| Compound ID |
Compound Name |
Compound Formula |
|
CP0452766
|
4-(2-((R)-2-(4-methylocta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C22H29NO3
|
2
|
| 1 |
EC50 = 0.1 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0380631
|
(S)-4-(1-(1-(3-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23F3N2O3
|
2
|
| 1 |
EC50 = 0.2 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0379617
|
(S)-4-(1-(1-(3,5-dibromobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H22Br2N2O3
|
2
|
| 1 |
EC50 = 0.36 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0457559
|
4-(2-((R)-2-oxo-5-(4-phenylpenta-1,3-dienyl)pyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C24H25NO3
|
2
|
| 1 |
EC50 = 0.5 nM
|
|
|
| 2 |
Ki = 29 nM
|
|
|
|
CP0379615
|
(S)-4-(1-(1-(3-chlorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H23ClN2O3
|
2
|
| 1 |
EC50 = 0.82 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0483781
|
4-(2-((R)-2-(octa-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C21H27NO3
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
Ki = 25 nM
|
|
|
|
CP0381433
|
(R)-5-((E)-(S)-3-Hydroxy-4-phenyl-but-1-enyl)-1-[6-(1H-tetrazol-5-yl)-hexyl]-pyrrolidin-2-one
Show/Hide
|
C21H29N5O2
|
1
|
| 1 |
EC50 = 2.5 nM
|
|
|
|
CP0055947
|
(15S)-prostaglandin E2
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|
C20H32O5
|
4
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
IC50 = 0.55 nM
|
|
|
| 3 |
Ki = 0.11 nM
|
|
|
| 4 |
Ki = 0.79 nM
|
|
|
|
CP0457560
|
4-(2-((R)-2-(4-methylhexa-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C20H25NO3
|
2
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
Ki = 24 nM
|
|
|
|
CP0464526
|
(R)-4-(2-(2-(4-methylpenta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C19H23NO3
|
2
|
| 1 |
EC50 = 4 nM
|
|
|
| 2 |
Ki = 45 nM
|
|
|
|
CP0423796
|
4-[2-[3,5-dichloro-2-(3-hydroxyoctyl)-6-oxopyridin-1-yl]ethyl]benzoic acid
Show/Hide
|
C22H27Cl2NO4
|
1
|
| 1 |
EC50 = 4.9 nM
|
|
|
|
CP0464527
|
4-(2-((R)-2-(4-methylocta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C22H29NO3
|
2
|
| 1 |
EC50 = 15 nM
|
|
|
| 2 |
Ki = 181 nM
|
|
|
|
CP0452767
|
4-(2-((R)-2-(3-methylocta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C22H29NO3
|
2
|
| 1 |
EC50 = 21 nM
|
|
|
| 2 |
Ki = 145 nM
|
|
|
|
CP0437308
|
4-[2-[3,5-dichloro-2-[(E)-3-hydroxy-3-methyloct-1-enyl]-6-oxopyridin-1-yl]ethyl]benzoic acid
Show/Hide
|
C23H27Cl2NO4
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0525833
|
7-[3,5-dichloro-2-[(E)-3-hydroxyoct-1-enyl]-6-oxopyridin-1-yl]heptanoic acid
Show/Hide
|
C20H29Cl2NO4
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0487510
|
7-[3,5-dibromo-2-[(E)-3-hydroxyoct-1-enyl]-6-oxopyridin-1-yl]heptanoic acid
Show/Hide
|
C20H29Br2NO4
|
1
|
| 1 |
EC50 = 360 nM
|
|
|
|
CP0437306
|
7-[2-(3-hydroxyoctyl)-6-oxopyridin-1-yl]heptanoic acid
Show/Hide
|
C20H33NO4
|
1
|
| 1 |
EC50 = 550 nM
|
|
|
|
CP0847236
|
5-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
Show/Hide
|
C23H29NO5S
|
3
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 6032 nM
|
|
|
| 3 |
Ki >= 6032 nM
|
|
|
|
CP0847237
|
5-{3-[(S)-1-(4-Hexanoyl-phenyl)-5-oxo-pyrrolidin-2-yl]-propyl}-thiophene-2-carboxylic acid
Show/Hide
|
C24H29NO4S
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0847239
|
5-{(R)-1-[4-(1-Hydroxy-propyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
Show/Hide
|
C20H23NO5S
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0847241
|
3-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-benzoic acid
Show/Hide
|
C23H27NO4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0847242
|
5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-thiophene-2-carboxylic acid
Show/Hide
|
C21H25NO4S
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0847243
|
5-{(R)-1-[4-(1-Hydroxy-heptyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
Show/Hide
|
C24H31NO5S
|
3
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 3288 nM
|
|
|
| 3 |
Ki >= 3288 nM
|
|
|
|
CP0852841
|
methyl 7-((1R,2S,3R)-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)heptanoate
Show/Hide
|
C27H40O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0856823
|
methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(hydroxymethyl)phenyl)cyclopentyl)heptanoate
Show/Hide
|
C20H29ClO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0856827
|
7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2,2-dimethylpropyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
|
C23H35ClO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866241
|
5-(3-{(S)-1-[4-(1-Hydroxy-heptyl)-phenyl]-5-oxo-pyrrolidin-2-yl}-propyl)-thiophene-2-carboxylic acid
Show/Hide
|
C25H33NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866245
|
7-((1R,2S)-2-(4-((R)-hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
|
C26H36O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866253
|
N-ethyl-7-((1R,2S,3R)-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)hept-5-enamide
Show/Hide
|
C26H37NO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866254
|
7-((1R,2S,3R,5R)-2-(4-tert-butylphenyl)-5-chloro-3-hydroxycyclopentyl)hept-5-enoic acid
Show/Hide
|
C22H31ClO3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866285
|
methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2,2-dimethylpropyl)phenyl)cyclopentyl)heptanoate
Show/Hide
|
C24H37ClO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866287
|
7-((1R,2S,3S,5R)-3,5-dichloro-2-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
|
C24H34Cl2O3
|
2
|
| 1 |
EC50 = 10000 nM
|
|
|
| 2 |
Ki = 2364 nM
|
|
|
|
CP0866394
|
methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropan-2-yl)phenyl)cyclopentyl)hept-5-enoate
Show/Hide
|
C23H33ClO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866431
|
methyl 7-((1R,2S,3R)-2-(4-tert-butylphenyl)-3-hydroxy-5-oxocyclopentyl)heptanoate
Show/Hide
|
C23H34O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866744
|
7-[(S)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-yl]-heptanoic acid
Show/Hide
|
C21H31NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0870239
|
5-(3-((1R,2S)-2-(4-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)propyl)thiophene-2-carboxylic acid
Show/Hide
|
C25H32O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0870431
|
5-(3-{(S)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-yl}-propyl)-thiophene-2-carboxylic acid
Show/Hide
|
C24H31NO4S
|
3
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki >= 3842 nM
|
|
|
| 3 |
Ki > 4849 nM
|
|
|
|
CP0882892
|
methyl 7-((1R,2S,3R)-2-(2,3-dihydro-1H-inden-5-yl)-3-hydroxy-5-oxocyclopentyl)heptanoate
Show/Hide
|
C22H30O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0883084
|
5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxy]-pentanoic acid
Show/Hide
|
C20H29NO4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0885328
|
5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-furan-2-carboxylic acid
Show/Hide
|
C21H25NO5
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0888294
|
methyl 7-((1R,2S,3R)-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoate
Show/Hide
|
C27H38O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0888315
|
7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2,2-dimethylpropyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
|
C23H33ClO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0895714
|
7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropan-2-yl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
|
C22H33ClO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0899422
|
methyl 7-((1R,2S,3R)-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxy-5-oxocyclopentyl)hept-5-enoate
Show/Hide
|
C26H36O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0920862
|
methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropyl)phenyl)cyclopentyl)hept-5-enoate
Show/Hide
|
C23H33ClO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0928827
|
methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropan-2-yl)phenyl)cyclopentyl)heptanoate
Show/Hide
|
C23H35ClO4
|
1
|
| 1 |
EC50 >= 10000 nM
|
|
|
|
CP0966505
|
methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropyl)phenyl)cyclopentyl)heptanoate
Show/Hide
|
C23H35ClO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0909260
|
methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(1-hydroxy-2,3-dihydro-1H-inden-5-yl)cyclopentyl)heptanoate
Show/Hide
|
C22H31ClO4
|
1
|
| 1 |
EC50 = 22457 nM
|
|
|
|
CP0542668
|
4-[[5-[3-(hydroxymethyl)phenyl]-2-methylbenzoyl]amino]-3,5-dimethylbenzoic acid
Show/Hide
|
C24H23NO4
|
1
|
| 1 |
IC50 = 0.28 nM
|
|
|
|
CP0473344
|
4-[(1S)-1-[[5-[(E)-prop-1-enyl]-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
|
C23H21F3N4O3
|
4
|
| 1 |
IC50 = 0.4 nM
|
|
|
| 2 |
IC50 = 5.2 nM
|
|
|
| 3 |
IC50 = 18.7 nM
|
|
|
| 4 |
Kd = 5.623 nM
|
|
|
|
CP0542669
|
4-[[6-[3-(hydroxymethyl)phenyl]-3-(trifluoromethyl)pyridine-2-carbonyl]amino]-3,5-dimethylbenzoic acid
Show/Hide
|
C23H19F3N2O4
|
1
|
| 1 |
IC50 = 0.67 nM
|
|
|
|
CP0566830
|
4-[[6-[3-(hydroxymethyl)phenyl]-3-methylpyridine-2-carbonyl]amino]-3,5-dimethylbenzoic acid
Show/Hide
|
C23H22N2O4
|
1
|
| 1 |
IC50 = 0.67 nM
|
|
|
|
CP0573581
|
4-[[2-fluoro-5-[3-(hydroxymethyl)phenyl]benzoyl]amino]-3,5-dimethylbenzoic acid
Show/Hide
|
C23H20FNO4
|
1
|
| 1 |
IC50 = 0.73 nM
|
|
|
|
CP0468170
|
(S)-4-(1-(1-(4-chlorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H23ClN2O3
|
1
|
| 1 |
IC50 = 0.92 nM
|
|
|
|
CP0473507
|
(S)-4-(1-(1-(3,4-dichlorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H22Cl2N2O3
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0048414
|
4-[[3-[3-(hydroxymethyl)phenyl]naphthalene-1-carbonyl]amino]-3,5-dimethylbenzoic acid
Show/Hide
|
C27H23NO4
|
1
|
| 1 |
IC50 = 1.11 nM
|
|
|
|
CP0388647
|
(S)-4-(1-(5-chloro-1-(4-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H20ClF3N2O3
|
1
|
| 1 |
IC50 = 1.12 nM
|
|
|
|
CP0372255
|
4-(1-(5-chloro-1-(4-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)cyclopropyl)benzoic acid
Show/Hide
|
C27H20ClF3N2O3
|
1
|
| 1 |
IC50 = 1.26 nM
|
|
|
|
CP0374156
|
4-(1-(1-(4-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)cyclopropyl)benzoic acid
Show/Hide
|
C27H21F3N2O3
|
2
|
| 1 |
IC50 = 1.3 nM
|
|
|
| 2 |
IC50 = 1.8 nM
|
|
|
|
CP0437430
|
(S)-4-(1-(1-(biphenyl-4-ylmethyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C31H28N2O3
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0388650
|
(S)-4-(1-(1-(3-chloro-5-(trifluoromethoxy)benzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H20ClF3N2O4
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0388649
|
(S)-4-(1-(5-chloro-1-(3-chlorobenzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H20Cl2N2O3
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0502291
|
1-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-3-(4-methylphenyl)sulfonylurea
Show/Hide
|
C35H37N3O6S
|
4
|
| 1 |
IC50 = 1.5 nM
|
|
|
| 2 |
IC50 = 17 nM
|
|
|
| 3 |
Ki = 0.11 nM
|
|
|
| 4 |
Ki = 10 nM
|
|
|
|
CP0462026
|
3-[[6-(3-chlorophenyl)-3-methylpyridine-2-carbonyl]amino]-2,4-dimethylbenzoic acid
Show/Hide
|
C22H19ClN2O3
|
1
|
