| Compound ID |
Compound Name |
Compound Formula |
|
CP0420613
|
4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C19H13NO3S
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0854430
|
(E,Z)-5-((2-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)thiazol-4-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C15H9N3O3S2
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0845047
|
(E,Z)-5-((6-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)benzo[b]thiophen-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C20H12N2O3S2
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0879857
|
(E,Z)-5-((6-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)-1H-indol-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C20H13N3O3S
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0893220
|
(E,Z)-5-((5-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)pyridin-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C17H11N3O3S
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0392745
|
5-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
Show/Hide
|
C17H10N2O4S2
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0395653
|
(5E)-5-[[5-(1-oxo-2,3-dihydroisoindol-5-yl)thiophen-2-yl]methylidene]imidazolidine-2,4-dione
Show/Hide
|
C16H11N3O3S
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0853998
|
(E,Z)-5-((6-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)quinolin-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C21H13N3O3S
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0852234
|
(E,Z)-5-((5-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)benzo[b]thiophen-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C20H12N2O3S2
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0915787
|
(E,Z)-5-((5-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)benzofuran-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C20H12N2O4S
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
|
CP0379907
|
2-methyl-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C17H13N3O2S2
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
|
CP0460345
|
2-(3-hydroxypropyl)-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C19H17N3O3S2
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0436030
|
ethyl 3-oxo-6-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-1H-isoindole-2-carboxylate
Show/Hide
|
C19H15N3O4S2
|
1
|
| 1 |
IC50 = 550 nM
|
|
|
|
CP0460347
|
2-ethyl-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C18H15N3O2S2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0379766
|
5-[6-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]pyridin-3-yl]-2,3-dihydroisoindol-1-one
Show/Hide
|
C17H12N4O2S
|
1
|
| 1 |
IC50 = 630 nM
|
|
|
|
CP0467021
|
7-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3,4-dihydro-2H-isoquinolin-1-one
Show/Hide
|
C17H13N3O2S2
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0406222
|
2-hydroxy-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C19H13NO4S
|
1
|
| 1 |
IC50 = 670 nM
|
|
|
|
CP0570159
|
4-[[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]sulfamoyl]benzoic acid
Show/Hide
|
C25H19N3O5S2
|
1
|
| 1 |
IC50 = 750 nM
|
|
|
|
CP0916491
|
(E,Z)-5-((5-(1-oxo-1,3-dihydroisobenzofuran-5-yl)thiophen-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C16H10N2O3S2
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0467020
|
2-(2-hydroxyethyl)-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C18H15N3O3S2
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0519081
|
N-[2-methoxy-5-[5-(6-methyl-7-oxo-5H-pyrrolo[3,4-b]pyridin-3-yl)thiophen-2-yl]pyridin-3-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H19F3N4O4S2
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0461881
|
3-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C15H11N3O2S2
|
1
|
| 1 |
IC50 = 790 nM
|
|
|
|
CP0392744
|
5-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]-1,3-diazinane-2,4,6-trione
Show/Hide
|
C17H10N2O5S
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0858671
|
(E,Z)-5-((5-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)-1H-indol-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C20H13N3O3S
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0429792
|
5-[5-[4-(hydroxymethyl)phenyl]thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
|
C19H14O3S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0531247
|
5-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]pyridine-2-carboxamide
Show/Hide
|
C18H12N2O3S
|
1
|
| 1 |
IC50 = 920 nM
|
|
|
|
CP0433102
|
2-acetyl-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C18H13N3O3S2
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0422975
|
