| Compound ID |
Compound Name |
Compound Formula |
|
CP0423240
|
N-[(1S)-3-[4-[[2-(3,4-dichlorophenyl)acetyl]-ethylamino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
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|
C30H39Cl2N3O2
|
1
|
| 1 |
IC50 = 0.05 nM
|
|
|
|
CP0478980
|
N-[(1S)-3-[4-[ethyl-[2-(4-methylsulfonylphenyl)acetyl]amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C31H43N3O4S
|
1
|
| 1 |
IC50 = 0.07 nM
|
|
|
|
CP0514717
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclopentanecarboxamide
Show/Hide
|
C27H41N5O
|
1
|
| 1 |
IC50 = 0.137 nM
|
|
|
|
CP0423241
|
N-[(1S)-3-[4-[benzylcarbamoyl(ethyl)amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
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|
C30H42N4O2
|
1
|
| 1 |
IC50 = 0.16 nM
|
|
|
|
CP0002124
|
4,4-Difluoro-cyclohexanecarboxylic acid {(S)-3-[(1S,5S)-3-(3-isopropyl-5-methyl-[1,2,4]triazol-4-yl)-8-aza-bicyclo[3.2.1]oct-8-yl]-1-phenyl-propyl}-amide
Show/Hide
|
C29H41F2N5O
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0478981
|
N-[(1S)-3-[4-[[2-(4-chlorophenyl)acetyl]-ethylamino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
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|
C30H40ClN3O2
|
1
|
| 1 |
IC50 = 0.34 nM
|
|
|
|
CP0468371
|
(+/-)-3,3-difluoro-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclobutanecarboxamide
Show/Hide
|
C26H37F2N5O
|
1
|
| 1 |
IC50 = 0.38 nM
|
|
|
|
CP0423242
|
N-[(1S)-3-[4-[ethyl-[2-[4-(trifluoromethyl)phenyl]acetyl]amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C31H40F3N3O2
|
1
|
| 1 |
IC50 = 0.48 nM
|
|
|
|
CP0493399
|
3,3-difluoro-N-((1S,3R)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclobutanecarboxamide
Show/Hide
|
C26H37F2N5O
|
1
|
| 1 |
IC50 = 0.48 nM
|
|
|
|
CP0508054
|
N-benzyl-N-[1-[1-(2,6-dimethylbenzoyl)-4-methylpiperidin-4-yl]piperidin-4-yl]cyclopropanecarboxamide
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|
C31H41N3O2
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0515715
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclohexanecarboxamide
Show/Hide
|
C28H43N5O
|
1
|
| 1 |
IC50 = 0.513 nM
|
|
|
|
CP0541362
|
(+/-)-4,4-difluoro-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclohexanecarboxamide
Show/Hide
|
C28H41F2N5O
|
1
|
| 1 |
IC50 = 0.84 nM
|
|
|
|
CP0418940
|
N-[(1S)-3-[4-[ethyl-[2-(4-fluorophenyl)acetyl]amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
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|
C30H40FN3O2
|
1
|
| 1 |
IC50 = 0.94 nM
|
|
|
|
CP0423728
|
(R)-N-benzyl-N-(1-(1-(2,6-dimethylbenzoyl)piperidin-4-yl)pyrrolidin-3-yl)cyclopropanecarboxamide
Show/Hide
|
C29H37N3O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0509413
|
N-benzyl-N-[(3R)-1-[(1R,5S)-8-(2,6-dimethylbenzoyl)-8-azabicyclo[3.2.1]octan-3-yl]pyrrolidin-3-yl]cyclopropanecarboxamide
Show/Hide
|
C31H39N3O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0852199
|
3,3-difluoro-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclobutanecarboxamide
Show/Hide
|
C26H38ClF2N5O