| 1 |
IC50 = 1.56 nM
|
|
|
|
CP0383780
|
4-[({[2,5-Dichloro-4-(3-chlorobenzyl)-3-thienyl]carbonyl}amino)methyl]benzoic acid
Show/Hide
|
C20H14Cl3NO3S
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0510062
|
4-[[6-(4,4-difluoropiperidin-1-yl)-3-methylpyridine-2-carbonyl]amino]-3,5-dimethylbenzoic acid
Show/Hide
|
C21H23F2N3O3
|
1
|
| 1 |
IC50 = 1.61 nM
|
|
|
|
CP0383779
|
4-[(1R)-1-({[2,5-Dichloro-4-(3-chlorobenzyl)-3-thienyl]carbonyl}amino)ethyl]benzoic acid
Show/Hide
|
C21H16Cl3NO3S
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0550583
|
3-[[6-[3-(hydroxymethyl)phenyl]-3-(trifluoromethyl)pyridine-2-carbonyl]amino]-2,4-dimethylbenzoic acid
Show/Hide
|
C23H19F3N2O4
|
1
|
| 1 |
IC50 = 1.94 nM
|
|
|
|
CP0424258
|
2,3-dichloro-N-(1-(4-(4,9-diethoxy-1-oxo-1H-benzo[f]isoindol-2(3H)-yl)-3-methylbenzyl)cyclopropylcarbamoyl)benzenesulfonamide
Show/Hide
|
C34H33Cl2N3O6S
|
4
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 28 nM
|
|
|
| 3 |
Ki = 0.4 nM
|
|
|
| 4 |
Ki = 64 nM
|
|
|
|
CP0091346
|
4-[(1S)-1-[[2-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzoxepine-10-carbonyl]amino]ethyl]benzoic acid
Show/Hide
|
C25H20F3NO4
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 20 nM
|
|
|
|
CP0393826
|
(S)-4-(1-(1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23F3N2O3
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1
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| 1 |
IC50 = 2.1 nM
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CP0402997
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(S)-4-(1-(5-fluoro-1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H22F4N2O3
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1
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| 1 |
IC50 = 2.1 nM
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CP0472248
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2-(2,4-dichlorophenyl)-N-(1-(4-(4,9-diethoxy-1-oxo-1H-benzo[f]isoindol-2(3H)-yl)-3-methylbenzyl)cyclopropyl)acetamide
Show/Hide
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C35H34Cl2N2O4
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4
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| 1 |
IC50 = 2.1 nM
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| 2 |
IC50 = 10.2 nM
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| 3 |
Ki = 0.34 nM
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| 4 |
Ki = 0.53 nM
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CP0377873
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(S)-4-(1-(5-chloro-1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H22ClF3N2O3
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1
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| 1 |
IC50 = 2.2 nM
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CP0465769
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2-bromo-N-(1-(4-(4,9-diethoxy-1-oxo-1H-benzo[f]isoindol-2(3H)-yl)-3-methylbenzyl)cyclopropylcarbamoyl)benzenesulfonamide
Show/Hide
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C34H34BrN3O6S
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4
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| 1 |
IC50 = 2.2 nM
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| 2 |
IC50 = 22 nM
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| 3 |
Ki = 0.49 nM
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| 4 |
Ki = 7.5 nM
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CP0469926
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US8969394, 14
Show/Hide
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C25H22F3N5OS
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1
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| 1 |
IC50 = 2.3 nM
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CP0458979
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3-[[5-[3-(hydroxymethyl)phenyl]-2-methylbenzoyl]amino]-2,4-dimethylbenzoic acid
Show/Hide
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C24H23NO4
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1
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| 1 |
IC50 = 2.31 nM
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CP0045472
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3-[[6-[3-(hydroxymethyl)phenyl]-3-methylpyridine-2-carbonyl]amino]-2,4-dimethylbenzoic acid
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C23H22N2O4
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1
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| 1 |
IC50 = 2.36 nM
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CP0474316
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2-chloro-N-(1-(4-(4,9-diethoxy-1-oxo-1H-benzo[f]isoindol-2(3H)-yl)-3-methylbenzyl)cyclopropylcarbamoyl)benzenesulfonamide
Show/Hide
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C34H34ClN3O6S
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4
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| 1 |
IC50 = 2.4 nM
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| 2 |
IC50 = 33 nM
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| 3 |
Ki = 0.16 nM
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| 4 |
Ki = 2.3 nM
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CP0082042
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4-[(1S)-1-[[5-chloro-2-(3-fluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H16ClFN2O4
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4
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| 1 |
IC50 = 2.4 nM
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| 2 |
IC50 = 16.3 nM
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| 3 |
Kd = 1.072 nM
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| 4 |
Ki = 0.97 nM
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CP0198309
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3-[[3-[3-(hydroxymethyl)phenyl]naphthalene-1-carbonyl]amino]-2,4-dimethylbenzoic acid
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C27H23NO4
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1
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| 1 |
IC50 = 2.42 nM
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CP0452755
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4-{1-[({2,5-Dimethyl-4-[4-(trifluoromethyl)benzyl]-3-thienyl}-carbonyl)amino]cyclopropyl}benzoic Acid
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C25H22F3NO3S
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2
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| 1 |
IC50 = 2.5 nM
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| 2 |
IC50 = 2.9 nM
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CP0490022
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1-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-3-naphthalen-2-ylsulfonylurea
Show/Hide
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C38H37N3O6S
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4
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| 1 |
IC50 = 2.5 nM
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| 2 |
IC50 = 37 nM
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| 3 |
Ki = 0.52 nM
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| 4 |
Ki = 6.3 nM
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CP0411079
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(S)-4-(1-(1-(4-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H21F3N2O3
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1
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| 1 |
IC50 = 2.7 nM
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CP0380630
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(S)-4-(1-(1-(4-(trifluoromethoxy)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H23F3N2O4
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1
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| 1 |
IC50 = 2.8 nM
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CP0718063
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(2R)-2-((S)-1-(4-carboxyphenyl)ethylcarbamoyl)-1-(2-(4-fluorophenoxy)ethyl)piperidinium chloride
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C23H28ClFN2O4
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3
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| 1 |
IC50 = 2.87 nM
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| 2 |
IC50 = 71.8 nM
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| 3 |
Ki = 40.4 nM
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CP0508827
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(S)-4-(1-(5-(trifluoromethyl)-1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C27H22F6N2O3
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1
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| 1 |
IC50 = 3 nM
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CP0459038
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2,6-dichloro-N-(1-(4-(4,9-diethoxy-1-oxo-1H-benzo[f]isoindol-2(3H)-yl)-3-methylbenzyl)cyclopropylcarbamoyl)benzenesulfonamide
Show/Hide
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C34H33Cl2N3O6S
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4
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| 1 |
IC50 = 3 nM
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| 2 |
IC50 = 14 nM
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| 3 |
Ki = 0.3 nM
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| 4 |
Ki = 3.1 nM
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CP0505590
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2-chloro-N-(1-(3-methyl-4-(6-oxo-5,9-bis(2,2,2-trifluoroethoxy)-6H-pyrrolo[3,4-g]quinolin-7(8H)-yl)benzyl)cyclopropylcarbamoyl)benzenesulfonamide
Show/Hide
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C33H27ClF6N4O6S
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4
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| 1 |
IC50 = 3 nM
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| 2 |
IC50 = 48 nM
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| 3 |
Ki = 0.48 nM
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| 4 |
Ki = 14 nM
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CP0048413
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4-[[2-[3-(hydroxymethyl)phenyl]quinoline-4-carbonyl]amino]-3,5-dimethylbenzoic acid
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C26H22N2O4
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1
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| 1 |
IC50 = 3.08 nM
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CP0499458
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2,6-dimethyl-N-(1-(4-(4,9-diethoxy-1-oxo-1H-benzo[f]isoindol-2(3H)-yl)-3-methylbenzyl)cyclopropylcarbamoyl)benzenesulfonamide
Show/Hide
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C36H39N3O6S
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4
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| 1 |
IC50 = 3.2 nM
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| 2 |
IC50 = 19 nM
