclopropylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H43N5O2
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0577692
|
(2S)-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H42N4O4
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0568333
|
(2S)-N-[(1S)-1-[5-(7-fluoro-2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H40FN5O2
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0569796
|
(2S)-N-[(1S)-1-[5-(7-methoxyquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O3
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0955940
|
(S)-6-ethyl-N-((S)-1-(5-(7-methoxyquinolin-6-yl)-1H-imidazol-2-yl)-7-oxononyl)-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C32H43N5O3
|
1
|
| 1 |
IC50 < 1.5 nM
|
|
|
|
CP0543658
|
(2S)-6-ethyl-N-[(1S)-1-(5-isoquinolin-6-yl-1H-imidazol-2-yl)-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O2
|
1
|
| 1 |
IC50 < 1.5 nM
|
|
|
|
CP0568220
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-[5-(2-oxo-1H-quinolin-3-yl)-1H-imidazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C30H39N5O3
|
1
|
| 1 |
IC50 < 1.5 nM
|
|
|
|
CP0577440
|
(2S)-6-methyl-N-[(1S)-1-[5-(2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O2
|
1
|
| 1 |
IC50 < 1.5 nM
|
|
|
|
CP0579476
|
(2S)-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H43N5O3
|
1
|
| 1 |
IC50 < 1.5 nM
|
|
|
|
CP0003676
|
N-hydroxy-2-[[2-(6-methoxypyridin-3-yl)-4-morpholin-4-ylthieno[3,2-d]pyrimidin-6-yl]methyl-methylamino]pyrimidine-5-carboxamide
Show/Hide
|
C23H24N8O4S
|
2
|
| 1 |
IC50 = 1.6 nM
|
|
|
| 2 |
IC50 = 5 nM
|
|
|
|
CP0832315
|
(S)-6-methyl-N-((S)-1-(5-(2-methyl-1-oxo-1,2-dihydroisoquinolin-6-yl)-1H-imidazol-2-yl)-7-oxononyl)-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C31H41N5O3
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0003580
|
Faridak
Show/Hide
|
C21H23N3O2
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 3.28 nM
|
|
|
|
CP0965642
|
(S)-N-((S)-1-(5-(7-methoxy-2-(pyrrolidin-1-yl)quinolin-6-yl)-1H-imidazol-2-yl)-7-oxononyl)-6-methyl-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C35H48N6O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0543659
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-[5-(2-pyrrolidin-1-ylquinolin-6-yl)-1H-imidazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C34H46N6O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0577443
|
(2S)-6-ethyl-N-[(1S)-1-[5-(2-ethyl-7-methoxy-1-oxoisoquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C34H46N4O5
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0577128
|
(2S)-6-methyl-N-[(1S)-1-[5-[2-(1,3-oxazol-2-yl)quinolin-6-yl]-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H40N6O3
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0547778
|
(2S)-6-ethyl-N-[(1S)-1-[5-(7-methoxyquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H42N4O4
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0568214
|
(2S)-N-[(1S)-1-[5-(2-methoxyquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O3
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0568320
|
(2S)-N-[(1S)-1-[5-(7-ethyl-2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H45N5O2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0579394
|
(2S)-6-ethyl-N-[(1S)-1-[5-(2-methoxy-1,8-naphthyridin-3-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O4
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0543657
|
(2S)-N-[(1S)-1-[5-(2-ethylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H43N5O2
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0579646
|
(2S)-N-[(1S)-1-[5-(2-methoxy-1,7-naphthyridin-3-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C30H40N6O3
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0578926
|
(2S)-6-ethyl-N-[(1S)-1-[5-(7-methoxy-1-methyl-2-oxoquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H44N4O5
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0014160
|
(5R,8S,11S)-11-[(Z)-2-fluoro-4-sulfanylbut-1-enyl]-5-methyl-8-propan-2-yl-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-triene-6,9,13-trione
Show/Hide
|
C21H27FN4O4S3
|
1
|
| 1 |
IC50 = 2.46 nM
|
|
|
|
CP0577438
|
(2S)-6-methyl-N-[(1S)-1-[5-(1-methyl-2-oxoquinolin-3-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O3
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0578925
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-[5-(4-pyridin-3-ylphenyl)-1H-imidazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H41N5O2
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0010223
|
2-[[2-(2-aminopyrimidin-5-yl)-9-methyl-6-morpholin-4-ylpurin-8-yl]methyl-methylamino]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C21H24N12O3
|
1
|
| 1 |
IC50 = 2.62 nM
|
|
|
|
CP0005479
|
CHEBI:46024
Show/Hide
|
C17H22N2O3
|
2
|
| 1 |
IC50 = 2.74 nM
|
|
|
| 2 |
IC50 = 5 nM
|
|
|
|
CP0004262
|
N-hydroxy-2-[methyl-[(9-methyl-6-morpholin-4-yl-2-pyridin-4-ylpurin-8-yl)methyl]amino]pyrimidine-5-carboxamide
Show/Hide
|
C22H24N10O3
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
|
CP0005544
|
2-[[2-(4-aminophenyl)-9-methyl-6-morpholin-4-ylpurin-8-yl]methyl-methylamino]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C23H26N10O3
|
1
|
| 1 |
IC50 = 2.9 nM
|
|
|
|
CP0136714
|
7-[6-(5-fluoro-6-methoxypyridin-3-yl)-4-methylquinazolin-8-yl]oxy-N-hydroxyheptanamide
Show/Hide
|
C22H25FN4O4
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0569431
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-(5-quinolin-6-yl-1H-imidazol-2-yl)nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C30H39N5O2
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0569795
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-[5-(4-pyridin-4-ylphenyl)-1H-imidazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H41N5O2
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0531517
|
(2S)-N-[(1S)-1-[5-(7-methoxyquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H40N4O4
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0569430
|
(2S)-6-ethyl-N-[(1S)-1-[5-(2-methoxy-1,7-naphthyridin-3-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O4
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0568325
|
(2S)-6-methyl-N-[(1S)-1-[5-(2-methylindazol-5-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C29H40N6O2
|
1
|
| 1 |
IC50 = 3.3 nM
|
|
|
|
CP0115609
|
N-hydroxy-2-[2-[6-(6-methoxypyridin-3-yl)-4-methylquinazolin-8-yl]oxyethyl-methylamino]pyrimidine-5-carboxamide
Show/Hide
|
C23H23N7O4
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0487666
|
N-[6-(2-fluoro-5-methoxyphenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C22H25FN4O4
|
1
|
| 1 |
IC50 = 3.5 nM
|
|
|
|
CP0527664
|
N-[6-(4-chlorophenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C21H23ClN4O3
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0004673
|
N-hydroxy-2-[[2-(4-methoxyphenyl)-9-methyl-6-morpholin-4-ylpurin-8-yl]methyl-methylamino]pyrimidine-5-carboxamide
Show/Hide
|
C24H27N9O4
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0565997
|
N'-hydroxy-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]octanediamide
Show/Hide
|
C22H26N4O4
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0426578
|
N-[6-(3-chlorophenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C21H23ClN4O3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0579557
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-[5-(4-pyrazin-2-ylphenyl)-1H-imidazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H40N6O2
|
1
|
| 1 |
IC50 = 4.1 nM
|
|
|
|
CP0426579
|
N-[6-(3-ethoxyphenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C23H28N4O4
|
1
|
| 1 |
IC50 = 4.2 nM
|
|
|
|
CP0531950
|
N'-hydroxy-N-[6-(4-methoxyphenyl)-1H-indazol-3-yl]octanediamide
Show/Hide
|
C22H26N4O4
|
1
|
| 1 |
IC50 = 4.2 nM
|
|
|
|
CP0568319
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-[5-(2-pyrazol-1-ylquinolin-6-yl)-1H-imidazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H41N7O2
|
1
|
| 1 |
IC50 = 4.2 nM
|
|
|
|
CP0531960
|
N-[6-(2-fluorophenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C21H23FN4O3
|
1
|
| 1 |
IC50 = 4.4 nM
|
|
|
|
CP0487052
|
N-[6-(3,4-dimethoxyphenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C23H28N4O5
|
1
|
| 1 |
IC50 = 4.6 nM
|
|
|
|
CP0531200
|
N-[6-(3,5-dimethoxyphenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C23H28N4O5
|
1
|
| 1 |
IC50 = 4.8 nM
|
|
|
|
CP0487675
|
N'-hydroxy-N-[6-[3-(trifluoromethyl)phenyl]-1H-indazol-3-yl]octanediamide
Show/Hide
|
C22H23F3N4O3
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0545443
|
(2S)-6-ethyl-N-[(1S)-7-oxo-1-[5-(2-oxo-6-phenyl-1H-pyridin-3-yl)-1H-imidazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H43N5O3