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0904500
|
4,4-difluoro-N-((1S)-3-(3-(5-isopropyl-3-methyl-1H-1,2,4-triazol-1-yl)-8-azabicyclo[3.2.1]octan-8-yl)-1-phenylpropyl)cyclohexanecarboxamide
Show/Hide
|
C29H41F2N5O
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0515639
|
N-[(1S)-3-[4-[[2-(3-chlorophenyl)acetyl]-ethylamino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C30H40ClN3O2
|
1
|
| 1 |
IC50 = 1.54 nM
|
|
|
|
CP0503482
|
N-[(1S)-3-[4-(3-methyl-5-propan-2-yl-1,2,4-triazol-4-yl)piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C26H39N5O
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0427113
|
N-[(1S)-3-[4-[[2-(2,4-dichlorophenyl)acetyl]-ethylamino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C30H39Cl2N3O2
|
1
|
| 1 |
IC50 = 2.33 nM
|
|
|
|
CP0428176
|
N-benzyl-N-[1-[1-(2,6-dimethylbenzoyl)piperidin-4-yl]piperidin-4-yl]cyclobutanecarboxamide
Show/Hide
|
C31H41N3O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0452628
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)isobutyramide
Show/Hide
|
C25H39N5O
|
1
|
| 1 |
IC50 = 3.11 nM
|
|
|
|
CP0514700
|
benzyl N-[1-[(4S)-4-(cyclobutanecarbonylamino)-4-phenylbutan-2-yl]piperidin-4-yl]-N-ethylcarbamate
Show/Hide
|
C30H41N3O3
|
1
|
| 1 |
IC50 = 3.16 nM
|
|
|
|
CP0493396
|
(+/-)-2-cyclopropyl-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)acetamide
Show/Hide
|
C26H39N5O
|
1
|
| 1 |
IC50 = 3.16 nM
|
|
|
|
CP0514701
|
4-chlorophenyl 1-((4S)-4-(cyclobutanecarboxamido)-4-phenylbutan-2-yl)piperidin-4-yl(ethyl)carbamate
Show/Hide
|
C29H38ClN3O3
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0504016
|
4-fluorophenyl 1-((4S)-4-(cyclobutanecarboxamido)-4-phenylbutan-2-yl)piperidin-4-yl(ethyl)carbamate
Show/Hide
|
C29H38FN3O3
|
1
|
| 1 |
IC50 = 3.63 nM
|
|
|
|
CP0419115
|
N-[(1S)-3-[4-[ethyl-[2-(4-methylphenyl)acetyl]amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C31H43N3O2
|
1
|
| 1 |
IC50 = 3.76 nM
|
|
|
|
CP0554450
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclopropanecarboxamide
Show/Hide
|
C25H37N5O
|
1
|
| 1 |
IC50 = 3.93 nM
|
|
|
|
CP0431532
|
N-[1-[(4S)-4-(cyclobutanecarbonylamino)-4-phenylbutan-2-yl]piperidin-4-yl]-N-ethyl-4-fluorobenzamide
Show/Hide
|
C29H38FN3O2
|
1
|
| 1 |
IC50 = 4.83 nM
|
|
|
|
CP0565562
|
(+/-)-1-Oxo-hexahydro-1lambda*4*-thiopyran-4-carboxylic acid{(S)-3-[4-(3-isopropyl-5-methyl-[1,2,4]triazol-4-yl)-piperidin-1-yl]-1-phenyl-butyl}-amide
Show/Hide
|
C27H41N5O2S
|
1
|
| 1 |
IC50 = 4.87 nM
|
|
|
|
CP0418943
|
N-[(1S)-3-[4-[ethyl-[2-(4-methoxyphenyl)acetyl]amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C31H43N3O3
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0511449
|
(+/-)-1,1-Dioxo-hexahydro-1lambda*6*-thiopyran-4-carboxylic acid{(S)-3-[4-(3-isopropyl-5-methyl-[1,2,4]triazol-4-yl)-piperidin-1-yl]-1-phenyl-butyl}-amide
Show/Hide
|
C27H41N5O3S
|
1
|
| 1 |
IC50 = 6.12 nM
|
|
|
|
CP0514370
|
(S)-4,4-difluoro-N-(3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylpropyl)cyclohexanecarboxamide
Show/Hide
|