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| 3 |
Ki = 0.4 nM
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| 4 |
Ki = 1.6 nM
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CP0372247
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(S)-4-(1-(1-(3-chlorobenzyl)-5-fluoro-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C25H20ClFN2O3
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1
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| 1 |
IC50 = 3.3 nM
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CP0465768
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1-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-3-[2-(trifluoromethyl)phenyl]sulfonylurea
Show/Hide
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C35H34F3N3O6S
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4
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| 1 |
IC50 = 3.3 nM
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| 2 |
IC50 = 28 nM
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| 3 |
Ki = 0.39 nM
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| 4 |
Ki = 8.9 nM
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CP0469274
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1-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-3-(2,6-dimethoxyphenyl)sulfonylurea
Show/Hide
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C36H39N3O8S
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4
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| 1 |
IC50 = 3.3 nM
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| 2 |
IC50 = 21 nM
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| 3 |
Ki = 0.34 nM
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| 4 |
Ki = 1.6 nM
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CP0502661
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1-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-3-(2-methylphenyl)sulfonylurea
Show/Hide
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C35H37N3O6S
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4
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| 1 |
IC50 = 3.3 nM
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| 2 |
IC50 = 14 nM
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| 3 |
Ki = 0.23 nM
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| 4 |
Ki = 3 nM
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CP0198225
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3,5-dimethyl-4-[(3-phenylnaphthalene-1-carbonyl)amino]benzoic acid
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C26H21NO3
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1
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| 1 |
IC50 = 3.48 nM
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CP0393828
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(S)-N-(1-(4-(2H-tetrazol-5-yl)phenyl)ethyl)-1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamide
Show/Hide
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C26H23F3N6O
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1
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| 1 |
IC50 = 3.5 nM
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CP0469928
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4-[(1S)-1-({[2,5-Dichloro-4-(3-chlorobenzyl)-3-thienyl]carbonyl}-amino)ethyl]benzoic Acid
Show/Hide
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C21H16Cl3NO3S
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1
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| 1 |
IC50 = 3.6 nM
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CP0048416
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3-[[3-(3-chlorophenyl)naphthalene-1-carbonyl]amino]-2,4-dimethylbenzoic acid
Show/Hide
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C26H20ClNO3
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1
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| 1 |
IC50 = 3.62 nM
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CP0441382
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3-(2-(1-(4-(4,9-diethoxy-1-oxo-1H-benzo[f]isoindol-2(3H)-yl)-3-methylbenzyl)cyclopropylamino)-2-oxoethyl)-4-methoxybenzoic acid
Show/Hide
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C37H38N2O7
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4
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| 1 |
IC50 = 3.8 nM
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| 2 |
IC50 = 60.6 nM
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| 3 |
Ki = 0.18 nM
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| 4 |
Ki = 6.2 nM
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CP0503018
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1-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-3-(2-methoxyphenyl)sulfonylurea
Show/Hide
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C35H37N3O7S
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4
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| 1 |
IC50 = 3.8 nM
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| 2 |
IC50 = 23 nM
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| 3 |
Ki = 0.17 nM
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| 4 |
Ki = 3 nM
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CP0060088
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4-[1-[[2-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzoxepine-10-carbonyl]amino]cyclopropyl]benzoic acid
Show/Hide
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C26H20F3NO4
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2
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 1000 nM
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CP0566829
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3-[[2-fluoro-5-[3-(hydroxymethyl)phenyl]benzoyl]amino]-2,4-dimethylbenzoic acid
Show/Hide
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C23H20FNO4
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1
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| 1 |
IC50 = 4.49 nM
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CP0489160
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4-{(1S)-1-[({2,5-Dimethyl-4-[4-(trifluoromethyl)benzyl]-3-thienyl}-carbonyl)amino]ethyl}benzoic acid
Show/Hide
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C24H22F3NO3S
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1
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| 1 |
IC50 = 4.5 nM
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CP0425392
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1-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-3-(4-fluorophenyl)sulfonylurea
Show/Hide
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C34H34FN3O6S
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4
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| 1 |
IC50 = 4.6 nM
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| 2 |
IC50 = 80 nM
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| 3 |
Ki = 0.48 nM
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| 4 |
Ki = 21 nM
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CP0489252
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N-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-2-(2-methoxyphenyl)acetamide
Show/Hide
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C36H38N2O5
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4
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| 1 |
IC50 = 4.6 nM
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| 2 |
IC50 = 16 nM
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| 3 |
Ki = 0.2 nM
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| 4 |
Ki = 0.68 nM
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CP0447496
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4-{(1S)-1-[({2,5-Dimethyl-4-[3-(trifluoromethyl)benzyl]-3-thienyl}carbonyl)amino]ethyl}benzoic Acid
Show/Hide
|
C24H22F3NO3S
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1
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| 1 |
IC50 = 4.7 nM
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CP0393829
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(S)-4-(1-(1-(2-bromo-4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H22BrF3N2O3
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1
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| 1 |
IC50 = 4.7 nM
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CP0489243
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N-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-2-(3-methoxypyridin-2-yl)acetamide
Show/Hide
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C35H37N3O5
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4
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| 1 |
IC50 = 4.9 nM
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| 2 |
IC50 = 23.6 nM
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| 3 |
Ki = 0.16 nM
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| 4 |
Ki = 1.44 nM
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CP0569215
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4-[[[2-[(4-fluorophenyl)methyl]-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carbonyl]amino]methyl]benzoic acid
Show/Hide
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C23H20FNO4S
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2
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| 1 |
IC50 = 5 nM
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| 2 |
Kd = 6.714 nM
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CP0238730
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4-[(1S)-1-[[5-chloro-2-(3-chlorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H16Cl2N2O4
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2
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| 1 |
IC50 = 5.02 nM
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| 2 |
IC50 = 21.8 nM
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CP0198224
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3-[[2-[3-(hydroxymethyl)phenyl]quinoline-4-carbonyl]amino]-2,4-dimethylbenzoic acid
Show/Hide
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C26H22N2O4
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1
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| 1 |
IC50 = 5.2 nM
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CP0447789
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4-[(1S)-1-({[4-(4-Chlorobenzyl)-2,5-dimethyl-3-thienyl]carbonyl}-amino)ethyl]benzoicAcid
Show/Hide
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C23H22ClNO3S
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1
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| 1 |
IC50 = 5.4 nM
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CP0801377
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(2R)-2-(1-(4-carboxyphenyl)cyclopropylcarbamoyl)-1-(2-phenoxyethyl)piperidinium chloride
Show/Hide
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C24H29ClN2O4
