| Compound ID |
Compound Name |
Compound Formula |
|
CP0048192
|
2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl)-5-(2-methyloctan-2-yl)phenol
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|
C24H40O3
|
7
|
| 1 |
EC50 = 0.28 nM
|
|
|
| 2 |
EC50 = 0.3 nM
|
|
|
| 3 |
EC50 = 0.437 nM
|
|
|
| 4 |
EC50 = 1.995 nM
|
|
|
| 5 |
IC50 = 0.77 nM
|
|
|
| 6 |
Ki = 0.5 nM
|
|
|
| 7 |
Ki = 0.7 nM
|
|
|
|
CP0461185
|
(6-fluoro-2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone
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|
C25H22FNO3
|
2
|
| 1 |
EC50 = 1.2 nM
|
|
|
| 2 |
Ki = 11 nM
|
|
|
|
CP0438382
|
AM4054
Show/Hide
|
C26H36O3
|
1
|
| 1 |
EC50 = 1.29 nM
|
|
|
|
CP0003146
|
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H21Cl3N4O
|
26
|
| 1 |
EC50 = 1.5 nM
|
|
|
| 2 |
EC50 = 4.1 nM
|
|
|
| 3 |
EC50 = 15.7 nM
|
|
|
| 4 |
EC50 = 18.2 nM
|
|
|
| 5 |
EC50 = 586 nM
|
|
|
| 6 |
IC50 = 2.8 nM
|
|
|
| 7 |
IC50 = 13.2 nM
|
|
|
| 8 |
IC50 = 15 nM
|
|
|
| 9 |
Kd = 1.8 nM
|
|
|
| 10 |
Kd = 2.57 nM
|
|
|
| 11 |
Ki = 0.9 nM
|
|
|
| 12 |
Ki = 1.1 nM
|
|
|
| 13 |
Ki = 1.18 nM
|
|
|
| 14 |
Ki = 1.8 nM
|
|
|
| 15 |
Ki = 1.9 nM
|
|
|
| 16 |
Ki = 1.995 nM
|
|
|
| 17 |
Ki = 2.1 nM
|
|
|
| 18 |
Ki = 2.4 nM
|
|
|
| 19 |
Ki = 6 nM
|
|
|
| 20 |
Ki = 6.18 nM
|
|
|
| 21 |
Ki = 7.1 nM
|
|
|
| 22 |
Ki = 8 nM
|
|
|
| 23 |
Ki = 12 nM
|
|
|
| 24 |
Ki = 16 nM
|
|
|
| 25 |
Ki = 18 nM
|
|
|
| 26 |
Ki = 40 nM
|
|
|
|
CP0125865
|
(6R)-N-[2-(cyclopropylamino)-2-oxoethyl]-N-ethyl-9-methyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C26H35N3O3
|
2
|
| 1 |
EC50 = 1.9 nM
|
|
|
| 2 |
Ki = 4.2 nM
|
|
|
|
CP0428045
|
(2-(2,4-dichlorophenyl)-6-fluoro-2-(2-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone
Show/Hide
|
C24H17Cl2F2NO4
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0461188
|
(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone
Show/Hide
|
C25H18F5NO3
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0893459
|
(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(4,4-difluoropiperidin-1-yl)methanone
Show/Hide
|
C25H16F7NO3
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
Ki = 6 nM
|
|
|
|
CP0400985
|
(8E)-8-[(5-chlorothiophen-2-yl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C27H23Cl3N4OS
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0176419
|
N-[4-(cyclopropylamino)-4-oxobutyl]-N-ethyl-9-methyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C28H39N3O3
|
2
|
| 1 |
EC50 = 2.9 nM
|
|
|
| 2 |
Ki = 2.8 nM
|
|
|
|
CP0382152
|
4-(2-(2,4-dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-ylsulfonyl)morpholine
Show/Hide
|
C23H17Cl2F2NO5S
|
2
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
Ki = 9 nM
|
|
|
|
CP0461186
|
1-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-ylsulfonyl)-4,4-difluoropiperidine
Show/Hide
|
C24H16F7NO4S
|
2
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0851724
|
5-(4-Chlorophenyl)-6-(cyclopropylmethoxy)-N-[(1R,2R)-2-hydroxycyclohexyl]-3-pyridinecarboxamide
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|
C22H25ClN2O3
|
1
|
| 1 |
EC50 = 3.9 nM
|
|
|
|
CP0458006
|
(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(morpholino)methanone
Show/Hide
|
C24H16F5NO4
|
2
|
| 1 |
EC50 = 4 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0411164
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C28H23Cl2FN4O
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0433000
|
(8E)-8-[(5-chloropyridin-2-yl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C28H24Cl3N5O
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0445998
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-[2-(triazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C33H29Cl2N7O3
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0570537
|
US9682955, 145
Show/Hide
|
C27H23Cl2F3N4O2S
|
1
|
| 1 |
EC50 = 4.6 nM
|
|
|
|
CP0466537
|
N-(azepan-1-yl)-1-(2,4-dichlorophenyl)-5-(5-hex-1-ynylthiophen-2-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C27H30Cl2N4OS
|
2
|
| 1 |
EC50 = 4.8 nM
|
|
|
| 2 |
IC50 = 1.7 nM
|
|
|
|
CP0461190
|
(2-(2,4-dichlorophenyl)-6-fluoro-2-(4-methoxyphenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone
Show/Hide
|
C26H22Cl2FNO4
|
2
|
| 1 |
EC50 = 5 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0484002
|
(2-(2,4-dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone
Show/Hide
|
C25H19Cl2F2NO3
|
2
|
| 1 |
EC50 = 5 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0433003
|
(7E)-1-(2,4-dichlorophenyl)-5-(2-imidazol-1-ylacetyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C34H30Cl2N6O3
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0576110
|
6-[(4-chlorophenyl)-imidazol-1-ylmethyl]-4-[[1-(trifluoromethylsulfonyl)piperidin-4-yl]amino]-1H-quinolin-2-one
Show/Hide
|
C25H23ClF3N5O3S
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0386647
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-thione
Show/Hide
|
C23H21Cl3N4S
|
2
|
| 1 |
EC50 = 5.1 nM
|
|
|
| 2 |
IC50 = 12 nM
|
|
|
|
CP0373861
|
1-(2,4-Dichlorophenyl)-5-(5-(hex-1-ynyl)thiophen-2-yl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C28H30Cl2N4OS
|
2
|
| 1 |
EC50 = 5.7 nM
|
|
|
| 2 |
IC50 = 1.3 nM
|
|
|
|
CP0400984
|
(8E)-1-(2,4-dichlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C30H26Cl2FN3O
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0385190
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-(3-sulfamoylpropanoyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H30Cl2N6O5S
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0411138
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-[2-(tetrazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H24Cl2FN9O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0451950
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-[2-(tetrazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C32H28Cl2N8O3
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0451951
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(3,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-5-[2-(1,2,4-triazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H25Cl3N8O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0190381
|
US9266835, 100
Show/Hide
|
C31H31Cl2F3N4O4S
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0256129
|
naphthalen-1-yl-(4-pentoxynaphthalen-1-yl)methanone
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|
C26H24O2
|
4
|
| 1 |
EC50 = 6.1 nM
|
|
|
| 2 |
EC50 = 73 nM
|
|
|
| 3 |
IC50 = 15 nM
|
|
|
| 4 |
Ki = 35 nM
|
|
|
|
CP0065778
|
N-[2-(cyclopropylamino)-2-oxoethyl]-N-ethyl-9-methyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C26H35N3O3
|
2
|
| 1 |
EC50 = 6.2 nM
|
|
|
| 2 |
Ki = 7.3 nM
|
|
|
|
CP0400982
|
(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-(1-pyridin-2-ylcyclopropyl)-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C29H24Cl2N4O
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0563716
|
(8E)-8-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H25Cl3N4O
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0433004
|
(7E)-1-(3,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-[2-(tetrazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H24Cl2FN9O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0486578
|
US9682955, 41
Show/Hide
|
C37H37Cl2N5O6S
|
1
|
| 1 |
EC50 = 7.8 nM
|
|
|
|
CP0373860
|
1-(2,4-Dichlorophenyl)-5-(5-(hex-1-ynyl)thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4OS
|
2
|
| 1 |
EC50 = 7.9 nM
|
|
|
| 2 |
IC50 = 1.4 nM
|
|
|
|
CP0425336
|
AM4089
Show/Hide
|
C26H30O3
|
1
|
| 1 |
EC50 = 7.97 nM
|
|
|
|
CP0941794
|
(R)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone
Show/Hide
|
C24H17Cl2F2NO4
|
2
|
| 1 |
EC50 = 8 nM
|
|
|
| 2 |
Ki = 3.3 nM
|
|
|
|
CP0400987
|
(8E)-8-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-(1-pyridin-2-ylcyclopropyl)-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H23Cl2F3N4OS
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0464143
|
(8E)-8-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C28H23Cl2F3N4OS
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0419667
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-(2-sulfamoylacetyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H28Cl2N6O5S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0451947
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-[2-(tetrazol-1-yl)acetyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H25Cl2FN8O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0219312
|
US9266835, 44
Show/Hide
|
C28H24Cl2F3N3O3S
|
1
|
| 1 |
EC50 = 8.2 nM
|
|
|
|
CP0772734
|
US9266835, 54
Show/Hide
|
C29H27ClF3N3O4S
|
1
|
| 1 |
EC50 = 8.4 nM
|
|
|
|
CP0455906
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazole-4-thio
Show/Hide
|
C22H19Cl3N4S
|
2
|
| 1 |
EC50 = 8.5 nM
|
|
|
| 2 |
IC50 = 6.3 nM
|
|
|
|
CP0433005
|
(7E)-5-(3-amino-3-oxopropanoyl)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H25Cl2FN6O3
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0388083
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C23H21Cl3N4O
|
2
|
| 1 |
EC50 = 9.8 nM
|
|
|
| 2 |
IC50 = 12.9 nM
|
|
|
|
CP0334445
|
(6R)-N-ethyl-N-[2-(2-fluoroethylamino)-2-oxoethyl]-9-methyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C25H34FN3O3
|
1
|
| 1 |
EC50 = 9.8 nM
|
|
|
|
CP0869705
|
US9266835, 55
Show/Hide
|
C29H25ClF3N3O5S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0565576
|
US9682955, 40
Show/Hide
|
C33H27Cl2F3N4O3
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0279480
|
US9266835, 57
Show/Hide
|
C31H27Cl2N5O
|
1
|
| 1 |
EC50 = 10.8 nM
|
|
|
|
CP0969771
|
US9266835, 72
Show/Hide
|
C27H23Cl2F3N4O3S
|
1
|
| 1 |
EC50 = 10.9 nM
|
|
|
|
CP0428044
|
4-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-ylsulfonyl)morpholine
Show/Hide
|
C23H16F5NO5S
|
2
|
| 1 |
EC50 = 11 nM
|
|
|
| 2 |
Ki = 25 nM
|
|
|
|
CP0458007
|
(R)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone
Show/Hide
|
C24H17Cl2F2NO4
|
2
|
| 1 |
EC50 = 11 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0400986
|
(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-(1-pyridin-2-ylcyclopropyl)-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C28H21Cl2F3N4OS
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0385182
|
3-[(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-3-[[(1R)-1-pyridin-2-ylethyl]carbamoyl]-4,6-dihydropyrazolo[4,3-c]pyridin-5-yl]-3-oxopropanoic acid
Show/Hide
|
C31H27Cl2N5O5
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0057830
|
5-(4-chlorophenyl)-N-[(1R,2R)-2-hydroxycyclohexyl]-6-(2-methoxyethoxy)pyridine-3-carboxamide
Show/Hide
|
C21H25ClN2O4
|
1
|
| 1 |
EC50 = 11.6 nM
|
|
|
|
CP0445997
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C31H28Cl2FN5O
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0475837
|
(7E)-1-(4-chlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C31H25ClFN7O2
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1
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| 1 |
EC50 = 12 nM
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CP0415444
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1-(2,4-Dichlorophenyl)-4-methyl-5-(5-(4-methylpent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C26H28Cl2N4OS
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3
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| 1 |
EC50 = 12.1 nM
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| 2 |
IC50 = 1.2 nM
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| 3 |
IC50 = 2.3 nM
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CP0495914
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2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(2-chlorobenzyl)acetamide
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C23H15Cl5N4O
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2
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| 1 |
EC50 = 12.2 nM
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| 2 |
IC50 = 48.9 nM
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CP0386648
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6-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-5,7-diaza-spiro[3.4]oct-5-en-8-one
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C23H19Cl3N4O
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2
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| 1 |
EC50 = 12.3 nM
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| 2 |
IC50 = 22.8 nM
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CP0050487
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(11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphthalen-1-ylcarbonyl)-9-oxa-1-azatricyclo[6.3.1.0^{4,12}]dodeca-2,4(12),5,7-tetraene
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C27H26N2O3
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8
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| 1 |
EC50 = 12.3 nM
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| 2 |
EC50 = 44 nM
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| 3 |
EC50 = 112 nM
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| 4 |
IC50 = 140 nM
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| 5 |
Ki = 9.2 nM
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| 6 |
Ki = 20 nM
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| 7 |
Ki = 21 nM
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| 8 |
Ki = 46 nM
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CP0065791
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(6R)-N-[4-(2-fluoroethylamino)-4-oxobutyl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
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C26H36FN3O3
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1
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| 1 |
EC50 = 12.9 nM
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CP0386505
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(8E)-1-(3,4-dichlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-(1-pyridin-2-ylcyclopropyl)-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
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C30H25Cl2FN4O
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1
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| 1 |
EC50 = 13 nM
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CP0321874
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US9266835, 140
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C32H32Cl2F3N3O4S
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1
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| 1 |
EC50 = 13 nM
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CP0517211
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US9732061, Compound 5
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C27H23Cl2F3N4O2S
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1
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| 1 |
EC50 = 13 nM
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CP0279468
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US9266835, 95
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C32H31Cl2N3O4
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1
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| 1 |
EC50 = 13.5 nM
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CP0375065
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1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(pent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C26H28Cl2N4OS
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3
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| 1 |
EC50 = 13.8 nM
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| 2 |
IC50 = 1.2 nM
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| 3 |
IC50 = 6.1 nM
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CP0219430
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US9266835, 80
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C33H29Cl2N3O3S
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1
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| 1 |
EC50 = 14 nM
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CP0373854
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N-(azepan-1-yl)-1-(2,4-dichlorophenyl)-4-methyl-5-(5-pent-1-ynylthiophen-2-yl)pyrazole-3-carboxamide
Show/Hide
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C26H28Cl2N4OS
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3
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| 1 |
EC50 = 14.1 nM
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| 2 |
IC50 = 1.2 nM
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| 3 |
IC50 = 7 nM
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CP0537810
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US9682955, 93
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C33H28Cl2N4O4S
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1
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| 1 |
EC50 = 14.2 nM
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CP0415446
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N-(azepan-1-yl)-1-(2,4-dichlorophenyl)-4-methyl-5-[5-(4-methylpent-1-ynyl)thiophen-2-yl]pyrazole-3-carboxamide
Show/Hide
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C27H30Cl2N4OS
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3
|
| 1 |
EC50 = 14.6 nM
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| 2 |
IC50 = 1.2 nM
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| 3 |
IC50 = 4.9 nM
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CP0433001
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(7E)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C31H24Cl2FN7O2
|
1
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| 1 |
EC50 = 15 nM
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CP0563751
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(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C32H27Cl2N7O3
|
1
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| 1 |
EC50 = 15 nM
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CP0803531
|
US9266835, 41
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C25H22ClF3N4O3S2
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1
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| 1 |
EC50 = 15 nM
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CP0434538
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4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[3,4-d][1,2]oxazol-9-ol
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C21H29NO3
|
1
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| 1 |
EC50 = 15.8 nM
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CP0334443
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N-[4-(cyclopropylamino)-4-oxobutyl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
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C27H37N3O3
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2
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| 1 |
EC50 = 16.2 nM
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| 2 |
Ki = 7.1 nM
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CP0460120
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N-(azepan-1-yl)-1-(2,4-dichlorophenyl)-4-ethyl-5-(5-pent-1-ynylthiophen-2-yl)pyrazole-3-carboxamide
Show/Hide
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C27H30Cl2N4OS
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3
|
| 1 |
EC50 = 16.5 nM
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| 2 |
IC50 = 1.2 nM
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| 3 |
IC50 = 8.9 nM
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CP0386471
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(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-5-[2-(methanesulfonamido)acetyl]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C30H27Cl3N6O4S
|
1
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| 1 |
EC50 = 17 nM
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CP0475838
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(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C31H25Cl2N7O2
|
1
|
| 1 |
EC50 = 17 nM
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CP0388774
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-chlorobenzyl)acetamide
Show/Hide
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C23H15Cl5N4O
|
2
|
| 1 |
EC50 = 17.8 nM
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|
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| 2 |
IC50 = 64.8 nM
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CP0400933
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(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
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C27H21Cl2F3N4OS
|
1
|
| 1 |
EC50 = 18 nM
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CP0433002
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-5-[(2S)-2,3-dihydroxypropanoyl]-N-[(1R)-1-phenylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C31H27Cl3N4O4
|
1
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| 1 |
EC50 = 18 nM
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CP0462577
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1-(2,4-Dichlorophenyl)-4-methyl-5-[5-(3-phenoxyprop-1-ynyl)-thiophen-2-yl]-1H-pyrazole-3-carboxylic Acid Piperidin-1-ylamide
Show/Hide
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C29H26Cl2N4O2S
|
2
|
| 1 |
EC50 = 18.7 nM
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| 2 |
IC50 = 43 nM
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CP0373855
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1-(2,4-Dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-5-(5-(pent-1-ynyl)thiophen-2-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C27H28Cl2N4OS
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2
|
| 1 |
EC50 = 19.2 nM
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| 2 |
IC50 = 7.9 nM
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CP0386470
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(7E)-5-(4-amino-4-oxobutanoyl)-1-(2,4-dichlorophenyl)-7-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C31H27Cl2FN6O3
|
1
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| 1 |
EC50 = 20 nM
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CP0467611
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-5,5-dimethyl-3,5-dihydro-imidazol-4-one
Show/Hide
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C22H19Cl3N4O
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2
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| 1 |
EC50 = 20.2 nM
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| 2 |
IC50 = 32.6 nM
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CP0373858
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1-(2,4-Dichlorophenyl)-4-methyl-5-(5-(4-phenylbut-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C30H28Cl2N4OS
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2
|
| 1 |
EC50 = 20.4 nM
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| 2 |
IC50 = 6.1 nM
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CP0713772
|
US9266835, 53
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C28H23Cl3F3N3O3S
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1
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| 1 |
EC50 = 20.4 nM
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CP0486648
|
US9682955, 54
Show/Hide
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C34H30Cl2F3N3O4
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1
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| 1 |
EC50 = 21.3 nM
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CP0444807
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(2,5-difluorobenzyl)acetamide
Show/Hide
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C23H14Cl4F2N4O
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2
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| 1 |
EC50 = 22 nM
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| 2 |
IC50 = 22.6 nM
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CP0447414
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(7E)-1-(4-chlorophenyl)-7-[(5-chloropyridin-2-yl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
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C27H23Cl2N5O
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1
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| 1 |
EC50 = 22 nM
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CP0419665
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(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-5-[(2S)-2,3-dihydroxypropanoyl]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C30H26Cl3N5O4
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1
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| 1 |
EC50 = 22 nM
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CP0426522
|
US9266835, 530
Show/Hide
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C31H30Cl2F3N3O4S
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1
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| 1 |
EC50 = 22 nM
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CP0467679
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1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(4-methylpent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C27H30Cl2N4OS
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2
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| 1 |
EC50 = 23 nM
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| 2 |
IC50 = 5.1 nM
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CP0388772
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2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(2-fluorobenzyl)acetamide
Show/Hide
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C23H15Cl4FN4O
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2
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| 1 |
EC50 = 23.5 nM
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| 2 |
IC50 = 19.3 nM
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CP0401021
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(7E)-5-(2-aminoacetyl)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C31H29Cl2N5O3
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1
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| 1 |
EC50 = 24 nM
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CP0243591
|
US9266835, 49
Show/Hide
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C29H26Cl2F3N3O3S
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1
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| 1 |
EC50 = 24 nM
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CP0175985
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(6S)-N-[2-(cyclopropylamino)-2-oxoethyl]-N-ethyl-9-methyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
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C26H35N3O3
|
2
|
| 1 |
EC50 = 24.2 nM
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| 2 |
Ki = 17.3 nM
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CP0415437
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5-(5-(Cyclopentylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C27H28Cl2N4OS
|
2
|
| 1 |
EC50 = 24.5 nM
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| 2 |
IC50 = 7.1 nM
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CP0375093
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3-(2,4-Dichlorophenyl)-4-(5-(3-ethoxyprop-1-ynyl)thiophen-2-yl)-5-methyl-N-(piperidin-1-yl)cyclopenta-1,4-dienecarboxamide
Show/Hide
|
C25H26Cl2N4O2S
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2
|
| 1 |
EC50 = 25.5 nM
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| 2 |
IC50 = 12.7 nM
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CP0483998
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(6-fluoro-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-ylmethanone
Show/Hide
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C24H20FNO4
|
2
|
| 1 |
EC50 = 26 nM
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| 2 |
Ki = 15 nM
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CP0411163
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(8E)-1-(4-chlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H26ClFN4O
|
1
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| 1 |
EC50 = 28 nM
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CP0573762
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(8E)-1-(2,4-dichlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-(1-pyridin-2-ylpiperidin-4-yl)-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C32H30Cl2FN5O
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1
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| 1 |
EC50 = 28 nM
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CP0545426
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(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5-(1H-1,2,4-triazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
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C30H24Cl2N8O2
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1
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| 1 |
EC50 = 28 nM
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CP0517210
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US9732061, Compound 36
Show/Hide
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C24H21ClF3N5O2S2
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1
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| 1 |
EC50 = 28 nM
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CP0386453
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1-(2,4-Dichlorophenyl)-4-methyl-5-(5-(pent-1-ynyl)thiophen-2-1-(2,4-Dichlorophenyl)-4-methyl-5-(5-(pent-1-ynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H26Cl2N4OS
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3
|
| 1 |
EC50 = 28.7 nM
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| 2 |
IC50 = 1.2 nM
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| 3 |
IC50 = 13.9 nM
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CP0386455
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1-(2,4-Dichlorophenyl)-5-(5-(3,3-dimethylbut-1-ynyl)thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4OS
|
2
|
| 1 |
EC50 = 28.9 nM
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| 2 |
IC50 = 32.7 nM
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CP0758258
|
US9266835, 62
Show/Hide
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C29H24ClF6N3O3S
|
1
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| 1 |
EC50 = 29 nM
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CP0375064
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N-butyl-1-(2,4-dichlorophenyl)-5-(5-hex-1-ynylthiophen-2-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H27Cl2N3OS
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2
|
| 1 |
EC50 = 29.8 nM
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| 2 |
IC50 = 3 nM
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CP0043110
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(2S)-N-(5-tert-butyl-1,2-oxazol-3-yl)-1-(4-chlorophenyl)pyrrolidine-2-carboxamide
Show/Hide
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C18H22ClN3O2
|
1
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| 1 |
EC50 = 30 nM
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CP0411161
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(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C28H23Cl3N4O
|
1
|
| 1 |
EC50 = 30 nM
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CP0451949
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(7E)-1-(4-chlorophenyl)-7-[(4-fluorophenyl)methylidene]-5-[2-(methanesulfonamido)acetyl]-N-[(1R)-1-pyridin-2-ylethyl]-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C30H28ClFN6O4S
|
1
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| 1 |
EC50 = 30 nM
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CP0385313
|
(6R)-N-ethyl-N-[4-(2-hydroxyethylamino)-4-oxobutyl]-9-methyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C27H39N3O4
|
1
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| 1 |
EC50 = 30.7 nM
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|
|
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CP0486580
|
US9682955, 114
Show/Hide
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C27H23Cl2F3N4O3S
|
1
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| 1 |
EC50 = 31.7 nM
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CP0451948
|
(7E)-1-(2,4-dichlorophenyl)-7-[(4-methoxyphenyl)methylidene]-N-[(1R)-1-phenylethyl]-5-(1H-pyrazole-5-carbonyl)-4,6-dihydropyrazolo[4,3-c]pyridine-3-carboxamide
Show/Hide
|
C33H28Cl2N6O3
|
1
|
| 1 |
EC50 = 32 nM
|
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CP0445931
|
(7E)-7-[(4-chlorophenyl)methylidene]-1-(2,4-dichlorophenyl)-N-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C31H28Cl3N5O
|
1
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| 1 |
EC50 = 34 nM
|
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CP0386504
|
(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-(2,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C26H21Cl3N4OS
|
1
|
| 1 |
EC50 = 35 nM
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CP0411165
|
(8E)-1-(3,4-dichlorophenyl)-8-[(4-fluorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
|
C29H25Cl2FN4O
|
1
|
| 1 |
EC50 = 35 nM
|
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|
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CP0388773
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(3-fluorobenzyl)acetamide
Show/Hide
|
C23H15Cl4FN4O
|
2
|
| 1 |
EC50 = 35.1 nM
|
|
|
| 2 |
IC50 = 25.7 nM
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CP0415442
|
5-(5-(But-1-ynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H26Cl2N4OS
|
2
|
| 1 |
EC50 = 35.5 nM
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|
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| 2 |
IC50 = 28.3 nM
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CP0415440
|
N-(azepan-1-yl)-5-(5-but-1-ynylthiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H26Cl2N4OS
|
2
|
| 1 |
EC50 = 36.4 nM
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| 2 |
IC50 = 24.2 nM
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CP0411162
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(8E)-8-[(4-chlorophenyl)methylidene]-1-(3,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
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C29H25Cl3N4O
|
1
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| 1 |
EC50 = 37 nM
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CP0509951
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(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-(3,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
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C26H21Cl3N4OS
|
1
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| 1 |
EC50 = 37 nM
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CP0175987
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(6R)-N-[2-(cyclopropylamino)-2-oxoethyl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
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C25H33N3O3
|
2
|
| 1 |
EC50 = 39.9 nM
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| 2 |
Ki = 24.5 nM
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CP0125866
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(6R)-N,9-dimethyl-6-(oxan-4-yl)-N-[4-(oxetan-3-ylamino)-4-oxobutyl]-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
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C27H37N3O4
|
1
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| 1 |
EC50 = 43.7 nM
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CP0373859
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N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(5-hex-1-ynylthiophen-2-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C27H29Cl2N3OS
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2
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| 1 |
EC50 = 43.9 nM
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| 2 |
IC50 = 2.1 nM
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CP0460128
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1-(2,4-Dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-5-(5-pentylthiophen-2-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C27H32Cl2N4OS
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2
|
| 1 |
EC50 = 48 nM
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| 2 |
IC50 = 20.6 nM
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CP0070269
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[5-ethylsulfonyl-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C25H35N3O4S
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2
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| 1 |
EC50 = 49 nM
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| 2 |
Ki = 120 nM
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CP0385362
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5-chloro-N-[2-[4-(dimethylamino)phenyl]ethyl]-3-ethyl-1H-indole-2-carboxamide
Show/Hide
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C21H24ClN3O
|
5
|
| 1 |
EC50 = 50 nM
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| 2 |
EC50 = 210 nM
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| 3 |
EC50 = 430 nM
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| 4 |
EC50 = 600 nM
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| 5 |
EC50 = 3430 nM
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CP0521468
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2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-fluorobenzyl)acetamide
Show/Hide
|
C23H15Cl4FN4O
|
2
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| 1 |
EC50 = 50.7 nM
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| 2 |
IC50 = 11.6 nM
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CP0119397
|
US9266835, 538
Show/Hide
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C33H33Cl2F3N4O4S
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1
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| 1 |
EC50 = 51 nM
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CP0460117
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5-(5-(But-1-ynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C24H24Cl2N4OS
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2
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| 1 |
EC50 = 51.4 nM
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| 2 |
IC50 = 65.4 nM
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CP0272283
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(6R)-N,9-dimethyl-N-[4-(methylamino)-4-oxobutyl]-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
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C25H35N3O3
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2
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| 1 |
EC50 = 51.4 nM
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| 2 |
Ki = 29.3 nM
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CP0205154
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1-(4-cyanophenyl)-3-[3-(6-pyrrolidin-1-ylpyridin-2-yl)phenyl]urea
Show/Hide
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C23H21N5O
|
1
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| 1 |
EC50 = 55.2 nM
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CP0451940
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(8E)-1-(3,4-dichlorophenyl)-N-[(1R)-1-pyridin-2-ylethyl]-8-[[4-(trifluoromethyl)phenyl]methylidene]-4,5,6,7-tetrahydrocyclohepta[c]pyrazole-3-carboxamide
Show/Hide
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C30H25Cl2F3N4O
|
1
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| 1 |
EC50 = 56 nM
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CP0566182
|
US9815790, 1
Show/Hide
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C37H42Cl2F3N3O7S
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1
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| 1 |
EC50 = 56 nM
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CP0504058
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2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-methoxybenzyl)acetamide
Show/Hide
|
C24H18Cl4N4O2
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2
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| 1 |
EC50 = 56.2 nM
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| 2 |
IC50 = 81.9 nM
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CP0375109
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1-(2,4-Dichlorophenyl)-5-(5-(3-isopropoxyprop-1-ynyl)thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H28Cl2N4O2S
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2
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| 1 |
EC50 = 57.4 nM
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| 2 |
IC50 = 23.2 nM
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CP0176000
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(6R)-N-[(2S)-5-(2-fluoroethylamino)-1-hydroxy-5-oxopentan-2-yl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C27H38FN3O4
|
1
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| 1 |
EC50 = 61.4 nM
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CP0078200
|
[5-hydroxy-1-(oxan-4-ylmethyl)indol-3-yl]-(4-methoxyphenyl)methanone
Show/Hide
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C22H23NO4
|
2
|
| 1 |
EC50 = 62.9 nM
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| 2 |
Ki = 1406 nM
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CP0713773
|
US9266835, 65
Show/Hide
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C29H24ClF3N4O3S2
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1
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| 1 |
EC50 = 64.2 nM
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CP0503126
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N-(azepan-1-yl)-5-(5-bromothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H21BrCl2N4OS
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2
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| 1 |
EC50 = 64.9 nM
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| 2 |
IC50 = 40.7 nM
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CP0388082
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1Hpyrazol-3-yl]-3,5,5-trimethyl-3,5-dihydro-imidazol-4-one
Show/Hide
|
C23H21Cl3N4O
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2
|
| 1 |
EC50 = 65.5 nM
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| 2 |
IC50 = 33.8 nM
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CP0572838
|
6-[(4-chlorophenyl)-imidazol-1-ylmethyl]-4-[(1R,2S)-2-phenylcyclopropyl]-1H-quinolin-2-one
Show/Hide
|
C28H22ClN3O
|
1
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| 1 |
EC50 = 66 nM
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CP0462567
|
5-(5-bromothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H19BrCl2N4OS
|
2
|
| 1 |
EC50 = 68.2 nM
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| 2 |
IC50 = 35.8 nM
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CP0334446
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(6R)-N-[4-(cyanomethylamino)-4-oxobutyl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C26H34N4O3
|
1
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| 1 |
EC50 = 70.6 nM
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CP0375062
|
1-(2,4-Dichlorophenyl)-4-methyl-5-[((E)-5-pent-1-enyl)-thiophen-2-yl]-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C27H30Cl2N4OS
|
2
|
| 1 |
EC50 = 71.4 nM
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| 2 |
IC50 = 27.5 nM
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CP0461191
|
(6-fluoro-2,2-bis(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone
Show/Hide
|
C25H20F3NO3
|
2
|
| 1 |
EC50 = 72 nM
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| 2 |
Ki = 7 nM
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CP0460118
|
5-(5-(Cyclopropylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H24Cl2N4OS
|
2
|
| 1 |
EC50 = 72.9 nM
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| 2 |
IC50 = 60.4 nM
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CP0460119
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1-(2,4-Dichlorophenyl)-5-(5-(hex-1-ynyl)thiophen-2-yl)-N-hexyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C27H31Cl2N3OS
|
2
|
| 1 |
EC50 = 74 nM
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| 2 |
IC50 = 2.6 nM
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CP0511854
|
US9682955, 107
Show/Hide
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C27H24Cl2F3N5O2S
|
1
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| 1 |
EC50 = 74.8 nM
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CP0813853
|
US9266835, 47
Show/Hide
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C24H20ClF3N4O3S2
|
1
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| 1 |
EC50 = 75 nM
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CP0489886
|
1-(2,4-Dichlorophenyl)-4-methyl-5-(5-pentylthiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H30Cl2N4OS
|
2
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| 1 |
EC50 = 75.9 nM
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| 2 |
IC50 = 57.9 nM
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CP0426521
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3-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[6-[bis(4-chlorophenyl)methyl]-4-[[1-(trifluoromethylsulfonyl)piperidin-4-yl]amino]quinolin-8-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoic acid
Show/Hide
|
C55H76Cl2F3N3O17S
|
1
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| 1 |
EC50 = 77 nM
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CP0134486
|
(6R)-N-[(2S)-5-(ethylamino)-1-hydroxy-5-oxopentan-2-yl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C27H39N3O4
|
1
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| 1 |
EC50 = 78.7 nM
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CP0314717
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N,9-dimethyl-N-[4-(methylamino)-4-oxobutyl]-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C25H35N3O3
|
2
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| 1 |
EC50 = 78.9 nM
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| 2 |
Ki = 53.7 nM
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CP0467612
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2-[1-(2,4-Dichloro-phenyl)-4-methyl-5-(4-trifluoromethylphenyl)-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C23H19Cl2F3N4O
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2
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| 1 |
EC50 = 81 nM
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| 2 |
IC50 = 15.9 nM
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CP0435287
|
N-benzyl-2-[4,5-bis(2,4-dichlorophenyl)triazol-2-yl]acetamide
Show/Hide
|
C23H16Cl4N4O
|
2
|
| 1 |
EC50 = 87 nM
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| 2 |
IC50 = 66.9 nM
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CP0385536
|
5-chloro-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
EC50 = 90 nM
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CP0250155
|
US9266835, 535
Show/Hide
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C34H34Cl2F3N3O5S
|
1
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| 1 |
EC50 = 92 nM
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CP0326974
|
US9266835, 63
Show/Hide
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C28H27Cl2N3O3S
|
1
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| 1 |
EC50 = 94.4 nM
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CP0804943
|
rac-N-(2-(cyclopropylamino)-2-oxoethyl)-N,9-dimethyl-3-(tetrahydro-2H-pyran-4-yl)-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
Show/Hide
|
C25H33N3O3
|
2
|
| 1 |
EC50 = 95.3 nM
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| 2 |
Ki = 44.5 nM
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CP0472557
|
4-N-[6-[bis(4-chlorophenyl)methyl]cinnolin-4-yl]-1-N-phenylcyclohexane-1,4-diamine
Show/Hide
|
C33H30Cl2N4
|
1
|
| 1 |
EC50 = 99 nM
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CP0460284
|
5-(5-(Cyclopentylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C29H30Cl2N4OS
|
2
|
| 1 |
EC50 = 99.3 nM
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| 2 |
IC50 = 10.5 nM
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CP0432243
|
(6R)-N-[(2S)-1-hydroxy-5-(methylamino)-5-oxopentan-2-yl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C26H37N3O4
|
1
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| 1 |
EC50 = 101 nM
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CP0386457
|
5-(5-(Cyclopropylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C27H26Cl2N4OS
|
2
|
| 1 |
EC50 = 104.8 nM
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| 2 |
IC50 = 21 nM
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CP0263236
|
US9266835, 537
Show/Hide
|
C33H32Cl2F3N3O5S
|
1
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| 1 |
EC50 = 108 nM
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CP0578088
|
6-[(4-chlorophenyl)-imidazol-1-ylmethyl]-4-[[4-(trifluoromethoxy)phenyl]methyl]-1H-quinolin-2-one
Show/Hide
|
C27H19ClF3N3O2
|
1
|
| 1 |
EC50 = 113 nM
|
|
|
|
CP0747958
|
US9266835, 11
Show/Hide
|
C27H20Cl2N2OS
|
1
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| 1 |
EC50 = 121 nM
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CP0437701
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-1-(piperidin-1-yl)ethanone
Show/Hide
|
C21H18Cl4N4O
|
2
|
| 1 |
EC50 = 122 nM
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| 2 |
IC50 = 168.9 nM
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CP0747957
|
US9266835, 136
Show/Hide
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C28H24Cl2F3N3O4S
|
1
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| 1 |
EC50 = 122 nM
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CP0467704
|
ethyl 2-[6-[bis(4-chlorophenyl)methyl]-4-[[1-(trifluoromethylsulfonyl)piperidin-4-yl]amino]quinolin-8-yl]oxyacetate
Show/Hide
|
C32H30Cl2F3N3O5S
|
1
|
| 1 |
EC50 = 126 nM
|
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CP0447415
|
(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
Show/Hide
|
C28H24Cl2N4O
|
1
|
| 1 |
EC50 = 127 nM
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|
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CP0375107
|
N-(azepan-1-yl)-5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C21H21Cl3N4OS
|
2
|
| 1 |
EC50 = 133.9 nM
|
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| 2 |
IC50 = 158.7 nM
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CP0428633
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-phenylacetamide
Show/Hide
|
C22H14Cl4N4O
|
2
|
| 1 |
EC50 = 136.2 nM
|
|
|
| 2 |
IC50 = 251.1 nM
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CP0387212
|
5-chloro-3-ethyl-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H28ClN3O
|
6
|
| 1 |
EC50 = 140 nM
|
|
|
| 2 |
EC50 = 640 nM
|
|
|
| 3 |
EC50 = 2090 nM
|
|
|
| 4 |
EC50 = 2240 nM
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| 5 |
EC50 = 10590 nM
|
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| 6 |
IC50 = 158.49 nM
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CP0415433
|
1-(2,4-Dichlorophenyl)-5-(5-(3-methoxyprop-1-ynyl)thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H24Cl2N4O2S
|
2
|
| 1 |
EC50 = 142.7 nM
|
|
|
| 2 |
IC50 = 65.3 nM
|
|
|
|
CP0279473
|
US9266835, 542
Show/Hide
|
C32H33Cl2F3N4O3S
|
1