C27H39F2N5O
|
1
|
| 1 |
IC50 = 7.5 nM
|
|
|
|
CP0423244
|
N-[(1S)-3-[4-[ethyl-(2-phenylacetyl)amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C30H41N3O2
|
1
|
| 1 |
IC50 = 13.4 nM
|
|
|
|
CP0503485
|
N-[(1S)-3-[(1R,5S)-3-[ethyl-[2-(4-methoxyphenyl)acetyl]amino]-8-azabicyclo[3.2.1]octan-8-yl]-1-phenylpropyl]cyclobutanecarboxamide
Show/Hide
|
C32H43N3O3
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0431533
|
N-[(1S)-3-[4-[ethyl-[2-(2-methoxyphenyl)acetyl]amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C31H43N3O3
|
1
|
| 1 |
IC50 = 17.9 nM
|
|
|
|
CP0419118
|
N-[(1S)-3-[4-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C23H32N4O2
|
1
|
| 1 |
IC50 = 21.4 nM
|
|
|
|
CP0423206
|
(4-((1-benzhydrylazetidin-3-yl)(methyl)amino)piperidin-1-yl)(2,4-dimethylpyridin-3-yl)methanone
Show/Hide
|
C30H36N4O
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0510218
|
4-chloro-N-(1-((4S)-4-(cyclobutanecarboxamido)-4-phenylbutan-2-yl)piperidin-4-yl)-N-ethylbenzamide
Show/Hide
|
C29H38ClN3O2
|
1
|
| 1 |
IC50 = 25.3 nM
|
|
|
|
CP0554451
|
(+/-)-1-acetyl-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)piperidine-4-carboxamide
Show/Hide
|
C29H44N6O2
|
1
|
| 1 |
IC50 = 28.7 nM
|
|
|
|
CP0506600
|
3,4-dichloro-N-(1-((4S)-4-(cyclobutanecarboxamido)-4-phenylbutan-2-yl)piperidin-4-yl)-N-ethylbenzamide
Show/Hide
|
C29H37Cl2N3O2
|
1
|
| 1 |
IC50 = 33.7 nM
|
|
|
|
CP0478982
|
N-[(1S)-3-[4-(3,5-dimethyl-1,2,4-triazol-4-yl)piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C24H35N5O
|
1
|
| 1 |
IC50 = 37.5 nM
|
|
|
|
CP0522542
|
(4-(3-benzhydryl-3,8-diazabicyclo[3.2.1]octan-8-yl)piperidin-1-yl)(2,4-dimethylpyridin-3-yl)methanone
Show/Hide
|
C32H38N4O
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0423246
|
(S)-N-(3-(4-(2-(4-methoxyphenyl)acetamido)piperidin-1-yl)-1-phenylpropyl)cyclobutanecarboxamide
Show/Hide
|
C28H37N3O3
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0555029
|
4,4-difluoro-N-((1S,3S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclohexanecarboxamide
Show/Hide
|
C28H41F2N5O
|
1
|
| 1 |
IC50 = 49.9 nM
|
|
|
|
CP0388630
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)-2-(2,2,2-trifluoroethoxy)acetamide
Show/Hide
|
C25H36F3N5O2
|
1
|
| 1 |
IC50 = 52.8 nM
|
|
|
|
CP0506027
|
N-[2-[3-(2,2-diphenylethyl)piperidin-1-yl]ethyl]-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C29H35N3O
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0904501
|
4,4-difluoro-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)cyclohexanecarboxamide
Show/Hide
|
C28H42ClF2N5O
|
1
|
| 1 |
IC50 = 62 nM
|
|
|
|
CP0503483
|
N-[1-[(4S)-4-(cyclobutanecarbonylamino)-4-phenylbutan-2-yl]piperidin-4-yl]-N-ethyl-4-methoxybenzamide
Show/Hide
|
C30H41N3O3
|
1
|
| 1 |
IC50 = 64.4 nM
|
|
|
|
CP0503484
|
N-[1-[(4S)-4-(cyclobutanecarbonylamino)-4-phenylbutan-2-yl]piperidin-4-yl]-N-ethylbenzamide
Show/Hide
|
C29H39N3O2
|
1
|
| 1 |
IC50 = 73.5 nM
|
|
|
|
CP0388632
|
(+/-)-3,3,3-trifluoro-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)propanamide
Show/Hide
|