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0570395
|
(2S)-N-[(1S)-1-[5-(7-fluoro-2-methylquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H39FN4O3
|
1
|
| 1 |
IC50 = 5.1 nM
|
|
|
|
CP0546114
|
N-[6-(2-chlorophenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C21H23ClN4O3
|
1
|
| 1 |
IC50 = 5.2 nM
|
|
|
|
CP0487672
|
N'-hydroxy-N-[6-(3-methoxyphenyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]octanediamide
Show/Hide
|
C21H25N5O4
|
1
|
| 1 |
IC50 = 5.3 nM
|
|
|
|
CP0015005
|
S-[(E)-4-[(4Z,7S,10S)-4-ethylidene-2,5,8,12-tetraoxo-7-propan-2-yl-9-oxa-16-thia-3,6,13,18-tetrazabicyclo[13.2.1]octadeca-1(17),15(18)-dien-10-yl]but-3-enyl] octanethioate
Show/Hide
|
C29H42N4O6S2
|
1
|
| 1 |
IC50 = 5.3 nM
|
|
|
|
CP0527665
|
N'-hydroxy-N-[6-(2-methoxyphenyl)-1H-indazol-3-yl]octanediamide
Show/Hide
|
C22H26N4O4
|
1
|
| 1 |
IC50 = 5.4 nM
|
|
|
|
CP0545445
|
(2S)-6-methyl-N-[(1S)-1-[5-(1-methyl-2-oxoquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O3
|
1
|
| 1 |
IC50 = 5.4 nM
|
|
|
|
CP0826898
|
(S)-6-methyl-N-((S)-7-oxo-1-(5-(quinolin-3-yl)-1H-imidazol-2-yl)nonyl)-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C30H39N5O2
|
1
|
| 1 |
IC50 = 5.8 nM
|
|
|
|
CP0570396
|
(2S)-N-[(1S)-1-[5-(2-cyclopropyl-7-fluoroquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C33H41FN4O3
|
1
|
| 1 |
IC50 = 5.9 nM
|
|
|
|
CP0564514
|
N-[6-(2-fluoro-3-methoxyphenyl)-1H-indazol-3-yl]-N'-hydroxyoctanediamide
Show/Hide
|
C22H25FN4O4
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0638655
|
(S)-N-(1-(5-(4-fluorophenyl)-1H-imidazol-2-yl)-7-(oxazol-2-yl)-7-oxoheptyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C24H28FN5O3
|
1
|
| 1 |
IC50 = 7.1 nM
|
|
|
|
CP0004747
|
(5R,8S,11S)-11-[(Z)-1-fluoro-4-sulfanylbut-1-enyl]-5-methyl-8-propan-2-yl-3,17-dithia-7,10,14,19,20-pentazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-triene-6,9,13-trione
Show/Hide
|
C21H28FN5O3S3
|
1
|
| 1 |
IC50 = 7.42 nM
|
|
|
|
CP0012571
|
(4Z,7S,10S)-7-(4-aminobutyl)-4-ethylidene-10-[(E)-4-(heptyldisulfanyl)but-1-enyl]-9-oxa-16-thia-3,6,13,18-tetrazabicyclo[13.2.1]octadeca-1(17),15(18)-diene-2,5,8,12-tetrone
Show/Hide
|
C29H45N5O5S3
|
1
|
| 1 |
IC50 = 7.5 nM
|
|
|
|
CP0638831
|
(S)-7-amino-7-(5-(2-fluorophenyl)-1H-imidazol-2-yl)-1-(isoxazol-3-yl)heptan-1-one
Show/Hide
|
C19H21FN4O2
|
1
|
| 1 |
IC50 = 8.5 nM
|
|
|
|
CP0531951
|
N'-hydroxy-N-[6-(4-methoxyphenyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]octanediamide
Show/Hide
|
C21H25N5O4
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0004960
|
(5R,8S,11R)-12,12-difluoro-5-methyl-8-propan-2-yl-11-[(E)-4-sulfanylbut-1-enyl]-3,17-dithia-7,10,14,19,20-pentazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-triene-6,9,13-trione
Show/Hide
|
C21H27F2N5O3S3
|
1
|
| 1 |
IC50 = 9.25 nM
|
|
|
|
CP0004955
|
(5R,8S,11S)-5-methyl-8-propan-2-yl-11-[(E)-4-sulfanylbut-1-enyl]-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-triene-6,9,13-trione
Show/Hide
|
C21H28N4O4S3
|
1
|
| 1 |
IC50 = 9.5 nM
|
|
|
|
CP0580117
|
(2S)-6-methyl-N-[(1S)-1-[5-(1,8-naphthyridin-3-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C29H38N6O2
|
1
|
| 1 |
IC50 = 9.9 nM
|
|
|
|
CP0572973
|
(2S)-N-[(1S)-1-[5-(3a,7a-dihydro-1,3-benzothiazol-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C28H39N5O2S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0005903
|
N-hydroxy-2-[[2-(6-methoxypyridin-3-yl)-9-methyl-6-morpholin-4-ylpurin-8-yl]methyl-methylamino]pyrimidine-5-carboxamide
Show/Hide
|
C23H26N10O4
|
1
|
| 1 |
IC50 = 11.46 nM
|
|
|
|
CP0034844
|
HDAC inhibitor, Compound 1
Show/Hide
|
C19H17N3O2S
|
2
|
| 1 |
IC50 = 13 nM
|
|
|
| 2 |
Ki = 1.5 nM
|
|
|
|
CP0003832
|
N'-hydroxy-N-phenyloctanediamide
Show/Hide
|
C14H20N2O3
|
12
|
| 1 |
IC50 = 13 nM
|
|
|
| 2 |
IC50 = 31 nM
|
|
|
| 3 |
IC50 = 51 nM
|
|
|
| 4 |
IC50 = 70 nM
|
|
|
| 5 |
IC50 = 91 nM
|
|
|
| 6 |
IC50 = 91.6 nM
|
|
|
| 7 |
IC50 = 146 nM
|
|
|
| 8 |
IC50 = 174 nM
|
|
|
| 9 |
IC50 = 200 nM
|
|
|
| 10 |
IC50 = 214 nM
|
|
|
| 11 |
IC50 = 230 nM
|
|
|
| 12 |
IC50 = 398.11 nM
|
|
|
|
CP0543663
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-[5-(4-pyridin-3-ylphenyl)-1,3-oxazol-2-yl]nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H40N4O3
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0558007
|
N'-hydroxy-N-(6-phenyl-1H-indazol-3-yl)octanediamide
Show/Hide
|
C21H24N4O3
|
1
|
| 1 |
IC50 = 13.1 nM
|
|
|
|
CP0012872
|
4-[[[2-(benzylamino)-2-oxoethyl]-[4-(dimethylamino)benzoyl]amino]methyl]-3-fluoro-N-hydroxybenzamide
Show/Hide
|
C26H27FN4O4
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0569794
|
(2S)-N-[(1S)-1-[5-(7-chloro-2-methylquinolin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H40ClN5O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0543660
|
(2S)-6-ethyl-N-[(1S)-1-[5-(7-methoxyquinoxalin-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H42N6O3
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0001838
|
N-[4-[2-(5,6-dimethoxyindol-1-yl)ethoxy]phenyl]-N'-hydroxyoctanediamide
Show/Hide
|
C26H33N3O6
|
1
|
| 1 |
IC50 = 16.6 nM
|
|
|
|
CP0012097
|
3-(4-fluorophenyl)-N-[[4-(hydroxycarbamoyl)phenyl]methyl]-1H-pyrazole-5-carboxamide
Show/Hide
|
C18H15FN4O3
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0010838
|
(5R,8S,11S)-11-[(E)-3,3-difluoro-4-sulfanylbut-1-enyl]-5-methyl-8-propan-2-yl-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-triene-6,9,13-trione
Show/Hide
|
C21H26F2N4O4S3
|
1
|
| 1 |
IC50 = 18.49 nM
|
|
|
|
CP0577444
|
(2S)-N-[(1S)-1-[5-(3a,7a-dihydro-1,3-benzoxazol-6-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C28H39N5O3
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0004956
|
(5R,8S,11S)-11-[(Z)-1-fluoro-4-sulfanylbut-1-enyl]-5-methyl-8-propan-2-yl-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-triene-6,9,13-trione
Show/Hide
|
C21H27FN4O4S3
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0003911
|
(7S)-7-amino-7-[5-(2-fluorophenyl)-1,2-oxazol-3-yl]-1-(1,2-oxazol-3-yl)heptan-1-one
Show/Hide
|
C19H20FN3O3
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0578924
|
(2S)-6-ethyl-N-[(1S)-1-(5-isoquinolin-7-yl-1H-imidazol-2-yl)-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0639103
|
(S)-N-(1-(5-(4-fluorophenyl)-1H-imidazol-2-yl)-7-oxo-7-(thiazol-2-yl)heptyl)-1-methylpiperidine-4-carboxamide
Show/Hide
|
C26H32FN5O2S
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0013501
|
N-hydroxy-6-(6-morpholin-4-yl-1,3-dioxobenzo[de]isoquinolin-2-yl)hexanamide
Show/Hide
|
C22H25N3O5
|
1
|
| 1 |
IC50 = 25.6 nM
|
|
|
|
CP0535181
|
N'-hydroxy-N-(6-pyridin-4-yl-1H-indazol-3-yl)octanediamide
Show/Hide
|
C20H23N5O3
|
1
|
| 1 |
IC50 = 25.9 nM
|
|
|
|
CP0749584
|
(S)-N-(5-(2-fluoro-6-hydroxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H26FN5O3S
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0840086
|
(S)-N-(5-(2-hydroxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H27N5O3S
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0543662
|
(2S)-6-ethyl-N-[(1S)-1-[5-(6-methoxy-2-methylindazol-5-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H43N5O4
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0546115
|
N'-hydroxy-N-(6-thiophen-3-yl-1H-indazol-3-yl)octanediamide
Show/Hide
|
C19H22N4O3S
|
1
|
| 1 |
IC50 = 31.6 nM
|
|
|
|
CP0634946
|
psammaplin A
Show/Hide
|
C22H24Br2N4O6S2
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0637650
|
(E)-3-(3-Bromo-4-hydroxyphenyl)-N-(3-(hydroxyamino)-3-oxopropyl)-2-(hydroxyimino)propanamide
Show/Hide
|
C12H14BrN3O5
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0013329
|
N'-hydroxy-N-[4-[2-(5-methoxyindol-1-yl)ethoxy]phenyl]octanediamide
Show/Hide
|
C25H31N3O5
|
1
|
| 1 |
IC50 = 33.1 nM
|
|
|
|
CP0545442
|
(2S)-N-[(1S)-1-(5-cinnolin-6-yl-1H-imidazol-2-yl)-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C29H38N6O2
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0577439
|
(2S)-6-methyl-N-[(1S)-7-oxo-1-(5-quinoxalin-6-yl-1H-imidazol-2-yl)nonyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C29H38N6O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0011193
|
3-(4-fluorophenyl)-N-[7-(hydroxyamino)-7-oxoheptyl]-1H-pyrazole-5-carboxamide
Show/Hide
|
C17H21FN4O3
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0013856
|
4-[[3-(1,3-benzodioxol-5-yl)-5-methylpyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C19H17N3O4
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0003093
|
N-hydroxy-4-[[5-methyl-3-(4-methylphenyl)pyrazol-1-yl]methyl]benzamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0579915
|
(2S)-6-methyl-N-[(1S)-1-[5-(1-methyl-4-oxoquinolin-3-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H41N5O3