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3
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| 1 |
IC50 = 5.42 nM
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| 2 |
IC50 = 77.8 nM
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| 3 |
Ki = 44.8 nM
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CP0663915
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4-((S)-1-((R)-1-(2-phenoxyethyl)piperidine-2-carboxamido)ethyl)benzoic acid hydrochloride
Show/Hide
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C23H29ClN2O4
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3
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| 1 |
IC50 = 5.62 nM
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| 2 |
IC50 = 68.8 nM
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| 3 |
Ki = 40.6 nM
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CP0045193
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US8933098, 1
Show/Hide
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C21H25N3O4
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1
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| 1 |
IC50 = 5.62 nM
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CP0233548
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2,4-dimethyl-3-[(3-phenylnaphthalene-1-carbonyl)amino]benzoic acid
Show/Hide
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C26H21NO3
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1
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| 1 |
IC50 = 5.65 nM
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CP0474166
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(S)-4-(1-(1-(4-methylbenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H26N2O3
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1
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| 1 |
IC50 = 5.8 nM
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CP0377878
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(S)-4-(1-(1-(3-chlorobenzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C25H21ClN2O3
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2
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| 1 |
IC50 = 5.9 nM
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| 2 |
IC50 = 6 nM
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CP0425391
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2-(2-chlorophenyl)-N-(1-(4-(4,9-diethoxy-1-oxo-1H-benzo[f]isoindol-2(3H)-yl)-3-methylbenzyl)cyclopropyl)acetamide
Show/Hide
|
C35H35ClN2O4
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4
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 35.1 nM
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| 3 |
Ki = 0.32 nM
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| 4 |
Ki = 1.3 nM
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CP0477213
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(S)-4-(1-(1-(4-fluorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H23FN2O3
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1
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| 1 |
IC50 = 6.2 nM
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CP0092571
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4-[(1S)-1-[[5-chloro-2-(4-fluorophenoxy)benzoyl]amino]ethyl]benzoic acid
Show/Hide
|
C22H17ClFNO4
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5
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| 1 |
IC50 = 6.59 nM
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| 2 |
IC50 = 10 nM
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| 3 |
IC50 = 13 nM
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| 4 |
IC50 = 38.2 nM
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| 5 |
Kd = 1.778 nM
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CP0522152
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(S)-4-(1-(1-(4-cyanobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H23N3O3
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1
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| 1 |
IC50 = 7.3 nM
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CP0475979
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(S)-4-(1-(1-(2-bromo-4-chlorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H22BrClN2O3
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1
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| 1 |
IC50 = 8.3 nM
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CP0490023
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1-[1-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methyl]cyclopropyl]-3-[4-(trifluoromethoxy)phenyl]sulfonylurea
Show/Hide
|
C35H34F3N3O7S
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4
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| 1 |
IC50 = 8.3 nM
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| 2 |
IC50 = 370 nM
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| 3 |
Ki = 0.66 nM
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| 4 |
Ki = 57 nM
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CP0371889
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4-[(1S)-1-({[4-(3-Chlorobenzyl)-2,5-dimethyl-3-thienyl]carbonyl}-amino)ethyl]benzoic Acid
Show/Hide
|
C23H22ClNO3S
|
1
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| 1 |
IC50 = 8.6 nM
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CP0092570
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4-[(1S)-1-[[5-chloro-2-(3-fluorophenoxy)benzoyl]amino]ethyl]benzoic acid
Show/Hide
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C22H17ClFNO4
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3
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| 1 |
IC50 = 8.76 nM
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| 2 |
IC50 = 30.6 nM
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| 3 |
Kd = 1.259 nM
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CP0469279
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1-[1-[[3-methyl-4-[6-oxo-5,9-bis(2,2,2-trifluoroethoxy)-8H-pyrrolo[3,4-g]quinolin-7-yl]phenyl]methyl]cyclopropyl]-3-naphthalen-2-ylsulfonylurea
Show/Hide
|
C37H30F6N4O6S
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4
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| 1 |
IC50 = 8.9 nM
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| 2 |
IC50 = 103 nM
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| 3 |
Ki = 1.2 nM
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| 4 |
Ki = 21 nM
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CP0118996
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4-[(1S)-1-[[5-chloro-2-(4-fluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
|
C21H16ClFN2O4
|
3
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| 1 |
IC50 = 9.68 nM
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| 2 |
IC50 = 25.9 nM
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| 3 |
Kd = 2.455 nM
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CP0572549
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3,5-dimethyl-4-[(2-phenylquinoline-4-carbonyl)amino]benzoic acid
Show/Hide
|
C25H20N2O3
|
1
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| 1 |
IC50 = 11.2 nM
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CP0065814
|
AAT-007
Show/Hide
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C26H29N5O3S
|
5
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| 1 |
IC50 = 11.7 nM
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| 2 |
IC50 = 689 nM
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| 3 |
Kd = 4.786 nM
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| 4 |
Ki = 13 nM
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| 5 |
Ki = 449 nM
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CP0388651
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(S)-4-(1-(1-(3-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
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C26H21F3N2O3
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1
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| 1 |
IC50 = 11.8 nM
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CP0481524
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4-[(1S)-1-({[4-(3-Chlorobenzyl)-3-thienyl]carbonyl}amino)ethyl]-benzoic Acid
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C21H18ClNO3S
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1
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| 1 |
IC50 = 12 nM
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CP0196909
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4-[(1S)-1-[[5-chloro-2-(3-cyanophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
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C22H16ClN3O4
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2
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| 1 |
IC50 = 13.4 nM
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| 2 |
IC50 = 36.2 nM
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CP0447995
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3-[[6-[3-(hydroxymethyl)piperidin-1-yl]-3-methylpyridine-2-carbonyl]amino]-2,4-dimethylbenzoic acid
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C22H27N3O4
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1
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| 1 |
IC50 = 14.2 nM
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CP0852327
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(2R)-2-((S)-1-(4-carboxyphenyl)propylcarbamoyl)-1-(2-phenoxyethyl)piperidinium chloride
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C24H31ClN2O4
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3
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| 1 |
IC50 = 14.4 nM
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| 2 |
IC50 = 232 nM
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| 3 |
Ki = 129 nM
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CP0510063
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4-[[6-[3-(hydroxymethyl)piperidin-1-yl]-3-methylpyridine-2-carbonyl]amino]-3,5-dimethylbenzoic acid
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C22H27N3O4
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1
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| 1 |
IC50 = 16.5 nM
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CP0719709
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(2R)-2-(4-carboxybenzylcarbamoyl)-1-(2-phenoxyethyl)piperidinium chloride
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C22H27ClN2O4
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3
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| 1 |
IC50 = 18.1 nM
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| 2 |
IC50 = 203 nM
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| 3 |
Ki = 126 nM
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CP0435681
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US8686018, 107
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C22H18F5N3O4
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1