|
| 1 |
EC50 = 144 nM
|
|
|
|
CP0375063
|
1-(2,4-Dichlorophenyl)-4-methyl-5-[((E)-5-pent-1-enyl)-thiophen-2-yl]-1H-pyrazole-3-carboxylic Acid Piperidin-1-ylamide
Show/Hide
|
C25H28Cl2N4OS
|
2
|
| 1 |
EC50 = 146.2 nM
|
|
|
| 2 |
IC50 = 21.6 nM
|
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CP0373856
|
5-(5-Chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H19Cl3N4OS
|
2
|
| 1 |
EC50 = 146.5 nM
|
|
|
| 2 |
IC50 = 50.2 nM
|
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|
|
CP0483996
|
(2-(2,4-dichlorophenyl)-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone
Show/Hide
|
C24H18Cl2FNO4
|
2
|
| 1 |
EC50 = 156 nM
|
|
|
| 2 |
Ki = 30 nM
|
|
|
|
CP0346676
|
US9266835, 129
Show/Hide
|
C35H31Cl2N3O3
|
1
|
| 1 |
EC50 = 157 nM
|
|
|
|
CP0454981
|
1-(2,4-Dichlorophenyl)-5-(5-(3,3-dimethylbut-1-ynyl)thiophen-2-yl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C28H30Cl2N4OS
|
2
|
| 1 |
EC50 = 158.4 nM
|
|
|
| 2 |
IC50 = 21.7 nM
|
|
|
|
CP0249763
|
US9266835, 122
Show/Hide
|
C34H29Cl2N3O5S
|
1
|
| 1 |
EC50 = 159 nM
|
|
|
|
CP0538076
|
6-[(4-chlorophenyl)-imidazol-1-ylmethyl]-4-[(E)-2-phenylethenyl]-1H-quinolin-2-one
Show/Hide
|
C27H20ClN3O
|
1
|
| 1 |
EC50 = 165 nM
|
|
|
|
CP0228439
|
1-(4-chlorophenyl)-3-[3-(6-pyrrolidin-1-ylpyridin-2-yl)phenyl]urea
Show/Hide
|
C22H21ClN4O
|
7
|
| 1 |
EC50 = 167 nM
|
|
|
| 2 |
IC50 = 1.47 nM
|
|
|
| 3 |
IC50 = 50 nM
|
|
|
| 4 |
IC50 = 230 nM
|
|
|
| 5 |
IC50 = 398.11 nM
|
|
|
| 6 |
IC50 = 455 nM
|
|
|
| 7 |
IC50 = 2620 nM
|
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|
CP0513379
|
(6R)-N-[4-(2-hydroxyethylamino)-4-oxobutyl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C26H37N3O4
|
1
|
| 1 |
EC50 = 173 nM
|
|
|
|
CP0421306
|
4,4-dimethyl-7-(2-methyloctan-2-yl)-9-phenylmethoxy-1H-chromeno[4,3-c]pyrazole
Show/Hide
|
C28H36N2O2
|
1
|
| 1 |
EC50 = 191 nM
|
|
|
|
CP0445458
|
2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-cyclohexylacetamide
Show/Hide
|
C22H20Cl4N4O
|
2
|
| 1 |
EC50 = 203.6 nM
|
|
|
| 2 |
IC50 = 144.4 nM
|
|
|
|
CP0880359
|
US9266835, 40
Show/Hide
|
C27H29ClN4O3S2
|
1
|
| 1 |
EC50 = 204 nM
|
|
|
|
CP0379222
|
1-(4-fluorophenyl)-3-[3-(6-pyrrolidin-1-ylpyridin-2-yl)phenyl]urea
Show/Hide
|
C22H21FN4O
|
1
|
| 1 |
EC50 = 207 nM
|
|
|
|
CP0486799
|
N-benzyl-2-[4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)triazol-2-yl]acetamide
Show/Hide
|
C23H17Cl3N4O
|
2
|
| 1 |
EC50 = 216.3 nM
|
|
|
| 2 |
IC50 = 203.5 nM
|
|
|
|
CP0266404
|
US9266835, 96
Show/Hide
|
C30H27Cl2N3O4
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0250148
|
US9266835, 110
Show/Hide
|
C31H30Cl2F3N3O4S
|
1
|
| 1 |
EC50 = 228 nM
|
|
|
|
CP0492352
|
5-chloro-3-methyl-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C23H26ClN3O
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0428634
|
2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-fluorobenzyl)acetamide
Show/Hide
|
C23H16Cl3FN4O
|
2
|
| 1 |
EC50 = 235.2 nM
|
|
|
| 2 |
IC50 = 449.2 nM
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|
|
|
CP0455069
|
2-(4-(4-chlorophenyl)-5-(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(2-fluorobenzyl)acetamide
Show/Hide
|
C23H16Cl3FN4O
|
2
|
| 1 |
EC50 = 256.1 nM
|
|
|
| 2 |
IC50 = 262.2 nM
|
|
|
|
CP0579010
|
6-[(4-chlorophenyl)methyl]-4-[[1-(trifluoromethylsulfonyl)piperidin-4-yl]amino]-1H-quinolin-2-one
Show/Hide
|
C22H21ClF3N3O3S
|
1
|
| 1 |
EC50 = 260 nM
|
|
|
|
CP0326975
|
US9266835, 84
Show/Hide
|
C34H29Cl2N3O5S
|
1
|
| 1 |
EC50 = 269 nM
|
|
|
|
CP0808704
|
US9266835, 137
Show/Hide
|
C32H33ClF3N5O3S
|
1
|
| 1 |
EC50 = 290 nM
|
|
|
|
CP0432244
|
(6R)-N-[4-(methoxyamino)-4-oxobutyl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C25H35N3O4
|
1
|
| 1 |
EC50 = 291 nM
|
|
|
|
CP0415434
|
5-(5-(Cyclohexylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C30H32Cl2N4OS
|
2
|
| 1 |
EC50 = 293.6 nM
|
|
|
| 2 |
IC50 = 7.8 nM
|
|
|
|
CP0434521
|
2-(2-hydroxyethyl)-4,4-dimethyl-7-(2-methyloctan-2-yl)chromeno[4,3-c]pyrazol-9-ol
Show/Hide
|
C23H34N2O3
|
1
|
| 1 |
EC50 = 298.8 nM
|
|
|
|
CP0563464
|
US9732061, Compound 12
Show/Hide
|
C34H30Cl2N4O2
|
1
|
| 1 |
EC50 = 302 nM
|
|
|
|
CP0250147
|
US9266835, 108
Show/Hide
|
C32H31Cl2F3N4O5S
|
1
|
| 1 |
EC50 = 310 nM
|
|
|
|
CP0543863
|
6-[(4-chlorophenyl)-(1,3-thiazol-2-yl)methyl]-4-[[4-(trifluoromethylsulfonyl)piperazin-1-yl]amino]-1H-quinolin-2-one
Show/Hide
|
C24H21ClF3N5O3S2
|
1
|
| 1 |
EC50 = 322 nM
|
|
|
|
CP0415438
|
1-(2,4-Dichlorophenyl)-5-(5-(3-(dimethylamino)prop-1-ynyl)-thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H27Cl2N5OS
|
2
|
| 1 |
EC50 = 348.8 nM
|
|
|
| 2 |
IC50 = 124.2 nM
|
|
|
|
CP0385361
|
5-chloro-3-ethyl-N-[2-(4-nitrophenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C19H18ClN3O3
|
5
|
| 1 |
EC50 = 360 nM
|
|
|
| 2 |
EC50 = 440 nM
|
|
|
| 3 |
EC50 = 660 nM
|
|
|
| 4 |
EC50 = 1140 nM
|
|
|
| 5 |
EC50 = 3590 nM
|
|
|
|
CP0373857
|
1-(2,4-Dichlorophenyl)-5-(5-(3-(isopropylamino)prop-1-ynyl)-thiophen-2-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C26H29Cl2N5OS
|
2
|
| 1 |
EC50 = 390.1 nM
|
|
|
| 2 |
IC50 = 82.4 nM
|
|
|
|
CP0838621
|
US9266835, 28
Show/Hide
|
C28H18ClF3N2OS
|
1
|
| 1 |
EC50 = 396 nM
|
|
|
|
CP0219426
|
US9266835, 541
Show/Hide
|
C28H24Cl2F3N3O3S
|
1
|
| 1 |
EC50 = 399 nM
|
|
|
|
CP0414613
|
1-(6-chloropyridin-3-yl)-3-[3-(6-pyrrolidin-1-ylpyridin-2-yl)phenyl]urea
Show/Hide
|
C21H20ClN5O
|
1
|
| 1 |
EC50 = 408 nM
|
|
|
|
CP0321871
|
US9266835, 116
Show/Hide
|
C35H29Cl2N3O4
|
1
|
| 1 |
EC50 = 438 nM
|
|
|
|
CP0489882
|
5-(5-(Cyclohexylethynyl)thiophen-2-yl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C28H30Cl2N4OS
|
2
|
| 1 |
EC50 = 442.4 nM
|
|
|
| 2 |
IC50 = 7.3 nM
|
|
|
|
CP0134485
|
(6S)-N-[2-(cyclopropylamino)-2-oxoethyl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C25H33N3O3
|
2
|
| 1 |
EC50 = 446 nM
|
|
|
| 2 |
Ki = 177 nM
|
|
|
|
CP0563833
|
US9732061, Compound 1
Show/Hide
|
C27H23Cl2F3N4O3S
|
1
|
| 1 |
EC50 = 455 nM
|
|
|
|
CP0440160
|
US9815790, 2
Show/Hide
|
C43H54Cl2F3N3O10S
|
1
|
| 1 |
EC50 = 457 nM
|
|
|
|
CP0876434
|
(S)-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(2-methoxypyrrolidin-1-yl)methanone
Show/Hide
|
C25H18F5NO4
|
2
|
| 1 |
EC50 = 466 nM
|
|
|
| 2 |
Ki = 46 nM
|
|
|
|
CP0395905
|
5-chloro-3-ethyl-N-[2-(4-methylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C20H21ClN2O
|
5
|
| 1 |
EC50 = 470 nM
|
|
|
| 2 |
EC50 = 550 nM
|
|
|
| 3 |
EC50 = 600 nM
|
|
|
| 4 |
EC50 = 790 nM
|
|
|
| 5 |
EC50 = 1010 nM
|
|
|
|
CP0548532
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-[6-(difluoromethoxy)pyridin-3-yl]piperazine-1-carboxamide
Show/Hide
|
C28H22Cl2F2N8O2
|
2
|
| 1 |
EC50 = 590 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0763370
|
US9266835, 39
Show/Hide
|
C24H23ClN4OS
|
1
|
| 1 |
EC50 = 604 nM
|
|
|
|
CP0241006
|
US9266835, 141
Show/Hide
|
C32H34Cl2F3N5O3S
|
1
|
| 1 |
EC50 = 625 nM
|
|
|
|
CP0149320
|
[7-hydroxy-1-(oxan-4-ylmethyl)indol-3-yl]-(4-methoxyphenyl)methanone
Show/Hide
|
C22H23NO4
|
2
|
| 1 |
EC50 = 632.5 nM
|
|
|
| 2 |
Ki = 3583 nM
|
|
|
|
CP0398854
|
1-(4-chlorophenyl)-3-[3-[6-(dimethylamino)pyridin-2-yl]phenyl]urea
Show/Hide
|
C20H19ClN4O
|
1
|
| 1 |
EC50 = 663 nM
|
|
|
|
CP0395907
|
5-chloro-N-[2-(4-chlorophenyl)ethyl]-3-ethyl-1H-indole-2-carboxamide
Show/Hide
|
C19H18Cl2N2O
|
5
|
| 1 |
EC50 = 760 nM
|
|
|
| 2 |
EC50 = 1840 nM
|
|
|
| 3 |
EC50 = 3420 nM
|
|
|
| 4 |
EC50 = 8180 nM
|
|
|
| 5 |
EC50 = 20000 nM
|
|
|
|
CP0529340
|
(2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(morpholino)methanone
Show/Hide
|
C24H21NO4
|
2
|
| 1 |
EC50 = 784 nM
|
|
|
| 2 |
Ki = 50 nM
|
|
|
|
CP0223129
|
(2-{4-[7-(benzylmethylamino)heptyloxy]phenyl}benzofuran-3-yl)phenylmethanone
Show/Hide
|
C36H37NO3
|
2
|
| 1 |
EC50 = 790 nM
|
|
|
| 2 |
Ki = 320 nM
|
|
|
|
CP0380710
|
3-ethyl-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H29N3O
|
5
|
| 1 |
EC50 = 810 nM
|
|
|
| 2 |
EC50 = 2990 nM
|
|
|
| 3 |
EC50 = 3550 nM
|
|
|
| 4 |
EC50 = 4010 nM
|
|
|
| 5 |
EC50 = 6840 nM
|
|
|
|
CP0772732
|
US9266835, 25
Show/Hide
|
C27H19ClN2OS
|
1
|
| 1 |
EC50 = 817 nM
|
|
|
|
CP0324009
|
US9266835, 127
Show/Hide
|
C35H31Cl2N3O3
|
1
|
| 1 |
EC50 = 876 nM
|
|
|
|
CP0399752
|
5-chloro-3-ethyl-N-[2-[4-(methylamino)phenyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C20H22ClN3O
|
1
|
| 1 |
EC50 = 960 nM
|
|
|
|
CP0402742
|
(2S,4S)-N-[(2S)-1-fluoro-3,3-dimethylbutan-2-yl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C18H22FN5O2
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0700560
|
US9266835, 135
Show/Hide
|
C29H26ClF4N3O3S
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0578045
|
6-[(4-chlorophenyl)-imidazol-1-ylmethyl]-4-phenylmethoxy-1H-quinolin-2-one
Show/Hide
|
C26H20ClN3O2
|
1
|
| 1 |
EC50 = 1150 nM
|
|
|
|
CP0795027
|
US9266835, 33
Show/Hide
|
C31H21ClF3NO
|
1
|
| 1 |
EC50 = 1210 nM
|
|
|
|
CP0471785
|
US9266835, 532
Show/Hide
|
C30H26Cl2F3N3O5S
|
1
|
| 1 |
EC50 = 1284 nM
|
|
|
|
CP0257209
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[4-(2-morpholin-4-ylethoxy)phenyl]methanone
Show/Hide
|
C42H48N2O5
|
2
|
| 1 |
EC50 = 1370 nM
|
|
|
| 2 |
Ki = 550 nM
|
|
|
|
CP0400642
|
5-chloro-3-(1-hydroxyethyl)-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H28ClN3O2
|
5
|
| 1 |
EC50 = 1510 nM
|
|
|
| 2 |
EC50 = 2660 nM
|
|
|
| 3 |
EC50 = 2970 nM
|
|
|
| 4 |
EC50 = 8450 nM
|
|
|
| 5 |
EC50 = 13370 nM
|
|
|
|
CP0398781
|
1-[3-[6-(butylamino)pyridin-2-yl]phenyl]-3-(4-chlorophenyl)urea
Show/Hide
|
C22H23ClN4O
|
1
|
| 1 |
EC50 = 1520 nM
|
|
|
|
CP0417341
|
5-chloro-N-[2-[4-(dimethylamino)phenyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C19H20ClN3O
|
1
|
| 1 |
EC50 = 1530 nM
|
|
|
|
CP0164723
|
US9266835, 106
Show/Hide
|
C30H28Cl2N4O3
|
1
|
| 1 |
EC50 = 1550 nM
|
|
|
|
CP0776704
|
US9266835, 42
Show/Hide
|
C28H29ClN4O3S
|
1
|
| 1 |
EC50 = 2330 nM
|
|
|
|
CP0382149
|
(4-chlorophenyl)-[4-(3,5-dichlorophenyl)-3-hydroxy-5-methoxyphenyl]methanone
Show/Hide
|
C20H13Cl3O3
|
1
|
| 1 |
EC50 = 2880 nM
|
|
|
|
CP0382148
|
(4-chlorophenyl)-[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]methanone
Show/Hide
|
C19H11Cl3O3
|
1
|
| 1 |
EC50 = 3280 nM
|
|
|
|
CP0803537
|
US9266835, 21
Show/Hide
|
C28H20ClNOS
|
1
|
| 1 |
EC50 = 4140 nM
|
|
|
|
CP0389340
|
5-chloro-3-ethyl-N-[2-(4-fluorophenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C19H18ClFN2O
|
5
|
| 1 |
EC50 = 4580 nM
|
|
|
| 2 |
EC50 = 4990 nM
|
|
|
| 3 |
EC50 = 7370 nM
|
|
|
| 4 |
EC50 = 8960 nM
|
|
|
| 5 |
EC50 > 10000 nM
|
|
|
|
CP0566181
|
2-[6-[bis(4-chlorophenyl)methyl]-4-[[1-(trifluoromethylsulfonyl)piperidin-4-yl]amino]quinolin-8-yl]oxyacetic acid
Show/Hide
|
C30H26Cl2F3N3O5S
|
1
|
| 1 |
EC50 = 4900 nM
|
|
|
|
CP0472556
|
US9732061, Compound 19
Show/Hide
|
C33H28Cl2N4O4S
|
1
|
| 1 |
EC50 = 5944 nM
|
|
|
|
CP0403234
|
(2S,4S)-N-[(2S)-1-fluoro-3-methylbutan-2-yl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C17H20FN5O2
|
1
|
| 1 |
EC50 = 6100 nM
|
|
|
|
CP0334844
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[3-[2-(diethylamino)ethoxy]phenyl]methanone
Show/Hide
|
C42H50N2O4
|
2
|
| 1 |
EC50 = 6380 nM
|
|
|
| 2 |
Ki = 2570 nM
|
|
|
|
CP0156123
|
7-[4-(1-benzofuran-2-yl)phenoxy]-N-benzyl-N-methylheptan-1-amine
Show/Hide
|
C29H33NO2
|
2
|
| 1 |
EC50 = 6950 nM
|
|
|
| 2 |
Ki = 2800 nM
|
|
|
|
CP0199912
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-(4-phenylphenyl)methanone
Show/Hide
|
C42H41NO3
|
2
|
| 1 |
EC50 = 7740 nM
|
|
|
| 2 |
Ki = 3120 nM
|
|
|
|
CP0241001
|
US9266835, 117
Show/Hide
|
C29H27Cl2N3O3
|
1
|
| 1 |
EC50 = 9700 nM
|
|
|
|
CP0380713
|
5-chloro-N-[2-(4-nitrophenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C17H14ClN3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0383427
|
5-chloro-N-[2-(4-chlorophenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C17H14Cl2N2O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0385535
|
N-[2-(4-aminophenyl)ethyl]-5-chloro-3-ethyl-1H-indole-2-carboxamide
Show/Hide
|
C19H20ClN3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0407748
|
5-chloro-3-ethyl-N-[2-(4-pyrrolidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C23H26ClN3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0410149
|
5-chloro-3-ethyl-N-[2-[4-(4-methylpiperazin-1-yl)phenyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H29ClN4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0087627
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[3-(diethylaminomethyl)phenyl]methanone
Show/Hide
|
C41H48N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0120662
|
anthracen-9-yl-[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]methanone
Show/Hide
|
C44H41NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0257210
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C40H39NO3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0259142
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[4-(diethylaminomethyl)phenyl]methanone
Show/Hide
|
C41H48N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0315950
|
[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-naphthalen-2-ylmethanone
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C40H39NO3
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2
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| 1 |
EC50 > 10000 nM
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| 2 |
Ki > 10000 nM
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CP0319745
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[2-[4-[7-[benzyl(methyl)amino]heptoxy]phenyl]-1-benzofuran-3-yl]-[4-[2-(diethylamino)ethoxy]phenyl]methanone
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C42H50N2O4
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2
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| 1 |
EC50 > 10000 nM
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| 2 |
Ki > 10000 nM
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CP0155571
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(2R,4R)-9-(2,4-difluorophenyl)-N-(1-hydroxy-2-methylpropan-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C18H19F2N3O2
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1
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| 1 |
EC50 > 10000 nM
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CP0204257
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APD-371
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C18H23N5O3
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1
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| 1 |
EC50 > 10000 nM
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CP0402740
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(2S,4S)-N-(1-methylcyclopropyl)-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C16H17N5O2
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1
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| 1 |
EC50 > 10000 nM
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CP0412791
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(2S,4S)-N-[(1S)-2-hydroxy-1-phenylethyl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C20H19N5O3
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1
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| 1 |
EC50 > 10000 nM
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CP0416862
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(2S,4S)-N-[(2R)-1-hydroxy-3,3-dimethylbutan-2-yl]-9-pyrazin-2-yl-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C18H23N5O2
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1
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| 1 |
EC50 > 10000 nM
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CP0416863
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(2R,4R)-N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-9-pyrazin-2-yl-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C18H23N5O2
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1
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| 1 |
EC50 > 10000 nM
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CP0416864
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(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-[(2R)-1,1,1-trifluoro-3-hydroxypropan-2-yl]-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C15H14F3N5O3
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1
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| 1 |
EC50 > 10000 nM
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CP0459091
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(2S,4S)-N-[1-(hydroxymethyl)cyclopentyl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C18H21N5O3
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1
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| 1 |
EC50 > 10000 nM
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CP0463801
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(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-[1-(trifluoromethyl)cyclobutyl]-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C17H16F3N5O2
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1
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| 1 |
EC50 > 10000 nM
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CP0473682
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(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-[1-(trifluoromethyl)cyclopropyl]-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C16H14F3N5O2
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1
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| 1 |
EC50 > 10000 nM
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CP0473684
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(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-(1,1,1-trifluoro-2-methylpropan-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
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C16H16F3N5O2
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1
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| 1 |
EC50 > 10000 nM
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CP0475675
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(2S,4S)-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-9-(4-oxidopyrazin-4-ium-2-yl)-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C17H21N5O3
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1
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| 1 |
EC50 > 10000 nM
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CP0477572
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(2S,4S)-N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-9-pyrazin-2-yl-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C18H23N5O2
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1
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| 1 |
EC50 > 10000 nM
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CP0482613
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(2S,4S)-9-(4-oxidopyrazin-4-ium-2-yl)-N-[(2S)-1,1,1-trifluoro-3-hydroxypropan-2-yl]-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
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C15H14F3N5O3
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1
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| 1 |
EC50 > 10000 nM
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CP0440175
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6-[(4-chlorophenyl)-hydroxymethyl]-4-[(E)-2-phenylethenyl]-1H-quinolin-2-one
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C24H18ClNO2
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1
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| 1 |
EC50 > 10000 nM
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CP0471828
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N-[6-[(4-chlorophenyl)-imidazol-1-ylmethyl]-2-oxo-1H-quinolin-4-yl]benzamide
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C26H19ClN4O2
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1
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| 1 |
EC50 > 10000 nM
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CP0579008
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6-[(4-chlorophenyl)-imidazol-1-ylmethyl]-4-(2-phenylethyl)-1H-quinolin-2-one
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C27H22ClN3O
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1
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| 1 |
EC50 > 10000 nM
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CP0258259
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5-tert-butyl-N-(1-hydroxy-2-methylpropan-2-yl)-1-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-3-carboxamide
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C18H23F3N4O2
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1
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| 1 |
EC50 > 10000 nM
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CP0385955
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[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]-[4-(trifluoromethyl)phenyl]methanone
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C20H11Cl2F3O3
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1
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| 1 |
EC50 > 5000 nM
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CP0450547
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cyclohexyl-[4-(3,5-dichlorophenyl)-3,5-dihydroxyphenyl]methanone
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C19H18Cl2O3
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1
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| 1 |
EC50 > 5000 nM
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CP0848668
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4-(methylamino)phenethyl 5-chloro-3-ethyl-1H-indole-2-carboxylate
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C20H21ClN2O2
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1
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| 1 |
EC50 < 10000 nM
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CP0106737
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N-[(2S,3S)-4-(4-chlorophenyl)-3-(3-cyanophenyl)butan-2-yl]-2-methyl-2-[5-(trifluoromethyl)pyridin-2-yl]oxypropanamide
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C27H25ClF3N3O2
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2
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| 1 |
IC50 = 0.3 nM
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| 2 |
Ki = 0.3 nM
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CP0045801
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(10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tetrahydro-6H-benzo[c]chromen-1-ol
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C21H30O2
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3
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| 1 |
IC50 = 2.8 nM
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| 2 |
Ki = 10 nM
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| 3 |
Ki = 18 nM
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CP0428706
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5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(3-methoxyphenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
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C27H28Cl2N2O2
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1
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| 1 |
IC50 = 6.8 nM
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CP0444451
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5-cyclohexyl-3-methyl-1-o-tolyl-2-(4-(trifluoromethyl)phenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
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C28H29F3N2O
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1
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| 1 |
IC50 = 9.3 nM
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CP0085568
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N-cyclohexyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
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C21H22Cl2N4O
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2
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| 1 |
IC50 = 10 nM
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| 2 |
Ki = 5.6 nM
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CP0465173
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2-(benzo[d][1,3]dioxol-5-yl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
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C27H26Cl2N2O3
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1
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| 1 |
IC50 = 12 nM
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CP0399820
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-1,3-diaza-spiro[4.5]dec-1-en-4-one
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C25H23Cl3N4O
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1
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| 1 |
IC50 = 12.3 nM
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CP0463993
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-1,3-diaza-spiro[4.4]non-1-en-4-one
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C24H21Cl3N4O
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1
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| 1 |
IC50 = 14.6 nM
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CP0528616
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-phenyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C26H26Cl2N2O
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1
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| 1 |
IC50 = 16 nM
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CP0455903
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2-[5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
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C23H21BrCl2N4O
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1
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| 1 |
IC50 = 16.3 nM
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CP0522321
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-m-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C27H28Cl2N2O
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1
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| 1 |
IC50 = 17 nM
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CP0444454
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(thiophen-2-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
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C24H24Cl2N2OS
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1
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| 1 |
IC50 = 19 nM
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CP0428704
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5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(furan-2-yl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C24H24Cl2N2O2
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1
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| 1 |
IC50 = 20 nM
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CP0501072
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5-cyclohexyl-2-(4-methoxyphenyl)-3-methyl-1-o-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C28H32N2O2
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1
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| 1 |
IC50 = 22 nM
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CP0444453
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2-(benzo[b]thiophen-2-yl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C28H26Cl2N2OS
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1
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| 1 |
IC50 = 23 nM
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CP0051325
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N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C23H26Cl2N4O
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2
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| 1 |
IC50 = 25 nM
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| 2 |
Ki = 14 nM
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CP0435955
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naphthalen-1-yl-[4-(pentylamino)naphthalen-1-yl]methanone
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C26H25NO
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1
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| 1 |
IC50 = 25 nM
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CP0511251
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-3,5,5-trimethyl-3,5-dihydro-imidazol-4-one
Show/Hide
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C22H19Cl3N4O
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1
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| 1 |
IC50 = 33.6 nM
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CP0439805
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(thiophen-3-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C24H24Cl2N2OS
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1
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| 1 |
IC50 = 37 nM
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CP0532376
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5-cyclohexyl-2-(4-fluorophenyl)-3-methyl-1-o-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C27H29FN2O
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1
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| 1 |
IC50 = 40 nM
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CP0456628
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2-[4-Bromo-5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
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C21H16BrCl3N4O
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1
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| 1 |
IC50 = 42.5 nM
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CP0417371
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2-[5-(4-Chloro-phenyl)-4-cyclopropyl-1-(2,4-dichloro-phenyl)-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
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C24H21Cl3N4O
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1
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| 1 |
IC50 = 43.9 nM
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CP0527090
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2-[5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
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C22H19BrCl2N4O
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1
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| 1 |
IC50 = 47.4 nM
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CP0434158
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(4-butoxynaphthalen-1-yl)-naphthalen-1-ylmethanone
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C25H22O2
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1
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| 1 |
IC50 = 48 nM
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CP0373045
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N-cyclohexyl-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
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C23H25Cl3N4O
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2
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| 1 |
IC50 = 50 nM
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| 2 |
Ki = 28 nM
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CP0405137
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1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C24H20Cl4N4O
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2
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| 1 |
IC50 = 50 nM
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| 2 |
Ki = 28 nM
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CP0433182
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1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H25Cl2N5O
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2
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| 1 |
IC50 = 50 nM
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| 2 |
Ki = 28 nM
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CP0398571
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-5,5-dimethyl-3,5-dihydro-imidazol-4-one
Show/Hide
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C21H17Cl3N4O
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1
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| 1 |
IC50 = 53.4 nM
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CP0102148
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1-(3,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C20H21Cl2N5O
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2
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| 1 |
IC50 = 54 nM
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| 2 |
Ki = 30 nM
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CP0455904
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
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C22H19Cl3N4O
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1
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| 1 |
IC50 = 54.7 nM
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CP0257790
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1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H16Cl4N4O
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2
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| 1 |
IC50 = 62 nM
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| 2 |
Ki = 35 nM
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CP0440923
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N-[(3,4-dichlorophenyl)methyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C24H20Cl2F2N4O
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2
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| 1 |
IC50 = 62 nM
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| 2 |
Ki = 35 nM
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CP0454268
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N-cyclohexyl-1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C23H26F2N4O
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2
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| 1 |
IC50 = 62 nM
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| 2 |
Ki = 35 nM
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CP0372929
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1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H16Cl4N4O
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2
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| 1 |
IC50 = 66 nM
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| 2 |
Ki = 37 nM
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CP0440912
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1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H25Cl2N5O
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2
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| 1 |
IC50 = 67 nM
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| 2 |
Ki = 38 nM
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CP0428705
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(3-(trifluoromethyl)phenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C27H25Cl2F3N2O
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1
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| 1 |
IC50 = 67 nM
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CP0440914
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N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C23H26Cl2N4O
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2
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| 1 |
IC50 = 74 nM
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| 2 |
Ki = 42 nM
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CP0230625
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[4-[(4-fluorophenyl)methyl-methylamino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
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C30H24FNO3
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2
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| 1 |
IC50 = 80 nM
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| 2 |
Ki = 20 nM
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CP0529812
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5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-N-(2-(dimethylamino)-2-methylpropanoyl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C23H23Cl3N4O2
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1
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| 1 |
IC50 = 82.9 nM
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CP0422587
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1-(4-chlorophenyl)-3-[5-(2,4-difluorophenyl)thiophen-2-yl]urea
Show/Hide
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C17H11ClF2N2OS
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2
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| 1 |
IC50 = 84 nM
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| 2 |
IC50 = 2290 nM
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CP0458229
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[(6aR,10aR)-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-yl] acetate
Show/Hide
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C23H32O3
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4
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| 1 |
IC50 = 87 nM
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| 2 |
IC50 = 88 nM
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| 3 |
Ki = 43 nM
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| 4 |
Ki = 44 nM
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CP0527089
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2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-1-cyclopropyl-5,5-dimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
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C24H21Cl3N4O
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1
|
| 1 |
IC50 = 95.2 nM
|
|
|
|
CP0446280
|
[(6aR,10aR)-9-hydroperoxy-6,6,9-trimethyl-3-pentyl-10,10a-dihydro-6aH-benzo[c]chromen-1-yl] 4-methylbenzenesulfonate
Show/Hide
|
C28H36O6S
|
4
|
| 1 |
IC50 = 97 nM
|
|
|
| 2 |
IC50 = 275 nM
|
|
|
| 3 |
Ki = 48 nM
|
|
|
| 4 |
Ki = 137 nM
|
|
|
|
CP0372927
|
N-cyclohexyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H22Cl2N4O
|
2
|
| 1 |
IC50 = 100 nM
|
|
|
| 2 |
Ki = 56 nM
|
|
|
|
CP0463994
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-1-ethyl-5,5-dimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C23H21Cl3N4O
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0396843
|
(E)-2-(benzenesulfonyl)-3-[1-(2-morpholin-4-ylethyl)indol-3-yl]prop-2-enenitrile
Show/Hide
|
C23H23N3O3S
|
2
|
| 1 |
IC50 = 155 nM
|
|
|
| 2 |
Ki = 62 nM
|
|
|
|
CP0451682
|
(4-hexyloxynaphthalen-1-yl)naphthalen-1-ylmethanone
Show/Hide
|
C27H26O2
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0404193
|
1-(4-chlorophenyl)-3-[3-[(6-pyrrolidin-1-ylpyridin-2-yl)amino]phenyl]urea
Show/Hide
|
C22H22ClN5O
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0522905
|
1-Benzyl-2-[5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-5,5-dimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C28H23Cl3N4O
|
1
|
| 1 |
IC50 = 197 nM
|
|
|
|
CP0372735
|
5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperidin-1-yl)-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H24Cl3N5O
|
2
|
| 1 |
IC50 = 200 nM
|
|
|
| 2 |
Ki = 110 nM
|
|
|
|
CP0372932
|
1-(4-chlorophenyl)-N-(cyclohexylmethyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H25ClN4O
|
2
|
| 1 |
IC50 = 200 nM
|
|
|
| 2 |
Ki = 110 nM
|
|
|
|
CP0422483
|
1-(4-chlorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H22ClN5O
|
2
|
| 1 |
IC50 = 200 nM
|
|
|
| 2 |
Ki = 110 nM
|
|
|
|
CP0455905
|
2-[1-(2,4-Dichloro-phenyl)-5-(4-methoxy-phenyl)-4-methyl-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C23H22Cl2N4O2
|
1
|
| 1 |
IC50 = 211.8 nM
|
|
|
|
CP0528596
|
1-Allyl-2-[5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-5,5-dimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C24H21Cl3N4O
|
1
|
| 1 |
IC50 = 248.9 nM
|
|
|
|
CP0426820
|
1-(4-chlorophenyl)-3-(5-pyridin-4-ylthiophen-2-yl)urea
Show/Hide
|
C16H12ClN3OS
|
2
|
| 1 |
IC50 = 263 nM
|
|
|
| 2 |
IC50 = 1800 nM
|
|
|
|
CP0422516
|
1-(4-chlorophenyl)-3-[5-(2-chlorophenyl)thiophen-2-yl]urea
Show/Hide
|
C17H12Cl2N2OS
|
2
|
| 1 |
IC50 = 272 nM
|
|
|
| 2 |
IC50 = 1190 nM
|
|
|
|
CP0404194
|
1-(4-chlorophenyl)-3-[3-(3-pyrrolidin-1-ylphenyl)phenyl]urea
Show/Hide
|
C23H22ClN3O
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0422623
|
1-(4-chlorophenyl)-3-(5-pyridin-3-ylthiophen-2-yl)urea
Show/Hide
|
C16H12ClN3OS
|
1
|
| 1 |
IC50 = 298 nM
|
|
|
|
CP0372383
|
naphthalen-1-yl-(4-propoxynaphthalen-1-yl)methanone
Show/Hide
|
C24H20O2
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0222933
|
[2-(4-methoxyphenyl)-1-benzofuran-3-yl]-[4-(pentylamino)phenyl]methanone
Show/Hide
|
C27H27NO3
|
2
|
| 1 |
IC50 = 300 nM
|
|
|
| 2 |
Ki = 80 nM
|
|
|
|
CP0506592
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyrazol-3-yl]-1,5,5-trimethyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C21H17Cl3N4O
|
1
|
| 1 |
IC50 = 325.1 nM
|
|
|
|
CP0446278
|
(6aR,9S,10aR)-6,6,9-trimethyl-3-pentyl-10,10a-dihydro-6aH-benzo[c]chromene-1,9-diol
Show/Hide
|
C21H30O3
|
4
|
| 1 |
IC50 = 387 nM
|
|
|
| 2 |
IC50 = 930 nM
|
|
|
| 3 |
Ki = 193 nM
|
|
|
| 4 |
Ki = 470 nM
|
|
|
|
CP0418412
|
1-(4-chlorophenyl)-3-[5-(3-fluorophenyl)thiophen-2-yl]urea
Show/Hide
|
C17H12ClFN2OS
|
1
|
| 1 |
IC50 = 425 nM
|
|
|
|
CP0426819
|
1-(4-chlorophenyl)-3-[5-(4-methoxyphenyl)thiophen-2-yl]urea
Show/Hide
|
C18H15ClN2O2S
|
2
|
| 1 |
IC50 = 449 nM
|
|
|
| 2 |
IC50 = 1850 nM
|
|
|
|
CP0497601
|
US9422235, 105
Show/Hide
|
C17H24F3N3O2S
|
2
|
| 1 |
IC50 = 459 nM
|
|
|
| 2 |
Ki = 325 nM
|
|
|
|
CP0379503
|
4-cyano-N-[(3,4-dichlorophenyl)methyl]-1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H15Cl2N5O
|
2
|
| 1 |
IC50 = 500 nM
|
|
|
| 2 |
Ki = 280 nM
|
|
|
|
CP0379504
|
1-(4-chlorophenyl)-N-cyclohexyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H21ClN4O
|
2
|
| 1 |
IC50 = 500 nM
|
|
|
| 2 |
Ki = 280 nM
|
|
|
|
CP0393710
|
N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(1H-pyrrol-1-yl)-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H15Cl5N4O
|
2
|
| 1 |
IC50 = 500 nM
|
|
|
| 2 |
Ki = 280 nM
|
|
|
|
CP0422466
|
1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H20Cl4N4O
|
2
|
| 1 |
IC50 = 500 nM
|
|
|
| 2 |
Ki = 280 nM
|
|
|
|
CP0439944
|
1-(4-chlorophenyl)-3-(5-phenylthiophen-2-yl)urea
Show/Hide
|
C17H13ClN2OS
|
2
|
| 1 |
IC50 = 524 nM
|
|
|
| 2 |
IC50 = 1760 nM
|
|
|
|
CP0426094
|
1-(4-chlorophenyl)-3-[5-(4-fluorophenyl)thiophen-2-yl]urea
Show/Hide
|
C17H12ClFN2OS
|
1
|
| 1 |
IC50 = 537 nM
|
|
|
|
CP0400705
|
N-[3-(3,3-difluoroazetidine-1-carbonyl)-5,7-dihydro-4H-thieno[2,3-c]pyran-2-yl]tricyclo[3.3.1.03,7]nonane-3-carboxamide
Show/Hide
|
C21H24F2N2O3S
|
1
|
| 1 |
IC50 = 549.54 nM
|
|
|
|
CP0421532
|
1-(4-chlorophenyl)-3-[5-(3-chlorophenyl)thiophen-2-yl]urea
Show/Hide
|
C17H12Cl2N2OS
|
1
|
| 1 |
IC50 = 553 nM
|
|
|
|
CP0519498
|
(9,9,13-trimethyl-5-pentyl-8,14-dioxatetracyclo[8.5.0.02,7.013,15]pentadeca-1(10),2(7),3,5-tetraen-3-yl) acetate
Show/Hide
|
C23H30O4
|
2
|
| 1 |
IC50 = 573 nM
|
|
|
| 2 |
Ki = 286 nM
|
|
|
|
CP0421531
|
1-(4-chlorophenyl)-3-(5-phenyl-1,3-thiazol-2-yl)urea
Show/Hide
|
C16H12ClN3OS
|
1
|
| 1 |
IC50 = 604 nM
|
|
|
|
CP0459716
|
1-(4-chlorophenyl)-3-(4-phenylthiophen-2-yl)urea
Show/Hide
|
C17H13ClN2OS
|
1
|
| 1 |
IC50 = 667 nM
|
|
|
|
CP0570047
|
1-(4-chlorophenyl)-3-[2-[3-(trifluoromethyl)phenyl]ethyl]urea
Show/Hide
|
C16H14ClF3N2O
|
1
|
| 1 |
IC50 = 676.08 nM
|
|
|
|
CP0542736
|
1-[2-(3-bromophenyl)ethyl]-3-(4-chlorophenyl)urea
Show/Hide
|
C15H14BrClN2O
|
1
|
| 1 |
IC50 = 724.44 nM
|
|
|
|
CP0422588
|
1-(4-chlorophenyl)-3-[5-(4-chlorophenyl)thiophen-2-yl]urea
Show/Hide
|
C17H12Cl2N2OS
|
1
|
| 1 |
IC50 = 774 nM
|
|
|
|
CP0415436
|
naphthalen-1-yl-(2-pentyl-1-benzothiophen-3-yl)methanone
Show/Hide
|
C24H22OS
|
2
|
| 1 |
IC50 = 800 nM
|
|
|
| 2 |
Ki = 500 nM
|
|
|
|
CP0463996
|
2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1Hpyrazol-3-yl]-5,5-dimethyl-1-propyl-1,5-dihydro-imidazol-4-one
Show/Hide
|
C24H23Cl3N4O
|
1
|
| 1 |
IC50 = 853.6 nM
|
|
|
|
CP0575797
|
1-(4-chlorophenyl)-3-[2-(3-cyanophenyl)ethyl]urea
Show/Hide
|
C16H14ClN3O
|
1
|
| 1 |
IC50 = 870.96 nM
|
|
|
|
CP0426101
|
1-(4-chlorophenyl)-3-(5-phenylthiophen-3-yl)urea
Show/Hide
|
C17H13ClN2OS
|
1
|
| 1 |
IC50 = 888 nM
|
|
|
|
CP0546146
|
1-(4-chlorophenyl)-3-[2-(3-methylphenyl)ethyl]urea
Show/Hide
|
C16H17ClN2O
|
1
|
| 1 |
IC50 = 912.01 nM
|
|
|
|
CP0445802
|
naphthalen-1-yl-[4-(2-phenylethoxy)naphthalen-1-yl]methanone
Show/Hide
|
C29H22O2
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0477868
|
US9422235, 28
Show/Hide
|
C19H22Cl2N2O5S
|
2
|
| 1 |
IC50 = 961 nM
|
|
|
| 2 |
Ki = 426 nM
|
|
|
|
CP0415470
|
naphthalen-1-yl-(2-propyl-1-benzothiophen-3-yl)methanone
Show/Hide
|
C22H18OS
|
2
|
| 1 |
IC50 = 1000 nM
|
|
|
| 2 |
Ki = 600 nM
|
|
|
|
CP0477194
|
[(6aR,10R,10aR)-10-hydroperoxy-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-yl] 4-methylbenzenesulfonate
Show/Hide
|
C28H36O6S
|
2
|
| 1 |
IC50 = 1024 nM
|
|
|
| 2 |
Ki = 512 nM
|
|
|
|
CP0458228
|
9-methoxy-6,6,9-trimethyl-3-pentyl-8,10-dihydro-7H-benzo[c]chromene-1,10-diol
Show/Hide
|
C22H32O4
|
2
|
| 1 |
IC50 = 1077 nM
|
|
|
| 2 |
Ki = 538 nM
|
|
|
|
CP0378554
|
[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C27H25NO3
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0308436
|
(4-methoxyphenyl)-[2-(4-methoxyphenyl)-1-benzothiophen-3-yl]methanone
Show/Hide
|
C23H18O3S
|
2
|
| 1 |
IC50 = 1100 nM
|
|
|
| 2 |
Ki = 700 nM
|
|
|
|
CP0506593
|
1-Butyl-2-[5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-5,5-dimethyl-1,5-dihydro-imidazol-4one
Show/Hide
|
C25H25Cl3N4O
|
1
|
| 1 |
IC50 = 1110.8 nM
|
|
|
|
CP0569657
|
1-(4-chlorophenyl)-3-[2-(3,4-dimethylphenyl)ethyl]urea
Show/Hide
|
C17H19ClN2O
|
1
|
| 1 |
IC50 = 1148.15 nM
|
|
|
|
CP0503233
|
butyl 2-[4,5-bis(2,4-dichlorophenyl)triazol-2-yl]acetate
Show/Hide
|
C20H17Cl4N3O2
|
1
|
| 1 |
IC50 = 1173.2 nM
|
|
|
|
CP0434074
|
1-(4-chlorophenyl)-3-[5-(3-methylphenyl)thiophen-2-yl]urea
Show/Hide
|
C18H15ClN2OS
|
1
|
| 1 |
IC50 = 1180 nM
|
|
|
|
CP0415435
|
[2-(2-methylpropyl)-1-benzothiophen-3-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C23H20OS
|
2
|
| 1 |
IC50 = 1200 nM
|
|
|
| 2 |
Ki = 700 nM
|
|
|
|
CP0451011
|
[(6aR,10S,10aR)-10-hydroxy-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-1-yl] 4-methylbenzenesulfonate
Show/Hide
|
C28H36O5S
|
2
|
| 1 |
IC50 = 1280 nM
|
|
|
| 2 |
Ki = 642 nM
|
|
|
|
CP0571149
|
1-(4-chlorophenyl)-3-[2-(3-fluorophenyl)ethyl]urea
Show/Hide
|
C15H14ClFN2O
|
1
|
| 1 |
IC50 = 1348.96 nM
|
|
|
|
CP0577016
|
1-(4-chlorophenyl)-3-[2-(3-chlorophenyl)ethyl]urea
Show/Hide
|
C15H14Cl2N2O
|
1
|
| 1 |
IC50 = 1513.56 nM
|
|
|
|
CP0134008
|
[4-[2-[benzyl(methyl)amino]ethoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C32H29NO4
|
2
|
| 1 |
IC50 = 1520 nM
|
|
|
| 2 |
Ki = 430 nM
|
|
|
|
CP0384803
|
US9422235, 88
Show/Hide
|
C19H27F3N2O2S
|
2
|
| 1 |
IC50 = 1669 nM
|
|
|
| 2 |
Ki = 930 nM
|
|
|
|
CP0327891
|
[4-(cyclopropylmethylamino)phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C26H23NO3
|
2
|
| 1 |
IC50 = 1670 nM
|
|
|
| 2 |
Ki = 470 nM
|
|
|
|
CP0576701
|
1-(4-chlorophenyl)-3-[2-(4-fluorophenyl)ethyl]urea
Show/Hide
|
C15H14ClFN2O
|
1
|
| 1 |
IC50 = 1698.24 nM
|
|
|
|
CP0426095
|
1-(4-chlorophenyl)-3-[5-(3,4-dichlorophenyl)thiophen-2-yl]urea
Show/Hide
|
C17H11Cl3N2OS
|
1
|
| 1 |
IC50 = 1720 nM
|
|
|
|
CP0542735
|
1-(4-chlorophenyl)-3-[2-(4-nitrophenyl)ethyl]urea
Show/Hide
|
C15H14ClN3O3
|
1
|
| 1 |
IC50 = 1778.28 nM
|
|
|
|
CP0482647
|
(6aR,9S)-9-ethoxy-6,6,9-trimethyl-3-pentyl-7,8-dihydro-6aH-benzo[c]chromene-1,4-dione
Show/Hide
|
C23H32O4
|
2
|
| 1 |
IC50 = 1840 nM
|
|
|
| 2 |
Ki = 919 nM
|
|
|
|
CP0511698
|
2-(4-chlorophenyl)-N-[3-(3-pyrrolidin-1-ylphenyl)phenyl]acetamide
Show/Hide
|
C24H23ClN2O
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0483301
|
US9422235, 17
Show/Hide
|
C19H23FN2O5S
|
2
|
| 1 |
IC50 = 2000 nM
|
|
|
| 2 |
Ki = 889 nM
|
|
|
|
CP0489601
|
US9422235, 7
Show/Hide
|
C17H17F3N2O2S
|
2
|
| 1 |
IC50 = 2000 nM
|
|
|
| 2 |
Ki = 1156 nM
|
|
|
|
CP0422517
|
1-(4-chlorophenyl)-3-[5-(2-methoxyphenyl)thiophen-2-yl]urea
Show/Hide
|
C18H15ClN2O2S
|
1
|
| 1 |
IC50 = 2020 nM
|
|
|
|
CP0578647
|
1-(4-chlorophenyl)-3-[2-(4-methylphenyl)ethyl]urea
Show/Hide
|
C16H17ClN2O
|
1
|
| 1 |
IC50 = 2041.74 nM
|
|
|
|
CP0211385
|
[4-[3-[benzyl(methyl)amino]propoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C33H31NO4
|
2
|
| 1 |
IC50 = 2060 nM
|
|
|
| 2 |
Ki = 500 nM
|
|
|
|
CP0461445
|
(E)-N-[(2R)-1-hydroxy-3-methoxypropan-2-yl]-N-methyloctadec-4-enamide
Show/Hide
|
C23H45NO3
|
2
|
| 1 |
IC50 = 2300 nM
|
|
|
| 2 |
Ki = 1300 nM
|
|
|
|
CP0534016
|
1-(4-chlorophenyl)-3-[2-[4-(dimethylamino)phenyl]ethyl]urea
Show/Hide
|
C17H20ClN3O
|
1
|
| 1 |
IC50 = 2511.89 nM
|
|
|
|
CP0426102
|
methyl 3-[5-[(4-chlorophenyl)carbamoylamino]thiophen-2-yl]benzoate
Show/Hide
|
C19H15ClN2O3S
|
1
|
| 1 |
IC50 = 2530 nM
|
|
|
|
CP0459715
|
1-(4-chlorophenyl)-3-(2-phenylpyridin-4-yl)urea
Show/Hide
|
C18H14ClN3O
|
1
|
| 1 |
IC50 = 2770 nM
|
|
|
|
CP0372944
|
N-cyclohexyl-1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H22F2N4O
|
2
|
| 1 |
IC50 = 2800 nM
|
|
|
| 2 |
Ki = 1600 nM
|
|
|
|
CP0440880
|
1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H25F2N5O
|
2
|
| 1 |
IC50 = 2800 nM
|
|
|
| 2 |
Ki = 1600 nM
|
|
|
|
CP0412001
|
(1-hydroxy-9-methoxy-6,6,9-trimethyl-3-pentyl-8,10-dihydro-7H-benzo[c]chromen-10-yl) acetate
Show/Hide
|
C24H34O5
|
2
|
| 1 |
IC50 = 2800 nM
|
|
|
| 2 |
Ki = 1400 nM
|
|
|
|
CP0490473
|
1-(4-chlorophenyl)-3-(2-phenylethyl)urea
Show/Hide
|
C15H15ClN2O
|
2
|
| 1 |
IC50 = 3162.28 nM
|
|
|
| 2 |
IC50 = 3467.37 nM
|
|
|
|
CP0379501
|
4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H20Cl3N5O
|
2
|
| 1 |
IC50 = 3200 nM
|
|
|
| 2 |
Ki = 1800 nM
|
|
|
|
CP0225671
|
[4-[(4-fluorophenyl)methylamino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C29H22FNO3
|
2
|
| 1 |
IC50 = 3210 nM
|
|
|
| 2 |
Ki = 780 nM
|
|
|
|
CP0422589
|
1-(4-chlorophenyl)-3-[5-(3-methylsulfonylphenyl)thiophen-2-yl]urea
Show/Hide
|
C18H15ClN2O3S2
|
1
|
| 1 |
IC50 = 3230 nM
|
|
|
|
CP0489361
|
1-(4-chlorophenyl)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]urea
Show/Hide
|
C16H14ClF3N2O
|
1
|
| 1 |
IC50 = 3235.94 nM
|
|
|
|
CP0418410
|
1-(4-chlorophenyl)-3-[5-(3-methoxyphenyl)thiophen-2-yl]urea
Show/Hide
|
C18H15ClN2O2S
|
2
|
| 1 |
IC50 = 3280 nM
|
|
|
| 2 |
IC50 = 6350 nM
|
|
|
|
CP0431778
|
1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H21Cl2N5O
|
2
|
| 1 |
IC50 = 3300 nM
|
|
|
| 2 |
Ki = 1850 nM
|
|
|
|
CP0474155
|
1-[5-(3-acetylphenyl)thiophen-2-yl]-3-(4-chlorophenyl)urea
Show/Hide
|
C19H15ClN2O2S
|
1
|
| 1 |
IC50 = 3430 nM
|
|
|
|
CP0400698
|
N-propyl-2-(tricyclo[3.3.1.03,7]nonane-3-carbonylamino)-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide
Show/Hide
|
C21H28N2O3S
|
1
|
| 1 |
IC50 = 3467.37 nM
|
|
|
|
CP0327835
|
[4-[4-[benzyl(methyl)amino]butoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C34H33NO4
|
2
|
| 1 |
IC50 = 3520 nM
|
|
|
| 2 |
Ki = 860 nM
|
|
|
|
CP0466611
|
US9422235, 26
Show/Hide
|
C19H25F3N2O3S
|
2
|
| 1 |
IC50 = 3808 nM
|
|
|
| 2 |
Ki = 1804 nM
|
|
|
|
CP0423528
|
1-(4-chlorophenyl)-3-(2-pyrrolidin-1-ylethyl)urea
Show/Hide
|
C13H18ClN3O
|
1
|
| 1 |
IC50 = 3981.07 nM
|
|
|
|
CP0908268
|
1-(4-chlorophenyl)-3-(4-methoxyphenethyl)urea
Show/Hide
|
C16H17ClN2O2
|
1
|
| 1 |
IC50 = 4168.69 nM
|
|
|
|
CP0542720
|