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0012287
|
3-(4-fluorophenyl)-N-[6-(hydroxyamino)-6-oxohexyl]-1H-pyrazole-5-carboxamide
Show/Hide
|
C16H19FN4O3
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0569432
|
(2S)-6-ethyl-N-[(1S)-1-[5-(6-methoxy-2-methylindazol-5-yl)-1H-imidazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H44N6O3
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0208472
|
N-(2-amino-5-thiophen-2-ylphenyl)-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C23H23N5O3S
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0012285
|
N-hydroxy-4-[[3-(4-methylphenyl)-5-(trifluoromethyl)pyrazol-1-yl]methyl]benzamide
Show/Hide
|
C19H16F3N3O2
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0004475
|
RICOLINOSTAT
Show/Hide
|
C24H27N5O3
|
3
|
| 1 |
IC50 = 48 nM
|
|
|
| 2 |
IC50 = 66 nM
|
|
|
| 3 |
IC50 = 379 nM
|
|
|
|
CP0638180
|
(S)-N-(1-(5-(4-fluorophenyl)-1H-imidazol-2-yl)-7-(4-methyloxazol-2-yl)-7-oxoheptyl)-1-methylpiperidine-4-carboxamide
Show/Hide
|
C27H34FN5O3
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0478984
|
6-[2-[4-[2-(dimethylamino)ethoxy]phenyl]-5-hydroxy-4-oxochromen-7-yl]oxy-N-hydroxyhexanamide;hydrochloride
Show/Hide
|
C25H31ClN2O7
|
1
|
| 1 |
IC50 = 58.46 nM
|
|
|
|
CP0004545
|
N-[2-(benzylamino)-2-oxoethyl]-N-[6-(hydroxyamino)-6-oxohexyl]-3,5-dimethylbenzamide
Show/Hide
|
C24H31N3O4
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0015198
|
(7S)-7-amino-7-[1-(4-fluorophenyl)pyrazol-4-yl]-1-(1,2-oxazol-3-yl)heptan-1-one
Show/Hide
|
C19H21FN4O2
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0955787
|
(S)-N-(5-(2-amino-6-fluorobenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H27FN6O2S
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0374534
|
N-[2-amino-5-(4-fluorophenyl)phenyl]oxane-4-carboxamide
Show/Hide
|
C18H19FN2O2
|
1
|
| 1 |
IC50 = 62 nM
|
|
|
|
CP0487053
|
N'-hydroxy-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]hexanediamide
Show/Hide
|
C20H22N4O4
|
1
|
| 1 |
IC50 = 62 nM
|
|
|
|
CP0535180
|
N'-hydroxy-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]heptanediamide
Show/Hide
|
C21H24N4O4
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0004543
|
N-[2-(benzylamino)-2-oxoethyl]-4-(dimethylamino)-N-[6-(hydroxyamino)-6-oxohexyl]benzamide
Show/Hide
|
C24H32N4O4
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0831925
|
(S)-N-(5-(3-hydroxypicolinamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C28H26N6O3S
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0554914
|
N-(4-(2-butylhydrazine-1- carbonyl)benzyl)cinnamamide
Show/Hide
|
C21H25N3O2
|
1
|
| 1 |
IC50 = 70.03 nM
|
|
|
|
CP0011194
|
N-hydroxy-4-[[3-methyl-5-(4-methylphenyl)pyrazol-1-yl]methyl]benzamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0553083
|
N-(4-(2-ethylhydrazine-1- carbonyl)benzyl)cinnamamide
Show/Hide
|
C19H21N3O2
|
1
|
| 1 |
IC50 = 76.57 nM
|
|
|
|
CP0013328
|
(7S)-7-amino-7-[2-(4-fluorophenyl)triazol-4-yl]-1-(1,2-oxazol-3-yl)heptan-1-one
Show/Hide
|
C18H20FN5O2
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0004235
|
N-[2-(cyclohexylamino)-2-oxoethyl]-N-[6-(hydroxyamino)-6-oxohexyl]-3,5-dimethylbenzamide
Show/Hide
|
C23H35N3O4
|
1
|
| 1 |
IC50 = 84 nM
|
|
|
|
CP0014401
|
(7S)-7-amino-7-[1-(4-fluorophenyl)pyrazol-3-yl]-1-(1,2-oxazol-3-yl)heptan-1-one
Show/Hide
|
C19H21FN4O2
|
1
|
| 1 |
IC50 = 86 nM
|
|
|
|
CP0395674
|
2-[4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]piperazin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C26H31N9O4
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
|
CP0030986
|
N-(4-(2-propylhydrazine-1- carbonyl)benzyl)cinnamamide
Show/Hide
|
C20H23N3O2
|
1
|
| 1 |
IC50 = 95.45 nM
|
|
|
|
CP0004957
|
(5R,8S,11R)-11-[(Z)-1-fluoro-4-sulfanylbut-1-enyl]-5-methyl-8-propan-2-yl-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-triene-6,9,13-trione
Show/Hide
|
C21H27FN4O4S3
|
1
|
| 1 |
IC50 = 95.51 nM
|
|
|
|
CP0455453
|
N-hydroxy-4-[(6-morpholin-4-yl-1,3-dioxobenzo[de]isoquinolin-2-yl)methyl]benzamide
Show/Hide
|
C24H21N3O5
|
1
|
| 1 |
IC50 = 98.8 nM
|
|
|
|
CP0514697
|
N-(4-(2-pentylhydrazine-1- carbonyl)benzyl)cinnamamide
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
IC50 = 99.56 nM
|
|
|
|
CP0011354
|
N-[(1S)-1-[5-(2-fluorophenyl)-1,3,4-oxadiazol-2-yl]-7-(1,2-oxazol-3-yl)-7-oxoheptyl]-1-methylazetidine-3-carboxamide
Show/Hide
|
C23H26FN5O4
|
1
|
| 1 |
IC50 = 101 nM
|
|
|
|
CP0010901
|
N'-hydroxy-N-[3-[2-(5,6,7-trimethoxyindol-1-yl)ethoxy]phenyl]octanediamide
Show/Hide
|
C27H35N3O7
|
1
|
| 1 |
IC50 = 111.2 nM
|
|
|
|
CP0374407
|
N'-hydroxy-N-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]octanediamide
Show/Hide
|
C17H20N4O5S
|
1
|
| 1 |
IC50 = 113 nM
|
|
|
|
CP0002498
|
4-[[3-(4-fluorophenyl)-5-methylpyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C18H16FN3O2
|
1
|
| 1 |
IC50 = 114 nM
|
|
|
|
CP0002022
|
2-[4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]sulfonylpiperazin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C26H31N9O6S
|
1
|
| 1 |
IC50 = 117 nM
|
|
|
|
CP0520599
|
N-[2-amino-5-(4-fluorophenyl)phenyl]-3,4-dihydro-1H-isochromene-3-carboxamide
Show/Hide
|
C22H19FN2O2
|
1
|
| 1 |
IC50 = 119 nM
|
|
|
|
CP0011388
|
4-[[5-(1,3-benzodioxol-5-yl)-3-methylpyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C19H17N3O4
|
1
|
| 1 |
IC50 = 135 nM
|
|
|
|
CP0514696
|
N-(4-(2-hexylhydrazine-1- carbonyl)benzyl)cinnamamide
Show/Hide
|
C23H29N3O2
|
1
|
| 1 |
IC50 = 139.2 nM
|
|
|
|
CP0010069
|
4-(dimethylamino)-N-[6-(hydroxyamino)-6-oxohexyl]-N-[2-(4-methylanilino)-2-oxoethyl]benzamide
Show/Hide
|
C24H32N4O4
|
1
|
| 1 |
IC50 = 146 nM
|
|
|
|
CP0111058
|
N-[4-[2-[[(2S)-2-amino-3-phenylpropanoyl]amino]phenyl]phenyl]-N'-hydroxyoctanediamide
Show/Hide
|
C29H34N4O4
|
1
|
| 1 |
IC50 = 156 nM
|
|
|
|
CP0427915
|
N-[2-amino-5-(4-fluorophenyl)phenyl]-3,4-dihydro-2H-chromene-3-carboxamide
Show/Hide
|
C22H19FN2O2
|
1
|
| 1 |
IC50 = 156 nM
|
|
|
|
CP0014421
|
2-[4-[4-ethoxy-N-methyl-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)anilino]piperidin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C28H35N9O4
|
1
|
| 1 |
IC50 = 166 nM
|
|
|
|
CP0436732
|
N-[4-[2-[[(2S)-2-amino-3-(1H-indol-3-yl)propanoyl]amino]phenyl]phenyl]-N'-hydroxyoctanediamide
Show/Hide
|
C31H35N5O4
|
1
|
| 1 |
IC50 = 167 nM
|
|
|
|
CP0447502
|
(1R,5S)-N-[2-amino-5-(4-fluorophenyl)phenyl]-8-oxabicyclo[3.2.1]octane-3-carboxamide
Show/Hide
|
C20H21FN2O2
|
2
|
| 1 |
IC50 = 168 nM
|
|
|
| 2 |
Ki = 519 nM
|
|
|
|
CP0426580
|
N'-hydroxy-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]pentanediamide
Show/Hide
|
C19H20N4O4
|
1
|
| 1 |
IC50 = 168 nM
|
|
|
|
CP0408928
|
N-[4-[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]phenyl]phenyl]-N'-hydroxyoctanediamide
Show/Hide
|
C29H34N4O5
|
1
|
| 1 |
IC50 = 205 nM
|
|
|
|
CP0634945
|
(E)-3-(3-bromo-4-hydroxyphenyl)-2-(hydroxyimino)-N-(2-mercaptoethyl)propanamide
Show/Hide
|
C11H13BrN2O3S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0379999
|
N-[2-amino-5-(4-fluorophenyl)phenyl]-3-oxabicyclo[3.1.0]hexane-6-carboxamide
Show/Hide
|
C18H17FN2O2
|
1
|
| 1 |
IC50 = 219 nM
|
|
|
|
CP0639104
|
(S)-1-methyl-N-(7-oxo-1-(4-phenyl-1H-imidazol-2-yl)-7-(pyridin-2-yl)heptyl)piperidine-4-carboxamide
Show/Hide
|
C28H35N5O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0004988
|
pyridin-3-ylmethyl N-[[4-[(2-aminophenyl)carbamoyl]phenyl]methyl]carbamate
Show/Hide
|
C21H20N4O3
|
2
|
| 1 |
IC50 = 247 nM
|
|
|
| 2 |
IC50 = 505 nM
|
|
|
|
CP0001056
|
N-hydroxy-7-[3-[4-[[(7-hydroxy-21-methyl-14-oxo-3,13,21-triazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-2(10),4(9),5,7,15(20),16,18-heptaen-17-yl)amino]methyl]phenyl]-1,2,4-oxadiazol-5-yl]heptanamide
Show/Hide
|
C35H37N7O5
|
1
|
| 1 |
IC50 = 275 nM
|
|
|
|
CP0010886
|
N-(2-aminophenyl)-4-[[[2-(benzylamino)-2-oxoethyl]-[4-(dimethylamino)benzoyl]amino]methyl]benzamide
Show/Hide
|
C32H33N5O3
|
1
|
| 1 |
IC50 = 283 nM
|
|
|
|
CP0545520
|
N-hydroxy-4-[[propan-2-yl-(2,3,4,5-tetrafluorophenyl)sulfonylamino]methyl]benzamide
Show/Hide
|
C17H16F4N2O4S
|
1
|
| 1 |
IC50 = 316 nM
|
|
|
|
CP0363242
|
US8609678, 2-((2-chlorophenyl)(phenyl)amino)-N-(7-(hydroxyamino)-7-oxoheptyl)pyrimidine-5-carboxamide [89]
Show/Hide
|
C24H26ClN5O3
|
2
|
| 1 |
IC50 = 318 nM
|
|
|
| 2 |
IC50 > 5000 nM
|
|
|
|
CP0005117
|
7-(3,4-dihydro-1H-isoquinolin-2-yl)-N-hydroxyheptanamide
Show/Hide
|
C16H24N2O2
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0010249
|
2-[4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]piperidin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C27H32N8O4
|
1
|
| 1 |
IC50 = 335 nM
|
|
|
|
CP0001244
|