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| 1 |
IC50 = 18.5 nM
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CP0407422
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3-[[6-(4-hydroxypiperidin-1-yl)-3-methylpyridine-2-carbonyl]amino]-2,4-dimethylbenzoic acid
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C21H25N3O4
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1
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| 1 |
IC50 = 19.5 nM
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CP0196940
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4-[[[5-chloro-2-(4-fluorophenoxy)benzoyl]amino]methyl]benzoic acid
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C21H15ClFNO4
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2
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| 1 |
IC50 = 21.6 nM
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| 2 |
IC50 = 101 nM
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CP0060089
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4-[1-[[3-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzoxepine-10-carbonyl]amino]cyclopropyl]benzoic acid
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C26H20F3NO4
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2
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| 1 |
IC50 = 27 nM
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| 2 |
IC50 = 34 nM
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CP0119018
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4-[(1S)-1-[[5-fluoro-2-(4-fluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
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C21H16F2N2O4
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2
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| 1 |
IC50 = 28.7 nM
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| 2 |
IC50 = 143 nM
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CP0801376
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(2R)-2-((S)-1-(4-carboxyphenyl)ethylcarbamoyl)-1-(2-(4-cyanophenoxy)ethyl)piperidinium chloride
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C24H28ClN3O4
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3
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| 1 |
IC50 = 35.8 nM
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| 2 |
IC50 = 621 nM
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| 3 |
Ki = 372 nM
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CP0196908
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4-[[[5-chloro-2-(4-fluorophenoxy)pyridine-3-carbonyl]amino]methyl]benzoic acid
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C20H14ClFN2O4
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2
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| 1 |
IC50 = 37.9 nM
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| 2 |
IC50 = 254 nM
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CP0407421
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4-[[6-(4-hydroxy-4-methylpiperidin-1-yl)-3-methylpyridine-2-carbonyl]amino]-3,5-dimethylbenzoic acid
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C22H27N3O4
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1
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| 1 |
IC50 = 39.8 nM
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CP0119016
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4-[(1S)-1-[[5-chloro-2-(3-chlorophenoxy)benzoyl]amino]ethyl]benzoic acid
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C22H17Cl2NO4
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1
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| 1 |
IC50 = 41.1 nM
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CP0060087
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4-[(1S)-1-[[3-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzoxepine-10-carbonyl]amino]ethyl]benzoic acid
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C25H20F3NO4
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2
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| 1 |
IC50 = 42 nM
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| 2 |
IC50 = 63 nM
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CP0454821
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4-[(1S)-1-[[5-chloro-2-(3,4-difluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
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C21H15ClF2N2O4
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1
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| 1 |
IC50 < 50 nM
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CP0476701
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4-[(1S)-1-[[5-chloro-2-(3,5-difluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H15ClF2N2O4
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1
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| 1 |
IC50 < 50 nM
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CP0564720
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4-[(1S)-1-[[5-chloro-2-(2,3-difluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H15ClF2N2O4
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1
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| 1 |
IC50 < 50 nM
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CP0564721
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4-[(1S)-1-[[5-chloro-2-(2,5-difluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H15ClF2N2O4
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1
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| 1 |
IC50 < 50 nM
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CP0114103
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4-[(1S)-1-[[5-chloro-2-[3-(trifluoromethyl)phenoxy]pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C22H16ClF3N2O4
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1
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| 1 |
IC50 = 60.4 nM
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CP0244132
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4-[(1S)-1-[[5-chloro-2-(2-fluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H16ClFN2O4
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1
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| 1 |
IC50 = 61.4 nM
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CP0402996
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(S)-4-(1-(1-(3-carbamoylbenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H25N3O4
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1
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| 1 |
IC50 = 72 nM
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CP0474165
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(S)-4-(1-(1-(4-carbamoylbenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H25N3O4
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1
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| 1 |
IC50 = 73 nM
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CP0414568
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4-[[6-[3-(hydroxymethyl)pyrrolidin-1-yl]-3-methylpyridine-2-carbonyl]amino]-3,5-dimethylbenzoic acid
Show/Hide
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C21H25N3O4
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1
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| 1 |
IC50 = 84 nM
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CP0414751
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3-[[6-(4-hydroxy-4-methylpiperidin-1-yl)-3-methylpyridine-2-carbonyl]amino]-2,4-dimethylbenzoic acid
Show/Hide
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C22H27N3O4
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1
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| 1 |
IC50 = 87.9 nM
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CP0081993
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4-[(1S)-1-[[5-chloro-2-(2-chlorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H16Cl2N2O4
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1
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| 1 |
IC50 = 93.5 nM
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CP0238731
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4-[(1S)-1-[[5-chloro-2-(4-chlorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H16Cl2N2O4
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1
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| 1 |
IC50 = 94.3 nM
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CP0474128
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4-[[6-(4-methoxypiperidin-1-yl)-3-methylpyridine-2-carbonyl]amino]-3,5-dimethylbenzoic acid
Show/Hide
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C22H27N3O4
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1
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| 1 |
IC50 = 96.7 nM
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CP0082041
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4-[[[5-fluoro-2-(4-fluorophenoxy)pyridine-3-carbonyl]amino]methyl]benzoic acid
Show/Hide
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C20H14F2N2O4
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3
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| 1 |
IC50 = 104 nM
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| 2 |
IC50 = 575 nM
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| 3 |
Ki = 73 nM
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CP0477214
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(S)-4-(1-(1-(4-tert-butylbenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C29H32N2O3
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1
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| 1 |
IC50 = 114 nM
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CP0119017
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4-[[[5-fluoro-2-(4-fluorophenoxy)benzoyl]amino]methyl]benzoic acid
Show/Hide
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C21H15F2NO4
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2
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| 1 |
IC50 = 124 nM
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| 2 |
IC50 = 317 nM
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CP0061222
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N-(2,6-dimethylphenyl)-2-phenylquinoline-4-carboxamide
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C24H20N2O
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1
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| 1 |
IC50 = 128 nM
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CP0196938
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4-[(1S)-1-[[5-chloro-2-(5-chloropyridin-3-yl)oxypyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C20H15Cl2N3O4
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1
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| 1 |
IC50 = 137 nM
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CP0119021