C24H34F3N5O
|
1
|
| 1 |
IC50 = 85.3 nM
|
|
|
|
CP0474798
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)acetamide
Show/Hide
|
C23H35N5O
|
1
|
| 1 |
IC50 = 89.2 nM
|
|
|
|
CP0504017
|
N-[(1S)-1-phenyl-3-[4-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]butyl]cyclobutanecarboxamide
Show/Hide
|
C25H36N4O2
|
1
|
| 1 |
IC50 = 94.6 nM
|
|
|
|
CP0506026
|
(3-((1-benzhydrylpiperidin-4-yl)(methyl)amino)azetidin-1-yl)(2,4-dimethylpyridin-3-yl)methanone
Show/Hide
|
C30H36N4O
|
1
|
| 1 |
IC50 = 102 nM
|
|
|
|
CP0373500
|
N-[[4-benzyl-1-[1-(2,6-dimethylbenzoyl)piperidin-4-yl]piperidin-4-yl]methyl]cyclopropanecarboxamide
Show/Hide
|
C31H41N3O2
|
1
|
| 1 |
IC50 = 145 nM
|
|
|
|
CP0474799
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)tetrahydro-2H-pyran-4-carboxamide
Show/Hide
|
C27H41N5O2
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0457693
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)morpholine-4-carboxamide
Show/Hide
|
C26H40N6O2
|
1
|
| 1 |
IC50 = 176 nM
|
|
|
|
CP0474800
|
(+/-)-N-((1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutyl)-4-methylpiperazine-1-carboxamide
Show/Hide
|
C27H43N7O
|
1
|
| 1 |
IC50 = 187 nM
|
|
|
|
CP0509412
|
(4-(8-benzhydryl-3,8-diazabicyclo[3.2.1]octan-3-yl)piperidin-1-yl)(2,4-dimethylpyridin-3-yl)methanone
Show/Hide
|
C32H38N4O
|
1
|
| 1 |
IC50 = 313 nM
|
|
|
|
CP0493397
|
(+/-)-methyl(1S)-3-(4-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)piperidin-1-yl)-1-phenylbutylcarbamate
Show/Hide
|
C23H35N5O2
|
1
|
| 1 |
IC50 = 315 nM
|
|
|
|
CP0419116
|
N-[(1S)-1-phenyl-3-[4-(4-pyridin-4-yl-1H-pyrazol-5-yl)piperidin-1-yl]butyl]cyclobutanecarboxamide
Show/Hide
|
C28H35N5O
|
1
|
| 1 |
IC50 = 382 nM
|
|
|
|
CP0503486
|
N-[(1S)-3-[4-[5-[(dimethylamino)methyl]-1,3,4-oxadiazol-2-yl]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C25H37N5O2
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0373501
|
(S)-N-benzyl-N-(1-(1-(2,6-dimethylbenzoyl)piperidin-4-yl)pyrrolidin-3-yl)cyclopropanecarboxamide
Show/Hide
|
C29H37N3O2
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
|
CP0478983
|
N-[(1S)-3-[4-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C23H32N4O2
|
1
|
| 1 |
IC50 = 1849 nM
|
|
|
|
CP0423245
|
N-[(1S)-3-[4-(2-oxo-5-phenyl-1H-imidazol-3-yl)piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C29H36N4O2
|
1
|
| 1 |
IC50 = 2310 nM
|
|
|
|
CP0504296
|
N-[[1-[1-(2,6-dimethylbenzoyl)piperidin-4-yl]azetidin-3-yl]-phenylmethyl]acetamide
Show/Hide
|
C26H33N3O2
|
1
|
| 1 |
IC50 = 2490 nM
|
|
|
|
CP0423207
|
N-benzyl-N-[1-[1-(2,6-dimethylbenzoyl)piperidin-4-yl]azetidin-3-yl]cyclopropanecarboxamide
Show/Hide
|
C28H35N3O2
|
1
|
| 1 |
IC50 = 5800 nM
|
|
|
|
CP0503487
|
N-[(1S)-3-[4-[ethyl-[methyl(phenyl)carbamoyl]amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C30H42N4O2
|
1
|
| 1 |
IC50 = 6430 nM
|
|
|
|
CP0419117
|
N-[(1S)-3-[4-[ethyl-(2-methyl-2-phenylpropanoyl)amino]piperidin-1-yl]-1-phenylbutyl]cyclobutanecarboxamide
Show/Hide
|
C32H45N3O2
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