2-[4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]sulfonylamino]piperidin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C27H33N9O6S
|
1
|
| 1 |
IC50 = 341 nM
|
|
|
|
CP0013110
|
4-[[3-(4-fluorophenyl)-5-propylpyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C20H20FN3O2
|
1
|
| 1 |
IC50 = 362 nM
|
|
|
|
CP0013857
|
4-[[5-ethyl-3-(4-fluorophenyl)pyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C19H18FN3O2
|
1
|
| 1 |
IC50 = 391 nM
|
|
|
|
CP0014885
|
N'-hydroxy-2-(3-imidazo[1,2-a]pyridin-2-ylphenyl)-3H-benzimidazole-5-carboximidamide
Show/Hide
|
C21H16N6O
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0385143
|
2-[4-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenoxy]piperidin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C26H30N8O5
|
1
|
| 1 |
IC50 = 432 nM
|
|
|
|
CP0637596
|
(S)-7-amino-1-(5-(hydroxymethyl)oxazol-2-yl)-7-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)heptan-1-one
Show/Hide
|
C24H27N5O4
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0013440
|
4-[(2-bromoacridin-9-yl)amino]-N-hydroxybenzamide
Show/Hide
|
C20H14BrN3O2
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0004189
|
N-[[4-[(2-aminophenyl)carbamoyl]phenyl]methyl]-N-[2-(benzylamino)-2-oxoethyl]-3,5-dimethylbenzamide
Show/Hide
|
C32H32N4O3
|
1
|
| 1 |
IC50 = 485 nM
|
|
|
|
CP0001245
|
2-[4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)anilino]piperidin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C27H33N9O4
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0007669
|
3-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxycyclobutane-1-carboxamide
Show/Hide
|
C22H27N5O4
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0424373
|
8-[3-(4-dimethylaminobenzyl)ureido]octanoic acid hydroxyamide
Show/Hide
|
C13H20N4O3
|
1
|
| 1 |
IC50 = 492 nM
|
|
|
|
CP0568663
|
[(2R,4S)-4-(3-chlorophenyl)pyrrolidin-2-yl]-(4-thieno[2,3-c]pyridin-7-ylpiperazin-1-yl)methanone
Show/Hide
|
C22H23ClN4OS
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0011389
|
N-hydroxy-4-[2-[3-(4-methylphenyl)-5-(trifluoromethyl)pyrazol-1-yl]ethyl]benzamide
Show/Hide
|
C20H18F3N3O2
|
1
|
| 1 |
IC50 = 549 nM
|
|
|
|
CP0014001
|
N-(2-aminophenyl)-4-[5-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]pentanoylamino]benzamide
Show/Hide
|
C33H33N7O7
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0013109
|
N-hydroxy-4-[2-[5-(4-methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]ethyl]benzamide
Show/Hide
|
C20H18F3N3O2
|
1
|
| 1 |
IC50 = 635 nM
|
|
|
|
CP0374405
|
1-(4-(dimethylamino)phenyl)-3-(7-(hydroxyamino)-7-oxoheptyl)urea
Show/Hide
|
C16H26N4O3
|
1
|
| 1 |
IC50 = 647 nM
|
|
|
|
CP0638821
|
(S)-7-amino-7-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)-1-(1H-pyrazol-3-yl)heptan-1-one
Show/Hide
|
C23H26N6O2
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0385177
|
2-[4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)anilino]methyl]piperidin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C28H35N9O4
|
1
|
| 1 |
IC50 = 712 nM
|
|
|
|
CP0007842
|
CHEMBL3955253
Show/Hide
|
C22H27N5O4
|
1
|
| 1 |
IC50 = 729 nM
|
|
|
|
CP0639105
|
(S)-7-amino-7-(5-(2-fluorophenyl)-1H-imidazol-2-yl)-1-(oxazol-4-yl)heptan-1-one
Show/Hide
|
C19H21FN4O2
|
1
|
| 1 |
IC50 = 740 nM
|
|
|
|
CP0015011
|
N-(2-aminophenyl)-4-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]heptanoylamino]benzamide
Show/Hide
|
C35H37N7O7
|
1
|
| 1 |
IC50 = 750 nM
|
|
|
|
CP0914610
|
(S)-N-(5-(2-hydroxy-5-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O4S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0003223
|
4-[[5-benzyl-3-(4-fluorophenyl)pyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C24H20FN3O2
|
1
|
| 1 |
IC50 = 763 nM
|
|
|
|
CP0012312
|
N-[[4-[(2-aminophenyl)carbamoyl]phenyl]methyl]-N-[2-(benzylamino)-2-oxoethyl]pyridine-3-carboxamide
Show/Hide
|
C29H27N5O3
|
1
|
| 1 |
IC50 = 786 nM
|
|
|
|
CP0456041
|
5-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)benzoyl]-N-hydroxythiophene-2-carboxamide
Show/Hide
|
C23H23N5O5S
|
1
|
| 1 |
IC50 = 799 nM
|
|
|
|
CP0014908
|
4-(acetylamino)-N-(2-amino-phenyl) benzamide
Show/Hide
|
C15H15N3O2
|
1
|
| 1 |
IC50 = 830 nM
|
|
|
|
CP0569146
|
2-[4-[(2R,4S)-4-(3-chlorophenyl)pyrrolidine-2-carbonyl]piperazin-1-yl]pyridine-3-carbonitrile
Show/Hide
|
C21H22ClN5O
|
1
|
| 1 |
IC50 = 850 nM
|
|
|
|
CP0012286
|
3-(4-fluorophenyl)-N-[5-(hydroxyamino)-5-oxopentyl]-1H-pyrazole-5-carboxamide
Show/Hide
|
C15H17FN4O3
|
1
|
| 1 |
IC50 = 883 nM
|
|
|
|
CP0011192
|
N-hydroxy-4-[5-(4-methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzamide
Show/Hide
|
C18H14F3N3O2
|
1
|
| 1 |
IC50 = 919 nM
|
|
|
|
CP0015290
|
N-(2-aminophenyl)-4-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexanoylamino]benzamide
Show/Hide
|
C32H32N6O6
|
1
|
| 1 |
IC50 = 970 nM
|
|
|
|
CP0001837
|
N'-hydroxy-N-[3-[4-(5,6,7-trimethoxyindol-1-yl)butoxy]phenyl]octanediamide
Show/Hide
|
C29H39N3O7
|
1
|
| 1 |
IC50 = 999.6 nM
|
|
|
|
CP0013434
|
N-(2-aminophenyl)-4-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentanoylamino]benzamide
Show/Hide
|
C31H30N6O6
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0053450
|
6-(3-adamantan-1-yl-ureido)hexanoic acid hydroxyamide
Show/Hide
|
C17H29N3O3
|
1
|
| 1 |
IC50 = 1050 nM
|
|
|
|
CP0410220
|
4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-methoxymethyl]-N-hydroxybenzamide
Show/Hide
|
C26H29N5O5
|
1
|
| 1 |
IC50 = 1110 nM
|
|
|
|
CP0489847
|
4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-hydroxymethyl]-N-hydroxybenzamide
Show/Hide
|
C25H27N5O5
|
1
|
| 1 |
IC50 = 1110 nM
|
|
|
|
CP0012142
|
N-(2-aminophenyl)-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoylamino]benzamide
Show/Hide
|
C30H28N6O6
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0011043
|
N-hydroxy-4-[[5-(4-methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]methyl]benzamide
Show/Hide
|
C19H16F3N3O2
|
1
|
| 1 |
IC50 = 1216 nM
|
|
|
|
CP0872331
|
(E)-N-Hydroxy-3-(4-oxo-3-phenethyl-3,4-dihydro-quinazolin-7-yl)-acrylamide
Show/Hide
|
C19H17N3O3
|
1
|
| 1 |
IC50 = 1220 nM
|
|
|
|
CP0014935
|
3-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxycyclobutane-1-carboxamide
Show/Hide
|
C22H27N5O4
|
1
|
| 1 |
IC50 = 1220 nM
|
|
|
|
CP0012954
|
N-[6-(2-aminoanilino)-6-oxohexyl]-N-[2-(benzylamino)-2-oxoethyl]-4-(dimethylamino)benzamide
Show/Hide
|
C30H37N5O3
|
1
|
| 1 |
IC50 = 1240 nM
|
|
|
|
CP0520711
|
(2R)-N-[2-amino-5-(4-fluorophenyl)phenyl]oxane-2-carboxamide
Show/Hide
|
C18H19FN2O2
|
1
|
| 1 |
IC50 = 1290 nM
|
|
|
|
CP0638862
|
(S)-7-amino-7-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)-1-(5-methylisoxazol-4-yl)heptan-1-one
Show/Hide
|
C24H27N5O3
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0455981
|
(E)-3-[4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]sulfonylamino]phenyl]-N-hydroxyprop-2-enamide
Show/Hide
|
C26H28N6O6S
|
1
|
| 1 |
IC50 = 1310 nM
|
|
|
|
CP0509880
|
(2S)-N-[2-amino-5-(4-fluorophenyl)phenyl]oxane-2-carboxamide
Show/Hide
|
C18H19FN2O2
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
|
CP0014542
|
N-(2-aminophenyl)-4-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]butanoylamino]benzamide
Show/Hide
|
C32H31N7O7
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0007688
|
4-[[3-ethyl-5-(4-fluorophenyl)pyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C19H18FN3O2
|
1
|
| 1 |
IC50 = 1503 nM
|
|
|
|
CP0004959
|
S-[(E)-4-[(5R,8S,11S)-5-methyl-6,9,13-trioxo-8-propan-2-yl-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-trien-11-yl]but-3-enyl] octanethioate
Show/Hide
|
C29H42N4O5S3
|
1
|
| 1 |
IC50 = 1520 nM
|
|
|
|
CP0014957
|
4-(acridin-9-ylamino)-N-hydroxybenzamide
Show/Hide
|
C20H15N3O2
|
1
|
| 1 |
IC50 = 1570 nM
|
|
|
|
CP0374538
|
CHEMBL3827055
Show/Hide
|
C20H21FN2O2
|
1
|
| 1 |
IC50 = 1590 nM
|
|
|
|
CP0015318
|
N-[6-(2-aminoanilino)-6-oxohexyl]-N-[2-(benzylamino)-2-oxoethyl]-3,5-dimethylbenzamide
Show/Hide
|
C30H36N4O3
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0703720
|
(E)-N-Hydroxy-3-(2-methyl-4-oxo-3-phenyl-3,4-dihydro-quinazolin-7-yl)-acrylamide
Show/Hide
|
C18H15N3O3
|
1
|
| 1 |
IC50 = 1610 nM
|
|
|
|
CP0578625
|
[(2R,4S)-4-phenylpyrrolidin-2-yl]-(4-thieno[2,3-c]pyridin-7-ylpiperazin-1-yl)methanone
Show/Hide
|
C22H24N4OS
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0572062
|
2-[4-[(2R,4S)-4-phenylpyrrolidine-2-carbonyl]piperazin-1-yl]pyridine-3-carbonitrile
Show/Hide
|
C21H23N5O
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0015319
|
N-[6-(2-amino-5-phenylanilino)-6-oxohexyl]-N-[2-(benzylamino)-2-oxoethyl]-3,5-dimethylbenzamide
Show/Hide
|
C36H40N4O3
|
1
|
| 1 |
IC50 = 1810 nM
|
|
|
|
CP0007715
|
