Brief Information of the Compound and Protein
Compound Name
(7E)-1-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-N-[(1R)-1-pyridin-2-ylethyl]-5,6-dihydro-4H-indazole-3-carboxamide
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PubChem ID
CID: 134157891
Canonical SMILES
C[C@@H](NC(=O)c1nn(c2c1CCC\C2=C/c1ccc(Cl)cc1)-c1ccc(Cl)cc1)c1ccccn1
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Compound Formula C28H24Cl2N4O
Compound Structure
Protein Name
Cannabinoid receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
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Cannabinoid receptor
Uniprot ID
P21554
Gene Name
CNR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 127 nM
   TI
   LI
   LO
   TS