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4-[(1S)-1-[[5-chloro-2-(5-fluoropyridin-3-yl)oxypyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C20H15ClFN3O4
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1
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| 1 |
IC50 = 175 nM
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CP0244131
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4-[1-[[5-fluoro-2-(4-fluorophenoxy)pyridine-3-carbonyl]amino]propyl]benzoic acid
Show/Hide
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C22H18F2N2O4
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1
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| 1 |
IC50 = 181 nM
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CP0380405
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(S)-4-(1-(1-(3-cyanobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C26H23N3O3
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1
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| 1 |
IC50 = 212 nM
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CP0380632
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(S)-4-(1-(1-(pyridin-3-ylmethyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
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C24H23N3O3
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1
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| 1 |
IC50 = 258 nM
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CP0533934
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N-[[4-[(3-chlorophenyl)sulfonylcarbamoyl]phenyl]methyl]-3-[(5-fluoro-1,3-benzothiazol-2-yl)methoxy]benzamide
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C29H21ClFN3O5S2
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1
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| 1 |
IC50 = 302 nM
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CP0082043
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4-[(1S)-1-[[5-chloro-2-(3-methoxyphenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C22H19ClN2O5
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1
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| 1 |
IC50 = 340 nM
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CP0533935
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4-[[[3-[(5-fluoro-1,3-benzothiazol-2-yl)methoxy]benzoyl]amino]methyl]benzoic acid
Show/Hide
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C23H17FN2O4S
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1
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| 1 |
IC50 = 370 nM
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CP0196910
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4-[(1S)-1-[[5-chloro-2-(3-methylsulfanylphenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C22H19ClN2O4S
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1
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| 1 |
IC50 = 400 nM
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CP0244567
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4-[2-[[5-fluoro-2-(4-fluorophenoxy)pyridine-3-carbonyl]amino]propan-2-yl]benzoic acid
Show/Hide
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C22H18F2N2O4
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1
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| 1 |
IC50 = 545 nM
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CP0119019
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4-[(1R)-1-[[5-chloro-2-(4-fluorophenoxy)pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C21H16ClFN2O4
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1
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| 1 |
IC50 = 1210 nM
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CP0323441
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4-[(1S)-1-[[5-chloro-2-[3-(trifluoromethoxy)phenoxy]pyridine-3-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C22H16ClF3N2O5
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1
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| 1 |
IC50 = 1790 nM
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CP0244566
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4-[[[2-(4-fluorophenoxy)-5-methylpyridine-3-carbonyl]amino]methyl]benzoic acid
Show/Hide
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C21H17FN2O4
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1
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| 1 |
IC50 = 2940 nM
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CP0042409
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2-[2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C28H26N2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0055418
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2-[6-chloro-2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C20H15Cl2FN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0055420
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2-[2-(3-chlorobenzoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C20H17ClN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0055873
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2-[8-fluoro-2-[2-(1H-indol-3-yl)acetyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C23H20FN3O3
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1
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| 1 |
IC50 > 10000 nM
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CP0086399
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2-[6-chloro-2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C28H25ClN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0086409
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2-[8-fluoro-2-(2-naphthalen-1-ylacetyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C25H21FN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0156867
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2-[2-(cyclohexanecarbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C20H24N2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0156868
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2-[6-chloro-8-fluoro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C24H18ClFN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0199029
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2-(2-benzoyl-8-propan-2-yl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
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C23H24N2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0199053
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2-(2-benzoyl-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
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C21H20N2O4
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1
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| 1 |
IC50 > 10000 nM
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CP0042410
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2-[8-chloro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C24H19ClN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0045673
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2-[2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C20H16ClFN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0055416
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2-[2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C24H20N2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0055874
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2-[8-fluoro-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C18H15FN2O3S
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1
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| 1 |
IC50 > 10000 nM
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CP0055877
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2-[2-benzoyl-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C21H17F3N2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0070143
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2-(2-benzoyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
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C20H18N2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0083568
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2-[8-fluoro-2-(3-naphthalen-1-ylpropanoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C26H23FN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0087804
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ACT-129968
Show/Hide
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C24H19FN2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0130562
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2-[8-methyl-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C25H22N2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0261961
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2-[2-(naphthalene-1-carbonyl)-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C25H19F3N2O3
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1
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| 1 |
IC50 > 10000 nM
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CP0863771
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methyl 7-((1R,2S,3R,5R)-5-chloro-2-(2,3-dihydro-1H-inden-5-yl)-3-hydroxycyclopentyl)heptanoate
Show/Hide
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C22H31ClO3
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1
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| 1 |
IC50 = 13100 nM
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CP0413856
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4-[4-[(2,6-dimethylphenyl)carbamoyl]quinolin-2-yl]benzoic acid
Show/Hide
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C25H20N2O3
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1
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| 1 |
IC50 > 25000 nM
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CP0196939
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4-[[[2-(4-fluorophenoxy)-6-methylpyridine-3-carbonyl]amino]methyl]benzoic acid
Show/Hide
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C21H17FN2O4
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1
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| 1 |
IC50 > 5000 nM
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CP0272414
|
US11149018, Example 34
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C26H27BrClN3O3
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1
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| 1 |
IC50 > 9400 nM
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CP0530784
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2-(2-acetyl-6-methoxyphenyl)-N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]acetamide
Show/Hide
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C34H35N3O8S
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2
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| 1 |
Ki = 0.12 nM
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| 2 |
Ki = 2.3 nM
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CP0426597