S-[(Z)-4-fluoro-4-[(5R,8S,11S)-5-methyl-6,9,13-trioxo-8-propan-2-yl-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-trien-11-yl]but-3-enyl] octanethioate
Show/Hide
|
C29H41FN4O5S3
|
1
|
| 1 |
IC50 = 1817 nM
|
|
|
|
CP0003094
|
3-(4-fluorophenyl)-N-[4-(hydroxyamino)-4-oxobutyl]-1H-pyrazole-5-carboxamide
Show/Hide
|
C14H15FN4O3
|
1
|
| 1 |
IC50 = 1835 nM
|
|
|
|
CP0385178
|
2-[2-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-2,8-diazaspiro[4.5]decan-8-yl]-N-hydroxypyrimidine-5-carboxamide
Show/Hide
|
C30H37N9O4
|
1
|
| 1 |
IC50 = 1850 nM
|
|
|
|
CP0395683
|
3-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxycyclobutane-1-carboxamide
Show/Hide
|
C21H25N5O4
|
1
|
| 1 |
IC50 = 1860 nM
|
|
|
|
CP0385176
|
6-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxypyridine-3-carboxamide
Show/Hide
|
C22H22N6O4
|
1
|
| 1 |
IC50 = 1870 nM
|
|
|
|
CP0008774
|
N-[6-(2-aminoanilino)-6-oxohexyl]-N-[2-(benzylamino)-2-oxoethyl]naphthalene-1-carboxamide
Show/Hide
|
C32H34N4O3
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0749709
|
(S)-N-(5-(2-hydroxy-4-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O4S
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0385171
|
3-[1-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]sulfonylpiperidin-4-yl]-N-hydroxypropanamide
Show/Hide
|
C25H34N6O6S
|
1
|
| 1 |
IC50 = 1940 nM
|
|
|
|
CP0008380
|
4-[[5-(4-fluorophenyl)-3-methylpyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C18H16FN3O2
|
1
|
| 1 |
IC50 = 1974 nM
|
|
|
|
CP0014760
|
N-hydroxy-4-[[3-(1-methylpyrrolidin-2-yl)indol-1-yl]methyl]benzamide
Show/Hide
|
C21H23N3O2
|
1
|
| 1 |
IC50 = 1995.26 nM
|
|
|
|
CP0470868
|
3-[1-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]piperidin-4-yl]-N-hydroxypropanamide
Show/Hide
|
C25H34N6O4
|
1
|
| 1 |
IC50 = 2030 nM
|
|
|
|
CP0872330
|
(E)-N-Hydroxy-3-{3-[2-(1H-indol-3-yl)-ethyl]-2-methyl-4-oxo-3,4-dihydro-quinazolin-7-yl}-acrylamide
Show/Hide
|
C22H20N4O3
|
1
|
| 1 |
IC50 = 2210 nM
|
|
|
|
CP0419590
|
4-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenoxy]-N-hydroxybenzamide
Show/Hide
|
C23H23N5O5
|
1
|
| 1 |
IC50 = 2250 nM
|
|
|
|
CP0427674
|
4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxybenzamide
Show/Hide
|
C24H25N5O4
|
1
|
| 1 |
IC50 = 2550 nM
|
|
|
|
CP0013650
|
7-(dibenzylamino)-N-hydroxyheptanamide
Show/Hide
|
C21H28N2O2
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0013651
|
N-hydroxy-5-(1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl)pentanamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0550038
|
[(2R,4S)-4-(3-chlorophenyl)pyrrolidin-2-yl]-(1,3-dihydroisoindol-2-yl)methanone
Show/Hide
|
C19H19ClN2O
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
|
CP0013640
|
4-[[5-(4-fluorophenyl)-3-propylpyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C20H20FN3O2
|
1
|
| 1 |
IC50 = 2883 nM
|
|
|
|
CP0419775
|
N-hydroxy-4-[(5-pyrimidin-2-yltetrazol-2-yl)methyl]benzamide
Show/Hide
|
C13H11N7O2
|
1
|
| 1 |
IC50 = 3007 nM
|
|
|
|
CP0013604
|
N-[6-(2-amino-5-fluoroanilino)-6-oxohexyl]-N-[2-(benzylamino)-2-oxoethyl]-4-(dimethylamino)benzamide
Show/Hide
|
C30H36FN5O3
|
1
|
| 1 |
IC50 = 3060 nM
|
|
|
|
CP0013674
|
7-(benzylamino)-N-hydroxyheptanamide
Show/Hide
|
C14H22N2O2
|
1
|
| 1 |
IC50 = 3100 nM
|
|
|
|
CP0014641
|
N-hydroxy-4-[[3-(3-methylimidazol-4-yl)indol-1-yl]methyl]benzamide
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 = 3162.28 nM
|
|
|
|
CP0875931
|
4-((2-Ethyl-4-oxo-3-phenethyl-3,4-dihydroquinazolin-6-yl)-methyl)-N-hydroxybenzamide
Show/Hide
|
C26H25N3O3
|
1
|
| 1 |
IC50 = 3610 nM
|
|
|
|
CP0544515
|
N-hydroxy-4-[(5-thiophen-2-yltetrazol-1-yl)methyl]benzamide
Show/Hide
|
C13H11N5O2S
|
1
|
| 1 |
IC50 = 3698 nM
|
|
|
|
CP0012519
|
5-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxythiophene-2-carboxamide
Show/Hide
|
C23H25N5O4S
|
1
|
| 1 |
IC50 = 3720 nM
|
|
|
|
CP0003090
|
4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxybenzamide
Show/Hide
|
C25H27N5O4
|
1
|
| 1 |
IC50 = 3860 nM
|
|
|
|
CP0860467
|
(E)-3-(3-Benzyl-2-methyl-4-oxo-3,4-dihydro-quinazolin-7-yl)-N-hydroxy-acrylamide
Show/Hide
|
C19H17N3O3
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0578624
|
[(2R,4S)-4-(4-chlorophenyl)pyrrolidin-2-yl]-(1,3-dihydroisoindol-2-yl)methanone
Show/Hide
|
C19H19ClN2O
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0008775
|
N-[6-(2-aminoanilino)-6-oxohexyl]-N-[2-[(3,5-dimethylphenyl)methylamino]-2-oxoethyl]-3,5-dimethylbenzamide
Show/Hide
|
C32H40N4O3
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0014909
|
N-(2-amino-4-fluorophenyl)-4-[5-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]pentanoylamino]benzamide
Show/Hide
|
C33H32FN7O7
|
1
|
| 1 |
IC50 = 4200 nM
|
|
|
|
CP0201347
|
5-[[4-ethoxy-3-(5-methyl-4-oxo-7-propyl-3H-imidazo[5,1-f][1,2,4]triazin-2-yl)phenyl]methyl]-N-hydroxythiophene-2-carboxamide
Show/Hide
|
C23H25N5O4S
|
1
|
| 1 |
IC50 = 4390 nM
|
|
|
|
CP0012873
|
4-[[[2-(tert-butylamino)-2-oxoethyl]-(2-propan-2-ylbenzoyl)amino]methyl]-3-fluoro-N-hydroxybenzamide
Show/Hide
|
C24H30FN3O4
|
1
|
| 1 |
IC50 = 4480 nM
|
|
|
|
CP0564513
|
4-N-hydroxy-1-N-[6-(3-methoxyphenyl)-1H-indazol-3-yl]cyclohexane-1,4-dicarboxamide
Show/Hide
|
C22H24N4O4
|
1
|
| 1 |
IC50 = 4630 nM
|
|
|
|
CP0435952
|
4-(dimethylamino)-N-(6-(2-mercaptoacetamido)hexyl)benzamide
Show/Hide
|
C17H27N3O2S
|
1
|
| 1 |
IC50 = 4640 nM
|
|
|
|
CP0470875
|
4-[4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]sulfonylpiperazin-1-yl]-N-hydroxybutanamide
Show/Hide
|
C25H35N7O6S
|
1
|
| 1 |
IC50 = 4640 nM
|
|
|
|
CP0406317
|
N-[2-amino-5-(4-fluorophenyl)phenyl]oxane-3-carboxamide
Show/Hide
|
C18H19FN2O2
|
1
|
| 1 |
IC50 = 4730 nM
|
|
|
|
CP0847869
|
(E)-3-(2-Ethyl-3-(4-methoxyphenethyl)-4-oxo-3,4-dihydroquinazolin-7-yl)-N-hydroxyacrylamide
Show/Hide
|
C22H23N3O4
|
1
|
| 1 |
IC50 = 4780 nM
|
|
|
|
CP0410225
|
5-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxythiophene-2-carboxamide
Show/Hide
|
C22H23N5O4S
|
1
|
| 1 |
IC50 = 4800 nM
|
|
|
|
CP0738916
|
(E)-3-(2-Ethyl-4-oxo-3-phenethyl-3,4-dihydro-quinazolin-7-yl)-N-hydroxy-acrylamide
Show/Hide
|
C21H21N3O3
|
1
|
| 1 |
IC50 = 4810 nM
|
|
|
|
CP0637595
|
(S)-7-amino-1-(1H-imidazol-2-yl)-7-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)heptan-1-one
Show/Hide
|
C23H26N6O2
|
1
|
| 1 |
IC50 = 4900 nM
|
|
|
|
CP0014516
|
N-[6-(2-aminoanilino)-6-oxohexyl]-3,5-dimethyl-N-[2-[(4-methylphenyl)methylamino]-2-oxoethyl]benzamide
Show/Hide
|
C31H38N4O3
|
1
|
| 1 |
IC50 = 5030 nM
|
|
|
|
CP0410227
|
4-[[4-ethoxy-3-(5-methyl-4-oxo-7-propyl-3H-imidazo[5,1-f][1,2,4]triazin-2-yl)phenyl]methyl]-N-hydroxybenzamide
Show/Hide
|
C25H27N5O4
|
1
|
| 1 |
IC50 = 5190 nM
|
|
|
|
CP0010752
|
N-[6-(2-aminoanilino)-6-oxohexyl]-N-[2-(cyclohexylamino)-2-oxoethyl]naphthalene-1-carboxamide
Show/Hide
|
C31H38N4O3
|
1
|
| 1 |
IC50 = 5380 nM
|
|
|
|
CP0013984
|
5-(dibenzylamino)-N-hydroxypentanamide
Show/Hide
|
C19H24N2O2
|
1
|
| 1 |
IC50 = 5400 nM
|
|
|
|
CP0731873
|
(E)-3-(2-Ethyl-7-fluoro-4-oxo-3-phenethyl-3,4-dihydroquinazolin-6-yl)-N-hydroxyacrylamide
Show/Hide
|
C21H20FN3O3
|
1
|
| 1 |
IC50 = 5680 nM
|
|
|
|
CP0010751
|
N-[6-(2-aminoanilino)-6-oxohexyl]-N-[2-(cyclohexylamino)-2-oxoethyl]benzamide
Show/Hide
|
C27H36N4O3
|
1
|
| 1 |
IC50 = 5950 nM
|
|
|
|
CP0004941
|
N-hydroxy-4-[[3-(pyrrolidin-1-ylmethyl)indol-1-yl]methyl]benzamide
Show/Hide
|
C21H23N3O2
|
1
|
| 1 |
IC50 = 6309.57 nM
|
|
|
|
CP0014425
|
4-[[3-[(dimethylamino)methyl]indol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C19H21N3O2
|
1
|
| 1 |
IC50 = 6309.57 nM
|
|
|
|
CP0572061
|
1,3-dihydroisoindol-2-yl-[(2R,4S)-4-phenylpyrrolidin-2-yl]methanone
Show/Hide
|
C19H20N2O
|
1
|
| 1 |
IC50 = 6400 nM
|
|
|
|
CP0385169
|
6-[4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]piperidin-1-yl]-N-hydroxypyridine-3-carboxamide
Show/Hide
|
C28H33N7O4
|
1
|
| 1 |
IC50 = 6430 nM
|
|
|
|
CP0133369
|
(E)-N-hydroxy-3-[2-methyl-4-oxo-3-(2-phenylethyl)quinazolin-7-yl]prop-2-enamide
Show/Hide
|
C20H19N3O3
|
1
|
| 1 |
IC50 = 6450 nM
|
|
|
|
CP0424371
|
4-(dimethylamino)-N-(5-(2-mercaptoacetamido)pentyl)benzamide
Show/Hide
|
C16H25N3O2S
|
1
|
| 1 |
IC50 = 6460 nM
|
|
|
|
CP0473570
|
N-[2-amino-5-(4-fluorophenyl)phenyl]-3,4-dihydro-2H-chromene-2-carboxamide
Show/Hide
|
C22H19FN2O2
|
1
|
| 1 |
IC50 = 6560 nM
|
|
|
|
CP0012311
|
N-[6-(2-aminoanilino)-6-oxohexyl]-N-[2-(cyclohexylamino)-2-oxoethyl]-3,5-dimethylbenzamide
Show/Hide
|
C29H40N4O3
|
1
|
| 1 |
IC50 = 6660 nM
|
|
|
|
CP0909248
|
(E)-3-(2-Ethyl-3-(4-fluorophenethyl)-4-oxo-3,4-dihydroquinazolin-7-yl)-N-hydroxyacrylamide
Show/Hide
|
C21H20FN3O3
|
1
|
| 1 |
IC50 = 6880 nM
|
|
|
|
CP0395676
|