1-(4-chlorophenyl)-3-[2-(3,5-dichlorophenyl)ethyl]urea
Show/Hide
|
C15H13Cl3N2O
|
1
|
| 1 |
IC50 = 4365.16 nM
|
|
|
|
CP0435286
|
4,5-Bis-(2,4-dichloro-phenyl)-[1,2,3]triazole-2-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C25H22Cl4N4O
|
1
|
| 1 |
IC50 = 4496.8 nM
|
|
|
|
CP0419750
|
1-benzothiophen-2-yl(naphthalen-1-yl)methanone
Show/Hide
|
C19H12OS
|
2
|
| 1 |
IC50 = 4500 nM
|
|
|
| 2 |
Ki = 2700 nM
|
|
|
|
CP0419754
|
(2-cyclohexylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C24H22N2O
|
2
|
| 1 |
IC50 = 4900 nM
|
|
|
| 2 |
Ki = 2900 nM
|
|
|
|
CP0372933
|
1-(4-chlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-3-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C22H17Cl3N4O
|
2
|
| 1 |
IC50 = 5000 nM
|
|
|
| 2 |
Ki = 2820 nM
|
|
|
|
CP0372945
|
1-(2,4-difluorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H21F2N5O
|
2
|
| 1 |
IC50 = 5000 nM
|
|
|
| 2 |
Ki = 2800 nM
|
|
|
|
CP0431799
|
1-(4-chlorophenyl)-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C19H20ClN5O
|
2
|
| 1 |
IC50 = 5000 nM
|
|
|
| 2 |
Ki = 2820 nM
|
|
|
|
CP0431800
|
1-(4-chlorophenyl)-4-cyano-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H19ClN6O
|
2
|
| 1 |
IC50 = 5000 nM
|
|
|
| 2 |
Ki = 2820 nM
|
|
|
|
CP0440911
|
N-[(3,4-dichlorophenyl)methyl]-1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H16Cl2F2N4O
|
2
|
| 1 |
IC50 = 5000 nM
|
|
|
| 2 |
Ki = 2800 nM
|
|
|
|
CP0426037
|
1-(4-chlorophenyl)-3-[5-[3-(dimethylamino)phenyl]thiophen-2-yl]urea
Show/Hide
|
C19H18ClN3OS
|
2
|
| 1 |
IC50 = 5020 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0412000
|
[(6aR,10aR)-8-hydroperoxy-6,6-dimethyl-9-methylidene-3-pentyl-7,8,10,10a-tetrahydro-6aH-benzo[c]chromen-1-yl] 4-methylbenzenesulfonate
Show/Hide
|
C28H36O6S
|
2
|
| 1 |
IC50 = 5700 nM
|
|
|
| 2 |
Ki = 2850 nM
|
|
|
|
CP0134010
|
[4-(heptylamino)phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C29H31NO3
|
2
|
| 1 |
IC50 = 5840 nM
|
|
|
| 2 |
Ki = 1660 nM
|
|
|
|
CP0451742
|
US9422235, 94
Show/Hide
|
C16H22F3N3O2S
|
2
|
| 1 |
IC50 = 6000 nM
|
|
|
| 2 |
Ki = 3000 nM
|
|
|
|
CP0471298
|
US9422235, 87
Show/Hide
|
C18H25F3N2O2S
|
2
|
| 1 |
IC50 = 6000 nM
|
|
|
| 2 |
Ki = 3000 nM
|
|
|
|
CP0477866
|
US9422235, 31
Show/Hide
|
C20H21F3N2O3S
|
2
|
| 1 |
IC50 = 6000 nM
|
|
|
| 2 |
Ki = 2680 nM
|
|
|
|
CP0483289
|
US9422235, 16
Show/Hide
|
C17H19F3N4O4S
|
2
|
| 1 |
IC50 = 6000 nM
|
|
|
| 2 |
Ki = 2666 nM
|
|
|
|
CP0483303
|
US9422235, 39
Show/Hide
|
C16H16F2N2O2S
|
1
|
| 1 |
IC50 = 6000 nM
|
|
|
|
CP0491079
|
US9422235, 32
Show/Hide
|
C19H27F3N2O3S
|
2
|
| 1 |
IC50 = 6000 nM
|
|
|
| 2 |
Ki = 2680 nM
|
|
|
|
CP0511964
|
US9422235, 92
Show/Hide
|
C17H23F3N2O2S
|
2
|
| 1 |
IC50 = 6000 nM
|
|
|
| 2 |
Ki = 3000 nM
|
|
|
|
CP0512366
|
US9422235, 108
Show/Hide
|
C19H27F3N2O2S
|
2
|
| 1 |
IC50 = 6000 nM
|
|
|
| 2 |
Ki = 6000 nM
|
|
|
|
CP0421533
|
1-(4-chlorophenyl)-3-[5-(3,5-dichlorophenyl)thiophen-2-yl]urea
Show/Hide
|
C17H11Cl3N2OS
|
2
|
| 1 |
IC50 = 6330 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0546122
|
1-(4-chlorophenyl)-3-[2-(3,5-dimethylphenyl)ethyl]urea
Show/Hide
|
C17H19ClN2O
|
1
|
| 1 |
IC50 = 6606.93 nM
|
|
|
|
CP0363236
|
[4-[5-[benzyl(methyl)amino]pentoxy]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C35H35NO4
|
2
|
| 1 |
IC50 = 7200 nM
|
|
|
| 2 |
Ki = 1760 nM
|
|
|
|
CP0458144
|
(4-methoxyphenyl)-[2-(2-methylpropyl)-1-benzothiophen-3-yl]methanone
Show/Hide
|
C20H20O2S
|
2
|
| 1 |
IC50 = 7600 nM
|
|
|
| 2 |
Ki = 4600 nM
|
|
|
|
CP0533305
|
1-(4-chlorophenyl)-3-[2-(3-methoxyphenyl)ethyl]urea
Show/Hide
|
C16H17ClN2O2
|
1
|
| 1 |
IC50 = 7762.47 nM
|
|
|
|
CP0385256
|
[2-(4-methoxyphenyl)benzimidazol-1-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C25H18N2O2
|
2
|
| 1 |
IC50 = 8100 nM
|
|
|
| 2 |
Ki = 4900 nM
|
|
|
|
CP0420581
|
(2-ethyl-1-benzothiophen-3-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C21H16OS
|
2
|
| 1 |
IC50 = 8400 nM
|
|
|
| 2 |
Ki = 5100 nM
|
|
|
|
CP0446597
|
[2-(4-methoxyphenyl)-1-benzothiophen-3-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C26H18O2S
|
2
|
| 1 |
IC50 = 8400 nM
|
|
|
| 2 |
Ki = 5100 nM
|
|
|
|
CP0491074
|
US9422235, 10
Show/Hide
|
C17H17Cl2F3N2O2S
|
2
|
| 1 |
IC50 = 8571 nM
|
|
|
| 2 |
Ki = 4757 nM
|
|
|
|
CP0262329
|
4-[[4-[2-(4-methoxyphenyl)-1-benzofuran-3-carbonyl]anilino]methyl]benzonitrile
Show/Hide
|
C30H22N2O3
|
2
|
| 1 |
IC50 = 9120 nM
|
|
|
| 2 |
Ki = 2600 nM
|
|
|
|
CP0519327
|
17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H27NO2
|
2
|
| 1 |
IC50 = 9350 nM
|
|
|
| 2 |
Ki = 3770 nM
|
|
|
|
CP0511699
|
1-(4-chlorophenyl)-3-[3-(3-pyrrolidin-1-ylanilino)phenyl]urea
Show/Hide
|
C23H23ClN4O
|
1
|
| 1 |
IC50 = 9600 nM
|
|
|
|
CP0446588
|
(2-cyclobutylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C22H18N2O
|
2
|
| 1 |
IC50 = 9700 nM
|
|
|
| 2 |
Ki = 5800 nM
|
|
|
|
CP0454683
|
(2-butylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C22H20N2O
|
2
|
| 1 |
IC50 = 9700 nM
|
|
|
| 2 |
Ki = 5900 nM
|
|
|
|
CP0373773
|
11-(4-hexyl-3-hydroxy-phenoxy)-undecanoic acid cyclopropylmethyl-amide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0378997
|
11-(4-hexyl-3-hydroxy-phenoxy)-undecanoic acid[2-(3,4-dihydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C31H47NO5
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0432937
|
12-(4-hexyl-3-hydroxy-phenoxy)-dodecanoic acidcyclopropylamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0437123
|
12-(4-hexyl-3-hydroxy-phenoxy)-dodecanoic acid(2-hydroxy-ethyl)-amide
Show/Hide
|
C26H45NO4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0437124
|
11-(4-hexyl-3-hydroxy-phenoxy)-undecanoic acid(3-methoxy-4-hydroxy-phenyl)-amide
Show/Hide
|
C31H47NO5
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0479102
|
(E)-6-Biphenyl-4-yl-4-oxohexanoic acid ethanolamide
Show/Hide
|
C20H23NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0493393
|
1-Biphenyl-4-yl-4-morpholin-4-yl-butane-1,4-dione
Show/Hide
|
C20H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858811
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid cyclopropamide
Show/Hide
|
C19H19NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858812
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid ethanolamide
Show/Hide
|
C19H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858813
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid(2-hydroxy-1(R)-methylethanolamide
Show/Hide
|
C20H23NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858814
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid
Show/Hide
|
C16H14O3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858815
|
(E)-6-(3,4-Dimethoxyphenyl)-4-oxohex-5-enoic acid ethanolamide
Show/Hide
|
C16H21NO5
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858816
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic piperidinamide
Show/Hide
|
C22H25NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858817
|
(E)-6-Biphenyl-4-yl-4-oxohex-5-enoic acid ethanolamide
Show/Hide
|
C20H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0861035
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid(4-hydroxyphenyl)-amide
Show/Hide
|
C22H19NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0878641
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid(2-hydroxy-1(R)-methylethanolamide
Show/Hide
|
C19H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0878642
|
(E)-7-Naphthalen-2-yl-5-oxo-hept-6-enoic acid glycinamide ethyl ester
Show/Hide
|
C21H23NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0884366
|
(E)-N-(4-Hydroxyphenyl)-6-(4-methoxyphenyl)-4-oxohex-5-enamide
Show/Hide
|
C19H19NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0890249
|
(E)-6-(3,4-Dimethoxyphenyl)4-oxohex-5-enoic acid piperedinamide
Show/Hide
|
C19H25NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0906698
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid cyclopropylamide
Show/Hide
|
C20H21NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0906700
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid piperidinamide
Show/Hide
|
C21H23NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0914916
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid glycinamide ethyl ester
Show/Hide
|
C20H21NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0914917
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid ethanolamide
Show/Hide
|
C18H19NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0918957
|
(E)-6-Naphthalen-2-yl-4-oxohex-5-enoic acid diethanolamide
Show/Hide
|
C20H23NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0918978
|
(E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid
Show/Hide
|
C17H16O3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0396842
|
ethyl (E)-2-benzoyl-3-[1-(2-piperidin-1-ylethyl)indol-3-yl]prop-2-enoate
Show/Hide
|
C27H30N2O3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0435957
|
ethyl (E)-2-benzoyl-3-[1-(2-morpholin-4-ylethyl)indol-3-yl]prop-2-enoate
Show/Hide
|
C26H28N2O4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0438035
|
[(Z)-3-acetyloxyprop-1-enyl] 5-methylideneoctadecanoate
Show/Hide
|
C24H42O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0380712
|
2-(4-piperidin-1-ylphenyl)ethyl 5-chloro-3-ethyl-1H-indole-2-carboxylate
Show/Hide
|
C24H27ClN2O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0383426
|
N-[2-(4-aminophenyl)ethyl]-5-chloro-1H-indole-2-carboxamide
Show/Hide
|
C17H16ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0400643
|
5-chloro-N-[2-[4-(methylamino)phenyl]ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C18H18ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0417342
|
2-(4-nitrophenyl)ethyl 5-chloro-3-ethyl-1H-indole-2-carboxylate
Show/Hide
|
C19H17ClN2O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0435063
|
2-[4-(dimethylamino)phenyl]ethyl 5-chloro-3-ethyl-1H-indole-2-carboxylate
Show/Hide
|
C21H23ClN2O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0436061
|
3-acetyl-5-chloro-N-[2-(4-piperidin-1-ylphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C24H26ClN3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0045030
|
(6aR,10aR)-3-(1,1-dimethylbutyl)-6a,7,10,10a-tetrahydro-6,6,9-trimethyl-6Hdibenzo[b,d]pyran
Show/Hide
|
C22H32O
|
4
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki = 116.8 nM
|
|
|
| 3 |
Ki = 677 nM
|
|
|
| 4 |
Ki > 10000 nM
|
|
|
|
CP0846986
|
1-(5-(benzo[d][1,3]dioxol-5-yloxy)pentyl)urea
Show/Hide
|
C13H18N2O4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846987
|
2-ethyl-5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)penta-2,4-dienamido)acetate
Show/Hide
|
C17H19NO5
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846988
|
N-(5-(naphthalen-2-yloxy)pentyl)ethanesulfonamide
Show/Hide
|
C17H23NO3S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846989
|
N-(5-(naphthalen-1-yloxy)pentyl)ethanesulfonamide
Show/Hide
|
C17H23NO3S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846990
|
1-ethyl-3-(5-(naphthalen-2-yloxy)pentyl)urea
Show/Hide
|
C18H24N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0846991
|
1-(5-(benzo[d][1,3]dioxol-5-yloxy)pentyl)-3-ethylurea
Show/Hide
|
C15H22N2O4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0852446
|
2-ethyl-(6-(naphthalen-1-yloxy)hexanamido)acetate
Show/Hide
|
C20H25NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853976
|
1-ethyl-3-(5-(naphthalen-1-yloxy)pentyl)urea
Show/Hide
|
C18H24N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853977
|
2-ethyl-5-(naphthalen-2-yl)penta-2,4-dienamido)acetate
Show/Hide
|
C19H19NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853978
|
N-cyclopropyl-5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)penta-2,4-dienamide
Show/Hide
|
C16H17NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853979
|
N-(5-(benzo[d][1,3]dioxol-5-yloxy)pentyl)ethanesulfonamide
Show/Hide
|
C14H21NO5S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853980
|
5-(9H-fluoren-3-yl)-N-(2-hydroxyethyl)penta-2,4-dienamide
Show/Hide
|
C20H19NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0853981
|
2-ethyl-(6-(naphthalen-2-yloxy)hexanamido)acetate
Show/Hide
|
C20H25NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858225
|
N-cyclopropyl-6-(naphthalen-2-yloxy)hexanamide
Show/Hide
|
C19H23NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0858226
|
N-(2-hydroxyethyl)-6-(naphthalen-2-yloxy)hexanamide
Show/Hide
|
C18H23NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0860293
|
N-(2-hydroxyethyl)-6-(naphthalen-1-yloxy)hexanamide
Show/Hide
|
C18H23NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0860294
|
N-cyclopropyl-5-(9H-fluoren-3-yl)penta-2,4-dienamide
Show/Hide
|
C21H19NO
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0860296
|
2-ethyl-5-(9H-fluoren-3-yl)penta-2,4-dienamido)acetate
Show/Hide
|
C22H21NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0876217
|
N-(5-(naphthalen-2-ylthio)pentyl)ethanesulfonamide
Show/Hide
|
C17H23NO2S2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0876218
|
N-cyclopropyl-6-(naphthalen-1-yloxy)hexanamide
Show/Hide
|
C19H23NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0876219
|
N-(2-hydroxyethyl)-5-(naphthalen-2-yl)penta-2,4-dienamide
Show/Hide
|
C17H17NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0876220
|
1-(5-(naphthalen-1-yloxy)pentyl)urea
Show/Hide
|
C16H20N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0882216
|
N-cyclopropyl-5-(naphthalen-2-yl)penta-2,4-dienamide
Show/Hide
|
C18H17NO
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0882217
|
1-ethyl-3-(5-(naphthalen-2-ylthio)pentyl)urea
Show/Hide
|
C18H24N2OS
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0401037
|
(2-methylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C19H14N2O
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0401056
|
naphthalen-1-yl-(2-propylbenzimidazol-1-yl)methanone
Show/Hide
|
C21H18N2O
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0401058
|
(4-methoxyphenyl)-(2-methylbenzimidazol-1-yl)methanone
Show/Hide
|
C16H14N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0415439
|
(2-cyclohexylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C21H22N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0415487
|
(2-ethyl-1-benzothiophen-3-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C18H16O2S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0415513
|
(4-methoxyphenyl)-[2-(2-methylpropyl)benzimidazol-1-yl]methanone
Show/Hide
|
C19H20N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0419748
|
(4-methoxyphenyl)-[2-(4-methoxyphenyl)benzimidazol-1-yl]methanone
Show/Hide
|
C22H18N2O3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0420649
|
(2-cyclopentylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C23H20N2O
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0420650
|
(4-methoxyphenyl)-(2-propylbenzimidazol-1-yl)methanone
Show/Hide
|
C18H18N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0446587
|
(2-cyclobutylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C19H18N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0446591
|
(2-tert-butylbenzimidazol-1-yl)-naphthalen-1-ylmethanone
Show/Hide
|
C22H20N2O
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0446595
|
2‐(4‐methoxyphenyl)‐1‐[(4‐methoxyphenyl)methyl]‐ 1,3‐benzodiazole (B14)
Show/Hide
|
C22H20N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0446663
|
(2-butylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C19H20N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0447449
|
[2-(2-methylpropyl)benzimidazol-1-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C22H20N2O
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0451448
|
(2-tert-butylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C19H20N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0452044
|
(4-methoxyphenyl)-(2-propyl-1-benzothiophen-3-yl)methanone
Show/Hide
|
C19H18O2S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0454680
|
(4-methoxyphenyl)-(2-pentyl-1-benzothiophen-3-yl)methanone
Show/Hide
|
C21H22O2S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0454681
|
(4-methoxyphenyl)-(2-propan-2-ylbenzimidazol-1-yl)methanone
Show/Hide
|
C18H18N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0454682
|
naphthalen-1-yl-(2-propan-2-ylbenzimidazol-1-yl)methanone
Show/Hide
|
C21H18N2O
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0458139
|
1-benzothiophen-3-yl(naphthalen-1-yl)methanone
Show/Hide
|
C19H12OS
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0510719
|
(2-cyclopentylbenzimidazol-1-yl)-(4-methoxyphenyl)methanone
Show/Hide
|
C20H20N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0436129
|
17-heptyl-1-methyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C26H29NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0436130
|
17-heptyl-1-[(heptylamino)methyl]-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C33H44N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0436131
|
17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C18H13NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0436132
|
4-chloro-17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2(7),3,5,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H26ClNO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0436133
|
1-chloro-17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H26ClNO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0441077
|
1-(heptoxymethyl)-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C26H29NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0477157
|
1-bromo-17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H26BrNO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0477160
|
17-hexyl-1-methyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C25H27NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0477162
|
1-[(heptylamino)methyl]-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C26H30N2O2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0491999
|
17-hexyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C24H25NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0492000
|
17-octyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C26H29NO2
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0492001
|
1-(heptoxymethyl)-17-heptyl-17-azapentacyclo[6.6.5.02,7.09,14.015,19]nonadeca-2,4,6,9,11,13-hexaene-16,18-dione
Show/Hide
|
C33H43NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0134007
|
[2-(4-methoxyphenyl)-1-benzofuran-3-yl]-[4-(pyridin-2-ylmethylamino)phenyl]methanone
Show/Hide
|
C28H22N2O3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0134009
|
[4-(dibenzylamino)phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C36H29NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0176623
|
[4-[4-[(3-fluorophenoxy)methyl]triazol-1-yl]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C31H22FN3O4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0176689
|
[4-(benzylamino)phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C29H23NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0211297
|
[4-[bis[(4-fluorophenyl)methyl]amino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C36H27F2NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0222934
|
[4-[(3,5-difluorophenyl)methylamino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C29H21F2NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0262330
|
[4-[bis[(3,5-difluorophenyl)methyl]amino]phenyl]-[2-(4-methoxyphenyl)-1-benzofuran-3-yl]methanone
Show/Hide
|
C36H25F4NO3
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0327836
|
[2-(4-methoxyphenyl)-1-benzofuran-3-yl]-[4-[(4-methoxyphenyl)methylamino]phenyl]methanone
Show/Hide
|
C30H25NO4
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0422515
|
1-(4-chlorophenyl)-3-[(3R)-1-phenylpiperidin-3-yl]urea
Show/Hide
|
C18H20ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0422585
|
1-(4-chlorophenyl)-3-(5-phenylpyridin-3-yl)urea
Show/Hide
|
C18H14ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0422586
|
1-(4-chlorophenyl)-3-[(1S,2R)-2-phenylcyclopropyl]urea
Show/Hide
|
C16H15ClN2O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0422620
|
1-(4-chlorophenyl)-3-(4-phenylpyridin-2-yl)urea
Show/Hide
|
C18H14ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0434078
|
1-(4-chlorophenyl)-3-(6-phenylpyridin-2-yl)urea
Show/Hide
|
C18H14ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0525584
|
1-(4-chlorophenyl)-3-[(1S,2S)-2-phenylcyclopropyl]urea
Show/Hide
|
C16H15ClN2O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0527980
|
1-(4-chlorophenyl)-3-[2-methoxy-5-(6-pyrrolidin-1-ylpyridin-2-yl)phenyl]urea
Show/Hide
|
C23H23ClN4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0542734
|
1-(4-chlorophenyl)-3-[2-(3,4-dimethoxyphenyl)ethyl]urea
Show/Hide
|
C17H19ClN2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0569264
|
1-[2-(4-tert-butylphenyl)ethyl]-3-(4-chlorophenyl)urea
Show/Hide
|
C19H23ClN2O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0573319
|
1-(4-chlorophenyl)-3-[2-[3-(trifluoromethoxy)phenyl]ethyl]urea
Show/Hide
|
C16H14ClF3N2O2
|
1
|
| 1 |
IC50 = 10715.19 nM
|
|
|
|
CP0489596
|
US9422235, 29
Show/Hide
|
C20H19F3N2O5S
|
2
|
| 1 |
IC50 = 11380 nM
|
|
|
| 2 |
Ki = 5045 nM
|
|
|
|
CP0419648
|
US9422235, 34
Show/Hide
|
C21H27F3N2O6S
|
2
|
| 1 |
IC50 = 12000 nM
|
|
|
| 2 |
Ki = 6000 nM
|
|
|
|
CP0445204
|
US9422235, 33
Show/Hide
|
C23H21F3N2O4S
|
2
|
| 1 |
IC50 = 12000 nM
|
|
|
| 2 |
Ki = 6000 nM
|
|
|
|
CP0507896
|
US9422235, 35
Show/Hide
|
C19H19Cl2F3N2O3S
|
2
|
| 1 |
IC50 = 13810 nM
|
|
|
| 2 |
Ki = 5841 nM
|
|
|
|
CP0451939
|
US9422235, 1
Show/Hide
|
C19H20Cl2F3N3O3S
|
2
|
| 1 |
IC50 = 34090 nM
|
|
|
| 2 |
Ki = 21020 nM
|
|
|
|
CP0372969
|
1-(4-chlorophenyl)-3-methyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C20H22ClN5O
|
2
|
| 1 |
IC50 > 5000 nM
|
|
|
| 2 |
Ki > 2820 nM
|
|
|
|
CP0384279
|
4-cyano-1-phenyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H20N6O
|
2
|
| 1 |
IC50 > 5000 nM
|
|
|
| 2 |
Ki > 2820 nM
|
|
|
|
CP0431801
|
1-phenyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C19H21N5O
|
2
|
| 1 |
IC50 > 5000 nM
|
|
|
| 2 |
Ki > 2820 nM
|
|
|
|
CP0458171
|
4-methyl-1-phenyl-N-(piperidin-1-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C20H23N5O
|
2
|
| 1 |
IC50 > 5000 nM
|
|
|
| 2 |
Ki > 2820 nM
|
|
|
|
CP0501941
|
1-(2,4-difluorophenyl)-4-methyl-N-(morpholin-4-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C19H19F2N5O2
|
2
|
| 1 |
IC50 > 5000 nM
|
|
|
| 2 |
Ki > 2820 nM
|
|
|
|
CP0415524
|
5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H23Cl3N4O
|
2
|
| 1 |
Kd = 12.02 nM
|
|
|
| 2 |
Ki = 16.1 nM
|
|
|
|
CP0418515
|
1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1Hpyrazole-3-carboxamide
Show/Hide
|
C22H20Cl4N4O
|
2
|
| 1 |
Kd = 19.05 nM
|
|
|
| 2 |
Ki = 34.2 nM
|
|
|
|
CP0501831
|
9-Chloro-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-4,5,6,7-tetrahydro-1H-benzo[7,8]cycloocta[1,2-c]pyrazole-3-carboxamide
Show/Hide
|
C25H25Cl3N4O
|
2
|
| 1 |
Kd = 40.74 nM
|
|
|
| 2 |
Ki = 40.9 nM
|
|
|
|
CP0419054
|
5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H22Cl4N4O
|
2
|
| 1 |
Kd = 77.62 nM
|
|
|
| 2 |
Ki = 251 nM
|
|
|
|
CP0465702
|
5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide
Show/Hide
|
C24H25Cl3N4O
|
2
|
| 1 |
Kd = 93.33 nM
|
|
|
| 2 |
Ki = 194 nM
|
|
|
|
CP0373943
|
5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H19Cl5N4O
|
2
|
| 1 |
Kd = 269.15 nM
|
|
|
| 2 |
Ki = 261 nM
|
|
|
|
CP0434132
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]oxane-4-carboxamide
Show/Hide
|
C25H25Cl2N3O3
|
1
|
| 1 |
Ki = 0.09 nM
|
|
|
|
CP0382775
|
N-(3-pentyl-1,3-benzothiazol-2-ylidene)adamantane-1-carboxamide
Show/Hide
|
C23H30N2OS
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0382825
|
N-(3-pentyl-1,3-benzothiazol-2-ylidene)naphthalene-1-carboxamide
Show/Hide
|
C23H22N2OS
|
1
|
| 1 |
Ki = 0.11 nM
|
|
|
|
CP0441039
|
1-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-3-ethylurea
Show/Hide
|
C22H22Cl2N4O2
|
1
|
| 1 |
Ki = 0.12 nM
|
|
|
|
CP0509763
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-1-cyanocyclopropane-1-carboxamide
Show/Hide
|
C24H20Cl2N4O2
|
1
|
| 1 |
Ki = 0.13 nM
|
|
|
|
CP0432518
|
N-[(8R)-2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-2-methylpropanamide
Show/Hide
|
C23H23Cl2N3O2
|
1
|
| 1 |
Ki = 0.14 nM
|
|
|
|
CP0895933
|
(R,S)-N-[2-(2-Chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydro-2H-oxepino[3,2-c]pyrazol-8-yl]-2-methylpropanamide
Show/Hide
|
C23H23Cl2N3O2
|
1
|
| 1 |
Ki = 0.16 nM
|
|
|
|
CP0124848
|
(6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-6,6-dimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C25H38O3
|
2
|
| 1 |
Ki = 0.18 nM
|
|
|
| 2 |
Ki = 1.5 nM
|
|
|
|
CP0035672
|
dibenzothiazepine, 12h
Show/Hide
|
C24H20ClFN2OS
|
1
|
| 1 |
Ki = 0.1995 nM
|
|
|
|
CP0035756
|
dibenzothiazepine, 12e
Show/Hide
|
C24H21ClN2OS
|
1
|
| 1 |
Ki = 0.1995 nM
|
|
|
|
CP0442489
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2-difluoropropyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
|
C20H14Cl2F2N4O
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0409089
|
methyl N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]carbamate
Show/Hide
|
C21H19Cl2N3O3
|
1
|
| 1 |
Ki = 0.25 nM
|
|
|
|
CP0425911
|
propan-2-yl N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]carbamate
Show/Hide
|
C23H23Cl2N3O3
|
1
|
| 1 |
Ki = 0.26 nM
|
|
|
|
CP0508356
|
3-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-1-(2-methoxyethyl)-1-methylurea
Show/Hide
|
C27H29Cl2N7O2
|
1
|
| 1 |
Ki = 0.26 nM
|
|
|
|
CP0457027
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
|
C19H11Cl2F3N4O
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0468462
|
dibenzothiazepine, 12b
Show/Hide
|
C26H24ClN3OS
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0416545
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-cyclopentylethanone
Show/Hide
|
C28H28Cl2N6O
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0462175
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]propanamide
Show/Hide
|
C22H21Cl2N3O2
|
1
|
| 1 |
Ki = 0.41 nM
|
|
|
|
CP0409567
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-2-methylsulfonylacetamide
Show/Hide
|
C22H21Cl2N3O4S
|
1
|
| 1 |
Ki = 0.54 nM
|
|
|
|
CP0467377
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-1,2-oxazole-5-carboxamide
Show/Hide
|
C23H18Cl2N4O3
|
1
|
| 1 |
Ki = 0.55 nM
|
|
|
|
CP0489872
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-2-ethoxyacetamide
Show/Hide
|
C23H23Cl2N3O3
|
1
|
| 1 |
Ki = 0.56 nM
|
|
|
|
CP0475994
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]cyclohexanecarboxamide
Show/Hide
|
C26H27Cl2N3O2
|
1
|
| 1 |
Ki = 0.59 nM
|
|
|
|
CP0136518
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-5-methyl-6-(2,2,2-trifluoroethyl)pyrazolo[4,3-d]pyrimidin-7-one
Show/Hide
|
C20H13Cl2F3N4O
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0435518
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2-difluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
|
C19H12Cl2F2N4O
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0552881
|
6-(4-butylsulfonylpiperazin-1-yl)-8-(2-chlorophenyl)-9-(4-chlorophenyl)purine
Show/Hide
|
C25H26Cl2N6O2S
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0295447
|
1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-4-(ethylamino)piperidine-4-carboxamide
Show/Hide
|
C25H25Cl2N7O
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0439886
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]acetamide
Show/Hide
|
C21H19Cl2N3O2
|
1
|
| 1 |
Ki = 0.75 nM
|
|
|
|
CP0372226
|
dibenzothiazepine, 12c
Show/Hide
|
C26H22ClF2N3OS
|
1
|
| 1 |
Ki = 0.7943 nM
|
|
|
|
CP0455587
|
3-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-1-methyl-1-(2-methylpropyl)urea
Show/Hide
|
C28H31Cl2N7O
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0420623
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(cyclohexylmethyl)urea
Show/Hide
|
C30H33Cl2N7O
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0447836
|
3-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-1-methyl-1-propylurea
Show/Hide
|
C27H29Cl2N7O
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0401262
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[3,4-c]pyridin-7(6H)-one
Show/Hide
|
C20H12Cl2F3N3O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0401263
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-5-ethyl-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
|
C21H15Cl2F3N4O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0859347
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-1-(2,2,2-trifluoroethyl)-4,9-dihydro-1H-purin-6(5H)-one
Show/Hide
|
C19H13Cl2F3N4O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0037081
|
PF-514273
Show/Hide
|
C21H17Cl2F2N3O2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0443610
|
1-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]pyrrolidin-2-one
Show/Hide
|
C23H21Cl2N3O2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0466292
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2,2,2-trifluoroethanone
Show/Hide
|
C23H17Cl2F3N6O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0462464
|
N-(3-pentyl-1,3-benzothiazol-2-ylidene)-3-(trifluoromethyl)benzamide
Show/Hide
|
C20H19F3N2OS
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0287055
|
(6aR,10aR)-6,6,9-trimethyl-3-(2-(thiophen-2-yl)propan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C23H28O2S
|
1
|
| 1 |
Ki = 1.08 nM
|
|
|
|
CP0431692
|
3-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-1-propyl-1-(2,2,2-trifluoroethyl)urea
Show/Hide
|
C28H28Cl2F3N7O
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0420376
|
N-cyclopropyl-8-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]octanamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0492172
|
(4-bromonaphthalen-1-yl)-(1-pentylindol-3-yl)methanone
Show/Hide
|
C24H22BrNO
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0391306
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-[4-(3,3,3-trifluoropropylsulfonyl)piperazin-1-yl]purine
Show/Hide
|
C24H21Cl2F3N6O2S
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0548533
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-propylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C24H24Cl2N6O2S
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0432073
|
N-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]piperidine-1-carboxamide
Show/Hide
|
C28H29Cl2N7O
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0510023
|
dibenzothiazepine, 12j
Show/Hide
|
C22H19ClN2OS2
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0459284
|
N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-2-methoxyacetamide
Show/Hide
|
C22H21Cl2N3O3
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0389941
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-propan-2-ylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C24H24Cl2N6O2S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0416547
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-cyclohexylpiperazine-1-carboxamide
Show/Hide
|
C28H29Cl2N7O
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0493585
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-cyclohexylurea
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C29H31Cl2N7O
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1
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| 1 |
Ki = 1.4 nM
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CP0485554
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dibenzothiazepine, 12k
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C24H23N3OS
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1
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| 1 |
Ki = 1.585 nM
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CP0257214
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(6aR,10aR)-3-(2-(3-bromophenyl)propan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C25H29BrO2
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1
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| 1 |
Ki = 1.59 nM
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CP0420951
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N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-1,2-oxazole-3-carboxamide
Show/Hide
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C23H18Cl2N4O3
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1
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| 1 |
Ki = 1.6 nM
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CP0443609
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N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-1,2,5-oxadiazole-3-carboxamide
Show/Hide
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C22H17Cl2N5O3
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1
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| 1 |
Ki = 1.7 nM
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CP0389942
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8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-[4-(cyclohexylmethylsulfonyl)piperazin-1-yl]purine
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C28H30Cl2N6O2S
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1
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| 1 |
Ki = 1.7 nM
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CP0157114
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(6aR,10aR)-6,6,9-trimethyl-3-(2-(4-propylphenyl)propan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C28H36O2
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1
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| 1 |
Ki = 1.77 nM
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CP0061669
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5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazole-3-carboxylic acid cyclohexylamide
Show/Hide
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C23H22Cl3N3O
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3
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| 1 |
Ki = 1.8 nM
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| 2 |
Ki = 3.7 nM
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| 3 |
Ki = 5 nM
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CP0371733
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2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(3,3,3-trifluoropropyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
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C20H13Cl2F3N4O
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1
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| 1 |
Ki = 1.8 nM
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CP0157108
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(6aR,10aR)-3-(2-(4-ethylphenyl)propan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C27H34O2
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1
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| 1 |
Ki = 1.85 nM
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CP0529740
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N-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-methylphenyl)imidazole-4-carboxamide
Show/Hide
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C23H23Cl2N3O
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1
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| 1 |
Ki = 1.9 nM
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CP0371734
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2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-propyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
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C20H16Cl2N4O
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1
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| 1 |
Ki = 2 nM
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CP0511273
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1-(2,4-Dichlorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(pyrrolidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H19Cl2N5O2
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1
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| 1 |
Ki = 2 nM
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CP0389945
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1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-3,3-dimethylbutan-1-one
Show/Hide
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C27H28Cl2N6O
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1
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| 1 |
Ki = 2 nM
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CP0466293
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[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-(thian-4-yl)methanone
Show/Hide
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C27H26Cl2N6OS
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1
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| 1 |
Ki = 2 nM
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CP0517588
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8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-[4-(2-methylpropylsulfonyl)piperazin-1-yl]purine
Show/Hide
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C25H26Cl2N6O2S
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1
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| 1 |
Ki = 2 nM
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CP0152977
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5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1H-pyrazole-3-carboxylic acid ((1S,2S,4R)-1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide
Show/Hide
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C29H34ClN3O
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5
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| 1 |
Ki = 2 nM
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| 2 |
Ki = 116 nM
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| 3 |
Ki = 116.79 nM
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| 4 |
Ki = 121.2 nM
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| 5 |
Ki = 5628 nM
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CP0502931
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N-(1-adamantyl)-1-pentyl-6-phenylindole-3-carboxamide
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C30H36N2O
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1
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| 1 |
Ki = 2.03 nM
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CP0417664
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2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C25H24Cl3N3O
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1
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| 1 |
Ki = 2.2 nM
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CP0384969
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-1H-imidazole-4-carboxamide
Show/Hide
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C22H21Cl2N3O
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1
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| 1 |
Ki = 2.2 nM
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CP0289084
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8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(piperidin-1-yl)-9H-purine
Show/Hide
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C22H19Cl2N5
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1
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| 1 |
Ki = 2.3 nM
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CP0102214
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1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H21Cl2IN4O
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1
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| 1 |
Ki = 2.3 nM
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CP0417230
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N-[11-(11-aminoundecylamino)undecyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C39H58Cl3N5O
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2
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| 1 |
Ki = 2.3 nM
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| 2 |
Ki = 4.56 nM
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CP0496088
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N-cyclohexyl-1-(2,4-dichlorophenyl)-4-methyl-5-(4,5,6,7-tetrahydroisoindol-2-yl)pyrazole-3-carboxamide
Show/Hide
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C25H28Cl2N4O
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1
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| 1 |
Ki = 2.3 nM
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CP0488465
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(4-chloronaphthalen-1-yl)-(1-pentylindol-3-yl)methanone
Show/Hide
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C24H22ClNO
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1
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| 1 |
Ki = 2.3 nM
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CP0447824
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[(2-fluorophenyl)methyl]urea
Show/Hide
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C30H26Cl2FN7O
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1
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| 1 |
Ki = 2.4 nM
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CP0410964
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4-oxo-1-pentyl-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C31H38N2O2S
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1
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| 1 |
Ki = 2.45 nM
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CP0524808
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(4-iodonaphthalen-1-yl)-(1-pentylindol-3-yl)methanone
Show/Hide
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C24H22INO
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1
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| 1 |
Ki = 2.5 nM
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CP0035757
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dibenzothiazepine, 12a
Show/Hide
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C25H29N3OS
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1
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| 1 |
Ki = 2.512 nM
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CP0286060
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(6aR,10aR)-6,6,9-trimethyl-3-(2-m-tolylpropan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C26H32O2
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1
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| 1 |
Ki = 2.53 nM
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CP0337138
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3-(2-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-3-yl)propan-2-yl)benzonitrile
Show/Hide
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C26H29NO2
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1
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| 1 |
Ki = 2.72 nM
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CP0471359
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11-[3-(5-azido-1,1-dimethylpentyl)phenoxy]undeca-5,8-dienoic acid [R-(1-hydroxypropan-2-yl)]-amide
Show/Hide
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C27H42N4O3
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1
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| 1 |
Ki = 2.74 nM
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CP0109122
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8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine
Show/Hide
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C22H20Cl2N6
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1
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| 1 |
Ki = 2.8 nM
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CP0432853
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1-(2-chlorophenyl)-2-(4-chlorophenyl)-5-cyclohexyl-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C26H26Cl2N2O
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1
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| 1 |
Ki = 2.8 nM
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CP0333956
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(6aR,10aR)-3-(2-(3-chlorophenyl)propan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C25H29ClO2
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1
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| 1 |
Ki = 2.8 nM
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CP0405615
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6-bromo-4-oxo-1-pentyl-N-((1R,2R,4S)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
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C25H33BrN2O2
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1
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| 1 |
Ki = 2.8 nM
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CP0111432
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quinolin-8-yl 4-methyl-3-piperidin-1-ylsulfonylbenzoate
Show/Hide
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C22H22N2O4S
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1
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| 1 |
Ki = 3 nM
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CP0392052
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2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2-fluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
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C19H13Cl2FN4O
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1
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| 1 |
Ki = 3 nM
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CP0392393
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N-cyclohexyl-1-(2,4-dichlorophenyl)-4-ethyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C22H24Cl2N4O
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1
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| 1 |
Ki = 3 nM
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CP0077457
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N-[1-(cyclohexylmethyl)-2-[(5-ethoxypyridin-2-yl)methyl]benzimidazol-5-yl]-N-methylthiophene-2-sulfonamide
Show/Hide
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C27H32N4O3S2
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1
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| 1 |
Ki = 3 nM
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CP0389943
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cyclobutylmethyl 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazine-1-carboxylate
Show/Hide
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C27H26Cl2N6O2
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1
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| 1 |
Ki = 3 nM
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CP0396584
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8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-ethylsulfonylpiperazin-1-yl)purine
Show/Hide
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C23H22Cl2N6O2S
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1
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| 1 |
Ki = 3 nM
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CP0411062
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8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-[4-(oxan-4-ylmethylsulfonyl)piperazin-1-yl]purine
Show/Hide
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C27H28Cl2N6O3S
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1
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| 1 |
Ki = 3 nM
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CP0416055
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1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-phenylpropan-1-one
Show/Hide
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C30H26Cl2N6O
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1
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| 1 |
Ki = 3 nM
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CP0466290
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cyclobutyl 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazine-1-carboxylate
Show/Hide
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C26H24Cl2N6O2
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1
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| 1 |
Ki = 3 nM
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CP0485555
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[(4-fluorophenyl)methyl]urea
Show/Hide
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C30H26Cl2FN7O
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1
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| 1 |
Ki = 3 nM
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CP0540524
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-cyclopentylurea
Show/Hide
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C28H29Cl2N7O
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1
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| 1 |
Ki = 3 nM
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CP0272343
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(6aR,10aR)-6,6,9-trimethyl-3-(2-p-tolylpropan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C26H32O2
|
1
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| 1 |
Ki = 3.13 nM
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CP0170798
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(S)-3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide
Show/Hide
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C23H20Cl2N4O2S
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4
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| 1 |
Ki = 3.162 nM
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| 2 |
Ki = 4.1 nM
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| 3 |
Ki = 7.8 nM
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| 4 |
Ki = 8 nM
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CP0376648
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(S)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C23H26Cl2N4O
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1
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| 1 |
Ki = 3.4 nM
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CP0501759
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1-(2-chlorophenyl)-2-(4-chlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C25H25Cl2N3O
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1
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| 1 |
Ki = 3.5 nM
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CP0469875
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N-cyclopropyl-11-(3-methoxy-5-pentylphenoxy)undecanamide
Show/Hide
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C26H43NO3
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1
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| 1 |
Ki = 3.5 nM
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CP0500978
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1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
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C24H25BrClN3O2
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1
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| 1 |
Ki = 3.7 nM
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CP0113406
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1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid cyclohexylamide
Show/Hide
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C22H20Cl3N3O
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1
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| 1 |