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US9180116, 9C
Show/Hide
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C19H31F2NO4
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1
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| 1 |
Ki = 0.2 nM
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CP0505112
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N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-[2-(trifluoromethoxy)phenyl]acetamide
Show/Hide
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C32H30F3N3O7S
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2
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| 1 |
Ki = 0.21 nM
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| 2 |
Ki = 56 nM
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CP0393733
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N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]methylsulfonyl]-2-phenylacetamide
Show/Hide
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C32H32N2O6S
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2
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| 1 |
Ki = 0.25 nM
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| 2 |
Ki = 29 nM
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CP0393746
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2-(2-chlorophenyl)-N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]acetamide
Show/Hide
|
C31H30ClN3O6S
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2
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| 1 |
Ki = 0.27 nM
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| 2 |
Ki = 37 nM
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CP0505149
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N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-(2-ethoxyphenyl)acetamide
Show/Hide
|
C33H35N3O7S
|
2
|
| 1 |
Ki = 0.27 nM
|
|
|
| 2 |
Ki = 8.9 nM
|
|
|
|
CP0393741
|
2-(2,6-dichlorophenyl)-N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]acetamide
Show/Hide
|
C31H29Cl2N3O6S
|
2
|
| 1 |
Ki = 0.28 nM
|
|
|
| 2 |
Ki = 4.8 nM
|
|
|
|
CP0562485
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-2-phenylacetamide
Show/Hide
|
C31H30N2O6S
|
2
|
| 1 |
Ki = 0.31 nM
|
|
|
| 2 |
Ki > 4000 nM
|
|
|
|
CP0382103
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-[2-(difluoromethoxy)phenyl]acetamide
Show/Hide
|
C32H31F2N3O7S
|
2
|
| 1 |
Ki = 0.32 nM
|
|
|
| 2 |
Ki = 13 nM
|
|
|
|
CP0505639
|
N-[2-[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)-3-methylphenyl]ethyl]-2-(2-methoxyphenyl)acetamide
Show/Hide
|
C34H36N2O5
|
2
|
| 1 |
Ki = 0.32 nM
|
|
|
| 2 |
Ki = 2.7 nM
|
|
|
|
CP0393739
|
2-(2-methoxyphenyl)-N-[[3-methyl-4-[6-oxo-5,9-di(propan-2-yloxy)-8H-pyrrolo[3,4-g]quinolin-7-yl]phenyl]methylsulfonyl]acetamide
Show/Hide
|
C34H37N3O7S
|
2
|
| 1 |
Ki = 0.36 nM
|
|
|
| 2 |
Ki = 26 nM
|
|
|
|
CP0393743
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-2-(2,5-dimethoxyphenyl)acetamide
Show/Hide
|
C33H34N2O8S
|
2
|
| 1 |
Ki = 0.37 nM
|
|
|
| 2 |
Ki = 38 nM
|
|
|
|
CP0426640
|
US9180116, 2C
Show/Hide
|
C21H31F2NO4
|
1
|
| 1 |
Ki = 0.378 nM
|
|
|
|
CP0422464
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-2-phenoxyacetamide
Show/Hide
|
C31H30N2O7S
|
2
|
| 1 |
Ki = 0.38 nM
|
|
|
| 2 |
Ki = 1200 nM
|
|
|
|
CP0433298
|
2-(2-methoxyphenyl)-N-[[3-methyl-4-[6-oxo-5,9-bis(2,2,2-trifluoroethoxy)-8H-pyrrolo[3,4-g]quinolin-7-yl]phenyl]methylsulfonyl]acetamide
Show/Hide
|
C32H27F6N3O7S
|
2
|
| 1 |
Ki = 0.38 nM
|
|
|
| 2 |
Ki = 17 nM
|
|
|
|
CP0224474
|
4-(2-((1R,2R,3R)-3-hydroxy-2-((S,E)-3-hydroxy-4-(3-(methoxymethyl)phenyl)but-1-enyl)-5-oxocyclopentyl)ethylthio)butanoic acid
Show/Hide
|
C23H32O6S
|
1
|
| 1 |
Ki = 0.396 nM
|
|
|
|
CP0378980
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-2-(2,4,6-trimethylphenyl)acetamide
Show/Hide
|
C34H36N2O6S
|
2
|
| 1 |
Ki = 0.43 nM
|
|
|
| 2 |
Ki = 380 nM
|
|
|
|
CP0501946
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-2-naphthalen-1-ylacetamide
Show/Hide
|
C35H32N2O6S
|
2
|
| 1 |
Ki = 0.43 nM
|
|
|
| 2 |
Ki = 4.8 nM
|
|
|
|
CP0505113
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-[2-(trifluoromethyl)phenyl]acetamide
Show/Hide
|
C32H30F3N3O6S
|
2
|
| 1 |
Ki = 0.43 nM
|
|
|
| 2 |
Ki = 350 nM
|
|
|
|
CP0525695
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-(2-fluorophenyl)acetamide
Show/Hide
|
C31H30FN3O6S
|
2
|
| 1 |
Ki = 0.48 nM
|
|
|
| 2 |
Ki = 34 nM
|
|
|
|
CP0440902
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-1-(2,6-dimethoxyphenyl)cyclopropane-1-carboxamide
Show/Hide
|
C35H37N3O8S
|
2
|
| 1 |
Ki = 0.54 nM
|
|
|
| 2 |
Ki = 2.3 nM
|
|
|
|
CP0433297
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-1-(2-methoxyphenyl)cyclopropane-1-carboxamide
Show/Hide
|
C34H35N3O7S
|
2
|
| 1 |
Ki = 0.55 nM
|
|
|
| 2 |
Ki = 4.2 nM
|
|
|
|
CP0503017
|
N-[1-[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]propan-2-yl]-2-(2-methoxyphenyl)acetamide
Show/Hide
|
C34H37N3O5
|
2
|
| 1 |
Ki = 0.67 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0454380
|
N-[2-[4-[4,9-bis(difluoromethoxy)-3-oxo-1H-benzo[f]isoindol-2-yl]-3-methylphenyl]ethyl]-2-(2-methoxyphenyl)acetamide
Show/Hide
|
C32H28F4N2O5
|
2
|
| 1 |
Ki = 0.71 nM
|
|
|
| 2 |
Ki = 8.4 nM
|
|
|
|
CP0393748
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-(2-methoxyphenyl)acetamide
Show/Hide
|
C32H33N3O7S
|
2
|
| 1 |
Ki = 0.74 nM
|
|
|
| 2 |
Ki = 3.6 nM
|
|
|
|
CP0530785
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-phenylacetamide
Show/Hide
|
C31H31N3O6S
|
2
|
| 1 |
Ki = 0.76 nM
|
|
|
| 2 |
Ki = 31 nM
|
|
|
|
CP0422463
|
1-(2,6-dimethoxyphenyl)-N-[[3-methyl-4-[6-oxo-5,9-bis(2,2,2-trifluoroethoxy)-8H-pyrrolo[3,4-g]quinolin-7-yl]phenyl]methylsulfonyl]cyclopropane-1-carboxamide
Show/Hide
|
C35H31F6N3O8S
|
2
|
| 1 |
Ki = 0.79 nM
|
|
|
| 2 |
Ki = 1.6 nM
|
|
|
|
CP0424452
|
N-[2-[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]ethyl]-2-(2-methoxyphenyl)acetamide
Show/Hide
|
C33H35N3O5
|
2
|
| 1 |
Ki = 0.87 nM
|
|
|
| 2 |
Ki = 2.6 nM
|
|
|
|
CP0393738
|
1-(2-methoxyphenyl)-N-[[3-methyl-4-[6-oxo-5,9-bis(2,2,2-trifluoroethoxy)-8H-pyrrolo[3,4-g]quinolin-7-yl]phenyl]methylsulfonyl]cyclopropane-1-carboxamide
Show/Hide
|
C34H29F6N3O7S
|
2
|
| 1 |
Ki = 0.95 nM
|
|
|
| 2 |
Ki = 12 nM
|
|
|
|
CP0404920
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-1,2,3,4-tetrahydronaphthalene-1-carboxamide
Show/Hide
|
C34H34N2O6S
|
2
|
| 1 |
Ki = 1 nM
|
|
|
| 2 |
Ki = 940 nM
|
|
|
|
CP0144553
|
7-[(R)-2-((E)-(S)-3-Hydroxy-oct-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C19H33NO4
|
1
|
| 1 |
Ki = 1.606 nM
|
|
|
|
CP0444299
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-2-(5-methylpyrazol-1-yl)acetamide
Show/Hide
|
C29H30N4O6S
|
2
|
| 1 |
Ki = 2 nM
|
|
|
| 2 |
Ki = 600 nM
|
|
|
|
CP0417632
|
7-[(2R)-2-[(E,3S,4S)-3-hydroxy-4-methylnon-1-en-6-ynyl]-5-oxopyrrolidin-1-yl]heptanoic acid
Show/Hide
|
C21H33NO4
|
1
|
| 1 |
Ki = 2.349 nM
|
|
|
|
CP0440904
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-pyridin-2-ylacetamide
Show/Hide
|
C30H30N4O6S
|
2
|
| 1 |
Ki = 2.4 nM
|
|
|
| 2 |
Ki = 13 nM
|
|
|
|
CP0530786
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-2-(3-methoxyphenyl)acetamide
Show/Hide
|
C32H32N2O7S
|
2
|
| 1 |
Ki = 2.4 nM
|
|
|
| 2 |
Ki = 1600 nM
|
|
|
|
CP0080235
|
4-(2-((R)-2-((S)-3-hydroxyhept-1-enyl)-5-oxopyrrolidin-1-yl)ethyl)benzoate
Show/Hide
|
C20H27NO4
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0440903
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-pyridin-3-ylacetamide
Show/Hide
|
C30H30N4O6S
|
2
|
| 1 |
Ki = 2.8 nM
|
|
|
| 2 |
Ki = 48 nM
|
|
|
|
CP0405168
|
N-[[4-(5,9-diethoxy-8-oxo-6H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-phenylacetamide
Show/Hide
|
C31H31N3O6S
|
2
|
| 1 |
Ki = 3.3 nM
|
|
|
| 2 |
Ki = 660 nM
|
|
|
|
CP0382084
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-3-thiophen-3-ylpropanamide
Show/Hide
|
C30H30N2O6S2
|
2
|
| 1 |
Ki = 4.2 nM
|
|
|
| 2 |
Ki > 4000 nM
|
|
|
|
CP0524076
|
2-(2-methoxyphenyl)-N-(3-methyl-4-(1-oxo-4,9-bis(2,2,2-trifluoroethoxy)-1H-benzo[f]isoindol-2(3H)-yl)phenethyl)acetamide
Show/Hide
|
C34H30F6N2O5
|
2
|
| 1 |
Ki = 4.4 nM
|
|
|
| 2 |
Ki = 104 nM
|
|
|
|
CP0393736
|
N-[[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]methylsulfonyl]-2,2-diphenylacetamide
Show/Hide
|
C37H34N2O6S
|
2
|
| 1 |
Ki = 7.9 nM
|
|
|
| 2 |
Ki > 4000 nM
|
|
|
|
CP0404875
|
N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-pyridin-4-ylacetamide
Show/Hide
|
C30H30N4O6S
|
2
|
| 1 |
Ki = 9.8 nM
|
|
|
| 2 |
Ki = 160 nM
|
|
|
|
CP0383173
|
2-[4-(5,9-diethoxy-6,8-dioxopyrrolo[3,4-g]quinolin-7-yl)phenyl]acetic acid
Show/Hide
|
C23H20N2O6
|
1
|
| 1 |
Ki = 31.62 nM
|
|
|
|
CP0459255
|
2-[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]acetic acid
Show/Hide
|
C24H23NO5
|
1
|
| 1 |
Ki = 79.43 nM
|
|
|
|
CP0536164
|
4-(2-((R)-2-(4-(cyclopentylmethyl)penta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C24H31NO3
|
1
|
| 1 |
Ki = 117 nM
|
|
|
|
CP0096991
|
2-[4-(4,9-diethoxy-1,3-dioxobenzo[f]isoindol-2-yl)phenyl]acetic acid
Show/Hide
|
C24H21NO6
|
1
|
| 1 |
Ki = 158.49 nM
|
|
|
|
CP0383176
|
2-[4-(4,9-diethoxy-6-methyl-1,3-dioxobenzo[f]isoindol-2-yl)phenyl]acetic acid
Show/Hide
|
C25H23NO6
|
1
|
| 1 |
Ki = 158.49 nM
|
|
|
|
CP0549817
|
2-[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]propanoic acid
Show/Hide
|
C25H25NO5
|
1
|
| 1 |
Ki = 199.53 nM
|
|
|
|
CP0181173
|
2-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl}-cyclopropanecarboxylic acid
Show/Hide
|
C27H22O3S
|
1
|
| 1 |
Ki = 300 nM
|
|
|
|
CP0412366
|
2-[4-[3-oxo-4,9-di(propan-2-yloxy)-1H-benzo[f]isoindol-2-yl]phenyl]acetic acid
Show/Hide
|
C26H27NO5
|
1
|
| 1 |
Ki = 398.11 nM
|
|
|
|
CP0441655
|
4-[3-(2-Benzyloxy-phenyl)-propyl]-benzoic acid
Show/Hide
|
C23H22O3
|
1
|
| 1 |
Ki = 440 nM
|
|
|
|
CP0457558
|
4-[2-[(2R)-2-[(1Z,3E)-3-methylocta-1,3-dienyl]-5-oxopyrrolidin-1-yl]ethyl]benzoic acid
Show/Hide
|
C22H29NO3
|
1
|
| 1 |
Ki = 443 nM
|
|
|
|
CP0466746
|
2-[2-[5-(2-phenylmethoxyphenyl)thiophen-3-yl]anilino]acetic acid
Show/Hide
|
C25H21NO3S
|
1
|
| 1 |
Ki = 460 nM
|
|
|
|
CP0383175
|
2-[4-(4,9-diethoxy-1,3-dihydrobenzo[f]isoindol-2-yl)phenyl]acetic acid
Show/Hide
|
C24H25NO4
|
1
|
| 1 |
Ki = 630.96 nM
|
|
|
|
CP0412364
|
2-[4-(3-oxo-4,9-dipropoxy-1H-benzo[f]isoindol-2-yl)phenyl]acetic acid
Show/Hide
|
C26H27NO5
|
1
|
| 1 |
Ki = 630.96 nM
|
|
|
|
CP0381724
|
3-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl}-propionic acid
Show/Hide
|
C26H22O3S
|
1
|
| 1 |
Ki = 650 nM
|
|
|
|
CP0424293
|
3-{2-[4-(2-Benzyloxy-phenyl)-thiophen-2-yl]-phenyl}-propionic acid
Show/Hide
|
C26H22O3S
|
1
|
| 1 |
Ki = 760 nM
|
|
|
|
CP0430206
|
3-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl}-2-methyl-propionic acid
Show/Hide
|
C27H24O3S
|
1
|
| 1 |
Ki = 980 nM
|
|
|
|
CP0404232
|
3-(2-Phenoxymethyl-[1,1';3',1'']terphenyl-2''-yl)-propionic acid
Show/Hide
|
C28H24O3
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0372972
|
3-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl}-butyric acid
Show/Hide
|
C27H24O3S
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0404532
|