(E)-3-[4-[[4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]sulfonylpiperazin-1-yl]methyl]phenyl]-N-hydroxyprop-2-enamide
Show/Hide
|
C31H37N7O6S
|
1
|
| 1 |
IC50 = 6970 nM
|
|
|
|
CP0053451
|
6-(2-Mercapto-acetylamino)-hexanoic acid quinolin-8-ylamide
Show/Hide
|
C17H21N3O2S
|
1
|
| 1 |
IC50 = 7380 nM
|
|
|
|
CP0853807
|
(E)-N-Hydroxy-3-(2-methyl-4-oxo-3-phenyl-3,4-dihydro-quinazolin-6-yl)-acrylamide
Show/Hide
|
C18H15N3O3
|
1
|
| 1 |
IC50 = 7480 nM
|
|
|
|
CP0961838
|
(S)-N-(5-(2-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O3S
|
1
|
| 1 |
IC50 = 7700 nM
|
|
|
|
CP0007527
|
4-[[3-[(dimethylamino)methyl]indazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C18H20N4O2
|
1
|
| 1 |
IC50 = 7943.28 nM
|
|
|
|
CP0011676
|
4-(3,4-dihydro-1H-pyrano[4,3-b]indol-5-ylmethyl)-N-hydroxybenzamide
Show/Hide
|
C19H18N2O3
|
1
|
| 1 |
IC50 = 7943.28 nM
|
|
|
|
CP0418465
|
11-iodo-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9IN2S2
|
1
|
| 1 |
IC50 = 8100 nM
|
|
|
|
CP0011520
|
(2E)-3-(3-bromo-4-hydroxyphenyl)-N-[2-(hydroxyamino)-2-oxoethyl]-2-hydroxyiminopropanamide
Show/Hide
|
C11H12BrN3O5
|
1
|
| 1 |
IC50 = 9210 nM
|
|
|
|
CP0512440
|
3,5-difluoro-N-hydroxy-4-[(5-thiophen-2-yltetrazol-1-yl)methyl]benzamide
Show/Hide
|
C13H9F2N5O2S
|
1
|
| 1 |
IC50 = 9232 nM
|
|
|
|
CP0013395
|
N-(2-aminophenyl)-5-[[(2E)-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanoyl]amino]pentanamide
Show/Hide
|
C20H23BrN4O4
|
1
|
| 1 |
IC50 = 9760 nM
|
|
|
|
CP0463887
|
4-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenoxy]-N-hydroxycyclohexane-1-carboxamide
Show/Hide
|
C23H29N5O5
|
1
|
| 1 |
IC50 = 9830 nM
|
|
|
|
CP0007846
|
N-hydroxy-4-[(2-methyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)methyl]benzamide
Show/Hide
|
C20H21N3O2
|
3
|
| 1 |
IC50 = 9970 nM
|
|
|
| 2 |
IC50 = 12589.25 nM
|
|
|
| 3 |
IC50 > 30000 nM
|
|
|
|
CP0073930
|
4-[[2-ethyl-4-oxo-3-(2-phenylethyl)quinazolin-8-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C26H25N3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0857858
|
(E)-N-Hydroxy-3-(2-methyl-4-oxo-3-phenyl-3,4-dihydro-quinazolin-5-yl)-acrylamide
Show/Hide
|
C18H15N3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0860465
|
(E)-3-(2-Ethyl-6-fluoro-4-oxo-3-phenethyl-3,4-dihydroquinazolin-7-yl)-N-hydroxyacrylamide
Show/Hide
|
C21H20FN3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0862024
|
(E)-N-Hydroxy-3-(2-methyl-4-oxo-3-phenyl-3,4-dihydro-quinazolin-8-yl)-acrylamide
Show/Hide
|
C18H15N3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0007405
|
3-[[(2E)-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanoyl]amino]propanoic acid
Show/Hide
|
C12H13BrN2O5
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0007406
|
(2E)-3-(3-bromo-4-hydroxyphenyl)-N-(2-hydroxyethyl)-2-hydroxyiminopropanamide
Show/Hide
|
C11H13BrN2O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0008251
|
N-(2-aminophenyl)-4-[[(2E)-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanoyl]amino]butanamide
Show/Hide
|
C19H21BrN4O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0009098
|
(2E)-N-[3-(2-aminoanilino)-3-oxopropyl]-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanamide
Show/Hide
|
C18H19BrN4O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0014643
|
(2E)-3-(3-bromo-4-hydroxyphenyl)-N-butyl-2-hydroxyiminopropanamide
Show/Hide
|
C13H17BrN2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0014644
|
(2E)-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyimino-N-propylpropanamide
Show/Hide
|
C12H15BrN2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0014891
|
(2E)-N-[2-(2-aminoanilino)-2-oxoethyl]-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanamide
Show/Hide
|
C17H17BrN4O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0014892
|
5-[[(2E)-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanoyl]amino]-N-hydroxypentanamide
Show/Hide
|
C14H18BrN3O5
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0636555
|
(E)-4-(3-(3-Bromo-4-hydroxyphenyl)-2-(hydroxyimino)-propanamido)-N-hydroxybutanamide
Show/Hide
|
C13H16BrN3O5
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0003577
|
N-(2-amino-4-fluorophenyl)-3-[3-(tert-butylamino)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C24H24FN5O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0012152
|
N-tert-butyl-2-[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H18F3N5O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0013013
|
N-tert-butyl-2-[3-[6-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]-1H-benzimidazol-2-yl]phenyl]imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C27H22F3N7O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0013240
|
N-tert-butyl-2-[3-[6-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]-1H-benzimidazol-2-yl]phenyl]imidazo[1,2-a]pyrazin-3-amine
Show/Hide
|
C26H21F3N8O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0410221
|
4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenoxy]methyl]-N-hydroxybenzamide
Show/Hide
|
C25H27N5O5
|
1
|
| 1 |
IC50 = 11400 nM
|
|
|
|
CP0666156
|
(E)-3-(2-Ethyl-4-oxo-3-(3-phenylpropyl)-3,4-dihydroquinazolin-7-yl)-N-hydroxyacrylamide
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
IC50 > 12000 nM
|
|
|
|
CP0860466
|
(E)-3-(7-Chloro-2-ethyl-4-oxo-3-phenethyl-3,4-dihydroquinazolin-6-yl)-N-hydroxyacrylamide
Show/Hide
|
C21H20ClN3O3
|
1
|
| 1 |
IC50 > 12000 nM
|
|
|
|
CP0007526
|
US9249087, 8
Show/Hide
|
C18H18N2O2
|
1
|
| 1 |
IC50 = 12589.25 nM
|
|
|
|
CP0012958
|
N-hydroxy-3-(1-naphthalen-1-yl-3,4-dihydro-1H-isoquinolin-2-yl)propanamide
Show/Hide
|
C22H22N2O2
|
1
|
| 1 |
IC50 = 13000 nM
|
|
|
|
CP0385180
|
3-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxycyclopentane-1-carboxamide
Show/Hide
|
C23H29N5O4
|
1
|
| 1 |
IC50 = 13900 nM
|
|
|
|
CP0143013
|
11-chloro-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9ClN2S2
|
1
|
| 1 |
IC50 = 14000 nM
|
|
|
|
CP0458113
|
2-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxycyclopropane-1-carboxamide
Show/Hide
|
C21H25N5O4
|
1
|
| 1 |
IC50 = 14100 nM
|
|
|
|
CP0411308
|
4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-3-fluoro-N-hydroxybenzamide
Show/Hide
|
C25H26FN5O4
|
1
|
| 1 |
IC50 = 14600 nM
|
|
|
|
CP0473393
|
3,5-difluoro-N-hydroxy-4-[(5-pyrimidin-2-yltetrazol-2-yl)methyl]benzamide
Show/Hide
|
C13H9F2N7O2
|
1
|
| 1 |
IC50 = 17196 nM
|
|
|
|
CP0458110
|
4-[4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)anilino]piperidin-1-yl]-N-hydroxybenzamide
Show/Hide
|
C29H35N7O4
|
1
|
| 1 |
IC50 = 17500 nM
|
|
|
|
CP0012955
|
5-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxyfuran-2-carboxamide
Show/Hide
|
C23H25N5O5
|
1
|
| 1 |
IC50 = 17500 nM
|
|
|
|
CP0902876
|
(S)-N-(5-(2-mercaptobenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H27N5O2S2
|
1
|
| 1 |
IC50 = 18000 nM
|
|
|
|
CP0003596
|
3-[4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]phenyl]-N-hydroxypropanamide
Show/Hide
|
C26H29N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0385168
|
2-[1-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]piperidin-4-yl]-N-hydroxyacetamide
Show/Hide
|
C24H32N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0385170
|
5-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxyfuran-2-carboxamide
Show/Hide
|
C21H21N5O5
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0385172
|
2-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxy-2-azaspiro[5.5]undecane-9-carboxamide
Show/Hide
|
C28H38N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0385173
|
4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)-N-hydroxybenzamide
Show/Hide
|
C17H19N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0385174
|
3-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxypropanamide
Show/Hide
|
C19H23N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0385175
|
4-[4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]piperidin-1-yl]-N-hydroxybenzamide
Show/Hide
|
C29H34N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0385179
|
3-[4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]piperidin-1-yl]-N-hydroxypropanamide
Show/Hide
|
C25H34N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0385181
|
1-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxyazetidine-3-carboxamide
Show/Hide
|
C21H26N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0395675
|
2-[4-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]cyclohexyl]-N-hydroxyacetamide
Show/Hide
|
C24H31N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0419618
|
4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxycyclohexane-1-carboxamide
Show/Hide
|
C24H31N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0419620