Ki = 3.9 nM
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CP0449529
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2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-ethyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
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C19H14Cl2N4O
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1
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| 1 |
Ki = 4 nM
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CP0435697
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7-fluoro-4-oxo-1-pentyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C25H33FN2O2
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1
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| 1 |
Ki = 4 nM
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CP0489576
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(2-fluorophenyl)urea
Show/Hide
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C29H24Cl2FN7O
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1
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| 1 |
Ki = 4 nM
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CP0547865
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-(2-fluorophenyl)urea
Show/Hide
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C30H26Cl2FN7O
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1
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| 1 |
Ki = 4 nM
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CP0532378
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(4-(trifluoromethyl)phenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C27H25Cl2F3N2O
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1
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| 1 |
Ki = 4.1 nM
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CP0400113
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5-(4-chlorophenyl)-N-[7-[7-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]heptylamino]heptyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C48H51Cl6N7O2
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2
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| 1 |
Ki = 4.41 nM
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| 2 |
Ki = 12.3 nM
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CP0453395
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N-[2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-N,2-dimethylpropanamide
Show/Hide
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C24H25Cl2N3O2
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1
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| 1 |
Ki = 4.5 nM
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CP0384966
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2-(2-chlorophenyl)-N-cyclohexyl-1-p-tolyl-1H-imidazole-4-carboxamide
Show/Hide
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C23H24ClN3O
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1
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| 1 |
Ki = 4.6 nM
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CP0383807
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1-(2-bromophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H22BrN5O2
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1
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| 1 |
Ki = 4.7 nM
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CP0500721
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1-butyl-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C30H36N2O2S
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1
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| 1 |
Ki = 4.7 nM
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CP0529739
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N-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-methoxyphenyl)imidazole-4-carboxamide
Show/Hide
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C23H23Cl2N3O2
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1
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| 1 |
Ki = 4.9 nM
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CP0379561
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5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzofuran-2-carboxamide
Show/Hide
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C27H32N2O4S
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1
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| 1 |
Ki = 5 nM
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CP0434259
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
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C24H25Cl2N3O2
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1
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| 1 |
Ki = 5 nM
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CP0441837
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6-benzyl-2-(2-chlorophenyl)-3-(4-chlorophenyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
|
C24H16Cl2N4O
|
1
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| 1 |
Ki = 5 nM
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CP0389946
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4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(2,4-difluorophenyl)piperazine-1-carboxamide
Show/Hide
|
C28H21Cl2F2N7O
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1
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| 1 |
Ki = 5 nM
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CP0391003
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tert-butyl 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazine-1-carboxylate
Show/Hide
|
C26H26Cl2N6O2
|
1
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| 1 |
Ki = 5 nM
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CP0391005
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4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(3,4-difluorophenyl)piperazine-1-carboxamide
Show/Hide
|
C28H21Cl2F2N7O
|
1
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| 1 |
Ki = 5 nM
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CP0416507
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4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-cyclopentylpiperazine-1-carboxamide
Show/Hide
|
C27H27Cl2N7O
|
1
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| 1 |
Ki = 5 nM
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CP0416595
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-cyclopropylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C24H22Cl2N6O2S
|
1
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| 1 |
Ki = 5 nM
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CP0466294
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[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-(2,3-dihydro-1,4-benzodioxin-3-yl)methanone
Show/Hide
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C30H24Cl2N6O3
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1
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| 1 |
Ki = 5 nM
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CP0484113
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(4,4-difluoro-1-methylcyclohexyl)urea
Show/Hide
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C30H31Cl2F2N7O
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1
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| 1 |
Ki = 5 nM
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CP0286058
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(6aR,10aR)-3-(2-(4-bromophenyl)propan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C25H29BrO2
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1
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| 1 |
Ki = 5.03 nM
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CP0517368
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N-[(8S)-2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydrooxepino[3,2-c]pyrazol-8-yl]-2-methylpropanamide
Show/Hide
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C23H23Cl2N3O2
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1
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| 1 |
Ki = 5.1 nM
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CP0339943
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9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine
Show/Hide
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C22H19Cl3N6
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1
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| 1 |
Ki = 5.2 nM
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CP0432931
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N-cyclopropyl-11-(3-hydroxy-4-pentylphenoxy)undecanamide
Show/Hide
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C25H41NO3
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1
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| 1 |
Ki = 5.2 nM
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CP0427591
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11-(3-hydroxy-5-pentylphenoxy)undecanoic acid cyclopropylamide
Show/Hide
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C25H41NO3
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1
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| 1 |
Ki = 5.2 nM
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CP0253788
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(6aR,10aR)-3-(2-(3-fluorophenyl)propan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C25H29FO2
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1
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| 1 |
Ki = 5.26 nM
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CP0072767
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(5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2-chloro-ethyl)-amide
Show/Hide
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C22H36ClNO
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1
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| 1 |
Ki = 5.3 nM
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CP0393334
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N-(1-adamantyl)-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
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C31H36N2O2S
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1
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| 1 |
Ki = 5.3 nM
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CP0474423
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N-[9-(9-aminononylamino)nonyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C35H50Cl3N5O
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2
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| 1 |
Ki = 5.44 nM
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| 2 |
Ki = 14 nM
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CP0505310
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5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(3,4-dimethoxyphenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C28H30Cl2N2O3
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1
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| 1 |
Ki = 5.5 nM
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CP0471358
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11-[3-(5-cyano-1,1-dimethylpentyl)phenoxy]-undeca-5,8-dienoic acid [R-(1-hydroxypropan-2-yl)]-amide
Show/Hide
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C27H40N2O3
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1
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| 1 |
Ki = 5.51 nM
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CP0375653
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N-[11-[11-aminoundecyl(methyl)amino]undecyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C40H60Cl3N5O
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2
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| 1 |
Ki = 5.51 nM
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| 2 |
Ki = 14.7 nM
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CP0376647
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N-(1-adamantyl)-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C27H30Cl2N4O
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1
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| 1 |
Ki = 5.6 nM
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CP0390569
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N-cycloheptyl-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C22H24Cl2N4O
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1
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| 1 |
Ki = 5.6 nM
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CP0440242
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N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-dichloropyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C21H20Cl4N4O
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1
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| 1 |
Ki = 5.6 nM
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CP0394622
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-propyl-1H-imidazole-4-carboxamide
Show/Hide
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C25H27Cl2N3O2
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1
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| 1 |
Ki = 5.7 nM
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CP0526835
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N-cyclopropyl-11-(3-pentylphenoxy)undecanamide
Show/Hide
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C25H41NO2
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1
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| 1 |
Ki = 5.9 nM
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CP0428707
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5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(4-fluorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C26H25Cl2FN2O
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1
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| 1 |
Ki = 6 nM
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CP0371732
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2-(2-chlorophenyl)-3-(4-chlorophenyl)-5-isopropyl-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
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C22H17Cl2F3N4O
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1
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| 1 |
Ki = 6 nM
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CP0416548
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4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-pyridin-2-ylpiperazine-1-carboxamide
Show/Hide
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C27H22Cl2N8O
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1
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| 1 |
Ki = 6 nM
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CP0466295
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4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(2-fluorophenyl)piperazine-1-carboxamide
Show/Hide
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C28H22Cl2FN7O
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1
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| 1 |
Ki = 6 nM
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CP0547412
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4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-phenylpiperazine-1-carboxamide
Show/Hide
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C28H23Cl2N7O
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1
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| 1 |
Ki = 6 nM
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CP0552882
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1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]pentan-1-one
Show/Hide
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C26H26Cl2N6O
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1
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| 1 |
Ki = 6 nM
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CP0431691
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-(2,4-difluorophenyl)urea
Show/Hide
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C30H25Cl2F2N7O
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1
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| 1 |
Ki = 6 nM
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CP0291135
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9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(piperidin-1-yl)-9H-purine
Show/Hide
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C22H18Cl3N5
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1
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| 1 |
Ki = 6.1 nM
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CP0386407
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N-(1-adamantyl)-7-(benzenesulfonyl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C31H36N2O4S
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1
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| 1 |
Ki = 6.1 nM
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CP0379530
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N-[9-[9-aminononyl(methyl)amino]nonyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C36H52Cl3N5O
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2
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| 1 |
Ki = 6.12 nM
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| 2 |
Ki = 10 nM
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CP0435620
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide
Show/Hide
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C25H19Cl2N3O2
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1
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| 1 |
Ki = 6.3 nM
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CP0553719
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[1-(trifluoromethyl)cyclopentyl]urea
Show/Hide
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C29H28Cl2F3N7O
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1
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| 1 |
Ki = 6.3 nM
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CP0379515
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5-(4-chlorophenyl)-N-[5-[5-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]pentyl-methylamino]pentyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C45H45Cl6N7O2
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2
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| 1 |
Ki = 6.35 nM
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| 2 |
Ki = 38.7 nM
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CP0395392
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N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-ethylpyrazole-3-carboxamide
Show/Hide
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C24H28Cl2N4O
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1
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| 1 |
Ki = 6.7 nM
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CP0437446
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-methyl-1H-imidazole-4-carboxamide
Show/Hide
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C23H23Cl2N3O2
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1
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| 1 |
Ki = 6.9 nM
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CP0420625
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-phenylurea
Show/Hide
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C29H25Cl2N7O
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1
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| 1 |
Ki = 7 nM
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CP0341653
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9-(4-chlorophenyl)-N-cyclohexyl-8-(2,4-dichlorophenyl)-9H-purin-6-amine
Show/Hide
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C23H20Cl3N5
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1
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| 1 |
Ki = 7.1 nM
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CP0384968
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1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-dimethylphenyl)-1H-imidazole-4-carboxamide
Show/Hide
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C24H26ClN3O
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1
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| 1 |
Ki = 7.2 nM
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CP0488128
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(4-fluoronaphthalen-1-yl)-(1-pentylindol-3-yl)methanone
Show/Hide
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C24H22FNO
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1
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| 1 |
Ki = 7.2 nM
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CP0379905
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8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]-N-prop-2-enyloctanamide
Show/Hide
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C26H43NO3
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1
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| 1 |
Ki = 7.22 nM
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CP0090273
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9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-9H-purin-6-amine
Show/Hide
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C22H19Cl3N6
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1
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| 1 |
Ki = 7.4 nM
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CP0465171
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1-(2-chlorophenyl)-5-cyclohexyl-2-(4-methoxyphenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C27H29ClN2O2
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1
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| 1 |
Ki = 7.5 nM
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CP0465176
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2-(4-chlorophenyl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C26H25Cl3N2O
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1
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| 1 |
Ki = 7.5 nM
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CP0548828
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8-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]-N-prop-2-enyloctanamide
Show/Hide
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C27H45NO3
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1
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| 1 |
Ki = 7.6 nM
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CP0395391
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5-(2-chloropyrrol-1-yl)-N-cyclohexyl-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C21H21Cl3N4O
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1
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| 1 |
Ki = 7.7 nM
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CP0208317
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5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide
Show/Hide
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C21H19Cl3N4O
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1
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| 1 |
Ki = 7.8 nM
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CP0501073
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5-cyclohexyl-1-(2,4-dichlorophenyl)-2-(4-methoxyphenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C27H28Cl2N2O2
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1
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| 1 |
Ki = 7.9 nM
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CP0441836
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2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[3,4-d]pyridazin-7(6H)-one
Show/Hide
|
C19H11Cl2F3N4O
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1
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| 1 |
Ki = 8 nM
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CP0416054
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1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-(oxolan-3-yl)ethanone
Show/Hide
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C27H26Cl2N6O2
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1
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| 1 |
Ki = 8 nM
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CP0406539
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N-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-fluorophenyl)imidazole-4-carboxamide
Show/Hide
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C22H20Cl2FN3O
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1
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| 1 |
Ki = 8.2 nM
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CP0416563
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ethyl 4-[[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]methyl]benzoate
Show/Hide
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C27H22Cl3N3O3
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1
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| 1 |
Ki = 8.2 nM
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CP0378453
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11-[3-(1,1-dimethylheptyl)phenoxy]undeca-5,8-dienoic acid [R(1-hydroxypropan-2-yl)]-amide
Show/Hide
|
C29H47NO3
|
1
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| 1 |
Ki = 8.55 nM
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CP0476372
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5-(2-chloropyrrol-1-yl)-N-cyclohexyl-1-(3,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C21H21Cl3N4O
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1
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| 1 |
Ki = 8.6 nM
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CP0381993
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5-bromo-N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
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C20H22BrFN2O2
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1
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| 1 |
Ki = 8.8 nM
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CP0372353
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11-[3-(5-bromo-1,1-dimethylpentyl)phenoxy]-undeca-5,8-dienoic acid [R-(1-hydroxypropan-2-yl)]-amide
Show/Hide
|
C27H42BrNO3
|
1
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| 1 |
Ki = 8.87 nM
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CP0513858
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(4-chloronaphthalen-1-yl)-(2-methyl-1-pentylindol-3-yl)methanone
Show/Hide
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C25H24ClNO
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1
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| 1 |
Ki = 8.9 nM
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CP0374422
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2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methoxyphenyl)-1H-imidazole-4-carboxamide
Show/Hide
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C23H24ClN3O2
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1
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| 1 |
Ki = 9 nM
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CP0387786
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(2-cyclopentyl-5-prop-2-enyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
Show/Hide
|
C26H35N3O
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1
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| 1 |
Ki = 9 nM
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CP0482402
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1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(cyclohexylsulfamoyl)-4-methylpiperidin-4-amine
Show/Hide
|
C29H33Cl2N7O2S
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1
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| 1 |
Ki = 9 nM
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CP0671680
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SID50107233
Show/Hide
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C28H30N2O6S
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1
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| 1 |
Ki = 9.2 nM
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CP0257213
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3-[1-(4-Cyano-phenyl)-1-methyl-ethyl]-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C26H29NO2
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1
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| 1 |
Ki = 9.25 nM
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CP0440706
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N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(2,5-dichloropyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C21H20Cl4N4O
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1
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| 1 |
Ki = 9.4 nM
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CP0454191
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N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C23H24FN3O2
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1
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| 1 |
Ki = 9.6 nM
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CP0420187
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(4-vinylphenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C28H28Cl2N2O
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1
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| 1 |
Ki = 9.8 nM
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CP0465174
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-p-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C27H28Cl2N2O
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1
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| 1 |
Ki = 10 nM
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CP0493058
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5-butyl-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C26H29Cl2N3O2
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1
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| 1 |
Ki = 10 nM
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CP0418900
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1,3-dihydroxypropan-2-yl 11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecanoate
Show/Hide
|
C29H50O6
|
1
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| 1 |
Ki = 10 nM
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CP0433967
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1-(2,4-Dichlorophenyl)-4-cyano-5-(4-(fluoromethoxy)phenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H20Cl2FN5O2
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1
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| 1 |
Ki = 10.3 nM
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CP0037555
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(5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-tetraenamide
Show/Hide
|
C22H37NO2
|
3
|
| 1 |
Ki = 11 nM
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| 2 |
Ki = 70 nM
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| 3 |
Ki = 72 nM
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CP0486888
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4-cyano-1-(2,4-dichlorophenyl)-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H21Cl2N5O2
|
1
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| 1 |
Ki = 11 nM
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CP0139483
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(6aR,10aR)-3-(2-(3,5-dimethylphenyl)propan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C27H34O2
|
1
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| 1 |
Ki = 11 nM
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CP0393333
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4-oxo-7-phenylsulfanyl-1-propyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C29H34N2O2S
|
1
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| 1 |
Ki = 11 nM
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CP0389944
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-ethoxyethanone
Show/Hide
|
C25H24Cl2N6O2
|
1
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| 1 |
Ki = 11 nM
|
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CP0554724
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4-[4-[2-(2,4-dichlorophenyl)-4-methyl-5-(piperidin-1-ylcarbamoyl)pyrazol-3-yl]phenyl]but-3-ynyl acetate
Show/Hide
|
C28H28Cl2N4O3
|
1
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| 1 |
Ki = 11 nM
|
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CP0420378
|
11-(3-butoxy-5-pentylphenoxy)-N-cyclopropylundecanamide
Show/Hide
|
C29H49NO3
|
1
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| 1 |
Ki = 11.3 nM
|
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CP0513751
|
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxoquinoline-3-carboxamide
Show/Hide
|
C24H25FN2O2
|
1
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| 1 |
Ki = 11.6 nM
|
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CP0569467
|
N-cyclopropyl-11-(3-ethoxy-5-pentylphenoxy)undecanamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 11.7 nM
|
|
|
|
CP0392053
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(piperidin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
|
C22H19Cl2N5O
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0396947
|
N-cycloheptyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C24H28Cl2N4O
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0042459
|
(6aR,10aR)-6,6,9-Trimethyl-3-(1-methyl-1-phenyl-ethyl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C25H30O2
|
1
|
| 1 |
Ki = 12.3 nM
|
|
|
|
CP0410867
|
8-(3-hydroxy-5-pentylphenoxy)-N-[(2R)-1-hydroxypropan-2-yl]octanamide
Show/Hide
|
C22H37NO4
|
1
|
| 1 |
Ki = 12.8 nM
|
|
|
|
CP0453386
|
4-oxo-1-pentyl-N-phenylmethoxy-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
|
C28H28N2O3S
|
1
|
| 1 |
Ki = 12.9 nM
|
|
|
|
CP0251560
|
1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-4-(4-fluoro-phenyl)-1,2,3,6-tetrahydro-pyridine
Show/Hide
|
C30H24FNO4S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0490572
|
(2,2-diphenyl-[1,3]dioxolo[4,5-c]pyridin-6-yl)-piperidin-1-ylmethanone
Show/Hide
|
C24H22N2O3
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0444413
|
12-(2-hexyl-5-hydroxy-phenoxy)-dodecanoic acidcyclopropylamide
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0441130
|
1-(2-Chloro-4-fluorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H21ClFN5O2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0411063
|
[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-pyrrolidin-1-ylmethanone
Show/Hide
|
C26H25Cl2N7O
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0432070
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-cyclohexylurea
Show/Hide
|
C30H33Cl2N7O
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0403140
|
methyl 6-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]hexanoate
Show/Hide
|
C24H24Cl3N3O3
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0548834
|
N-cyclopropyl-11-(3-pentyl-5-prop-2-enoxyphenoxy)undecanamide
Show/Hide
|
C28H45NO3
|
1
|
| 1 |
Ki = 13.6 nM
|
|
|
|
CP0493669
|
4-[2-[(6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydrobenzo[c]chromen-3-yl]propan-2-yl]benzamide
Show/Hide
|
C26H31NO3
|
1
|
| 1 |
Ki = 13.7 nM
|
|
|
|
CP0553941
|
1-(2,4-Dichlorophenyl)-4-cyano-5-(4-bromophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H18BrCl2N5O
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0473858
|
(R)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C23H26Cl2N4O
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0496604
|
(4-fluoronaphthalen-1-yl)-(2-methyl-1-pentylindol-3-yl)methanone
Show/Hide
|
C25H24FNO
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0524809
|
(4-bromonaphthalen-1-yl)-(2-methyl-1-pentylindol-3-yl)methanone
Show/Hide
|
C25H24BrNO
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0539751
|
(4-iodonaphthalen-1-yl)-(2-methyl-1-pentylindol-3-yl)methanone
Show/Hide
|
C25H24INO
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0452689
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(2,4-difluorophenyl)urea
Show/Hide
|
C29H23Cl2F2N7O
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0457644
|
(R)-7-Fluoro-4-oxo-1-pentyl-N-(1-phenylethyl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C23H25FN2O2
|
1
|
| 1 |
Ki = 14.3 nM
|
|
|
|
CP0480040
|
1-butyl-7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C24H31FN2O2
|
1
|
| 1 |
Ki = 14.4 nM
|
|
|
|
CP0496323
|
(2-cyclopentyl-5-propyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
Show/Hide
|
C26H37N3O
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0484112
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-[(2-fluorophenyl)methyl]urea
Show/Hide
|
C31H28Cl2FN7O
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0476297
|
N-cyclohexyl-1-(3,4-dichlorophenyl)-4-ethyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H24Cl2N4O
|
1
|
| 1 |
Ki = 15.3 nM
|
|
|
|
CP0410105
|
N-[7-[7-aminoheptyl(methyl)amino]heptyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C32H44Cl3N5O
|
2
|
| 1 |
Ki = 15.5 nM
|
|
|
| 2 |
Ki = 37.5 nM
|
|
|
|
CP0432935
|
8-(3-hydroxy-5-pentyl-phenoxy)-octanoic acid cyclopropylamide
Show/Hide
|
C22H35NO3
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0537625
|
N-cyclohexyl-1-[(4-fluorophenyl)methyl]-2-oxoquinoline-3-carboxamide
Show/Hide
|
C23H23FN2O2
|
1
|
| 1 |
Ki = 16.5 nM
|
|
|
|
CP0394223
|
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-3-[(E)-piperidinoiminomethyl]-1H-pyrazole
Show/Hide
|
C22H21Cl3N4
|
3
|
| 1 |
Ki = 17 nM
|
|
|
| 2 |
Ki = 19 nM
|
|
|
| 3 |
Ki = 57 nM
|
|
|
|
CP0522363
|
1-benzyl-N-cycloheptyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C24H26N2O2
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0406536
|
2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methylcyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C23H30ClN3O
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0493059
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-[(1R,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl]imidazole-4-carboxamide
Show/Hide
|
C25H19Cl2N3O2
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0397208
|
(2-cyclopentyl-5-ethylsulfonyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
Show/Hide
|
C25H35N3O3S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0544189
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-(4,4-difluorocyclohexyl)urea
Show/Hide
|
C30H31Cl2F2N7O
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0415354
|
8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]-N-[(2R)-1-hydroxypropan-2-yl]octanamide
Show/Hide
|
C26H45NO4
|
1
|
| 1 |
Ki = 17.2 nM
|
|
|
|
CP0474427
|
5-(4-chlorophenyl)-N-[7-[7-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]heptyl-methylamino]heptyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C49H53Cl6N7O2
|
2
|
| 1 |
Ki = 17.3 nM
|
|
|
| 2 |
Ki = 27.5 nM
|
|
|
|
CP0454189
|
N-cycloheptyl-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H30N4O3
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0483997
|
(6-fluoro-2,2-bis(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone
Show/Hide
|
C24H18F3NO4
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0435608
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide
Show/Hide
|
C25H19Cl2N3O2
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0536626
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-isopropyl-1H-imidazole-4-carboxamide
Show/Hide
|
C25H27Cl2N3O2
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0565197
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(4,4-difluorocyclohexyl)urea
Show/Hide
|
C29H29Cl2F2N7O
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0145758
|
8-Chloro-1-(2,4-dichloro-phenyl)-1,3a,4,5,6,10b-hexahydro-1,2-diaza-benzo[e]azulene-3-carboxylic acid piperidin-1-ylamide
Show/Hide
|
C24H23Cl3N4O
|
1
|
| 1 |
Ki = 18.4 nM
|
|
|
|
CP0353026
|
(6aR,10aR)-3-(2-(4-chlorophenyl)propan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
|
C25H29ClO2
|
1
|
| 1 |
Ki = 18.8 nM
|
|
|
|
CP0529789
|
5-bromo-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C22H20BrCl2N3O2
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0391007
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(4-fluorophenyl)piperazine-1-carboxamide
Show/Hide
|
C28H22Cl2FN7O
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0455586
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(cyclopentylmethyl)urea
Show/Hide
|
C29H31Cl2N7O
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0529572
|
1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxoquinoline-3-carboxamide
Show/Hide
|
C24H25FN2O2
|
1
|
| 1 |
Ki = 19.4 nM
|
|
|
|
CP0374241
|
N-[7-(7-aminoheptylamino)heptyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C31H42Cl3N5O
|
2
|
| 1 |
Ki = 19.5 nM
|
|
|
| 2 |
Ki = 46.7 nM
|
|
|
|
CP0398425
|
cyclopropanolamide, 14a
Show/Hide
|
C23H37NO2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0501760
|
1-(2-chlorophenyl)-2-(4-methoxyphenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C26H28ClN3O2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0486201
|
2-(2-chlorophenyl)-N-cyclohexyl-1-(4-fluorophenyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C22H21ClFN3O
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0371731
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-cyclohexyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
|
C23H20Cl2N4O
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0430148
|
N-cycloheptyl-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C22H24Cl2N4O
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0158863
|
2-[((11Z,14Z)-Icosa-5,8,11,14-tetraenyl)oxy]-propane-1,3-diol
Show/Hide
|
C23H40O3
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0469872
|
N-cyclopropyl-11-(3-pentyl-5-propan-2-yloxyphenoxy)undecanamide
Show/Hide
|
C28H47NO3
|
1
|
| 1 |
Ki = 20.7 nM
|
|
|
|
CP0498313
|
4-oxo-1-pentyl-7-phenylsulfanyl-N-propan-2-ylquinoline-3-carboxamide
Show/Hide
|
C24H28N2O2S
|
1
|
| 1 |
Ki = 20.9 nM
|
|
|
|
CP0486261
|
1-(4-chlorophenyl)-N-cyclohexyl-2-o-tolyl-1H-imidazole-4-carboxamide
Show/Hide
|
C23H24ClN3O
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0449530
|
2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-isopropyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
|
C20H16Cl2N4O
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0507173
|
(8-bromonaphthalen-1-yl)-(1-pentylindol-3-yl)methanone
Show/Hide
|
C24H22BrNO
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0526326
|
1-[4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperazin-1-yl]-2-piperidin-1-ylethanone
Show/Hide
|
C28H29Cl2N7O
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0486202
|
1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(2-hydroxycyclohexyl)imidazole-4-carboxamide
Show/Hide
|
C22H20Cl3N3O2
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0553901
|
2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-[(1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]imidazole-4-carboxamide
Show/Hide
|
C25H19Cl2N3O2
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0397210
|
2-cyclopentyl-N,N-dimethyl-8-(4-methylpiperidine-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indole-5-sulfonamide
Show/Hide
|
C25H36N4O3S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0495591
|
(2-cyclopentyl-5-propylsulfonyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
Show/Hide
|
C26H37N3O3S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0022072
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[6-(difluoromethoxy)pyridin-3-yl]urea
Show/Hide
|
C29H24Cl2F2N8O2
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0489575
|
1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(4-fluorophenyl)urea
Show/Hide
|
C29H24Cl2FN7O
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0496608
|
(8-chloronaphthalen-1-yl)-(1-pentylindol-3-yl)methanone
Show/Hide
|
C24H22ClNO
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0395641
|
5-bromo-1-butyl-N-cycloheptyl-2-oxopyridine-3-carboxamide
Show/Hide
|
C17H25BrN2O2
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0550757
|
11-(3-methoxy-5-pentylphenoxy)-N-prop-2-enylundecanamide
Show/Hide
|
C26H43NO3
|
1
|
| 1 |
Ki = 23.7 nM
|
|
|
|
CP0378066
|
1-(2-methoxyethyl)-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C29H34N2O3S
|
1
|
| 1 |
Ki = 23.8 nM
|
|
|
|
CP0441149
|
5-(4-chlorophenyl)-4-cyano-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H18Cl3N5O
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0381992
|
N-cycloheptyl-5-(4-fluorophenyl)-1-[(4-fluorophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
|
C26H26F2N2O2
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0458672
|
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxo-5-[(E)-2-phenylethenyl]pyridine-3-carboxamide
Show/Hide
|
C28H29FN2O2
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0466291
|
4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-[1-(trifluoromethyl)cyclopentyl]piperazine-1-carboxamide
Show/Hide
|
C28H26Cl2F3N7O
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0559842
|
8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylsulfonylpiperazin-1-yl)purine
Show/Hide
|
C22H20Cl2N6O2S
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0381990
|
ethyl (E)-3-[5-(cycloheptylcarbamoyl)-1-[(4-fluorophenyl)methyl]-6-oxopyridin-3-yl]prop-2-enoate
Show/Hide
|
C25H29FN2O4
|
1
|
| 1 |
Ki = 24.8 nM
|
|
|
|
CP0435619
|
1-(4-chlorophenyl)-N-cyclohexyl-2-(2,5-dichlorophenyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C22H20Cl3N3O
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0382776
|
N-(3-pentyl-1,3-benzothiazol-2-ylidene)-4-(trifluoromethyl)benzamide
Show/Hide
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C20H19F3N2OS
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1
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| 1 |
Ki = 25 nM
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CP0456605
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dibenzothiazepine, 12g
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C24H21ClN2OS
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1
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| 1 |
Ki = 25.12 nM
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CP0392392
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5-(2-chloropyrrol-1-yl)-1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methylpyrazole-3-carboxamide
Show/Hide
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C22H15Cl5N4O
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1
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| 1 |
Ki = 25.2 nM
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CP0441838
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2-(2-chlorophenyl)-3-(4-chlorophenyl)-6-(pentan-3-yl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
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C22H20Cl2N4O
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1
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| 1 |
Ki = 26 nM
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CP0476543
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[(4,4-difluorocyclohexyl)methyl]urea
Show/Hide
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C30H31Cl2F2N7O
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1
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| 1 |
Ki = 26 nM
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CP0382145
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(3',5'-dichloro-2,6-dihydroxybiphenyl-4-yl)(phenyl)methanone
Show/Hide
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C19H12Cl2O3
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1
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| 1 |
Ki = 27 nM
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CP0298207
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cyclopropanolamide, 11a
Show/Hide
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C23H37NO2
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1
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| 1 |
Ki = 28 nM
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CP0433751
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(2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone
Show/Hide
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C25H23NO3
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1
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| 1 |
Ki = 28 nM
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CP0442487
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3-(2-chlorophenyl)-2-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
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C19H11Cl2F3N4O
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1
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| 1 |
Ki = 28 nM
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CP0457647
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N-(1-adamantyl)-7-(benzenesulfinyl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C31H36N2O3S
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1
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| 1 |
Ki = 28 nM
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CP0037364
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(-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C21H30O2
|
2
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| 1 |
Ki = 28.5 nM
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| 2 |
Ki = 78 nM
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CP0435747
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1-[2-(dimethylamino)ethyl]-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C30H37N3O2S
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1
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| 1 |
Ki = 28.8 nM
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CP0498311
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4-oxo-1-pentyl-7-phenylsulfanyl-N-piperidin-1-ylquinoline-3-carboxamide
Show/Hide
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C26H31N3O2S
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1
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| 1 |
Ki = 28.9 nM
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CP0394621
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
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C22H21Cl2N3O2
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1
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| 1 |
Ki = 29 nM
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CP0467955
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide
Show/Hide
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C21H19Cl2N3O2
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1
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| 1 |
Ki = 29 nM
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CP0388546
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(R)-7-Ethoxy-4-oxo-1-pentyl-N-(1-phenylethyl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
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C25H30N2O3