3-[2''-(2,6-Dichloro-benzyloxy)-[1,1';3',1'']terphenyl-2-yl]-propionic acid
Show/Hide
|
C28H22Cl2O3
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0441093
|
(2''-Benzyloxy-[1,1';3',1'']terphenyl-2-yl)-acetic acid
Show/Hide
|
C27H22O3
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0466770
|
3-{2-[5-(2-Benzyloxy-phenyl)-thiophen-2-yl]-phenyl}-propionic acid
Show/Hide
|
C26H22O3S
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0406374
|
3-(2''-Benzyloxy-[1,1';3',1'']terphenyl-2-yl)-2-methyl-propionic acid
Show/Hide
|
C29H26O3
|
1
|
| 1 |
Ki = 1200 nM
|
|
|
|
CP0870434
|
7-((1R,2S,3R,5R)-3,5-dichloro-2-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
|
C24H34Cl2O3
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0404585
|
3-[2-[3-(2-phenylmethoxyphenyl)phenyl]phenyl]-N-thiophen-2-ylsulfonylpropanamide
Show/Hide
|
C32H27NO4S2
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0496137
|
(E)-3-(2-Benzyloxy-[1,1';3',1'']terphenyl-2''-yl)-acrylic acid
Show/Hide
|
C28H22O3
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0436538
|
3-(2-Benzyloxy-[1,1';3',1'']terphenyl-2''-yl)-propionic acid
Show/Hide
|
C28H24O3
|
1
|
| 1 |
Ki = 1800 nM
|
|
|
|
CP0277044
|
(E)-3-{2-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-allyl]-phenyl}-acrylic acid
Show/Hide
|
C26H24O3
|
1
|
| 1 |
Ki = 1900 nM
|
|
|
|
CP0469671
|
2-[4-(4,9-dibutoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]acetic acid
Show/Hide
|
C28H31NO5
|
1
|
| 1 |
Ki = 1995.26 nM
|
|
|
|
CP0437614
|
4-(2-Benzyloxy-[1,1';3',1'']terphenyl-2''-yl)-butyric acid
Show/Hide
|
C29H26O3
|
1
|
| 1 |
Ki = 2000 nM
|
|
|
|
CP0866746
|
7-((1R,2S,3R)-2-(4-hexanoylphenyl)-3-hydroxy-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
|
C24H32O5
|
1
|
| 1 |
Ki = 2809 nM
|
|
|
|
CP0160939
|
(E)-3-[2-(3,4-dichlorophenyl)phenyl]-N-thiophen-2-ylsulfonylprop-2-enamide
Show/Hide
|
C19H13Cl2NO3S2
|
1
|
| 1 |
Ki = 3700 nM
|
|
|
|
CP0374187
|
2-[(3R)-5-bromo-4-[(4-chlorophenyl)methyl]-7-fluoro-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acid
Show/Hide
|
C20H16BrClFNO2
|
1
|
| 1 |
Ki = 4400 nM
|
|
|
|
CP0381706
|
3-[1,1';3',1'']Terphenyl-2-yl-propionic acid
Show/Hide
|
C21H18O2
|
1
|
| 1 |
Ki = 6000 nM
|
|
|
|
CP0866243
|
4-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxy}-benzoic acid
Show/Hide
|
C24H29NO5
|
1
|
| 1 |
Ki = 8752 nM
|
|
|
|
CP0415118
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(E)-3-(3',4'-Dichloro-biphenyl-2-yl)-acrylic acid
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C15H10Cl2O2
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1
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| 1 |
Ki > 10000 nM
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CP0847233
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3-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-benzoic acid
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C25H31NO5
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1
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| 1 |
Ki > 10000 nM
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CP0847234
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5-{(R)-1-[4-(1-Hydroxy-butyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
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C21H25NO5S
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1
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| 1 |
Ki > 10000 nM
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CP0847235
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5-((E/Z)-3-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-yl}-allyl)-thiophene-2-carboxylic acid
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C24H29NO4S
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1
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| 1 |
Ki > 10000 nM
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CP0847238
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5-[(R)-1-(4-Hexanoyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-thiophene-2-carboxylic acid
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C23H27NO5S
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1
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| 1 |
Ki > 10000 nM
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CP0847240
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5-{(R)-1-[4-(1-Hydroxy-2-phenyl-ethyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-furan-2-carboxylic acid
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C25H25NO6
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1
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| 1 |
Ki > 10000 nM
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CP0850987
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5-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-furan-2-carboxylic acid
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C23H29NO6
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1
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| 1 |
Ki > 10000 nM
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CP0850988
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5-{(R)-1-[4-(1-Hydroxy-pentyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
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C22H27NO5S
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1
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| 1 |
Ki > 10000 nM
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CP0870416
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5-{(R)-1-[4-(1-Hydroxy-2-methyl-propyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-furan-2-carboxylic acid
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C21H25NO6
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1
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| 1 |
Ki > 10000 nM
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CP0895715
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5-(3-((2R)-1-(4-(1-hydroxyhexyl)phenyl)-5-oxopyrrolidin-2-yl)allyl)thiophene-2-carboxylic acid
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C24H29NO4S
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1
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| 1 |
Ki > 10000 nM
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CP0899507
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7-((1S,2S,3R,5R)-5-cyano-3-hydroxy-2-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)hept-5-enoic acid
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C25H35NO4
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1
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| 1 |
Ki > 10000 nM
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CP0174264
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7-[(1R,2S)-2-[4-(1-hydroxyhexyl)phenyl]-5-oxocyclopentyl]heptanoic acid
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C24H36O4
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1
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| 1 |
Ki = 15000 nM
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CP0852855
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7-((1R,2S)-2-(4-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
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C24H34O4
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1
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| 1 |
Ki = 15000 nM
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CP0856833
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methyl 7-((1R,2S)-2-(4-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)heptanoate
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C25H38O4
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1
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| 1 |
Ki = 15000 nM
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CP0863699
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methyl 7-((1R,2S)-2-(4-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)hept-5-enoate
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C25H36O4
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1
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| 1 |
Ki = 15000 nM
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CP0343798
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2-[(3R)-4-[(4-chlorophenyl)methyl]-7-fluoro-5-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acid
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C21H19ClFNO4S
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1
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| 1 |
Ki > 15200 nM
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CP0041889
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2-((R)-4-(4-chlorobenzyl)-5-(1-hydroxyethyl)-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid
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C23H24ClNO5S
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1
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| 1 |
Ki > 20000 nM
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CP0108218
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(R)-2-(4-(4-chlorobenzyl)-5-acetyl-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid
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C23H22ClNO5S
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1
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| 1 |
Ki > 20000 nM
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CP0372074
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2-[(3R)-5-acetyl-4-[(4-chlorophenyl)methyl]-7-fluoro-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acid
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C22H19ClFNO3
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1
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| 1 |
Ki > 20000 nM
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CP0404233
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3-(4''-Benzyloxy-[1,1';3',1'']terphenyl-2-yl)-propionic acid
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C28H24O3
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1
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| 1 |
Ki = 21000 nM
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CP0388282
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2-(4-(4-(butylcarbamoyl)-2-(2,4-dichlorophenylsulfonamido)phenoxy)-3-methoxyphenyl)acetic acid
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C26H26Cl2N2O7S
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1
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| 1 |
Ki = 44000 nM
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CP0517668
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2-[4-(4,9-dihexoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]acetic acid
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C32H39NO5
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1
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| 1 |
Ki > 6309.57 nM
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