|
2-[4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]cyclohexyl]-N-hydroxyacetamide
Show/Hide
|
C25H33N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0446576
|
5-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxypyridine-2-carboxamide
Show/Hide
|
C22H22N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0458108
|
3-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)anilino]-N-hydroxypropanamide
Show/Hide
|
C20H26N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0458109
|
8-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxy-8-azaspiro[4.5]decane-3-carboxamide
Show/Hide
|
C27H36N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0458111
|
4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxycyclohexane-1-carboxamide
Show/Hide
|
C24H31N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0458112
|
4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)anilino]-N-hydroxycyclohexane-1-carboxamide
Show/Hide
|
C24H32N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0463889
|
2-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxycyclopropane-1-carboxamide
Show/Hide
|
C20H23N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0470869
|
3-[4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]sulfonylpiperazin-1-yl]-N-hydroxypropanamide
Show/Hide
|
C24H33N7O6S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0470874
|
(E)-3-[4-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]phenyl]-N-hydroxyprop-2-enamide
Show/Hide
|
C26H27N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0477630
|
1-[[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxypiperidine-4-carboxamide
Show/Hide
|
C23H30N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0525405
|
2-[4-ethoxy-3-(3-ethyl-1-methyl-7-oxo-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxyacetamide
Show/Hide
|
C18H21N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0003091
|
2-[4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]phenyl]-N-hydroxyacetamide
Show/Hide
|
C26H29N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0396658
|
2-[4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]phenyl]-N-hydroxyacetamide
Show/Hide
|
C25H27N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0409165
|
4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-2-fluoro-N-hydroxybenzamide
Show/Hide
|
C25H26FN5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0411310
|
4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxy-3-methoxybenzamide
Show/Hide
|
C26H29N5O5
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0411311
|
4-[4-ethoxy-3-(5-methyl-4-oxo-7-propyl-3H-imidazo[5,1-f][1,2,4]triazin-2-yl)phenyl]-N-hydroxybenzamide
Show/Hide
|
C24H25N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0413948
|
1-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxypiperidine-4-carboxamide
Show/Hide
|
C23H30N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0413950
|
4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxycyclohex-3-ene-1-carboxamide
Show/Hide
|
C24H29N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0427293
|
4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)anilino]-N-hydroxybenzamide
Show/Hide
|
C24H26N6O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0456039
|
4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxycyclohexane-1-carboxamide
Show/Hide
|
C24H31N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0477735
|
4-[[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]methyl]-N-hydroxy-2-methoxybenzamide
Show/Hide
|
C26H29N5O5
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0489845
|
4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxycyclohexane-1-carboxamide
Show/Hide
|
C24H31N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0489846
|
4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]-N-hydroxycyclohexane-1-carboxamide
Show/Hide
|
C24H31N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0526726
|
2-[4-[4-ethoxy-3-(1-methyl-7-oxo-3-propyl-6H-pyrazolo[4,3-d]pyrimidin-5-yl)phenyl]cyclohex-3-en-1-yl]-N-hydroxyacetamide
Show/Hide
|
C25H31N5O4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0011675
|
N-hydroxy-4-[(2-methyl-3,4-dihydro-1H-pyrido[3,4-b]indol-9-yl)methyl]benzamide
Show/Hide
|
C20H21N3O2
|
1
|
| 1 |
IC50 = 25118.86 nM
|
|
|
|
CP0577167
|
[(2R,4S)-4-phenylpyrrolidin-2-yl]-pyrrolidin-1-ylmethanone
Show/Hide
|
C15H20N2O
|
1
|
| 1 |
IC50 = 26000 nM
|
|
|
|
CP0012490
|
3-[1-(4-tert-butylphenyl)-3,4-dihydro-1H-isoquinolin-2-yl]-N-hydroxypropanamide
Show/Hide
|
C22H28N2O2
|
1
|
| 1 |
IC50 = 29000 nM
|
|
|
|
CP0955788
|
(S)-N-(5-(2-cyclopropylbenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C32H31N5O2S
|
1
|
| 1 |
IC50 = 29000 nM
|
|
|
|
CP0374410
|
1-(6-(2-mercaptoacetamido)hexyl)-3-phenylurea
Show/Hide
|
C15H23N3O2S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0394609
|
4-Dimethylamino-N-[3-(2-mercapto-acetylamino)-propyl]-benzamide
Show/Hide
|
C14H21N3O2S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0435947
|
4-Dimethylamino-N-[4-(2-mercapto-acetylamino)-butyl]-benzamide
Show/Hide
|
C15H23N3O2S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0014148
|
N-hydroxy-1-[(4-methoxyphenyl)methyl]indole-6-carboxamide
Show/Hide
|
C17H16N2O3
|
1
|
| 1 |
IC50 = 31000 nM
|
|
|
|
CP0742396
|
(S)-N-(5-(2-(methylthio)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O2S2
|
1
|
| 1 |
IC50 = 31000 nM
|
|
|
|
CP0001717
|
N-hydroxy-3-(1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl)propanamide
Show/Hide
|
C18H20N2O2
|
1
|
| 1 |
IC50 = 40000 nM
|
|
|
|
CP0914609
|
(S)-N-(5-(2-fluoro-6-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H28FN5O3S
|
1
|
| 1 |
IC50 = 40000 nM
|
|
|
|
CP0902998
|
N-((1S)-5-(2-(methylsulfinyl)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O3S2
|
1
|
| 1 |
IC50 = 43000 nM
|
|
|
|
CP0418461
|
10-bromo-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7BrN2S2
|
1
|
| 1 |
IC50 = 45000 nM
|
|
|
|
CP0350774
|
N-[(1S)-1-[5-(2-methoxyquinolin-3-yl)-1,3,4-oxadiazol-2-yl]-5-[(2-methylsulfanylbenzoyl)amino]pentyl]-1,3-thiazole-5-carboxamide
Show/Hide
|
C29H28N6O4S2
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0767213
|
(S)-N-(5-(2-hydroxy-3-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O4S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0835239
|
(S)-N-(5-(2-(methylamino)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H30N6O2S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0840085
|
(S)-N-(5-(3-aminopicolinamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C28H27N7O2S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0882461
|
(S)-N-(1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)-5-(2-(trifluoromethoxy)benzamido)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H26F3N5O3S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0882462
|
(S)-N-(1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)-5-(2-(2,2,2-trifluoroethoxy)benzamido)pentyl)thiazole-5-carboxamide
Show/Hide
|
C31H28F3N5O3S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0882463
|
(S)-N-(5-(2-cyanobenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H26N6O2S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0898602
|
(S)-N-(5-(2-hydroxy-6-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O4S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0902996
|
(S)-N-(5-(2-(dimethylamino)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C31H32N6O2S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0902997
|
(S)-N-(5-(2-chlorobenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H26ClN5O2S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0928234
|
(S)-N-(5-(2,3-dihydro-1H-indene-4-carboxamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C32H31N5O2S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0928238
|
(S)-N-(5-(2-(ethylthio)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C31H31N5O2S2
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0942943
|
(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)-5-(2-(methylthio)benzamido)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H30N6O3S2
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0946826
|
(S)-N-(5-(2-(1H-pyrrol-1-yl)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C33H30N6O2S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0958717
|
(S)-N-(5-(2-ethylbenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C31H31N5O2S
|
1
|
| 1 |
IC50 > 45000 nM
|
|
|
|
CP0013653
|
N-hydroxy-3-[1-(4-phenylphenyl)-3,4-dihydro-1H-isoquinolin-2-yl]propanamide
Show/Hide
|
C24H24N2O2
|
1
|
| 1 |
IC50 = 47000 nM
|
|
|
|
CP0418462
|