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1
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| 1 |
Ki = 29.7 nM
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CP0493054
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4-Oxo-1-pentyl-6-pyrrol-1-yl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
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C29H35N3O2
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1
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| 1 |
Ki = 29.7 nM
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CP0267790
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5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazole-3-carboxylic acid cyclohexyl-methyl-amide
Show/Hide
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C24H24Cl3N3O
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3
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| 1 |
Ki = 30 nM
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| 2 |
Ki = 54 nM
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| 3 |
Ki = 107 nM
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CP0439166
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N-[2-(4-chlorophenyl)ethyl]-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H23Cl3N4O
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1
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| 1 |
Ki = 30 nM
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CP0374242
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5-(4-chlorophenyl)-N-[5-[5-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]pentylamino]pentyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C44H43Cl6N7O2
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2
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| 1 |
Ki = 30.4 nM
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| 2 |
Ki = 68.1 nM
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CP0436996
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N-(1-adamantyl)-7-fluoro-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C25H31FN2O2
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1
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| 1 |
Ki = 30.5 nM
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CP0396949
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N-(1-adamantyl)-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C25H26Cl2N4O
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1
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| 1 |
Ki = 31 nM
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CP0510139
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[5-(benzenesulfonyl)-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C29H35N3O4S
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1
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| 1 |
Ki = 31 nM
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CP0858250
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10alpha-Hydroxy-Delta8-tetrahydrocannabinol
Show/Hide
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C21H30O3
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1
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| 1 |
Ki = 31 nM
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CP0282078
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5-(4-chlorophenyl)-3-[(E)-2-cyclohexylethenyl]-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole
Show/Hide
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C24H23Cl3N2
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3
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| 1 |
Ki = 31.3 nM
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| 2 |
Ki = 60 nM
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| 3 |
Ki = 85 nM
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CP0376757
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N-(1-adamantyl)-2-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C25H32N2O2
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1
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| 1 |
Ki = 31.3 nM
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CP0441131
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1-(2-Bromo-4-fluorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C23H21BrFN5O2
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1
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| 1 |
Ki = 32 nM
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CP0496324
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(2-cyclopentyl-5-methyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C24H33N3O
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1
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| 1 |
Ki = 32 nM
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CP0383808
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1-(2,4-Dichlorophenyl)-4-cyano-5-(4-iodophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H18Cl2IN5O
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1
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| 1 |
Ki = 33 nM
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CP0516603
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N-(1-adamantyl)-7-hydroxy-2-methyl-5-oxo-4-pentylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C23H32N4O3
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1
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| 1 |
Ki = 33.5 nM
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CP0394618
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-N-methyl-1H-imidazole-4-carboxamide
Show/Hide
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C23H23Cl2N3O
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1
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| 1 |
Ki = 34 nM
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CP0397207
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(2-cyclopentyl-5-ethyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C25H35N3O
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1
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| 1 |
Ki = 34 nM
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CP0302795
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(6aR,10aR)-6,6,9-trimethyl-3-(2-o-tolylpropan-2-yl)-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C26H32O2
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1
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| 1 |
Ki = 34.4 nM
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CP0940324
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(S)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone
Show/Hide
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C24H17Cl2F2NO4
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1
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| 1 |
Ki = 35 nM
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CP0435741
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N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxo-5-phenylpyridine-3-carboxamide
Show/Hide
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C26H27FN2O2
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1
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| 1 |
Ki = 35 nM
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CP0384967
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1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-difluorophenyl)-1H-imidazole-4-carboxamide
Show/Hide
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C22H20ClF2N3O
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1
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| 1 |
Ki = 36 nM
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CP0401296
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N-cyclopentyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C22H24Cl2N4O
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1
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| 1 |
Ki = 36 nM
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CP0448347
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(2-cyclopentyl-5-methylsulfonyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C24H33N3O3S
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1
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| 1 |
Ki = 36 nM
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CP0374244
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5-(4-chlorophenyl)-N-[11-[11-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]undecylamino]undecyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C56H67Cl6N7O2
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2
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| 1 |
Ki = 37 nM
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| 2 |
Ki = 99.3 nM
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CP0498793
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-N-(3,3-dimethylbutyl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C23H28Cl2N4O
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1
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| 1 |
Ki = 37.5 nM
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CP0433752
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1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-piperidine
Show/Hide
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C24H23NO4S
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1
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| 1 |
Ki = 38 nM
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CP0435517
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3-(2-chlorophenyl)-2-(4-chlorophenyl)-6-cyclohexyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
Show/Hide
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C23H20Cl2N4O
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1
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| 1 |
Ki = 38 nM
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CP0453371
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1-(4-hydroxybutyl)-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C30H36N2O3S
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1
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| 1 |
Ki = 38.6 nM
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CP0467953
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1-(4-chlorophenyl)-N-cyclohexyl-2-(2-ethylphenyl)-1H-imidazole-4-carboxamide
Show/Hide
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C24H26ClN3O
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1
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| 1 |
Ki = 39 nM
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CP0560406
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N-(1-adamantyl)-4-(4-fluorobutyl)-7-hydroxy-1-methyl-5-oxo-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C22H31FN4O3
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1
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| 1 |
Ki = 39.3 nM
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CP0417505
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dibenzothiazepine, 13
Show/Hide
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C23H18ClNOS
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1
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| 1 |
Ki = 39.81 nM
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CP0518050
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-[(1S,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl]imidazole-4-carboxamide
Show/Hide
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C25H19Cl2N3O2
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1
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| 1 |
Ki = 41 nM
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CP0439162
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N-[2-(2,4-dichlorophenyl)ethyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H22Cl2F2N4O
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1
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| 1 |
Ki = 41 nM
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CP0410104
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5-(4-chlorophenyl)-N-[3-[3-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]propylamino]propyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C40H35Cl6N7O2
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2
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| 1 |
Ki = 41.9 nM
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| 2 |
Ki = 174 nM
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CP0085406
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4-Oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
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C25H32N2O2
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1
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| 1 |
Ki = 42.1 nM
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CP0395172
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N-cycloheptyl-1-[(4-fluorophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
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C20H23FN2O2
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1
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| 1 |
Ki = 43 nM
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CP0547413
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4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(cyclohexylmethyl)piperazine-1-carboxamide
Show/Hide
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C29H31Cl2N7O
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1
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| 1 |
Ki = 43 nM
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CP0444255
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6-O-tert-butyl 1-O-[4-[4-[2-(2,4-dichlorophenyl)-4-methyl-5-(piperidin-1-ylcarbamoyl)pyrazol-3-yl]phenyl]but-3-ynyl] hexanedioate
Show/Hide
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C36H42Cl2N4O5
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1
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| 1 |
Ki = 45 nM
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CP0501840
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1-(2,4-Dichlorophenyl)-N-(3,3-dimethylbutyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C21H24Cl2N4O
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1
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| 1 |
Ki = 45.6 nM
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CP0390454
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1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(4,5,6,7-tetrahydroisoindol-2-yl)pyrazole-3-carboxamide
Show/Hide
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C26H22Cl4N4O
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1
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| 1 |
Ki = 45.9 nM
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CP0875825
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(R,S)-2-(2-Chlorophenyl)-3-(4-chlorophenyl)-N-methyl-5,6,7,8-tetrahydro-2H-oxepino[3,2-c]pyrazol-8-amine hydrochloride
Show/Hide
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C20H20Cl3N3O
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1
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| 1 |
Ki = 46 nM
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CP0436242
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(6aR,10aR)-9-(acetyloxymethyl)-1-hydroxy-6,6-dimethyl-3-pentyl-6a,7,8,10a-tetrahydrobenzo[c]chromene-2-carboxylic acid
Show/Hide
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C24H32O6
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1
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| 1 |
Ki = 47 nM
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CP0380261
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1-(2,4-Dichlorophenyl)-4-methyl-N-tert-pentyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C20H22Cl2N4O
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1
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| 1 |
Ki = 47.6 nM
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CP0456245
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N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-ethylpyrazole-3-carboxamide
Show/Hide
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C24H28Cl2N4O
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1
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| 1 |
Ki = 48 nM
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CP0481084
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N-(1-adamantyl)-5-phenyl-1-prop-2-enylindole-3-carboxamide
Show/Hide
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C28H30N2O
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1
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| 1 |
Ki = 48.2 nM
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CP0390455
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1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-ethyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H18Cl4N4O
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1
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| 1 |
Ki = 48.7 nM
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CP0376645
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N-[2-(4-chlorophenyl)ethyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H23ClF2N4O
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1
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| 1 |
Ki = 50 nM
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CP0453835
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N-cyclopentyl-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C20H20Cl2N4O
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1
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| 1 |
Ki = 50 nM
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CP0495590
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[5-[(4-ethoxyphenyl)methyl]-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C32H41N3O3
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1
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| 1 |
Ki = 51 nM
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CP0485556
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-[6-(trifluoromethyl)pyridin-3-yl]urea
Show/Hide
|
C29H23Cl2F3N8O
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1
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| 1 |
Ki = 51 nM
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CP0920867
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S-(R)-1-((2S,3R)-1-(4-fluorophenyl)-2-(4-hydroxyphenyl)-4-oxoazetidin-3-yl)-3-phenylpropyl ethanethioate
Show/Hide
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C26H24FNO3S
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1
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| 1 |
Ki = 52.8 nM
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CP0392395
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1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dimethylpyrrol-1-yl)-4-ethylpyrazole-3-carboxamide
Show/Hide
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C25H22Cl4N4O
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1
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| 1 |
Ki = 53.1 nM
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CP0548830
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8-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]-N-(2,2,2-trifluoroethyl)octanamide
Show/Hide
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C26H42F3NO3
|
1
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| 1 |
Ki = 53.5 nM
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CP0453828
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N-[2-(3,4-dichlorophenyl)ethyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H22Cl2F2N4O
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1
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| 1 |
Ki = 54 nM
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CP0381511
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(8-bromonaphthalen-1-yl)-(2-methyl-1-pentylindol-3-yl)methanone
Show/Hide
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C25H24BrNO
|
1
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| 1 |
Ki = 54 nM
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CP0386430
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5-(4-chlorophenyl)-N-[9-[9-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]nonylamino]nonyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C52H59Cl6N7O2
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2
|
| 1 |
Ki = 54.1 nM
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| 2 |
Ki = 57.4 nM
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CP0395647
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1-[(4-chlorophenyl)methyl]-N-cycloheptyl-2-oxopyridine-3-carboxamide
Show/Hide
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C20H23ClN2O2
|
1
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| 1 |
Ki = 55 nM
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CP0459063
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1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dichloropyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H14Cl6N4O
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1
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| 1 |
Ki = 55.6 nM
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CP0498832
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N-cyclohexyl-1-[(4-fluorophenyl)methyl]-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C22H22FN3O2
|
1
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| 1 |
Ki = 56 nM
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CP0444410
|
8-(4-hexyl-3-hydroxy-phenoxy)-octanoic acidcyclopropylamide
Show/Hide
|
C23H37NO3
|
1
|
| 1 |
Ki = 56 nM
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CP0390565
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N-[(4-chlorophenyl)methyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C24H21ClF2N4O
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1
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| 1 |
Ki = 56 nM
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CP0396951
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N-cycloheptyl-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C24H28F2N4O
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1
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| 1 |
Ki = 56 nM
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CP0480063
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N-cycloheptyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C24H28Cl2N4O
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1
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| 1 |
Ki = 56 nM
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CP0390836
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(2-cyclohexyl-5-prop-2-enyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C27H37N3O
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1
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| 1 |
Ki = 56 nM
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CP0458673
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1-benzyl-N-cycloheptyl-2-oxopyridine-3-carboxamide
Show/Hide
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C20H24N2O2
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1
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| 1 |
Ki = 56 nM
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CP0560405
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N-(1-adamantyl)-7-hydroxy-1-methyl-5-oxo-4-pentyl-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C23H34N4O3
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1
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| 1 |
Ki = 56 nM
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CP0899711
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(R,S)-2-(2-Chlorophenyl)-3-(4-chlorophenyl)-5,6,7,8-tetrahydro-2H-oxepino[3,2-c]pyrazol-8-amine Hydrochloride
Show/Hide
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C19H18Cl3N3O
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1
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| 1 |
Ki = 57 nM
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CP0371805
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CAS_15998383
Show/Hide
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C25H30N2O5S
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1
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| 1 |
Ki = 58 nM
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CP0528170
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CAS_22422464
Show/Hide
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C24H27ClN2O4S
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1
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| 1 |
Ki = 58 nM
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CP0372352
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N-(3,3-diphenylpropyl)-2,2-diphenylacetamide
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C29H27NO
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1
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| 1 |
Ki = 58 nM
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CP0372970
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(4-methylpiperidin-1-yl)-[2-(oxan-4-yl)-5-propyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]methanone
Show/Hide
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C26H37N3O2
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1
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| 1 |
Ki = 58 nM
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CP0453373
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N-(1-hydroxybutan-2-yl)-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
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C25H30N2O3S
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1
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| 1 |
Ki = 58.2 nM
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CP0386991
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methyl 2-(adamantane-1-carbonylamino)-5-butyl-4-methylthiophene-3-carboxylate
Show/Hide
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C22H31NO3S
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1
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| 1 |
Ki = 58.89 nM
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CP0398973
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CAS_11496202
Show/Hide
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C25H30N2O4S
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1
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| 1 |
Ki = 59 nM
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CP0427162
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12-(3-hydroxy-5-pentyl-phenoxy)-dodecanoic acid(2-hydroxy-ethyl)-amide
Show/Hide
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C25H43NO4
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1
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| 1 |
Ki = 60 nM
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CP0432796
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1,3-dihydroxypropan-2-yl 11-(2-hexyl-5-hydroxyphenoxy)undecanoate
Show/Hide
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C26H44O6
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1
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| 1 |
Ki = 60 nM
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CP0379559
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CAS_22422466
Show/Hide
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C24H27FN2O4S
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1
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| 1 |
Ki = 62 nM
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CP0443539
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N-cycloheptyl-1-[(4-fluorophenyl)methyl]-5-(4-methoxyphenyl)-2-oxopyridine-3-carboxamide
Show/Hide
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C27H29FN2O3
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1
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| 1 |
Ki = 63 nM
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CP0525504
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N-(2-morpholin-4-ylethyl)-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
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C27H33N3O3S
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1
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| 1 |
Ki = 63.2 nM
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CP0426923
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N-cyclohexyl-4-hydroxy-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C21H28N4O4
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1
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| 1 |
Ki = 64.6 nM
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CP0380792
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THC, 8 beta-OH
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C21H30O3
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1
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| 1 |
Ki = 65 nM
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CP0392391
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1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dichloropyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C22H14Cl6N4O
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1
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| 1 |
Ki = 66.1 nM
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CP0513447
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1-benzyl-N-cyclohexyl-2-oxoquinoline-3-carboxamide
Show/Hide
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C23H24N2O2
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1
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| 1 |
Ki = 67 nM
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CP0516604
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N-(1-adamantyl)-4-butyl-7-hydroxy-1-methyl-5-oxo-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C22H32N4O3
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1
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| 1 |
Ki = 69 nM
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CP0376650
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N-[(4-chlorophenyl)methyl]-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C22H17Cl3N4O
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1
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| 1 |
Ki = 70 nM
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CP0376697
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N-[2-(4-chlorophenyl)ethyl]-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H19Cl3N4O
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1
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| 1 |
Ki = 70 nM
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CP0432138
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N-cyclohexyl-1-[(4-fluorophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
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C19H21FN2O2
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1
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| 1 |
Ki = 70 nM
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CP0434013
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1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
Show/Hide
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C20H23FN2O2
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1
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| 1 |
Ki = 70 nM
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CP0488466
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(8-iodonaphthalen-1-yl)-(1-pentylindol-3-yl)methanone
Show/Hide
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C24H22INO
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1
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| 1 |
Ki = 73 nM
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CP0465170
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2-(4-methoxyphenyl)-3-methyl-5-(piperidin-1-yl)-1-o-tolyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C27H31N3O2
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1
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| 1 |
Ki = 74 nM
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CP0495980
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5-(2-chloropyrrol-1-yl)-1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-methylpyrazole-3-carboxamide
Show/Hide
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C22H15Cl5N4O
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1
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| 1 |
Ki = 74.1 nM
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CP0486199
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide
Show/Hide
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C21H19Cl2N3O2
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1
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| 1 |
Ki = 75 nM
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CP0527864
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11-(3-methoxy-5-pentylphenoxy)-N-(2,2,2-trifluoroethyl)undecanamide
Show/Hide
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C25H40F3NO3
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1
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| 1 |
Ki = 75.5 nM
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CP0275006
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[5-methyl-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C24H33N3O2
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1
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| 1 |
Ki = 76 nM
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CP0157111
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(6aR,10aR)-3-(2-(4-fluorophenyl)propan-2-yl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromen-1-ol
Show/Hide
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C25H29FO2
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1
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| 1 |
Ki = 76.1 nM
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CP0526831
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N-(2-hydroxyethyl)-8-(3-methoxy-5-pentylphenoxy)octanamide
Show/Hide
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C22H37NO4
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1
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| 1 |
Ki = 76.1 nM
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CP0371806
|
CAS_15991674
Show/Hide
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C24H28N2O4S
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1
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| 1 |
Ki = 77 nM
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CP0412747
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11-[3-(5-hydroxy-1,1-dimethylpentyl)phenoxy]-undeca-5,8-dienoic acid [R-(1-hydroxypropan-2-yl)]amide
Show/Hide
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C27H43NO4
|
1
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| 1 |
Ki = 78.97 nM
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CP0528073
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5-(3,5-dimethyl-piperidine-1-sulfonyl)-3-methyl-benzofuran-2-carboxylic acid 4-methyl-benzylamide
Show/Hide
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C25H30N2O4S
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1
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| 1 |
Ki = 79 nM
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CP0453833
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N-[2-(4-chlorophenyl)ethyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H19ClF2N4O
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1
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| 1 |
Ki = 80 nM
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CP0506341
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1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methyl-N-(1-phenylethyl)pyrazole-3-carboxamide
Show/Hide
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C25H24Cl2N4O
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1
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| 1 |
Ki = 80 nM
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CP0498791
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1-(2,4-Dichlorophenyl)-4-methyl-N-pentyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C20H22Cl2N4O
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1
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| 1 |
Ki = 81 nM
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CP0535473
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-[6-(difluoromethoxy)pyridin-3-yl]urea
Show/Hide
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C30H26Cl2F2N8O2
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1
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| 1 |
Ki = 81 nM
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CP0402060
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N-(1-adamantyl)-1,3-benzothiazole-2-carboxamide
Show/Hide
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C18H20N2OS
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1
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| 1 |
Ki = 82 nM
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CP0430955
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N-cyclopentyl-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C20H20Cl2N4O
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1
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| 1 |
Ki = 84 nM
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CP0478120
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12-[2-(1,1-dimethylheptyl)phenyl]dodeca-5,8,11-trienoic acid [R-(1-hydroxypropan-2-yl)]-amide
Show/Hide
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C30H47NO2
|
1
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| 1 |
Ki = 86.33 nM
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CP0393335
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N',N'-dimethyl-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carbohydrazide
Show/Hide
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C23H27N3O2S
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1
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| 1 |
Ki = 86.6 nM
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CP0572166
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4-butyl-7-hydroxy-N-(3-hydroxy-1-adamantyl)-1-methyl-5-oxo-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C22H32N4O4
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1
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| 1 |
Ki = 86.9 nM
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CP0527861
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N-(2-hydroxyethyl)-11-(3-methoxy-5-pentylphenoxy)undecanamide
Show/Hide
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C25H43NO4
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1
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| 1 |
Ki = 87.6 nM
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CP0375654
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N-[5-[5-aminopentyl(methyl)amino]pentyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C28H36Cl3N5O
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2
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| 1 |
Ki = 88.8 nM
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| 2 |
Ki = 162 nM
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CP0420377
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N-(2-hydroxyethyl)-8-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]octanamide
Show/Hide
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C26H45NO4
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1
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| 1 |
Ki = 89.1 nM
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CP0472387
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N-tert-butyl-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C19H20Cl2N4O
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1
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| 1 |
Ki = 89.5 nM
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CP0394012
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CAS_15998702
Show/Hide
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C22H30N2O4S
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1
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| 1 |
Ki = 90 nM
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CP0439167
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N-[(4-chlorophenyl)methyl]-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C24H21Cl3N4O
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1
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| 1 |
Ki = 90 nM
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CP0376687
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1-(2,4-Difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-N-(3,3-dimethylbutyl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C23H28F2N4O
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1
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| 1 |
Ki = 90.7 nM
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CP0371809
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CAS_4055807
Show/Hide
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C26H32N2O4S
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1
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| 1 |
Ki = 92 nM
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CP0488647
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(4-chloronaphthalen-1-yl)-(1-propylindol-3-yl)methanone
Show/Hide
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C22H18ClNO
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1
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| 1 |
Ki = 93 nM
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CP0510098
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3',5'-dichloro-4-(2-phenylpropan-2-yl)biphenyl-2,6-diol
Show/Hide
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C21H18Cl2O2
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1
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| 1 |
Ki = 93.66 nM
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CP0399367
|
CAS_4621779
Show/Hide
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C21H30N2O4S
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1
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| 1 |
Ki = 94 nM
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CP0379528
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5-(4-chlorophenyl)-N-[2-[2-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]ethylamino]ethyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C38H31Cl6N7O2
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2
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| 1 |
Ki = 94 nM
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| 2 |
Ki = 229 nM
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CP0406055
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5-(4-chlorophenyl)-N-[9-[9-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]nonyl-methylamino]nonyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C53H61Cl6N7O2
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2
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| 1 |
Ki = 94.1 nM
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| 2 |
Ki = 247 nM
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CP0529737
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1-(4-chlorophenyl)-N-cyclohexyl-2-(2-methoxyphenyl)-1H-imidazole-4-carboxamide
Show/Hide
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C23H24ClN3O2
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1
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| 1 |
Ki = 95 nM
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CP0496213
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N-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C23H19Cl3N4O
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1
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| 1 |
Ki = 96 nM
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CP0440571
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CAS_15998061
Show/Hide
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C26H32N2O5S
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1
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| 1 |
Ki = 97 nM
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CP0486200
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2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
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C22H21Cl2N3O2
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1
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| 1 |
Ki = 97 nM
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CP0567241
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4-[4-[2-(2,4-dichlorophenyl)-4-methyl-5-(piperidin-1-ylcarbamoyl)pyrazol-3-yl]phenyl]but-3-ynyl 11-aminoundecanoate;2,2,2-trifluoroacetic acid
Show/Hide
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C39H48Cl2F3N5O5
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1
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| 1 |
Ki = 97 nM
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CP0382509
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-Nheptyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C24H30Cl2N4O
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1
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| 1 |
Ki = 97.2 nM
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CP0453827
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N-[2-(3-chloro-4-methoxyphenyl)ethyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C26H25ClF2N4O2
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1
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| 1 |
Ki = 99 nM
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CP0453834
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N-[(4-chlorophenyl)methyl]-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C24H21Cl3N4O
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1
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| 1 |
Ki = 100 nM
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CP0432137
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N-cycloheptyl-2-[(4-fluorophenyl)methoxy]pyridine-3-carboxamide
Show/Hide
|
C20H23FN2O2
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1
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| 1 |
Ki = 100 nM
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CP0431129
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1-[8-(4-methylpiperidine-1-carbonyl)-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]butan-1-one
Show/Hide
|
C27H37N3O3
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1
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| 1 |
Ki = 102 nM
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CP0465952
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(octan-2-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H32Cl2N4O
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1
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| 1 |
Ki = 104.7 nM
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CP0416564
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4-[4-[2-(2,4-dichlorophenyl)-4-methyl-5-(piperidin-1-ylcarbamoyl)pyrazol-3-yl]phenyl]but-3-ynyl 6-[(2-methylpropan-2-yl)oxycarbonylamino]hexanoate
Show/Hide
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C37H45Cl2N5O5
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1
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| 1 |
Ki = 106 nM
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CP0371808
|
CAS_3379236
Show/Hide
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C23H32N2O4S
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1
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| 1 |
Ki = 108 nM
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CP0564717
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N-(1-adamantyl)-7-hydroxy-2-(2-hydroxyethyl)-5-oxo-4-pentylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C24H34N4O4
|
1
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| 1 |
Ki = 108 nM
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CP0433753
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(6-(methylsulfonyl)-1-pentyl-1H-indol-3-yl)(naphthalen-2-yl)methanone
Show/Hide
|
C25H25NO3S
|
1
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| 1 |
Ki = 110 nM
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CP0495588
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N,N-dimethyl-8-(4-methylpiperidine-1-carbonyl)-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indole-5-sulfonamide
Show/Hide
|
C25H36N4O4S
|
1
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| 1 |
Ki = 110 nM
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CP0453830
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N-[2-(3-chloro-4-methoxyphenyl)ethyl]-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C26H25Cl3N4O2
|
1
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| 1 |
Ki = 112 nM
|
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CP0069603
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(4-methylpiperidin-1-yl)-[2-(oxan-4-yl)-5-propylsulfonyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]methanone
Show/Hide
|
C26H37N3O4S
|
1
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| 1 |
Ki = 115 nM
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CP0520163
|
(8-chloronaphthalen-1-yl)-(2-methyl-1-pentylindol-3-yl)methanone
Show/Hide
|
C25H24ClNO
|
1
|
| 1 |
Ki = 116 nM
|
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CP0453831
|
1-(2,4-dichlorophenyl)-N-[2-(3,4-dichlorophenyl)ethyl]-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C25H22Cl4N4O
|
1
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| 1 |
Ki = 117 nM
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CP0876344
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10alpha-Hydroxy-Delta9,11-hexahydrocannabinol
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C21H30O3
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1
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| 1 |
Ki = 117 nM
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CP0376698
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N-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
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C21H15Cl3N4O
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1
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| 1 |
Ki = 120 nM
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CP0535474
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-methylpiperidin-4-yl]-3-(2-fluorophenyl)sulfonylurea
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C30H26Cl2FN7O3S
