Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(7E)-7-[(5-chlorothiophen-2-yl)methylidene]-1-[2-chloro-4-(trifluoromethyl)phenyl]-N-(1-pyridin-2-ylcyclopropyl)-5,6-dihydro-4H-indazole-3-carboxamide
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 PubChem ID
CID: 134155808
Canonical SMILES
FC(F)(F)c1ccc(c(Cl)c1)-n1nc(C(=O)NC2(CC2)c2ccccn2)c2CCC\C(=C/c3ccc(Cl)s3)c12
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Compound Formula C28H21Cl2F3N4OS
Compound Structure
Protein Name
 Protein Info 
Cannabinoid receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
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Cannabinoid receptor
Uniprot ID
P21554
Gene Name
CNR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 11 nM
   TI
   LI
   LO
   TS