10-chloro-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9ClN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0418463
|
8-fluoro-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9FN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0418464
|
5-sulfanylidene-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-8-carbonitrile
Show/Hide
|
C11H7N3S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0418467
|
8-(dimethylamino)-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C12H13N3S2
|
1
|
| 1 |
IC50 = 50000 nM
|
|
|
|
CP0418468
|
8-methyl-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C12H12N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0422674
|
6-sulfanylidene-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-9-carbonitrile
Show/Hide
|
C12H9N3S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0422675
|
10-bromo-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9BrN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0422676
|
9-chloro-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9ClN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0422677
|
9-bromo-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7BrN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0422678
|
9-fluoro-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9FN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426103
|
9-iodo-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7IN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426105
|
9-methyl-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C11H10N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426106
|
3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H10N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426107
|
9-fluoro-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7FN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426108
|
10-(trifluoromethyl)-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C12H9F3N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426109
|
9-bromo-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9BrN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426110
|
11-fluoro-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9FN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426111
|
8-bromo-10-fluoro-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H6BrFN2S2
|
1
|
| 1 |
IC50 = 50000 nM
|
|
|
|
CP0426112
|
7-methyl-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C11H10N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426113
|
10-methyl-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C12H12N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426114
|
8-bromo-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7BrN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426115
|
10-iodo-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9IN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0426116
|
9-(dimethylamino)-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C13H15N3S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0439954
|
10-fluoro-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7FN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0439955
|
11-bromo-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9BrN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0439956
|
8-chloro-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9ClN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0439958
|
10-fluoro-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C11H9FN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0473304
|
10-iodo-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7IN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0473315
|
7-chloro-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7ClN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0473316
|
2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H8N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0473317
|
9-methyl-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C12H12N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0473318
|
10-chloro-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7ClN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0488055
|
9-chloro-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7ClN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0488064
|
8-methyl-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C11H10N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0528002
|
8-chloro-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7ClN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0528005
|
7-fluoro-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C10H7FN2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0533759
|
8-methoxy-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C11H10N2OS2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0540902
|
11-methyl-3,4-dihydro-2H-pyrimido[1,2-c][1,3]benzothiazine-6-thione
Show/Hide
|
C12H12N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0542076
|
9-methoxy-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C11H10N2OS2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0549146
|
10-methyl-2,3-dihydroimidazo[1,2-c][1,3]benzothiazine-5-thione
Show/Hide
|
C11H10N2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0001716
|
5-(benzylamino)-N-hydroxypentanamide
Show/Hide
|
C12H18N2O2
|
1
|
| 1 |
IC50 = 58000 nM
|
|
|
|
CP0014113
|
N-hydroxy-3-[1-(3-methoxyphenyl)-3,4-dihydro-1H-isoquinolin-2-yl]propanamide
Show/Hide
|
C19H22N2O3
|
1
|
| 1 |
IC50 = 69000 nM
|
|
|
|
CP0012488
|
3-[1-(4-ethoxyphenyl)-3,4-dihydro-1H-isoquinolin-2-yl]-N-hydroxypropanamide
Show/Hide
|
C20H24N2O3
|
1
|
| 1 |
IC50 = 99000 nM
|
|
|
|
CP0227283
|
N-hydroxy-4-[2-(6-morpholin-4-yl-1,3-dioxobenzo[de]isoquinolin-2-yl)ethyl]benzamide
Show/Hide
|
C25H23N3O5
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0005364
|
N-hydroxy-2-(1-phenyl-3,4-dihydro-1H-isoquinolin-2-yl)acetamide
Show/Hide
|
C17H18N2O2
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0010479
|
N-hydroxy-3-[1-(4-methoxyphenyl)-3,4-dihydro-1H-isoquinolin-2-yl]propanamide
Show/Hide
|
C19H22N2O3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0012487
|
3-(benzylamino)-N-hydroxypropanamide
Show/Hide
|
C10H14N2O2
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0012489
|
N-hydroxy-3-[1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinolin-2-yl]propanamide
Show/Hide
|
C19H19F3N2O2
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0013652
|
3-(1-cyclohexyl-3,4-dihydro-1H-isoquinolin-2-yl)-N-hydroxypropanamide
Show/Hide
|
C18H26N2O2
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0013675
|
3-(3,4-dihydro-1H-isoquinolin-2-yl)-N-hydroxypropanamide
Show/Hide
|
C12H16N2O2
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0014112
|
3-(dibenzylamino)-N-hydroxypropanamide
Show/Hide
|
C17H20N2O2
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0014147
|
N-hydroxy-3-[1-[3-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinolin-2-yl]propanamide
Show/Hide
|
C19H19F3N2O2
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0417643
|
4-tert-butyl-N-[4-(hydroxycarbamoyl)phenyl]benzamide
Show/Hide
|
C18H20N2O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0007404
|
(E)-N-(2-amino-4-fluorophenyl)-3-[1-[(E)-3-phenylprop-2-enyl]pyrazol-4-yl]prop-2-enamide
Show/Hide
|
C21H19FN4O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0011853
|
N-(2-aminophenyl)-8-[[(2E)-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanoyl]amino]octanamide
Show/Hide
|
C23H29BrN4O4
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0013313
|
N-(2-aminophenyl)-7-[[(2E)-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanoyl]amino]heptanamide
Show/Hide
|
C22H27BrN4O4
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0014890
|
N-(2-aminophenyl)-6-[[(2E)-3-(3-bromo-4-hydroxyphenyl)-2-hydroxyiminopropanoyl]amino]hexanamide
Show/Hide
|
C21H25BrN4O4
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0421417
|
2,3,4,5,6-pentafluoro-N-[[4-(hydroxycarbamoyl)phenyl]methyl]benzamide
Show/Hide
|
C15H9F5N2O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0542777
|
4-[[cyclopropyl-(2,3,4,5-tetrafluorophenyl)sulfonylamino]methyl]-N-hydroxybenzamide
Show/Hide
|
C17H14F4N2O4S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0007689
|
4-[[3-benzyl-5-(4-fluorophenyl)pyrazol-1-yl]methyl]-N-hydroxybenzamide
Show/Hide
|
C24H20FN3O2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0011048
|
3-(4-fluorophenyl)-N-[3-(hydroxyamino)-3-oxopropyl]-1H-pyrazole-5-carboxamide
Show/Hide
|
C13H13FN4O3
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