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1
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| 1 |
Ki = 120 nM
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CP0527604
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N-butyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
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C21H24Cl2N4O
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1
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| 1 |
Ki = 123.1 nM
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CP0500041
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1-(2,4-Dichlorophenyl)-N-hexyl-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
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C21H24Cl2N4O
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1
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| 1 |
Ki = 124.1 nM
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CP0427500
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8-(3-hydroxy-5-pentyl-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide
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C21H35NO4
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1
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| 1 |
Ki = 130 nM
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CP0529738
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1-(4-chlorophenyl)-N-cyclohexyl-2-phenyl-1H-imidazole-4-carboxamide
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C22H22ClN3O
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1
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| 1 |
Ki = 130 nM
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CP0383810
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1-(2,4-Dichlorophenyl)-4-cyano-5-(4-iodophenyl)-N-morpholino-1H-pyrazole-3-carboxamide
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C21H16Cl2IN5O2
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1
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| 1 |
Ki = 131 nM
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CP0438260
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methyl 4-[4-[2-(2,4-dichlorophenyl)-4-methyl-5-(piperidin-1-ylcarbamoyl)pyrazol-3-yl]phenyl]benzoate
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C30H28Cl2N4O3
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1
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| 1 |
Ki = 131 nM
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CP0515131
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(5Z,8Z,11Z)-N-((R)-1-hydroxypropan-2-yl)-14-(3-(2-methyloctan-2-yl)phenoxy)tetradeca-5,8,11-trienamide
Show/Hide
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C32H51NO3
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1
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| 1 |
Ki = 131.33 nM
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CP0410866
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11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]-N-[(2R)-1-hydroxypropan-2-yl]undecanamide
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C29H51NO4
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1
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| 1 |
Ki = 132.2 nM
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CP0440708
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N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-diethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H30Cl2N4O
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1
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| 1 |
Ki = 136.3 nM
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CP0400886
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11-(3-hydroxy-5-pentylphenoxy)-N-prop-2-enylundecanamide
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C25H41NO3
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1
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| 1 |
Ki = 136.3 nM
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CP0449956
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1-[(4-fluorophenyl)methyl]-4-hydroxy-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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C23H24FN3O3
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1
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| 1 |
Ki = 138.5 nM
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CP0386405
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N-(1-adamantyl)-6-fluoro-4-oxo-1-pentyl-7-pyrrol-1-ylquinoline-3-carboxamide
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C29H34FN3O2
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1
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| 1 |
Ki = 139.8 nM
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CP0453832
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N-[(4-chlorophenyl)methyl]-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C22H17Cl3N4O
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1
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| 1 |
Ki = 140 nM
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CP0488127
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(4-iodonaphthalen-1-yl)-(1-propylindol-3-yl)methanone
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C22H18INO
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1
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| 1 |
Ki = 140 nM
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CP0087210
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[2-(cyclopropylmethyl)-5-prop-2-enyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C25H33N3O
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1
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| 1 |
Ki = 143 nM
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CP0430953
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N-[(2-bromo-3,4,5-trimethoxyphenyl)methyl]-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C27H27BrCl2N4O4
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1
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| 1 |
Ki = 144 nM
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CP0401267
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N-cyclopentyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
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C22H24Cl2N4O
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1
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| 1 |
Ki = 150 nM
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CP0376686
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N-tert-butyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C21H24Cl2N4O
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1
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| 1 |
Ki = 150.7 nM
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CP0404947
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N-(1-azabicyclo[2.2.2]octan-3-yl)-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
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C28H33N3O2S
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1
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| 1 |
Ki = 151.1 nM
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CP0376652
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1-(2,4-dichlorophenyl)-N-[2-(2,4-dichlorophenyl)ethyl]-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H22Cl4N4O
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1
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| 1 |
Ki = 156 nM
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CP0450845
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1-(2,4-dichlorophenyl)-N-[2-(3,4-dichlorophenyl)ethyl]-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H18Cl4N4O
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1
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| 1 |
Ki = 157 nM
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CP0412798
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1-(2,4-Dichlorophenyl)-4-methyl-N-(octan-2-yl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C23H28Cl2N4O
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1
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| 1 |
Ki = 157.5 nM
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CP0457643
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(R)-4-Oxo-1-pentyl-N-(1-phenylethyl)-7-(pyrrolidin-1-yl)-1,4-dihydroquinoline-3-carboxamide
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C27H33N3O2
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1
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| 1 |
Ki = 160 nM
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CP0379382
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N-cycloheptyl-5-(4-fluorophenyl)-2-methoxy-3-methylbenzamide
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C22H26FNO2
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1
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| 1 |
Ki = 160 nM
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CP0496605
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(4-bromonaphthalen-1-yl)-(1-propylindol-3-yl)methanone
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C22H18BrNO
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1
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| 1 |
Ki = 161 nM
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CP0516606
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4-(4-fluorobutyl)-7-hydroxy-N-(3-hydroxy-1-adamantyl)-1-methyl-5-oxo-3a,7a-dihydropyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C22H31FN4O4
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1
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| 1 |
Ki = 161 nM
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CP0506340
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N-[(2-bromo-3,4,5-trimethoxyphenyl)methyl]-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C27H27BrF2N4O4
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1
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| 1 |
Ki = 165 nM
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CP0510584
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1-benzyl-N-cyclohexyl-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxamide
Show/Hide
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C24H26N2O3
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1
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| 1 |
Ki = 170 nM
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CP0432932
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12-(2-hexyl-5-hydroxy-phenoxy)-dodecanoic acid(2-hydroxy-ethyl)-amide
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C26H45NO4
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1
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| 1 |
Ki = 170 nM
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CP0419836
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2-[6-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]hexoxy]propane-1,3-diol
Show/Hide
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C24H42O5
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1
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| 1 |
Ki = 170 nM
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CP0496103
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(4-methylpiperidin-1-yl)-[2-(oxan-4-yl)-5-propan-2-ylsulfonyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]methanone
Show/Hide
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C26H37N3O4S
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1
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| 1 |
Ki = 170 nM
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CP0458168
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5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N,3-dimethyl-N-phenethylbenzofuran-2-carboxamide
Show/Hide
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C26H32N2O4S
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1
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| 1 |
Ki = 172 nM
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CP0533214
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N-(1,3-dihydroxypropan-2-yl)-8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]octanamide
Show/Hide
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C26H45NO5
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1
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| 1 |
Ki = 177.8 nM
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CP0452471
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1-[2-(dimethylamino)ethyl]-7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C24H32FN3O2
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1
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| 1 |
Ki = 178.7 nM
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CP0388920
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5-(4-fluorophenyl)-2-methoxy-3-methyl-N-(4-methylcyclohexyl)benzamide
Show/Hide
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C22H26FNO2
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1
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| 1 |
Ki = 180 nM
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CP0469454
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1-(2,4-dichlorophenyl)-5-[4-(4-hydroxybut-1-ynyl)phenyl]-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide
Show/Hide
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C26H26Cl2N4O2
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1
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| 1 |
Ki = 180 nM
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CP0404949
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1-ethyl-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C28H32N2O2S
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1
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| 1 |
Ki = 181.3 nM
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CP0465950
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-pentyl-1H-pyrazole-3-carboxamide
Show/Hide
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C22H26Cl2N4O
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1
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| 1 |
Ki = 182.1 nM
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CP0425247
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methyl 2-(adamantane-1-carbonylamino)-4-ethyl-5-methylthiophene-3-carboxylate
Show/Hide
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C20H27NO3S
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1
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| 1 |
Ki = 185.14 nM
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CP0488646
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(4-chloronaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone
Show/Hide
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C23H20ClNO
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1
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| 1 |
Ki = 187 nM
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CP0427501
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8-(4-hexyl-3-hydroxy-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide
Show/Hide
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C22H37NO4
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1
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| 1 |
Ki = 190 nM
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CP0371807
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CAS_3340785
Show/Hide
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C23H32N2O4S
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1
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| 1 |
Ki = 193 nM
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CP0404948
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7-fluoro-4-oxo-1-propyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C23H29FN2O2
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1
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| 1 |
Ki = 193 nM
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CP0465951
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-tert-pentyl-1H-pyrazole-3-carboxamide
Show/Hide
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C22H26Cl2N4O
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1
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| 1 |
Ki = 193.5 nM
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CP0412748
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11-[4-(1,1-dimethylheptyl)phenoxy]undeca-5,8-dienoic acid [R(1-hydroxypropan-2-yl)]-amide
Show/Hide
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C29H47NO3
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1
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| 1 |
Ki = 194.85 nM
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CP0087211
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[5-ethylsulfonyl-2-(oxolan-3-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C24H33N3O4S
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1
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| 1 |
Ki = 197 nM
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CP0394013
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5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-phenethylbenzofuran-2-carboxamide
Show/Hide
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C25H30N2O4S
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1
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| 1 |
Ki = 198 nM
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CP0051372
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1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C23H24FN3O2
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1
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| 1 |
Ki = 200 nM
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CP0471931
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1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C23H24FN3O2
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1
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| 1 |
Ki = 200 nM
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CP0444452
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2-(4-chlorophenyl)-5-cyclohexyl-1-(2,6-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C26H25Cl3N2O
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1
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| 1 |
Ki = 200 nM
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CP0471598
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N-(1-adamantyl)-8-nitro-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C25H31N3O4
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1
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| 1 |
Ki = 200 nM
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CP0409164
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N-cycloheptyl-1-(2-morpholin-4-ylethyl)-2-oxoquinoline-3-carboxamide
Show/Hide
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C23H31N3O3
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1
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| 1 |
Ki = 206 nM
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CP0376688
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1-(2,4-Dichlorophenyl)-N-heptyl-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C22H26Cl2N4O
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1
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| 1 |
Ki = 211 nM
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CP0394225
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1-[2-(5-(4-chlorophenyl)-1(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-yl)-(E)-vinyl]-piperidine
Show/Hide
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C23H22Cl3N3
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3
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| 1 |
Ki = 213 nM
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| 2 |
Ki = 223 nM
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| 3 |
Ki = 258 nM
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CP0433750
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(6-chloro-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone
Show/Hide
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C24H20ClNO4
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1
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| 1 |
Ki = 216 nM
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CP0506396
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1-(2,4-dichlorophenyl)-N-[2-(2,4-dichlorophenyl)ethyl]-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H18Cl4N4O
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1
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| 1 |
Ki = 218 nM
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CP0372609
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2-(4-Bromophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
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C29H26BrNO
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1
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| 1 |
Ki = 220 nM
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CP0849493
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9beta,10beta-Epoxyhexahydrocannabinol
Show/Hide
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C21H30O3
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1
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| 1 |
Ki = 224 nM
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CP0275040
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[5-methyl-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]-piperidin-1-ylmethanone
Show/Hide
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C23H31N3O2
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1
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| 1 |
Ki = 226 nM
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CP0431070
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1-(1-(4-chlorophenyl)-4-(3-methoxyphenyl)-5-(4-morpholinophenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethanone
Show/Hide
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C27H27ClN4O3
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1
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| 1 |
Ki = 227 nM
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CP0388378
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N-[(2-bromo-3,4,5-trimethoxyphenyl)methyl]-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C25H23BrCl2N4O4
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1
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| 1 |
Ki = 227 nM
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CP0410517
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N-(4-methylcyclohexyl)-2-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C22H30N2O2
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1
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| 1 |
Ki = 227 nM
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CP0374243
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N-[5-(5-aminopentylamino)pentyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C27H34Cl3N5O
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2
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| 1 |
Ki = 230 nM
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| 2 |
Ki = 349 nM
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CP0526748
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N-(1-adamantyl)-4-butyl-7-hydroxy-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C22H30N4O3
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1
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| 1 |
Ki = 231 nM
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CP0527077
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-Nisopropyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C20H22Cl2N4O
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1
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| 1 |
Ki = 233.5 nM
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CP0513750
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N-cycloheptyl-4-hydroxy-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C22H30N4O4
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1
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| 1 |
Ki = 234 nM
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CP0387785
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(4-methylpiperidin-1-yl)-[5-methylsulfonyl-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]methanone
Show/Hide
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C24H33N3O4S
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1
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| 1 |
Ki = 239 nM
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CP0465172
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C20H22Cl2N2O
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1
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| 1 |
Ki = 240 nM
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CP0376649
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N-[2-(4-chlorophenyl)ethyl]-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H19Cl3N4O
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1
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| 1 |
Ki = 240 nM
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CP0517625
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(4-fluoronaphthalen-1-yl)-(1-propylindol-3-yl)methanone
Show/Hide
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C22H18FNO
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1
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| 1 |
Ki = 240 nM
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CP0443537
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5-bromo-N-cycloheptyl-1-(2-morpholin-4-ylethyl)-2-oxopyridine-3-carboxamide
Show/Hide
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C19H28BrN3O3
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1
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| 1 |
Ki = 243 nM
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CP0880973
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(3R,4S)-4-(4-methoxyphenyl)-1-phenyl-3-(3-(pyridin-3-yl)propyl)azetidin-2-one
Show/Hide
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C24H24N2O2
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1
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| 1 |
Ki = 243.8 nM
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CP0501629
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6-(1-Isobutyl-1H-pyrazol-4-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
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C32H42N4O2
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1
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| 1 |
Ki = 245.7 nM
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CP0548567
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4-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-N-(2-fluorophenyl)sulfonylpiperazine-1-carboxamide
Show/Hide
|
C28H22Cl2FN7O3S
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1
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| 1 |
Ki = 250 nM
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CP0507878
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4-(indolin-1-ylsulfonyl)-N-(2-phenoxyphenyl)benzamide
Show/Hide
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C27H22N2O4S
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1
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| 1 |
Ki = 256 nM
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CP0378995
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8-(2-hexyl-5-hydroxy-phenoxy)-octanoic acid (2-hydroxy-ethyl)-amide
Show/Hide
|
C22H37NO4
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1
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| 1 |
Ki = 260 nM
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CP0396891
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N-(1-adamantyl)-4-oxo-8-pentoxy-1H-quinoline-3-carboxamide
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C25H32N2O3
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1
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| 1 |
Ki = 260 nM
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CP0557473
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4-[4-[2-(2,4-dichlorophenyl)-4-methyl-5-(piperidin-1-ylcarbamoyl)pyrazol-3-yl]phenyl]but-3-ynyl 6-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-carbothioyl)amino]hexanoate
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C53H47Cl2N5O8S
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1
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| 1 |
Ki = 260 nM
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CP0490713
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2-(7,7-dimethyl-2-p-tolyl-7,8-dihydro-5H-pyrano[4,3-d]pyrimidin-4-ylthio)-N-(2-methoxyphenyl)propanamide
Show/Hide
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C26H29N3O3S
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1
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| 1 |
Ki = 264 nM
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CP0431130
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(2-cyclopentyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-8-yl)-(4-methylpiperidin-1-yl)methanone
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C23H31N3O
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1
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| 1 |
Ki = 264 nM
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CP0567082
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11-(3-hydroxy-5-pentylphenoxy)-N-[(2R)-1-hydroxypropan-2-yl]undecanamide
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C25H43NO4
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1
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| 1 |
Ki = 264.4 nM
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CP0439659
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N-[(1S,2S)-2-aminocyclohexyl]-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)imidazole-4-carboxamide
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C22H21Cl3N4O
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1
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| 1 |
Ki = 270 nM
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CP0477443
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N-(1-adamantyl)-6-(furan-2-yl)-4-hydroxy-2-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C29H34N2O4
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1
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| 1 |
Ki = 270 nM
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CP0452193
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2-[8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]octoxy]propane-1,3-diol
Show/Hide
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C26H46O5
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1
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| 1 |
Ki = 270 nM
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CP0382752
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N-(1,3-benzothiazol-2-yl)adamantane-1-carboxamide
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C18H20N2OS
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1
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| 1 |
Ki = 272 nM
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CP0465953
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N-butyl-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C19H20Cl2N4O
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1
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| 1 |
Ki = 272.6 nM
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CP0507879
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ethyl 2-[6-bromo-2-(4-fluorophenyl)-4-phenyl-2,4-dihydro-1H-quinazolin-3-yl]acetate
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C24H22BrFN2O2
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1
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| 1 |
Ki = 273 nM
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CP0428047
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6-(morpholine-4-carbonyl)-2,2-diphenyl-benzo[1,3]dioxole-5-carbonitrile
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C25H20N2O4
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1
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| 1 |
Ki = 277 nM
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CP0509078
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2-chloro-N-(3,3-diphenylpropyl)-2,2-diphenylacetamide
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C29H26ClNO
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1
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| 1 |
Ki = 280 nM
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CP0469873
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N-cyclopropyl-11-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
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C30H51NO3
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1
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| 1 |
Ki = 280 nM
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CP0446046
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2,5-dimethyl-N-naphthalen-2-yl-1-phenylpyrrole-3-carboxamide
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C23H20N2O
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1
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| 1 |
Ki = 281.06 nM
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CP0431071
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ethyl 4-[5-(2-chlorophenyl)-2-(2,4-dimethylphenyl)pyrazole-3-carbonyl]piperazine-1-carboxylate
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C25H27ClN4O3
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1
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| 1 |
Ki = 287 nM
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CP0382824
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N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-benzothiazole-2-carboxamide
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C18H16N2OS
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1
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| 1 |
Ki = 288 nM
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CP0455045
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N-cycloheptyl-1-(2-morpholin-4-ylethyl)-4-oxoquinoline-3-carboxamide
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C23H31N3O3
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1
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| 1 |
Ki = 290 nM
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CP0498789
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-propyl-1H-pyrazole-3-carboxamide
Show/Hide
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C20H22Cl2N4O
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1
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| 1 |
Ki = 290.1 nM
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CP0455246
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7-fluoro-1-(2-methoxyethyl)-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C23H29FN2O3
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1
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| 1 |
Ki = 296.8 nM
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CP0527862
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N-(cyclopropylmethyl)-11-(3-methoxy-5-pentylphenoxy)undecanamide
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C27H45NO3
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1
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| 1 |
Ki = 297.4 nM
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CP0454190
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1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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C23H24FN3O2
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1
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| 1 |
Ki = 300 nM
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CP0410760
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N-cyclohexyl-1-(2-morpholin-4-ylethyl)-2-oxoquinoline-3-carboxamide
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C22H29N3O3
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1
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| 1 |
Ki = 300 nM
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CP0855252
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(3S,4R)-1-(4-fluorophenyl)-3-(3-(4-fluorophenyl)-3-hydroxypropyl)-4-(4-hydroxyphenyl)azetidin-2-one
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C24H21F2NO3
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1
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| 1 |
Ki = 301.4 nM
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CP0509860
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3-tert-butyl-1-isopropyl-1-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]quinoxalin-5(4H)-yl)-2-oxoethyl)urea
Show/Hide
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C28H34N4O3
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1
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| 1 |
Ki = 308 nM
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CP0428675
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8-(2-hexyl-5-hydroxy-phenoxy)-octanoic acidcyclopropylamide
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C23H37NO3
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1
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| 1 |
Ki = 310 nM
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CP0376646
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N-[2-(3,4-dichlorophenyl)ethyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H18Cl2F2N4O
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1
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| 1 |
Ki = 310 nM
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CP0527080
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1-(2,4-Difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-Nhexyl-4-methyl-1H-pyrazole-3-carboxamide
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C23H28F2N4O
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1
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| 1 |
Ki = 311.4 nM
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CP0455975
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2,5-dimethyl-N-naphthalen-1-yl-1-phenylpyrrole-3-carboxamide
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C23H20N2O
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1
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| 1 |
Ki = 317.03 nM
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CP0222092
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(4-methylpiperidin-1-yl)-[2-(oxolan-3-yl)-5-propylsulfonyl-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]methanone
Show/Hide
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C25H35N3O4S
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1
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| 1 |
Ki = 320 nM
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CP0496490
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2-[2-(2,4,6-Trimethyl-phenoxy)-acetylamino]-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid (1,1-dioxo-tetrahydro-1lambda*6*-thiophen-3-yl)-amide
Show/Hide
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C24H30N2O5S2
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1
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| 1 |
Ki = 325 nM
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CP0509784
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N-[(4-chlorophenyl)methyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C22H17ClF2N4O
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1
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| 1 |
Ki = 340 nM
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CP0429455
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N-(1-adamantyl)-5-(furan-2-yl)-1-pentylindole-3-carboxamide
Show/Hide
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C28H34N2O2
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1
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| 1 |
Ki = 341.6 nM
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CP0453121
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N-(1-adamantyl)-2-[5-(furan-2-yl)-1-pentylindol-3-yl]-2-oxoacetamide
Show/Hide
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C29H34N2O3
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1
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| 1 |
Ki = 344.9 nM
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CP0390568
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N-[(2-bromo-3,4,5-trimethoxyphenyl)methyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C25H23BrF2N4O4
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1
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| 1 |
Ki = 345 nM
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CP0553772
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N-(1,3-dihydroxypropan-2-yl)-11-(3-methoxy-5-pentylphenoxy)undecanamide
Show/Hide
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C26H45NO5
|
1
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| 1 |
Ki = 349.7 nM
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CP0411868
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6-(6-Methoxy-naphthalen-2-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
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C36H40N2O3
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1
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| 1 |
Ki = 360 nM
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CP0390564
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N-[2-(3-chloro-4-methoxyphenyl)ethyl]-1-(2,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C24H21Cl3N4O2
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1
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| 1 |
Ki = 368 nM
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CP0500040
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1-(2,4-Difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-Nheptyl-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C24H30F2N4O
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1
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| 1 |
Ki = 368.2 nM
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CP0379578
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1-(2,4-Dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-N-(5-hydroxypentyl)-4-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C22H26Cl2N4O2
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1
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| 1 |
Ki = 372.3 nM
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CP0513861
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(4-bromonaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone
Show/Hide
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C23H20BrNO
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1
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| 1 |
Ki = 373 nM
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CP0390567
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N-[2-(2,4-dichlorophenyl)ethyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H18Cl2F2N4O
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1
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| 1 |
Ki = 380 nM
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CP0432075
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1-[1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]piperidin-4-yl]-3-(2-fluorophenyl)sulfonylurea
Show/Hide
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C29H24Cl2FN7O3S
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1
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| 1 |
Ki = 380 nM
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CP0395646
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1-benzyl-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
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C20H24N2O2
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1
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| 1 |
Ki = 386 nM
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CP0497153
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5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(pyridin-3-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C25H25Cl2N3O
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1
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| 1 |
Ki = 390 nM
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CP0396948
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N-[2-(4-chlorophenyl)ethyl]-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C25H23Cl3N4O
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1
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| 1 |
Ki = 390 nM
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CP0498310
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N-[(3,4-dichlorophenyl)methyl]-4-oxo-1-pentyl-7-phenylquinoline-3-carboxamide
Show/Hide
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C28H26Cl2N2O2
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1
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| 1 |
Ki = 390 nM
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CP0382826
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N-(1-adamantyl)-2-tert-butyl-4-methyl-1,3-thiazole-5-carboxamide
Show/Hide
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C19H28N2OS
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1
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| 1 |
Ki = 395 nM
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CP0555106
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8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]-N-(2,2,2-trifluoroethyl)octanamide
Show/Hide
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C25H40F3NO3
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1
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| 1 |
Ki = 397 nM
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CP0393332
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7-fluoro-1-(4-hydroxybutyl)-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C24H31FN2O3
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1
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| 1 |
Ki = 398.5 nM
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CP0193415
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N-[(3,4-dichlorophenyl)methyl]-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
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C28H26Cl2N2O2S
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1
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| 1 |
Ki = 420 nM
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CP0042287
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1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C21H19Cl2IN4O2
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1
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| 1 |
Ki = 422 nM
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CP0448348
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N-ethyl-8-(4-methylpiperidine-1-carbonyl)-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indole-5-sulfonamide
Show/Hide
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C25H36N4O4S
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1
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| 1 |
Ki = 424 nM
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CP0419835
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2-[6-(3-hydroxy-5-pentylphenoxy)hexoxy]propane-1,3-diol
Show/Hide
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C20H34O5
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1
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| 1 |
Ki = 430 nM
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CP0048193
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5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1H-pyrazole-3-carboxylic acid (1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide
Show/Hide
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C29H34ClN3O
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4
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| 1 |
Ki = 437 nM
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| 2 |
Ki > 2820 nM
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| 3 |
Ki > 5000 nM
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| 4 |
Ki > 5600 nM
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CP0548584
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11-(3-hydroxy-5-pentylphenoxy)-N-(2,2,2-trifluoroethyl)undecanamide
Show/Hide
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C24H38F3NO3
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1
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| 1 |
Ki = 438 nM
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CP0437116
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2-(3-aminophenyl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
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C26H27Cl2N3O
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1
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| 1 |
Ki = 450 nM
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CP0427554
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N-(1-adamantyl)-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C21H24N2OS
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1
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| 1 |
Ki = 450 nM
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CP0441547
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4-(4-methoxyphenyl)-1-phenyl-3-(2-(phenylsulfonyl)ethyl)azetidin-2-one
Show/Hide
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C24H23NO4S
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1
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| 1 |
Ki = 451.5 nM
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CP0440707
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1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-4-ethyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C23H18Cl4N4O
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1
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| 1 |
Ki = 454 nM
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CP0406214
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N-(1-adamantyl)-6-(benzenesulfinyl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C31H36N2O3S
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1
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| 1 |
Ki = 460 nM
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CP0043807
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1,3-dihydroxypropan-2-yl (5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoate
Show/Hide
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C23H38O4
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1
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| 1 |
Ki = 470 nM
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CP0497271
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6-(furan-2-yl)-4-oxo-1-pentyl-N-((1R,2R,4S)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
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C29H36N2O3
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1
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| 1 |
Ki = 480 nM
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CP0416221
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N-(1-adamantyl)-2-(1-methyl-5-phenylindol-3-yl)acetamide
Show/Hide
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C27H30N2O
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1
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| 1 |
Ki = 488 nM
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CP0443426
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N-methoxy-4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carboxamide
Show/Hide
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C22H24N2O3S
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1
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| 1 |
Ki = 490 nM
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CP0564718
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7-hydroxy-N-(3-hydroxy-1-adamantyl)-2-(2-hydroxyethyl)-5-oxo-4-pentylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C24H34N4O5
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1
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| 1 |
Ki = 492 nM
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CP0458710
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(4-iodonaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone
Show/Hide
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C23H20INO
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1
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| 1 |
Ki = 501 nM
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CP0401720
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(4-methoxyphenyl)-[1-(oxan-4-ylmethyl)-7-propoxyindol-3-yl]methanone
Show/Hide
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C25H29NO4
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1
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| 1 |
Ki = 504.6 nM
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CP0395711
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2-ethyl-5-methyl-N-naphthalen-1-yl-1-phenylpyrrole-3-carboxamide
Show/Hide
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C24H22N2O
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1
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| 1 |
Ki = 505.03 nM
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CP0379529
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N-[2-(2-aminoethylamino)ethyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C21H22Cl3N5O
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2
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| 1 |
Ki = 506 nM
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| 2 |
Ki = 1225 nM
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CP0458008
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(6-methyl-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone
Show/Hide
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C25H23NO4
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1
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| 1 |
Ki = 509 nM
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CP0432934
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11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid cyclopropylmethyl-amide
Show/Hide
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C26H43NO3
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1
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| 1 |
Ki = 510 nM
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CP0102145
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6-(4-Methoxy-3,5-dimethyl-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
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C34H42N2O3
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1
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| 1 |
Ki = 510 nM
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CP0400951
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N-(1-adamantyl)-2,5-dimethyl-1-phenylpyrrole-3-carboxamide
Show/Hide
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C23H28N2O
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1
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| 1 |
Ki = 518.2 nM
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CP0425255
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methyl 2-(adamantane-1-carbonylamino)-5-pentyl-4-phenylthiophene-3-carboxylate
Show/Hide
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C28H35NO3S
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1
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| 1 |
Ki = 518.57 nM
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CP0500042
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1-(2,4-Dichlorophenyl)-N-isopropyl-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C18H18Cl2N4O
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1
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| 1 |
Ki = 518.9 nM
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CP0429470
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2-(1-(4-(4-chlorophenyl)-2,2,4-trimethyl-3,4-dihydroquinolin-1(2H)-yl)-1-oxopropan-2-yl)hexahydro-1H-isoindole-1,3(2H)-dione
Show/Hide
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C29H33ClN2O3
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1
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| 1 |
Ki = 520 nM
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CP0490714
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N-cyclopropyl-N-[2-[4-(4-methylphenyl)-4H-pyrrolo[1,2-a]quinoxalin-5-yl]-2-oxoethyl]cyclopentanecarboxamide
Show/Hide
|
C29H31N3O2
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1
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| 1 |
Ki = 520 nM
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CP0513857
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(8-iodonaphthalen-1-yl)-(2-methyl-1-pentylindol-3-yl)methanone
Show/Hide
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C25H24INO
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1
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| 1 |
Ki = 522 nM
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CP0416198
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N-(1-adamantyl)-2-(5-phenyl-1-prop-2-enylindol-3-yl)acetamide
Show/Hide
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C29H32N2O
|
1
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| 1 |
Ki = 530 nM
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CP0481751
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(4-fluoronaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone
Show/Hide
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C23H20FNO
|
1
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| 1 |
Ki = 530 nM
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CP0525855
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N-(1-adamantyl)-4-(4-fluorobutyl)-7-hydroxy-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
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C22H29FN4O3
|
1
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| 1 |
Ki = 532 nM
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CP0501839
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1-(2,4-Dichlorophenyl)-N-(5-hydroxypentyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C20H22Cl2N4O2
|
1
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| 1 |
Ki = 534.4 nM
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CP0380260
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1-(2,4-Dichlorophenyl)-4-methyl-N-propyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C18H18Cl2N4O
|
1
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| 1 |
Ki = 550.3 nM
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CP0499727
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1-butyl-N-(4-methylcyclohexyl)-2-oxoquinoline-3-carboxamide
Show/Hide
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C21H28N2O2
|
1
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| 1 |
Ki = 551 nM
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CP0498354
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N-cyclohexyl-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C21H28N4O3
|
1
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| 1 |
Ki = 560 nM
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CP0498940
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1-benzyl-N-cyclohexyl-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C22H23N3O2
|
1
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| 1 |
Ki = 560 nM
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CP0454092
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5-benzyl-7-chloro-2-cyclohexyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one
Show/Hide
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C23H22ClN3O
|
1
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| 1 |
Ki = 560 nM
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CP0522361
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1-benzyl-N-cyclohexyl-7-methoxy-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
Show/Hide
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C23H25N3O3
|
1
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| 1 |
Ki = 560 nM
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CP0428635
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11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid [2-(3,4-dihydroxy-phenyl)-ethyl]-amide
Show/Hide
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C30H45NO5
|
1
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| 1 |
Ki = 560 nM
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CP0396952
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N-(4-chlorophenyl)-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
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C23H19ClF2N4O
|
1
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| 1 |
Ki = 560 nM
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CP0430952
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N-cycloheptyl-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
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C22H24F2N4O
|
1
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| 1 |
Ki = 560 nM
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CP0372349
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2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
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C29H26ClNO
|
1
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| 1 |
Ki = 560 nM
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CP0400884
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N-(3,3-diphenylpropyl)-2,2-diphenylpropanamide
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C30H29NO
|
1
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| 1 |
Ki = 560 nM
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CP0493783
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2-(4-Nitrophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
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C29H26N2O3
|
1
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| 1 |
Ki = 560 nM
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CP0493784
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2-(4-Methylphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
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C30H29NO
|
1
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| 1 |
Ki = 560 nM
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CP0496637
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N-(3,3-diphenylpropyl)-2-phenylacetamide
Show/Hide
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C23H23NO
|
1
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| 1 |
Ki = 560 nM
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CP0524192
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2-(4-Methoxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
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C30H29NO2
|
1
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| 1 |
Ki = 560 nM
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CP0542696
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2-(4-Hydroxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
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C29H27NO2
|
1
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| 1 |
Ki = 560 nM
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CP0450454
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1-benzyl-N-cyclohexyl-4-hydroxy-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C22H23N3O3
|
1
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| 1 |
Ki = 560 nM
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CP0514780
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N-(1-adamantyl)-2-[5-(furan-2-yl)-1-prop-2-enylindol-3-yl]acetamide
Show/Hide
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C27H30N2O2
|
1
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| 1 |
Ki = 560 nM
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CP0175984
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(6S)-N,9-dimethyl-N-[4-(methylamino)-4-oxobutyl]-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
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C25H35N3O3
|
1
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| 1 |
Ki = 576 nM
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CP0397209
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[5-imidazol-1-ylsulfonyl-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indol-8-yl]-(4-methylpiperidin-1-yl)methanone
Show/Hide
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C26H33N5O4S
|
1
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| 1 |
Ki = 592 nM
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CP0417551
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N-benzhydryl-5-(3,5-dimethylpiperidin-1-yl)sulfonyl-2-fluorobenzamide
Show/Hide
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C27H29FN2O3S
|
1
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| 1 |
Ki = 611 nM
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CP0444362
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5-benzyl-2-cyclohexyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one
Show/Hide
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C23H23N3O
|
1
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| 1 |
Ki = 620 nM
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CP0505366
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1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1S,2S)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
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C23H23Cl3N4O
|
1
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| 1 |
Ki = 620 nM
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CP0379381
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5-(4-fluorophenyl)-2-methoxy-3-methyl-N-(4-methylcyclohexyl)benzamide
Show/Hide
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C22H26FNO2
|
1
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| 1 |
Ki = 620 nM
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CP0499113
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4-hydroxy-N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C22H30N4O4
|
1
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| 1 |
Ki = 630.3 nM
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CP0395708
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2-ethyl-5-methyl-N-naphthalen-2-yl-1-phenylpyrrole-3-carboxamide
Show/Hide
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C24H22N2O
|
1
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| 1 |
Ki = 633.03 nM
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CP0290316
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N-(1-adamantyl)-4-oxo-1-pentyl-6-phenylsulfanylquinoline-3-carboxamide
Show/Hide
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C31H36N2O2S
|
1
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| 1 |
Ki = 640 nM
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CP0511004
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(8-chloronaphthalen-1-yl)-(1-propylindol-3-yl)methanone
Show/Hide
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C22H18ClNO
|
1
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| 1 |
Ki = 642 nM
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CP0334444
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N-[3-(cyclopropylamino)-3-oxopropyl]-N,9-dimethyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
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C26H35N3O3
|
1
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| 1 |
Ki = 655 nM
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CP0443425
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7-bromo-N-[(3,4-dichlorophenyl)methyl]-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C22H21BrCl2N2O2
|
1
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| 1 |
Ki = 660 nM
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CP0404950
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1-[(3-methylphenyl)methyl]-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C34H36N2O2S
|
1
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| 1 |
Ki = 669.3 nM
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CP0516622
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N-(cyclopropylmethyl)-11-(2-hexyl-5-methoxyphenoxy)undecanamide
Show/Hide
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C28H47NO3
|
1
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| 1 |
Ki = 693.5 nM
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CP0460327
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N-(1-adamantyl)-6-bromo-4-oxo-1-pent-4-enylquinoline-3-carboxamide
Show/Hide
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C25H29BrN2O2
|
1
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| 1 |
Ki = 696 nM
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CP0542424
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N-(1-adamantyl)-2-(1-ethyl-5-phenylindol-3-yl)acetamide
Show/Hide
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C28H32N2O
|
1
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| 1 |
Ki = 698 nM
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CP0557205
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1-butyl-4-hydroxy-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C20H27N3O3
|
1
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| 1 |
Ki = 701.5 nM
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CP0538198
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1-[1-[8-(2-chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]purin-6-yl]piperidin-4-yl]-3-(cyclohexylmethyl)urea
Show/Hide
|
C30H32ClF3N8O
|
1
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| 1 |
Ki = 730 nM
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CP0436216
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N-(1-adamantyl)-6-(3-chloro-4-fluorophenoxy)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
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C31H34ClFN2O3
|
1
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| 1 |
Ki = 739 nM
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CP0428636
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12-(3-hydroxy-5-pentyl-phenoxy)-dodecanoic acidcyclopropylamide
Show/Hide
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C26H43NO3
|
1
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| 1 |
Ki = 750 nM
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CP0444415
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11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acidcyclopropylmethyl-amide
Show/Hide
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C27H45NO3
|
1
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| 1 |
Ki = 750 nM
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CP0479506
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2-(4-bromophenyl)-N-(3,3-diphenylpropyl)acetamide
Show/Hide
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C23H22BrNO
|
1
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| 1 |
Ki = 800 nM
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CP0392072
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1,3-dihydroxypropan-2-yl 8-(2-hexyl-5-hydroxyphenoxy)octanoate
Show/Hide
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C23H38O6
|
1
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| 1 |
Ki = 800 nM
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CP0450453
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1-benzyl-N-cyclohexyl-2-oxopyridine-3-carboxamide
Show/Hide
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C19H22N2O2
|
1
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| 1 |
Ki = 800 nM
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CP0415214
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N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxoquinoline-3-carboxamide
Show/Hide
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C23H31N3O3
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1
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| 1 |
Ki = 800 nM
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CP0919485
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(1R,2S)-N-Oleoylcyclopropanolamide
Show/Hide
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C19H37NO2
|
1
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| 1 |
Ki = 820 nM
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CP0149319
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[5-hydroxy-1-(oxan-4-ylmethyl)indol-3-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C25H23NO3
|
1
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| 1 |
Ki = 823.8 nM
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CP0381996
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3-[12-(cyclopropylamino)dodecoxy]-5-pentylphenol
Show/Hide
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C26H45NO2
|
1
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| 1 |
Ki = 830 nM
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CP0877895
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10beta-Hydroxy-Delta8-tetrahydrocannabinol
Show/Hide
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C21H30O3
|
1
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| 1 |
Ki = 830 nM
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CP0877723
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(3R,4S)-3-(benzofuran-2-ylmethyl)-4-(4-methoxyphenyl)-1-phenylazetidin-2-one
Show/Hide
|
C25H21NO3
|
1
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| 1 |
Ki = 839 nM
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CP0044659
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(6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-indol-3-yl)(4-methoxyphenyl)methanone
Show/Hide
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C23H25IN2O3
|
2
|
| 1 |
Ki = 840 nM
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| 2 |
Ki = 5152 nM
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CP0453826
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N-cyclopentyl-1-(2,4-difluorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C22H24F2N4O
|
1
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| 1 |
Ki = 840 nM
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CP0526833
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11-(3-methoxy-5-pentylphenoxy)-N-phenylundecanamide
Show/Hide
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C29H43NO3
|
1
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| 1 |
Ki = 844.5 nM
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CP0566882
|
11-(3-hydroxy-5-pentylphenoxy)-N',N'-dimethylundecanehydrazide
Show/Hide
|
C24H42N2O3
|
1
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| 1 |
Ki = 845.5 nM
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CP0383135
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N-cycloheptyl-2-methoxy-3-methyl-5-phenylbenzamide
Show/Hide
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C22H27NO2
|
1
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| 1 |
Ki = 870 nM
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CP0428043
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(6-bromo-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone
Show/Hide
|
C24H20BrNO4
|
1
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| 1 |
Ki = 873 nM
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CP0422853
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N-[2-[4-(4-fluorophenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-N-(2-methylpropyl)furan-2-carboxamide
Show/Hide
|
C24H25FN2O3S
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1
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| 1 |
Ki = 875 nM
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CP0388259
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2-[(4-fluorophenyl)methoxy]-N-(4-methylcyclohexyl)pyridine-3-carboxamide
Show/Hide
|
C20H23FN2O2
|
1
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| 1 |
Ki = 884 nM
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CP0372348
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2-(4-Aminophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide
Show/Hide
|
C29H28N2O
|
1
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| 1 |
Ki = 900 nM
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CP0195802
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N-(1-adamantyl)-6-ethyl-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C27H36N2O2
|
1
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| 1 |
Ki = 900 nM
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CP0384509
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N-[11-(2-hexyl-5-hydroxyphenoxy)undecyl]cyclopropanecarboxamide
Show/Hide
|
C27H45NO3
|
1
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| 1 |
Ki = 900 nM
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CP0405572
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2-(4-aminophenyl)-5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C26H27Cl2N3O
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1
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| 1 |
Ki = 920 nM
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CP0435963
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1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1R,2R)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide
Show/Hide
|
C23H23Cl3N4O
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1
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| 1 |
Ki = 920 nM
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CP0480324
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N-[(1R,2R)-2-aminocyclohexyl]-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)imidazole-4-carboxamide
Show/Hide
|
C22H21Cl3N4O
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1
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| 1 |
Ki = 940 nM
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CP0491341
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N-[2-(3-chloro-4-methoxyphenyl)ethyl]-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C24H21ClF2N4O2
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1
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| 1 |
Ki = 948 nM
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CP0432135
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N-cycloheptyl-1-(2-morpholin-4-ylethyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C19H29N3O3
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1
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| 1 |
Ki = 950 nM
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CP0257260
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1-ethyl-7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C22H27FN2O2
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1
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| 1 |
Ki = 959.7 nM
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CP0454192
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1-benzyl-N-cycloheptyl-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H25N3O2
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1
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| 1 |
Ki = 960 nM
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CP0489050
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1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-dimethylpyrrol-1-yl)-4-ethylpyrazole-3-carboxamide
Show/Hide
|
C25H22Cl4N4O
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1
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| 1 |
Ki = 965.7 nM
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CP0141726
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N-(1-adamantyl)-6-bromo-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C25H31BrN2O2
|
1
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| 1 |
Ki = 996 nM
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CP0120450
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N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C22H30N4O3
|
1
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| 1 |
Ki = 1000 nM
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CP0429473
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methyl (1Z)-N-[4-[5-thiophen-2-yl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]sulfonylpyrrolidine-1-carboximidothioate
Show/Hide
|
C20H19F3N4O2S3
|
1
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| 1 |
Ki = 1000 nM
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CP0169639
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N-(1-adamantyl)-2-ethyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),11-tetraene-11-carboxamide
Show/Hide
|
C24H28N2O3
|
1
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| 1 |
Ki = 1000 nM
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CP0385072
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ethyl 2-(adamantane-1-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C22H29NO3S
|
1
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| 1 |
Ki = 1008.48 nM
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CP0502191
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N-[2-[4-(4-fluorophenyl)-4H-pyrrolo[1,2-a]quinoxalin-5-yl]-2-oxoethyl]-3,3-dimethyl-N-propan-2-ylbutanamide
Show/Hide
|
C28H32FN3O2
|
1
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| 1 |
Ki = 1030 nM
|
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CP0427943
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2-[12-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]dodecoxy]propane-1,3-diol
Show/Hide
|
C30H54O5
|
1
|
| 1 |
Ki = 1040 nM
|
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CP0507880
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N-phenyl-N-[1-(phenylcarbamoyl)cyclohexyl]-4-(tetrazol-1-yl)benzamide
Show/Hide
|
C27H26N6O2
|
1
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| 1 |
Ki = 1049 nM
|
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CP0535273
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N-(1-adamantyl)-1-pentyl-5-phenylindole-3-carboxamide
Show/Hide
|
C30H36N2O
|
1
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| 1 |
Ki = 1052 nM
|
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CP0543211
|
3-[9-[[(2R)-1-hydroxypropan-2-yl]amino]nonoxy]-5-pentylphenol
Show/Hide
|
C23H41NO3
|
1
|
| 1 |
Ki = 1060 nM
|
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CP0382783
|
N-[(2-chlorophenyl)methyl]-1,3-benzothiazole-2-carboxamide
Show/Hide
|
C15H11ClN2OS
|
1
|
| 1 |
Ki = 1084 nM
|
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CP0918783
|
ethyl 6'-amino-1-benzyl-5',5',7'-tricyano-2-oxo-5',8a'-dihydro-1'H-spiro[indoline-3,8'-isoquinoline]-2'(3'H)-carboxylate
Show/Hide
|
C29H24N6O3
|
1
|
| 1 |
Ki = 1086 nM
|
|
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CP0419213
|
2-methoxy-3-methyl-N-(4-methylcyclohexyl)-5-phenylbenzamide
Show/Hide
|
C22H27NO2
|
1
|
| 1 |
Ki = 1090 nM
|
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|
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CP0035557
|
(Z)-N-(2-hydroxyethyl)octadec-9-enamide
Show/Hide
|
C20H39NO2
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0486260
|
2-(2-chlorophenyl)-N-cyclohexyl-1-(pyridin-3-yl)-1H-imidazole-4-carboxamide
Show/Hide
|
C21H21ClN4O
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0425254
|
methyl 2-(adamantane-1-carbonylamino)-5-methyl-4-propylthiophene-3-carboxylate
Show/Hide
|
C21H29NO3S
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0492411
|
1,3-dihydroxypropan-2-yl 8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]octanoate
Show/Hide
|
C26H44O6
|
1
|
| 1 |
Ki = 1120 nM
|
|
|
|
CP0410859
|
3-pentyl-5-[11-(prop-2-enylamino)undecoxy]phenol
Show/Hide
|
C25H43NO2
|
1
|
| 1 |
Ki = 1140 nM
|
|
|
|
CP0417552
|
N-benzhydryl-6-(2,6-dimethylmorpholin-4-yl)-5-nitropyrimidin-4-amine
Show/Hide
|
C23H25N5O3
|
1
|
| 1 |
Ki = 1177 nM
|
|
|
|
CP0856485
|
2-Ethyl-5-methyl-1-phenyl-1H-pyrrole-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C24H30N2O
|
1
|
| 1 |
Ki = 1196.7 nM
|
|
|
|
CP0409163
|
N-cyclohexyl-2-[(4-fluorophenyl)methoxy]quinoline-3-carboxamide
Show/Hide
|
C23H23FN2O2
|
1
|
| 1 |
Ki = 1200 nM
|
|
|
|
CP0195829
|
6-Isopropyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C28H38N2O2
|
1
|
| 1 |
Ki = 1220 nM
|
|
|
|
CP0494513
|
3-[11-(benzylamino)undecoxy]-5-pentylphenol
Show/Hide
|
C29H45NO2
|
1
|
| 1 |
Ki = 1240 nM
|
|
|
|
CP0442970
|
N-cycloheptyl-1-[(4-iodophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
|
C20H23IN2O2
|
1
|
| 1 |
Ki = 1270 nM
|
|
|
|
CP0431630
|
N-(1,3-benzothiazol-2-yl)naphthalene-1-carboxamide
Show/Hide
|
C18H12N2OS
|
1
|
| 1 |
Ki = 1288 nM
|
|
|
|
CP0375900
|
5-(4-chlorophenyl)-N-[11-[11-[[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carbonyl]amino]undecyl-methylamino]undecyl]-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C57H69Cl6N7O2
|
2
|
| 1 |
Ki = 1292 nM
|
|
|
| 2 |
Ki = 1885 nM
|
|
|
|
CP0376651
|
N-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C21H15Cl3N4O
|
1
|
| 1 |
Ki = 1300 nM
|
|
|
|
CP0382828
|
N-(cyclohexylmethyl)-1,3-benzothiazole-2-carboxamide
Show/Hide
|
C15H18N2OS
|
1
|
| 1 |
Ki = 1324 nM
|
|
|
|
CP0429267
|
methyl 2-(adamantane-1-carbonylamino)-5-propylthiophene-3-carboxylate
Show/Hide
|
C20H27NO3S
|
1
|
| 1 |
Ki = 1339.29 nM
|
|
|
|
CP0455976
|
ethyl 2-(naphthalene-1-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C22H21NO3S
|
1
|
| 1 |
Ki = 1373.03 nM
|
|
|
|
CP0920451
|
(1S,2S)-N-Oleoylcyclopropanolamide
Show/Hide
|
C19H37NO2
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0154028
|
N-[4-(cyclopropylamino)-4-oxobutyl]-9-methyl-6-(oxan-4-yl)-5,6,7,8-tetrahydrocarbazole-3-carboxamide
Show/Hide
|
C26H35N3O3
|
1
|
| 1 |
Ki = 1440 nM
|
|
|
|
CP0515229
|
3-(benzo[d][1,3]dioxol-5-yl)-N-(2-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-2-oxo-1-p-tolylethyl)-N-methylacrylamide
Show/Hide
|
C28H26N2O6
|
1
|
| 1 |
Ki = 1473 nM
|
|
|
|
CP0453372
|
(2S)-1-(4-oxo-1-pentyl-7-phenylsulfanylquinoline-3-carbonyl)pyrrolidine-2-carboxamide
Show/Hide
|
C26H29N3O3S
|
1
|
| 1 |
Ki = 1490 nM
|
|
|
|
CP0379401
|
3-butyl-N-cycloheptyl-2-methoxy-5-(4-methoxyphenyl)benzamide
Show/Hide
|
C26H35NO3
|
1
|
| 1 |
Ki = 1494 nM
|
|
|
|
CP0490554
|
1-(4-(4-chlorophenyl)-5,6-dihydropyridin-1(2H)-yl)-3,3-diphenylpropan-1-one
Show/Hide
|
C26H24ClNO
|
1
|
| 1 |
Ki = 1500 nM
|
|
|
|
CP0429451
|
N-(1-adamantyl)-2-(5-phenyl-1-propylindol-3-yl)acetamide
Show/Hide
|
C29H34N2O
|
1
|
| 1 |
Ki = 1508 nM
|
|
|
|
CP0454196
|
1-benzyl-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
Ki = 1519 nM
|
|
|
|
CP0388919
|
2-methoxy-3-methyl-N-(4-methylcyclohexyl)-5-phenylbenzamide
Show/Hide
|
C22H27NO2
|
1
|
| 1 |
Ki = 1530 nM
|
|
|
|
CP0382821
|
N-(1-adamantyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
Show/Hide
|
C16H22N2OS
|
1
|
| 1 |
Ki = 1530 nM
|
|
|
|
CP0388921
|
3-butyl-2-methoxy-5-(4-methoxyphenyl)-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C26H35NO3
|
1
|
| 1 |
Ki = 1550 nM
|
|
|
|
CP0401724
|
methyl 5-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxypentanoate
Show/Hide
|
C28H33NO6
|
1
|
| 1 |
Ki = 1583 nM
|
|
|
|
CP0498834
|
1-benzyl-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
Ki = 1600 nM
|
|
|
|
CP0372347
|
2-(4-chlorophenyl)-N-(3,3-diphenylpropyl)acetamide
Show/Hide
|
C23H22ClNO
|
1
|
| 1 |
Ki = 1600 nM
|
|
|
|
CP0502192
|
methyl 4-[4-(9H-fluoren-9-yl)piperazin-1-yl]sulfonyl-2,5-dimethylfuran-3-carboxylate
Show/Hide
|
C25H26N2O5S
|
1
|
| 1 |
Ki = 1606 nM
|
|
|
|
CP0443540
|
1-butyl-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C17H26N2O2
|
1
|
| 1 |
Ki = 1623 nM
|
|
|
|
CP0514781
|
N-(1-adamantyl)-2-[5-(furan-2-yl)-1-pentylindol-3-yl]acetamide
Show/Hide
|
C29H36N2O2
|
1
|
| 1 |
Ki = 1660 nM
|
|
|
|
CP0489860
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-1-formylpyrrolidine-2-carboxylate
Show/Hide
|
C28H49NO5
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0415324
|
6-Bromo-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid cyclohexylamide
Show/Hide
|
C21H27BrN2O2
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0506021
|
N-[2,6-di(propan-2-yl)phenyl]-4-[3-[(4-methylphenyl)methyl]-1,2,4-thiadiazol-5-yl]-1,4-diazepane-1-carboxamide
Show/Hide
|
C28H37N5OS
|
1
|
| 1 |
Ki = 1764 nM
|
|
|
|
CP0567079
|
11-(3-hydroxy-5-pentylphenoxy)-N-piperidin-1-ylundecanamide
Show/Hide
|
C27H46N2O3
|
1
|
| 1 |
Ki = 1782 nM
|
|
|
|
CP0558528
|
4-[4-[2-(2,4-dichlorophenyl)-4-methyl-5-(piperidin-1-ylcarbamoyl)pyrazol-3-yl]phenyl]but-3-ynyl 6-aminohexanoate;2,2,2-trifluoroacetic acid
Show/Hide
|
C34H38Cl2F3N5O5
|
1
|
| 1 |
Ki = 1810 nM
|
|
|
|
CP0525975
|
N-cyclohexyl-2-[(4-fluorophenyl)methoxy]pyridine-3-carboxamide
Show/Hide
|
C19H21FN2O2
|
1
|
| 1 |
Ki = 1811 nM
|
|
|
|
CP0536700
|
N-(1-adamantyl)-2-(1-but-3-enyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C30H34N2O
|
1
|
| 1 |
Ki = 1827 nM
|
|
|
|
CP0388258
|
N-cycloheptyl-1-[(3-iodophenyl)methyl]-2-oxopyridine-3-carboxamide
Show/Hide
|
C20H23IN2O2
|
1
|
| 1 |
Ki = 1830 nM
|
|
|
|
CP0456682
|
2-[8-(3-hydroxy-5-pentylphenoxy)octoxy]propane-1,3-diol
Show/Hide
|
C22H38O5
|
1
|
| 1 |
Ki = 1860 nM
|
|
|
|
CP0480041
|
1-methyl-4-oxo-7-phenylsulfanyl-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
|
C27H30N2O2S
|
1
|
| 1 |
Ki = 1866.9 nM
|
|
|
|
CP0487935
|
N-(1,3-dihydroxypropan-2-yl)-11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
|
C29H51NO5
|
1
|
| 1 |
Ki = 1890 nM
|
|
|
|
CP0465926
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] 3-formamidopropanoate
Show/Hide
|
C26H47NO5
|
1
|
| 1 |
Ki = 1900 nM
|
|
|
|
CP0418048
|
2-(4-bromophenyl)-2-phenyl-N-(3-phenylpropyl)acetamide
Show/Hide
|
C23H22BrNO
|
1
|
| 1 |
Ki = 1900 nM
|
|
|
|
CP0401975
|
6-Bromo-4-oxo-1-pentyl-N-(piperidin-1-yl)-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C20H26BrN3O2
|
1
|
| 1 |
Ki = 1900 nM
|
|
|
|
CP0877894
|
8alpha-Hydroxy-Delta9-tetrahydrocannabinol
Show/Hide
|
C21H30O3
|
1
|
| 1 |
Ki = 1906 nM
|
|
|
|
CP0434010
|
N-cycloheptyl-2-phenylmethoxypyridine-3-carboxamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
Ki = 1920 nM
|
|
|
|
CP0452468
|
1-(4-(3-(2,4-dimethoxyphenyl)-1-m-tolyl-1H-pyrazole-5-carbonyl)piperazin-1-yl)ethanone
Show/Hide
|
C25H28N4O4
|
1
|
| 1 |
Ki = 1943 nM
|
|
|
|
CP0400887
|
N-[11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecyl]cyclopropanecarboxamide
Show/Hide
|
C30H51NO3
|
1
|
| 1 |
Ki = 2070 nM
|
|
|
|
CP0195798
|
6-Iodo-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C25H31IN2O2
|
1
|
| 1 |
Ki = 2080 nM
|
|
|
|
CP0379903
|
3-[11-(cyclopropylamino)undecoxy]-5-pentylphenol
Show/Hide
|
C25H43NO2
|
1
|
| 1 |
Ki = 2080 nM
|
|
|
|
CP0427498
|
11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acid[2-(3,4-dihydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C31H47NO5
|
1
|
| 1 |
Ki = 2100 nM
|
|
|
|
CP0528608
|
11-(3-hydroxy-5-pentyl-phenoxy)-undecanoic acid (3-methoxy-4-hydroxy-phenyl)-amide
Show/Hide
|
C30H45NO5
|
1
|
| 1 |
Ki = 2100 nM
|
|
|
|
CP0453829
|
N-(4-chlorophenyl)-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C21H15ClF2N4O
|
1
|
| 1 |
Ki = 2100 nM
|
|
|
|
CP0386406
|
N-(1-adamantyl)-5,8-dimethoxy-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C27H36N2O4
|
1
|
| 1 |
Ki = 2100 nM
|
|
|
|
CP0557475
|
4-[4-[2-(2,4-dichlorophenyl)-4-methyl-5-(piperidin-1-ylcarbamoyl)pyrazol-3-yl]phenyl]but-3-ynyl 11-[(3',6'-dihydroxy-3-oxospiro[2-benzofuran-1,9'-xanthene]-5-carbothioyl)amino]undecanoate
Show/Hide
|
C58H57Cl2N5O8S
|
1
|
| 1 |
Ki = 2110 nM
|
|
|
|
CP0481802
|
methyl 2-(adamantane-1-carbonylamino)-5-ethyl-4-methylthiophene-3-carboxylate
Show/Hide
|
C20H27NO3S
|
1
|
| 1 |
Ki = 2120 nM
|
|
|
|
CP0502229
|
2-(4-chlorophenyl)-2-phenyl-N-(3-phenylpropyl)acetamide
Show/Hide
|
C23H22ClNO
|
1
|
| 1 |
Ki = 2200 nM
|
|
|
|
CP0528142
|
N-(3,3-diphenylpropyl)-2-hydroxy-2,2-diphenylacetamide
Show/Hide
|
C29H27NO2
|
1
|
| 1 |
Ki = 2200 nM
|
|
|
|
CP0507882
|
2-(5-benzyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)-N-isopropylpropanamide
Show/Hide
|
C22H23N5OS
|
1
|
| 1 |
Ki = 2269 nM
|
|
|
|
CP0413292
|
3-butyl-2-methoxy-5-(4-methoxyphenyl)-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C26H35NO3
|
1
|
| 1 |
Ki = 2294 nM
|
|
|
|
CP0888599
|
(3-((2-(4,6-dimorpholino-1,3,5-triazin-2-yl)hydrazono)methyl)-1H-indol-1-yl)(p-tolyl)methanone
Show/Hide
|
C28H30N8O3
|
1
|
| 1 |
Ki = 2299 nM
|
|
|
|
CP0423366
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] 2-acetamidoacetate
Show/Hide
|
C26H47NO5
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0427561
|
4-methyl-2-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-thiazole-5-carboxamide
Show/Hide
|
C21H20N2OS
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0417553
|
1-(4-(2-methoxyphenyl)piperazin-1-yl)-2-(4-phenyl-6-(trifluoromethyl)pyrimidin-2-ylthio)propan-1-one
Show/Hide
|
C25H25F3N4O2S
|
1
|
| 1 |
Ki = 2314 nM
|
|
|
|
CP0418727
|
N,N-dimethyl-8-(4-methylpiperidine-1-carbonyl)-2-(oxan-4-yl)-3,4-dihydro-1H-pyrido[4,3-b]indole-5-carboxamide
Show/Hide
|
C26H36N4O3
|
1
|
| 1 |
Ki = 2380 nM
|
|
|
|
CP0436073
|
N-(1-adamantyl)-2-(1-pentyl-5-phenylindol-3-yl)acetamide
Show/Hide
|
C31H38N2O
|
1
|
| 1 |
Ki = 2380 nM
|
|
|
|
CP0417554
|
2-cyclohexyl-3-(4-methoxyphenyl)-N-(6-methylpyridin-2-yl)-1-oxo-1,2,3,4-tetrahydroisoquinoline-4-carboxamide
Show/Hide
|
C29H31N3O3
|
1
|
| 1 |
Ki = 2396 nM
|
|
|
|
CP0390566
|
N-cyclopentyl-1-(2,4-difluorophenyl)-4-methyl-5-pyrrol-1-ylpyrazole-3-carboxamide
Show/Hide
|
C20H20F2N4O
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0058220
|
(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl (2S)-2-formamido-4-methylpentanoate
Show/Hide
|
C29H53NO5
|
1
|
| 1 |
Ki = 2500 nM
|
|
|
|
CP0139727
|
N-(1-adamantyl)-4-oxo-1-pentyl-6-(trifluoromethyl)quinoline-3-carboxamide
Show/Hide
|
C26H31F3N2O2
|
1
|
| 1 |
Ki = 2520 nM
|
|
|
|
CP0431073
|
N-[2-[4-(4-methoxyphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-N-propan-2-ylcyclohexanecarboxamide
Show/Hide
|
C26H34N2O3S
|
1
|
| 1 |
Ki = 2593 nM
|
|
|
|
CP0433844
|
5-oxo-L-Proline-(1S)-1-[[(2S,3S)-3-hexyl-4-oxo-2-oxetanyl]methyl]dodecyl Ester
Show/Hide
|
C27H47NO5
|
1
|
| 1 |
Ki = 2600 nM
|
|
|
|
CP0446041
|
N-(4-methylcyclohexyl)-2-oxo-1-propylquinoline-3-carboxamide
Show/Hide
|
C20H26N2O2
|
1
|
| 1 |
Ki = 2609 nM
|
|
|
|
CP0395712
|
2,5-dimethyl-1-phenyl-N-(1-phenylethyl)pyrrole-3-carboxamide
Show/Hide
|
C21H22N2O
|
1
|
| 1 |
Ki = 2621.82 nM
|
|
|
|
CP0051463
|
(E)-N-(Adamant-1-yl)-6-[2-(4-methoxyphenyl)vinyl]-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C34H40N2O3
|
1
|
| 1 |
Ki = 2630 nM
|
|
|
|
CP0423081
|
N-(1-adamantyl)-6-bromo-1-but-3-enyl-4-oxoquinoline-3-carboxamide
Show/Hide
|
C24H27BrN2O2
|
1
|
| 1 |
Ki = 2680 nM
|
|
|
|
CP0400439
|
1,3-dihydroxypropan-2-yl 12-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]dodecanoate
Show/Hide
|
C30H52O6
|
1
|
| 1 |
Ki = 2710 nM
|
|
|
|
CP0490716
|
1-benzyl-4-methyl-6-phenyl-3-(phenylsulfonyl)pyridin-2(1H)-one
Show/Hide
|
C25H21NO3S
|
1
|
| 1 |
Ki = 2716 nM
|
|
|
|
CP0484631
|
N-cycloheptyl-5-(4-fluorophenyl)-1-(2-morpholin-4-ylethyl)-2-oxopyridine-3-carboxamide
Show/Hide
|
C25H32FN3O3
|
1
|
| 1 |
Ki = 2734 nM
|
|
|
|
CP0410896
|
N-[11-(3-hydroxy-5-pentylphenoxy)undecyl]cyclopropanecarboxamide
Show/Hide
|
C26H43NO3
|
1
|
| 1 |
Ki = 2770 nM
|
|
|
|
CP0429472
|
2-chloro-N-(2,6-dimethylphenyl)-N-(2-morpholino-2-(4-nitrophenyl)acetyl)benzamide
Show/Hide
|
C27H26ClN3O5
|
1
|
| 1 |
Ki = 2785 nM
|
|
|
|
CP0383647
|
N-(1-adamantyl)-5-(furan-2-yl)-1-prop-2-enylindole-3-carboxamide
Show/Hide
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C26H28N2O2
|
1
|
| 1 |
Ki = 2794 nM
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CP0522362
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5-(2-morpholinoethyl)-2-phenyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one
Show/Hide
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C22H22N4O2
|
1
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| 1 |
Ki = 2800 nM
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CP0444412
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11-(2-hexyl-5-hydroxy-phenoxy)-undecanoic acid(3-methoxy-4-hydroxy-phenyl)-amide
Show/Hide
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C31H47NO5
|
1
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| 1 |
Ki = 2820 nM
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CP0450989
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[5-hydroxy-1-(2-morpholin-4-ylethyl)indol-3-yl]-naphthalen-1-ylmethanone
Show/Hide
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C25H24N2O3
|
1
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| 1 |
Ki = 2838 nM
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CP0382785
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(4-methyl-2-phenyl-1,3-thiazol-5-yl)-morpholin-4-ylmethanone
Show/Hide
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C15H16N2O2S
|
1
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| 1 |
Ki = 2860 nM
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CP0454320
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N-cyclohexyl-7-methoxy-1-(2-morpholin-4-ylethyl)-4-oxoquinoline-3-carboxamide
Show/Hide
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C23H31N3O4
|
1
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| 1 |
Ki = 2920 nM
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CP0492363
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2-[10-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]decoxy]propane-1,3-diol
Show/Hide
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C28H50O5
|
1
|
| 1 |
Ki = 2940 nM
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CP0520162
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(8-iodonaphthalen-1-yl)-(1-propylindol-3-yl)methanone
Show/Hide
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C22H18INO
|
1
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| 1 |
Ki = 2960 nM
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CP0395644
|
N-(4-methylcyclohexyl)-2-phenylmethoxypyridine-3-carboxamide
Show/Hide
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C20H24N2O2
|
1
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| 1 |
Ki = 3093 nM
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CP0485042
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[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-formamidopropanoate
Show/Hide
|
C26H47NO5
|
1
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| 1 |
Ki = 3100 nM
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CP0550756
|
N-(2-hydroxyethyl)-11-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
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C29H51NO4
|
1
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| 1 |
Ki = 3157 nM
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CP0469874
|
N-(cyclopropylmethyl)-11-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
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C31H53NO3
|
1
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| 1 |
Ki = 3193.5 nM
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CP0051324
|
6-Bromo-4-oxo-1-prop-2-ynyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
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C23H23BrN2O2
|
1
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| 1 |
Ki = 3210 nM
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CP0516621
|
N-(cyclopropylmethyl)-11-(4-hexyl-3-methoxyphenoxy)undecanamide
Show/Hide
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C28H47NO3
|
1
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| 1 |
Ki = 3250 nM
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CP0372351
|
2,2-diphenyl-N-(3-phenylpropyl)acetamide
Show/Hide
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C23H23NO
|
1
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| 1 |
Ki = 3400 nM
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CP0500720
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1-ethenyl-7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C22H25FN2O2
|
1
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| 1 |
Ki = 3572.6 nM
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CP0434997
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N-(1-adamantyl)-2-[5-(furan-2-yl)-1-prop-2-enylindol-3-yl]-2-oxoacetamide
Show/Hide
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C27H28N2O3
|
1
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| 1 |
Ki = 3617 nM
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CP0435085
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N-(1-adamantyl)-1-pentyl-5-thiophen-2-ylindole-3-carboxamide
Show/Hide
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C28H34N2OS
|
1
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| 1 |
Ki = 3621 nM
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CP0395713
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2-ethyl-5-methyl-1-phenyl-N-(1-phenylethyl)pyrrole-3-carboxamide
Show/Hide
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C22H24N2O
|
1
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| 1 |
Ki = 3736.7 nM
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CP0499114
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1-(3-hydroxypropyl)-N-(4-methylcyclohexyl)-2-oxoquinoline-3-carboxamide
Show/Hide
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C20H26N2O3
|
1
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| 1 |
Ki = 3761 nM
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CP0418898
|
2-[12-(3-hydroxy-5-pentylphenoxy)dodecoxy]propane-1,3-diol
Show/Hide
|
C26H46O5
|
1
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| 1 |
Ki = 3780 nM
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CP0502917
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N-(1-adamantyl)-2-oxo-2-(5-phenyl-1-prop-2-enylindol-3-yl)acetamide
Show/Hide
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C29H30N2O2
|
1
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| 1 |
Ki = 3915 nM
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CP0394387
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N-[6-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxyhexyl]acetamide
Show/Hide
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C30H38N2O5
|
1
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| 1 |
Ki = 3918 nM
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CP0439368
|
4-(8-benzyl-5-cyano-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-N-propylpiperazine-1-carboxamide
Show/Hide
|
C26H33N5O2
|
1
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| 1 |
Ki = 3949 nM
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CP0488645
|
(8-iodonaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone
Show/Hide
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C23H20INO
|
1
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| 1 |
Ki = 4290 nM
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CP0078199
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(4-methoxyphenyl)-[1-(oxan-4-ylmethyl)-5-propoxyindol-3-yl]methanone
Show/Hide
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C25H29NO4
|
1
|
| 1 |
Ki = 4527 nM
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CP0446146
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N-cyclohexyl-2-ethyl-5-methyl-1-phenylpyrrole-3-carboxamide
Show/Hide
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C20H26N2O
|
1
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| 1 |
Ki = 4571.51 nM
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CP0454197
|
1-benzyl-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C23H25N3O2
|
1
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| 1 |
Ki = 5255 nM
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CP0542425
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N-(1-adamantyl)-2-(5-bromo-1-pentylindol-3-yl)acetamide
Show/Hide
|
C25H33BrN2O
|
1
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| 1 |
Ki = 5510 nM
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CP0498835
|
1-butyl-N-cyclohexyl-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C19H25N3O2
|
1
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| 1 |
Ki = 5600 nM
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CP0501752
|
7-amino-1-benzyl-N-cyclohexyl-4-oxo-1,4-dihydro-1,8-naphthyridine-2-carboxamide
Show/Hide
|
C22H24N4O2
|
1
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| 1 |
Ki = 5600 nM
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CP0394718
|
1,3-dihydroxypropan-2-yl 8-(3-hydroxy-5-pentylphenoxy)octanoate
Show/Hide
|
C22H36O6
|
1
|
| 1 |
Ki = 5600 nM
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CP0467435
|
1,3-dihydroxypropan-2-yl 11-(3-hydroxy-5-pentylphenoxy)undecanoate
Show/Hide
|
C25H42O6
|
1
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| 1 |
Ki = 5600 nM
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CP0433616
|
(6aR,9S,10S,10aR)-6,6,9-trimethyl-3-pentyl-7,8,10,10a-tetrahydro-6aH-benzo[c]chromene-1,9,10-triol
Show/Hide
|
C21H32O4
|
1
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| 1 |
Ki = 5668 nM
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CP0439729
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-formamido-3-methylbutanoate
Show/Hide
|
C28H51NO5
|
1
|
| 1 |
Ki = 5700 nM
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CP0395707
|
2,5-dimethyl-1-phenyl-N-(2-phenylethyl)pyrrole-3-carboxamide
Show/Hide
|
C21H22N2O
|
1
|
| 1 |
Ki = 5926.7 nM
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CP0423365
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-formamido-3-methylpentanoate
Show/Hide
|
C29H53NO5
|
1
|
| 1 |
Ki = 6000 nM
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CP0498833
|
1-benzyl-N-[2-(4-fluorophenyl)ethyl]-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C24H20FN3O2
|
1
|
| 1 |
Ki = 6947 nM
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CP0490717
|
3-(4-tert-butylbenzoyl)-2-(3-fluorophenyl)-N-(pyridin-2-ylmethyl)thiazolidine-4-carboxamide
Show/Hide
|
C27H28FN3O2S
|
1
|
| 1 |
Ki = 7490 nM
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CP0506288
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-acetamido-3-methylbutanoate
Show/Hide
|
C29H53NO5
|
1
|
| 1 |
Ki = 8400 nM
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CP0511846
|
[(2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-2-yl] (2S)-2-acetamido-3-methylpentanoate
Show/Hide
|
C30H55NO5
|
1
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| 1 |
Ki = 8600 nM
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CP0049976
|
(6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methylnon-6-enamide
Show/Hide
|
C18H27NO3
|
1
|
| 1 |
Ki > 10000 nM
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CP0395030
|
cyclopropanolamide, rac-10c
Show/Hide
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C19H37NO2
|
1
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| 1 |
Ki > 10000 nM
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CP0493725
|
cyclopropanolamide, rac-9c
Show/Hide
|
C19H37NO2
|
1
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| 1 |
Ki > 10000 nM
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CP0485066
|
(1R)-1-{[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]methyl}dodecyl N-formylglycinate
Show/Hide
|
C25H45NO5
|
1
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| 1 |
Ki > 10000 nM
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CP0408018
|
4-(benzyloxy)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole
Show/Hide
|
C29H35NO3
|
1
|
| 1 |
Ki > 10000 nM
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CP0506262
|
1-(2-Bromophenyl)-5-(4-methoxyphenyl)-N3-(piperidin-1-yl)-1H-pyrazole-3,4-dicarboxamide
Show/Hide
|
C23H24BrN5O3
|
1
|
| 1 |
Ki > 10000 nM
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CP0195828
|
N-(1-adamantyl)-4-oxo-1-pentyl-6-phenylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0436994
|
N-(1-adamantyl)-7-chloro-8-methyl-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C26H33ClN2O2
|
1
|
| 1 |
Ki > 10000 nM
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CP0436999
|
N-(1-adamantyl)-5,8-dimethoxy-4-oxo-1-prop-2-enylquinoline-3-carboxamide
Show/Hide
|
C25H30N2O4
|
1
|
| 1 |
Ki > 10000 nM
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CP0048140
|
N-(1-adamantyl)-6-(furan-2-yl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C29H34N2O3
|
1
|
| 1 |
Ki > 10000 nM
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CP0054395
|
6-(4-Cyano-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C32H35N3O2
|
1
|
| 1 |
Ki > 10000 nM
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CP0054397
|
1-But-3-enyl-6-furan-2-yl-4-oxo-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C28H30N2O3
|
1
|
| 1 |
Ki > 10000 nM
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CP0085407
|
6-(4-Hydroxy-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylicacid adamantan-1-ylamide
Show/Hide
|
C31H36N2O3
|
1
|
| 1 |
Ki > 10000 nM
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CP0102143
|
6-(2,4-Difluoro-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H34F2N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0102144
|
6-(5-Chloro-thiophen-2-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C29H33ClN2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0102146
|
6-Cyclohexyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H42N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0102216
|
N-(1-adamantyl)-4-oxo-1-pentyl-6-(2-phenylethynyl)quinoline-3-carboxamide
Show/Hide
|
C33H36N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0103197
|
N-(1-adamantyl)-6-imidazol-1-yl-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C28H34N4O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0190974
|
6-(2-Ethyl-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C33H40N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0195800
|
4-Oxo-1-pentyl-6-thiophen-2-yl-1,4-dihydro-quinoline-3-carboxylic acidadamantan-1-ylamide
Show/Hide
|
C29H34N2O2S
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0225272
|
6-Cyclohex-1-enyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H40N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0257793
|
6-(2,4-Dichloro-benzyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C32H36Cl2N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0281047
|
N-(1-adamantyl)-6-ethynyl-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C27H32N2O2
|
1
|
| 1 |
Ki > 10000 nM
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CP0292304
|
6-Biphenyl-4-yl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acidadamantan-1-ylamide
Show/Hide
|
C37H40N2O2
|
1
|
| 1 |
Ki > 10000 nM
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CP0313817
|
6-(4-Chloro-phenyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H35ClN2O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0398771
|
1-Allyl-6-furan-2-yl-4-oxo-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C27H28N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0401971
|
6-(6-Methoxy-pyridin-3-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H37N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0402075
|
N-(1-adamantyl)-6-(benzenesulfonyl)-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C31H36N2O4S
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0406215
|
(E)-N-(Adamantan-1-yl)-4-oxo-1-pentyl-6-styryl-1,4-dihydroquinoline-3-carboxamide
Show/Hide
|
C33H38N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
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CP0418513
|
6-(3,5-Dimethyl-isoxazol-4-yl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C30H37N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
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CP0493047
|
6-((E)-3,3-Dimethyl-but-1-enyl)-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C31H42N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
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CP0051827
|
8-Methyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic acid adamantan-1-ylamide
Show/Hide
|
C26H34N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0376756
|
N-(1-adamantyl)-8-methoxy-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C21H24N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0396892
|
N-(1-adamantyl)-2-butyl-6-(furan-2-yl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C28H32N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0425469
|
N-(1-adamantyl)-6-(furan-2-yl)-8-methoxy-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C30H36N2O4
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0428319
|
N-(1-adamantyl)-6-bromo-8-methoxy-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C26H33BrN2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0471599
|
N-(1-adamantyl)-8-methoxy-4-oxo-1-pentyl-6-phenylquinoline-3-carboxamide
Show/Hide
|
C32H38N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0471601
|
N-(1-adamantyl)-6-bromo-4-hydroxy-2-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C25H31BrN2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0480579
|
N-(1-adamantyl)-8-methoxy-4-oxo-1-pentylquinoline-3-carboxamide
Show/Hide
|
C26H34N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0498367
|
N-(1-adamantyl)-6-bromo-2-butyl-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C24H29BrN2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0506638
|
N-(1-adamantyl)-4-oxo-8-phenyl-1H-quinoline-3-carboxamide
Show/Hide
|
C26H26N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0459053
|
1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-5-(2,5-diethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C26H24Cl4N4O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0400477
|
2-[6-(4-hexyl-3-hydroxyphenoxy)hexoxy]propane-1,3-diol
Show/Hide
|
C21H36O5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0418896
|
2,3-dihydroxypropyl 11-(3-hydroxy-5-pentylphenoxy)undecanoate
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C25H42O6
|
1
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| 1 |
Ki > 10000 nM
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CP0418897
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2-[10-(3-hydroxy-5-pentylphenoxy)decoxy]propane-1,3-diol
Show/Hide
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C24H42O5
|
1
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| 1 |
Ki > 10000 nM
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CP0418899
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2,3-dihydroxypropyl 11-(4-hexyl-3-hydroxyphenoxy)undecanoate
Show/Hide
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C26H44O6
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1
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| 1 |
Ki > 10000 nM
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CP0428008
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1,3-dihydroxypropan-2-yl 8-(4-hexyl-3-hydroxyphenoxy)octanoate
Show/Hide
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C23H38O6
|
1
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| 1 |
Ki > 10000 nM
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CP0432794
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2-[10-(4-hexyl-3-hydroxyphenoxy)decoxy]propane-1,3-diol
Show/Hide
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C25H44O5
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1
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| 1 |
Ki > 10000 nM
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CP0440291
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1,3-dihydroxypropan-2-yl 11-(4-hexyl-3-hydroxyphenoxy)undecanoate
Show/Hide
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C26H44O6
|
1
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| 1 |
Ki > 10000 nM
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CP0461991
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2,3-dihydroxypropyl 11-(2-hexyl-5-hydroxyphenoxy)undecanoate
Show/Hide
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C26H44O6
|
1
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| 1 |
Ki > 10000 nM
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CP0461992
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2,3-dihydroxypropyl 11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecanoate
Show/Hide
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C29H50O6
|
1
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| 1 |
Ki > 10000 nM
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CP0438030
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(2S)-3-hydroxy-2-[[(5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoyl]amino]propanoic acid
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C23H37NO4
|
1
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| 1 |
Ki > 10000 nM
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CP0432133
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N-cyclohexyl-2-phenylmethoxypyridine-3-carboxamide
Show/Hide
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C19H22N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0432136
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N-cyclohexyl-1-(2-morpholin-4-ylethyl)-2-oxopyridine-3-carboxamide
Show/Hide
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C18H27N3O3
|
1
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| 1 |
Ki > 10000 nM
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CP0383283
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N-(1-adamantyl)-2-(5-bromo-1-prop-2-enylindol-3-yl)acetamide
Show/Hide
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C23H27BrN2O
|
1
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| 1 |
Ki > 10000 nM
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CP0412556
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N-cyclohexyl-2-[5-[(3-methoxyphenyl)methoxy]-1-prop-2-enylindol-3-yl]acetamide
Show/Hide
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C27H32N2O3
|
1
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| 1 |
Ki > 10000 nM
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CP0416199
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N-(1-adamantyl)-5-(4-hydroxyphenyl)-1-prop-2-enylindole-3-carboxamide
Show/Hide
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C28H30N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0424026
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N-(1-adamantyl)-2-(1-benzyl-5-phenylindol-3-yl)acetamide
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C33H34N2O
|
1
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| 1 |
Ki > 10000 nM
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CP0434998
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N-(1-adamantyl)-2-(1-butyl-5-phenylindol-3-yl)acetamide
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C30H36N2O
|
1
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| 1 |
Ki > 10000 nM
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CP0436076
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N-(1-adamantyl)-2-oxo-2-(1-pentyl-5-phenylindol-3-yl)acetamide
Show/Hide
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C31H36N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0514782
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N-cycloheptyl-2-[5-(furan-2-yl)-1-prop-2-enylindol-3-yl]acetamide
Show/Hide
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C24H28N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0525904
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N-(1-adamantyl)-2-(5-phenyl-1H-indol-3-yl)acetamide
Show/Hide
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C26H28N2O
|
1
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| 1 |
Ki > 10000 nM
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CP0548881
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N-cyclohexyl-2-oxo-2-(1-pentyl-5-phenylindol-3-yl)acetamide
Show/Hide
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C27H32N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0404951
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4-oxo-7-phenylsulfanyl-1-(4-phenylsulfanylbutyl)-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C36H40N2O2S2
|
1
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| 1 |
Ki > 10000 nM
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CP0404952
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1-(4-chlorophenyl)-7-fluoro-4-oxo-N-piperidin-1-ylquinoline-3-carboxamide
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C21H19ClFN3O2
|
1
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| 1 |
Ki > 10000 nM
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CP0453384
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7-fluoro-1-[(3-methylphenyl)methyl]-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C28H31FN2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0455325
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7-fluoro-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]-1H-quinoline-3-carboxamide
Show/Hide
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C20H23FN2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0498312
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7-fluoro-1-methyl-4-oxo-N-[(1R,2S)-1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl]quinoline-3-carboxamide
Show/Hide
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C21H25FN2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0525501
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1-(4-fluorophenyl)-4-oxo-7-phenylsulfanyl-N-piperidin-1-ylquinoline-3-carboxamide
Show/Hide
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C27H24FN3O2S
|
1
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| 1 |
Ki > 10000 nM
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CP0447490
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(8-bromonaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone
Show/Hide
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C23H20BrNO
|
1
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| 1 |
Ki > 10000 nM
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CP0488644
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(8-chloronaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone
Show/Hide
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C23H20ClNO
|
1
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| 1 |
Ki > 10000 nM
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CP0511003
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(8-bromonaphthalen-1-yl)-(1-propylindol-3-yl)methanone
Show/Hide
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C22H18BrNO
|
1
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| 1 |
Ki > 10000 nM
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CP0395642
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ethyl 4-[3-(cycloheptylcarbamoyl)-2-oxopyridin-1-yl]butanoate
Show/Hide
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C19H28N2O4
|
1
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| 1 |
Ki > 10000 nM
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CP0395643
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5-bromo-2-butoxy-N-cycloheptylpyridine-3-carboxamide
Show/Hide
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C17H25BrN2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0395645
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1-(2-hydroxyethyl)-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
Show/Hide
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C15H22N2O3
|
1
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| 1 |
Ki > 10000 nM
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CP0435742
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N-(4-methylcyclohexyl)-2-oxo-1-propylpyridine-3-carboxamide
Show/Hide
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C16H24N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0435743
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4-[3-(cycloheptylcarbamoyl)-2-oxopyridin-1-yl]butanoic acid
Show/Hide
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C17H24N2O4
|
1
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| 1 |
Ki > 10000 nM
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CP0481037
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1-(3-hydroxypropyl)-N-(4-methylcyclohexyl)-2-oxopyridine-3-carboxamide
Show/Hide
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C16H24N2O3
|
1
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| 1 |
Ki > 10000 nM
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CP0385040
|
11-(3-hydroxy-5-pentylphenoxy)-N-phenylundecanamide
Show/Hide
|
C28H41NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0410861
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N-[11-(4-hexyl-3-hydroxyphenoxy)undecyl]cyclopropanecarboxamide
Show/Hide
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C27H45NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0410863
|
N-benzyl-11-(3-hydroxy-5-pentylphenoxy)undecanamide
Show/Hide
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C29H43NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0411873
|
N-(1-adamantyl)-11-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
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C36H59NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0445847
|
N-(1,3-dihydroxypropan-2-yl)-11-(2-hexyl-5-hydroxyphenoxy)undecanamide
Show/Hide
|
C26H45NO5
|
1
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| 1 |
Ki > 10000 nM
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CP0494535
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N-(1,3-dihydroxypropan-2-yl)-11-(4-hexyl-3-hydroxyphenoxy)undecanamide
Show/Hide
|
C26H45NO5
|
1
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| 1 |
Ki > 10000 nM
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CP0543214
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N-(1-adamantyl)-11-(3-hydroxy-5-pentylphenoxy)undecanamide
Show/Hide
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C32H51NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0555102
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N-(1-adamantyl)-8-[3-hydroxy-5-(2-methyloctan-2-yl)phenoxy]octanamide
Show/Hide
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C33H53NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0555103
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N-(1,3-dihydroxypropan-2-yl)-11-(3-hydroxy-5-pentylphenoxy)undecanamide
Show/Hide
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C25H43NO5
|
1
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| 1 |
Ki > 10000 nM
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CP0555105
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N-(1-adamantyl)-11-(4-hexyl-3-hydroxyphenoxy)undecanamide
Show/Hide
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C33H53NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0556362
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N-(1-adamantyl)-11-(2-hexyl-3-hydroxyphenoxy)undecanamide
Show/Hide
|
C33H53NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0419212
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N-cycloheptyl-2-methoxy-5-(4-methoxyphenyl)-3-methylbenzamide
Show/Hide
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C23H29NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0444875
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2-methoxy-5-(4-methoxyphenyl)-3-methyl-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C23H29NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0481742
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2-methoxy-5-(4-methoxyphenyl)-3-methyl-N-(4-methylcyclohexyl)benzamide
Show/Hide
|
C23H29NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0499726
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4-hydroxy-1-(3-hydroxypropyl)-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
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C19H25N3O4
|
1
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| 1 |
Ki > 10000 nM
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CP0085437
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(3-benzyl-3-methyl-2,3-dihydrobenzofuran-6-yl)(piperidin-1-yl)methanone
Show/Hide
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C22H25NO2
|
1
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| 1 |
Ki > 10000 nM
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CP0163467
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ethyl 2-amino-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C11H15NO2S
|
1
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| 1 |
Ki > 10000 nM
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CP0395709
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ethyl 2-(naphthalene-1-carbonylamino)-5-phenylthiophene-3-carboxylate
Show/Hide
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C24H19NO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0395710
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ethyl 2-(methanesulfonamido)-5-phenylthiophene-3-carboxylate
Show/Hide
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C14H15NO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0395714
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ethyl 2-(naphthalene-2-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C22H21NO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0400947
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ethyl 2-(3-phenylpropanoylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C20H23NO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0400948
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ethyl 2-[bis(naphthalen-2-ylsulfonyl)amino]-5-phenylthiophene-3-carboxylate
Show/Hide
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C33H25NO6S3
|
1
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| 1 |
Ki > 10000 nM
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CP0400949
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2-ethyl-5-methyl-1-phenyl-N-(2-phenylethyl)pyrrole-3-carboxamide
Show/Hide
|
C22H24N2O
|
1
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| 1 |
Ki > 10000 nM
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CP0400950
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N-cyclohexyl-2,5-dimethyl-1-phenylpyrrole-3-carboxamide
Show/Hide
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C19H24N2O
|
1
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| 1 |
Ki > 10000 nM
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CP0400952
|
ethyl 2-(naphthalene-2-carbonylamino)-5-phenylthiophene-3-carboxylate
Show/Hide
|
C24H19NO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0424492
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ethyl 2-(benzenesulfonamido)-5-phenylthiophene-3-carboxylate
Show/Hide
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C19H17NO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0446044
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ethyl 2-(methanesulfonamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C12H17NO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0446052
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ethyl 2-(naphthalen-1-ylsulfonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C21H21NO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0446147
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2,5-dimethyl-1-phenylpyrrole-3-carboxylic acid
Show/Hide
|
C13H13NO2
|
1
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| 1 |
Ki > 10000 nM
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CP0446148
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ethyl 2-(naphthalen-2-ylsulfonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C21H21NO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0446149
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ethyl 2-[(4-chlorophenyl)sulfonylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C17H18ClNO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0455958
|
ethyl 2-[(4-chlorophenyl)sulfonylamino]-5-phenylthiophene-3-carboxylate
Show/Hide
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C19H16ClNO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0477627
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2-ethyl-5-methyl-1-phenylpyrrole-3-carboxylic acid
Show/Hide
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C14H15NO2
|
1
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| 1 |
Ki > 10000 nM
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CP0514481
|
ethyl 2-(naphthalen-1-ylsulfonylamino)-5-phenylthiophene-3-carboxylate
Show/Hide
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C23H19NO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0518083
|
ethyl 2-(benzenesulfonamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C17H19NO4S2
|
1
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| 1 |
Ki > 10000 nM
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CP0392261
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2-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxyacetic acid
Show/Hide
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C24H25NO6
|
1
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| 1 |
Ki > 10000 nM
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CP0401718
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2-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-5-yl]oxyacetic acid
Show/Hide
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C24H25NO6
|
1
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| 1 |
Ki > 10000 nM
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CP0401726
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N-[2-[2-(2-acetamidoethoxy)ethoxy]ethyl]-5-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxypentanamide
Show/Hide
|
C35H47N3O8
|
1
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| 1 |
Ki > 10000 nM
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CP0405460
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5-[3-(4-methoxybenzoyl)-1-(oxan-4-ylmethyl)indol-7-yl]oxypentanoic acid
Show/Hide
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C27H31NO6
|
1
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| 1 |
Ki > 10000 nM
|
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CP0457571
|
cyclohexyl-[5-hydroxy-1-(2-morpholin-4-ylethyl)indol-3-yl]methanone
Show/Hide
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C21H28N2O3
|
1
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| 1 |
Ki > 10000 nM
|
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CP0458125
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2-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyacetic acid
Show/Hide
|
C24H26N2O6
|
1
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| 1 |
Ki > 10000 nM
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CP0469353
|
[5-hydroxy-1-(2-morpholin-4-ylethyl)indol-3-yl]-(4-methoxyphenyl)methanone
Show/Hide
|
C22H24N2O4
|
1
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| 1 |
Ki > 10000 nM
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CP0494059
|
2-[1-(2-morpholin-4-ylethyl)-3-(naphthalene-1-carbonyl)indol-5-yl]oxyacetic acid
Show/Hide
|
C27H26N2O5
|
1
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| 1 |
Ki > 10000 nM
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CP0517908
|
6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]-N-[2-[2-[2-[5-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxypentanoylamino]ethoxy]ethoxy]ethyl]hexanamide
Show/Hide
|
C62H72BF2N7O10S
|
1
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| 1 |
Ki > 10000 nM
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CP0536539
|
N-[2-[2-[2-[6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]hexanoylamino]ethoxy]ethoxy]ethyl]-7-[3-(4-methoxybenzoyl)-1-(2-morpholin-4-ylethyl)indol-5-yl]oxyheptanamide
Show/Hide
|
C64H76BF2N7O10S
|
1
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| 1 |
Ki > 10000 nM
|
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CP0386988
|
methyl 2-(adamantane-1-carbonylamino)-5-phenylthiophene-3-carboxylate
Show/Hide
|
C23H25NO3S
|
1
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| 1 |
Ki > 10000 nM
|
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CP0386990
|
methyl 2-[(4-chlorobenzoyl)amino]-4-ethyl-5-methylthiophene-3-carboxylate
Show/Hide
|
C16H16ClNO3S
|
1
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| 1 |
Ki > 10000 nM
|
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CP0386992
|
methyl 4-(adamantane-1-carbonylamino)-1-methylpyrazole-3-carboxylate
Show/Hide
|
C17H23N3O3
|
1
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| 1 |
Ki > 10000 nM
|
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CP0386993
|
methyl 2-(adamantane-1-carbonylamino)pyridine-3-carboxylate
Show/Hide
|
C18H22N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
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CP0394001
|
methyl 3-(adamantane-1-carbonylamino)-1H-pyrrole-2-carboxylate
Show/Hide
|
C17H22N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
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CP0394003
|
methyl 2-(adamantane-1-carbonylamino)-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
Show/Hide
|
C20H25NO3S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
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CP0394005
|
methyl 2-(adamantane-1-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
|
C21H27NO3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0425248
|
methyl 2-(piperidine-1-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C16H22N2O3S
|
1
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| 1 |
Ki > 10000 nM
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CP0425249
|
methyl 2-(morpholine-4-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C15H20N2O4S
|
1
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| 1 |
Ki > 10000 nM
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CP0425250
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methyl 2-(adamantane-1-carbonylamino)-4-phenylthiophene-3-carboxylate
Show/Hide
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C23H25NO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0425251
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methyl 4-ethyl-2-[(4-fluorobenzoyl)amino]-5-methylthiophene-3-carboxylate
Show/Hide
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C16H16FNO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0425252
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methyl 2-(adamantane-1-carbonylamino)thiophene-3-carboxylate
Show/Hide
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C17H21NO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0425253
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methyl 2-(adamantane-1-carbonylamino)-4,5-dimethylthiophene-3-carboxylate
Show/Hide
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C19H25NO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0429266
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methyl 5-(adamantane-1-carbonylamino)-3-methyl-1,2-oxazole-4-carboxylate
Show/Hide
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C17H22N2O4
|
1
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| 1 |
Ki > 10000 nM
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CP0466696
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methyl 2-(adamantane-1-carbonylamino)-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
Show/Hide
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C20H25NO5S2
|
1
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| 1 |
Ki > 10000 nM
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CP0479032
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methyl 2-(1-adamantylcarbamoylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C21H28N2O3S
|
1
|
| 1 |
Ki > 10000 nM
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CP0482759
|
methyl 2-(adamantane-1-carbonylamino)-5-methylthiophene-3-carboxylate
Show/Hide
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C18H23NO3S
|
1
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| 1 |
Ki > 10000 nM
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CP0482760
|
methyl 2-(phenoxycarbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
Show/Hide
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C17H17NO4S
|
1
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| 1 |
Ki > 10000 nM
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CP0482765
|
methyl 4-(adamantane-1-carbonylamino)-2-methylpyrazole-3-carboxylate
Show/Hide
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C17H23N3O3
|
1
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| 1 |
Ki > 10000 nM
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CP0382754
|
N-hexyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C17H22N2OS
|
1
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| 1 |
Ki > 10000 nM
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CP0382755
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N-cyclopentyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C16H18N2OS
|
1
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| 1 |
Ki > 10000 nM
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CP0382756
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N-benzyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H16N2OS
|
1
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| 1 |
Ki > 10000 nM
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CP0382757
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N-[(2-fluorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H15FN2OS
|
1
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| 1 |
Ki > 10000 nM
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CP0382758
|
N-benzyl-1,3-benzothiazole-2-carboxamide
Show/Hide
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C15H12N2OS
|
1
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| 1 |
Ki > 10000 nM
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|
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CP0382759
|
N-(1,3-benzothiazol-2-yl)-4-(trifluoromethyl)benzamide
Show/Hide
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C15H9F3N2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
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CP0382778
|
N-naphthalen-1-yl-1,3-benzothiazole-2-carboxamide
Show/Hide
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C18H12N2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0382781
|
N-cyclopropyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C14H14N2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0382820
|
N-(cyclohexylmethyl)-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H22N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0382822
|
N-butyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C15H18N2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0382823
|
N-[(4-fluorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H15FN2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0382827
|
N-benzyl-2,4-dimethyl-1,3-thiazole-5-carboxamide
Show/Hide
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C13H14N2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0427553
|
N-cyclohexyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C17H20N2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0427555
|
N-[(2-chlorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
Show/Hide
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C18H15ClN2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0427556
|
N-naphthalen-2-yl-1,3-benzothiazole-2-carboxamide
Show/Hide
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C18H12N2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0431627
|
N-(1,3-benzothiazol-2-yl)-3-(trifluoromethyl)benzamide
Show/Hide
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C15H9F3N2OS
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0870378
|
2-(2-((1H-benzo[d][1,2,3]triazol-1-yl)methyl)-5-methyl-1H-benzo[d]imidazol-1-yl)-N,N-dimethylethanamine
Show/Hide
|
C19H22N6
|
1
|
| 1 |
Ki > 10000 nM
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|
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CP0877580
|
1-(1-(2-(diethylamino)ethyl)-2-(4-methoxybenzyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
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C23H29N3O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0879200
|
1-Butyl-2-(3,4-dichlorobenzyl)-5-trifluoromethylbenzimidazole
Show/Hide
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C19H17Cl2F3N2
|
1
|
| 1 |
Ki = 10000 nM
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|
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CP0879201
|
(1S,9aR)-1-((2-(4-methoxybenzyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)methyl)octahydro-1H-quinolizine
Show/Hide
|
C26H30F3N3O
|
1
|
| 1 |
Ki > 10000 nM
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|
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CP0902321
|
N,N-diethyl-3-(2-(4-methoxybenzyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)propan-1-amine
Show/Hide
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C23H28F3N3O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0902322
|
5-acetyl-1-(2-diethylaminoethyl)-2-(4-ethoxybenzyl)benzimidazole
Show/Hide
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C24H31N3O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0902323
|
N,N-diethyl-2-(2-(4-methoxyphenyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)ethanamine
Show/Hide
|
C21H24F3N3O
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0902324
|
1-[2-(Diethylamino)ethyl]-2-(4-ethoxybenzyl)-5-(1-hydrazonoethyl)-1H-benzimidazole
Show/Hide
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C24H33N5O
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0902325
|
N,N-diethyl-2-(2-(4-methoxybenzyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)ethanamine
Show/Hide
|
C22H26F3N3O
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0902326
|
2-[(3,4-Dichloro)benzyl]-1-[(2-dimethylamino)ethyl]-5-trifluoromethylbenzimidazole
Show/Hide
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C19H18Cl2F3N3
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0902327
|
1-(2-((2H-benzo[d][1,2,3]triazol-2-yl)methyl)-1-(3-(diethylamino)propyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
|
C23H28N6O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0905762
|
2-(2-benzyl-5-(trifluoromethyl)-1H-benzo[d]imidazol-1-yl)-N,N-diethylethanamine
Show/Hide
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C21H24F3N3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0905763
|
(1S,9aR)-1-(2-(2-((2H-benzo[d][1,2,3]triazol-2-yl)methyl)-5-chloro-1H-benzo[d]imidazol-1-yl)ethyl)octahydro-1H-quinolizine
Show/Hide
|
C25H29ClN6
|
1
|
| 1 |
Ki > 10000 nM
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|
|
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CP0905764
|
1-(2-((1H-benzo[d][1,2,3]triazol-1-yl)methyl)-1-(2-(diethylamino)ethyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
|
C22H26N6O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0929327
|
1-(2-(4-methoxybenzyl)-1-(((1S,9aR)-octahydro-1H-quinolizin-1-yl)methyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
|
C27H33N3O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0929328
|
2-(3,4-Dichlorobenzyl)-1-[(2-methoxy)ethyl]-5-trifluoromethylbenzimidazole
Show/Hide
|
C18H15Cl2F3N2O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0942687
|
1-(2-(4-chlorobenzyl)-1-(2-(diethylamino)ethyl)-1H-benzo[d]imidazol-5-yl)ethanone
Show/Hide
|
C22H26ClN3O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0943932
|
1-(2-diethylaminoethyl)-2-(4-ethoxybenzyl)-5-trifluoromethylbenzimidazole
Show/Hide
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C23H28F3N3O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0548838
|
N-(1,3-dihydroxypropan-2-yl)-11-[3-methoxy-5-(2-methyloctan-2-yl)phenoxy]undecanamide
Show/Hide
|
C30H53NO5
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0039728
|
2-fluorophenyl N-[6-(2-methyl-4,5-diphenyl-1H-imidazol-1-yl)hexyl]carbamate
Show/Hide
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C29H30FN3O2
|
1
|
| 1 |
Ki = 23000 nM
|
|
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CP0428048
|
4-[6-fluoro-2,2-bis-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-ylmethyl]-morpholine
Show/Hide
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C24H20F3NO3
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
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CP0085567
|
1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-5-amine
Show/Hide
|
C22H30N2O2
|
1
|
| 1 |
Ki > 1000 nM
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|
|
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CP0398722
|
(3',5'-dichloro-2-hydroxy-6-methoxybiphenyl-4-yl)(phenyl)methanone
Show/Hide
|
C20H14Cl2O3
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0517506
|
(3',5'-dichloro-2,6-dimethoxybiphenyl-4-yl)(phenyl)methanol
Show/Hide
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C21H18Cl2O3
|
1
|
| 1 |
Ki > 1000 nM
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|
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CP0441132
|
1-(2,4-Dichlorophenyl)-4-cyano-5-(4-bromophenyl)-N-morpholino-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H16BrCl2N5O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
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CP0420323
|
2-[6-(1-adamantylcarbamoyl)-7-hydroxy-5-oxo-4-propylpyrazolo[4,3-b]pyridin-2-yl]ethyl acetate
Show/Hide
|
C24H32N4O5
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0423778
|
N-(1-adamantyl)-4-butyl-7-hydroxy-2-(2-hydroxyethyl)-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C23H32N4O4
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
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CP0516605
|
N-(1-adamantyl)-4-butyl-7-hydroxy-1-(2-hydroxyethyl)-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C23H32N4O4
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
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CP0516608
|
N-(1-adamantyl)-7-hydroxy-4-(4-hydroxybutyl)-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H30N4O4
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
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CP0525854
|
4-[6-(1-adamantylcarbamoyl)-7-hydroxy-2-methyl-5-oxopyrazolo[4,3-b]pyridin-4-yl]butyl acetate
Show/Hide
|
C24H32N4O5
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0531748
|
4-(4-fluorobutyl)-7-hydroxy-N-(3-hydroxy-1-adamantyl)-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H29FN4O4
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
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CP0531749
|
4-butyl-7-hydroxy-N-(3-hydroxy-1-adamantyl)-2-methyl-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H30N4O4
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
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CP0532218
|
N-(1-adamantyl)-7-hydroxy-2-(2-hydroxyethyl)-5-oxo-4-propylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C22H30N4O4
|
1
|
| 1 |
Ki > 1000 nM
|
|
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CP0444457
|
4-(5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-4-oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl)benzoic acid
Show/Hide
|
C27H26Cl2N2O3
|
1
|
| 1 |
Ki > 2500 nM
|
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|
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CP0444459
|
1-(4-chlorophenyl)-5-cyclohexyl-2-(2,4-dichlorophenyl)-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C26H25Cl3N2O
|
1
|
| 1 |
Ki > 2500 nM
|
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CP0465175
|
1,2-bis(4-chlorophenyl)-5-cyclohexyl-3-methyl-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C26H26Cl2N2O
|
1
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| 1 |
Ki > 2500 nM
|
|
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CP0532377
|
5-cyclohexyl-1-(2,4-dichlorophenyl)-3-methyl-2-(4-(methylthio)phenyl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one
Show/Hide
|
C27H28Cl2N2OS
|
1
|
| 1 |
Ki > 2500 nM
|
|
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CP0410102
|
N-[3-(3-aminopropylamino)propyl]-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C23H26Cl3N5O
|
1
|
| 1 |
Ki > 2500 nM
|
|
|
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CP0396953
|
N-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C23H19Cl3N4O
|
1
|
| 1 |
Ki > 2820 nM
|
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CP0494321
|
N-[(4-chlorophenyl)-phenylmethyl]-1-(3,4-dichlorophenyl)-5-(2,5-dimethylpyrrol-1-yl)-4-methylpyrazole-3-carboxamide
Show/Hide
|
C30H25Cl3N4O
|
1
|
| 1 |
Ki > 2820 nM
|
|
|
|
CP0098948
|
Impulsin
Show/Hide
|
C18H37NO2
|
1
|
| 1 |
Ki > 5000 nM
|
|
|
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CP0454319
|
N-cyclohexyl-7-(dimethylamino)-1-(2-morpholin-4-ylethyl)-4-oxo-1,8-naphthyridine-3-carboxamide
Show/Hide
|
C23H33N5O3
|
1
|
| 1 |
Ki > 5600 nM
|
|
|
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CP0461224
|
2-cyclohexyl-5-(2-morpholinoethyl)-2H-pyrazolo[4,3-c]quinolin-3(5H)-one
Show/Hide
|
C22H28N4O2
|
1
|
| 1 |
Ki > 5600 nM
|
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