(Z)-1-(Benzo[b]thiophen-3-ylmethylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C17H11NO2S2
|
1
|
| 1 |
IC50 = 970 nM
|
|
|
|
CP0410670
|
N-[2-chloro-5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-2,4-difluorobenzenesulfonamide
Show/Hide
|
C24H16ClF2N3O3S2
|
1
|
| 1 |
IC50 = 1030 nM
|
|
|
|
CP0504773
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-methylbenzamide
Show/Hide
|
C21H14N6O
|
1
|
| 1 |
IC50 = 1040 nM
|
|
|
|
CP0919192
|
(E,Z)-5-((4-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)thiophen-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C16H10N2O3S2
|
1
|
| 1 |
IC50 = 1050 nM
|
|
|
|
CP0570160
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]pyridine-2-sulfonamide
Show/Hide
|
C23H18N4O3S2
|
1
|
| 1 |
IC50 = 1070 nM
|
|
|
|
CP0571111
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]thiophene-2-sulfonamide
Show/Hide
|
C22H17N3O3S3
|
1
|
| 1 |
IC50 = 1070 nM
|
|
|
|
CP0395075
|
N-[4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]phenyl]methanesulfonamide
Show/Hide
|
C19H15NO4S2
|
1
|
| 1 |
IC50 = 1090 nM
|
|
|
|
CP0393027
|
(5E)-5-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C16H9NO4S2
|
1
|
| 1 |
IC50 = 1120 nM
|
|
|
|
CP0190435
|
6-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3,4-dihydro-2H-isoquinolin-1-one
Show/Hide
|
C17H13N3O2S2
|
1
|
| 1 |
IC50 = 1140 nM
|
|
|
|
CP0467022
|
(5E)-5-[[5-(4-methylsulfanylphenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C15H12N2OS3
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
|
CP0491272
|
2-[3-oxo-6-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-1H-isoindol-2-yl]ethyl acetate
Show/Hide
|
C20H17N3O4S2
|
1
|
| 1 |
IC50 = 1170 nM
|
|
|
|
CP0432663
|
2-butyl-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C20H19N3O2S2
|
1
|
| 1 |
IC50 = 1180 nM
|
|
|
|
CP0461456
|
(5E)-5-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]imidazolidine-2,4-dione
Show/Hide
|
C16H10N2O4S
|
1
|
| 1 |
IC50 = 1190 nM
|
|
|
|
CP0540807
|
2-amino-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C19H14N2O3S
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0520927
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-3-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H18F3N3O3S2
|
1
|
| 1 |
IC50 = 1220 nM
|
|
|
|
CP0395661
|
2-(2,3-dihydroxypropyl)-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C19H17N3O4S2
|
1
|
| 1 |
IC50 = 1260 nM
|
|
|
|
CP0434778
|
(Z)-1-((1H-Indol-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C17H12N2O2S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0854002
|
(E,Z)-5-((3-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)isoxazol-5-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C15H9N3O4S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0485658
|
3,4-dichloro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H17Cl2N3O3S2
|
1
|
| 1 |
IC50 = 1320 nM
|
|
|
|
CP0451675
|
6-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-2,3-dihydroisoindol-1-one
Show/Hide
|
C16H11N3O2S2
|
1
|
| 1 |
IC50 = 1380 nM
|
|
|
|
CP0476299
|
N-[5-[5-(6-methyl-7-oxo-5H-pyrrolo[3,4-b]pyridin-3-yl)thiophen-2-yl]pyridin-3-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C24H17F3N4O3S2
|
1
|
| 1 |
IC50 = 1380 nM
|
|
|
|
CP0918023
|
(E,Z)-5-((4-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)thiazol-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C15H9N3O3S2
|
1
|
| 1 |
IC50 = 1410 nM
|
|
|
|
CP0574874
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-3-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C25H18F3N3O4S2
|
1
|
| 1 |
IC50 = 1420 nM
|
|
|
|
CP0854260
|
(E,Z)-5-((3-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)isothiazol-5-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C15H9N3O3S2
|
1
|
| 1 |
IC50 = 1440 nM
|
|
|
|
CP0451674
|
CHEMBL3103900
Show/Hide
|
C21H16N4O2S
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
|
CP0489138
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H18F3N3O3S2
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
|
CP0461880
|
5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-2-propyl-3H-isoindol-1-one
Show/Hide
|
C19H17N3O2S2
|
1
|
| 1 |
IC50 = 1520 nM
|
|
|
|
CP0444285
|
4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C15H11N3O2S2
|
1
|
| 1 |
IC50 = 1560 nM
|
|
|
|
CP0444296
|
CHEMBL3103897
Show/Hide
|
C20H14N4O2S
|
1
|
| 1 |
IC50 = 1580 nM
|
|
|
|
CP0525380
|
methyl 4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzoate
Show/Hide
|
C16H12N2O3S2
|
1
|
| 1 |
IC50 = 1620 nM
|
|
|
|
CP0491271
|
CHEMBL3103899
Show/Hide
|
C21H16N4O2S
|
1
|
| 1 |
IC50 = 1660 nM
|
|
|
|
CP0894717
|
(E,Z)-5-((5-(4-Acetylphenyl)thiophen-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C16H12N2O2S2
|
1
|
| 1 |
IC50 = 1670 nM
|
|
|
|
CP0467023
|
(5E)-5-[[5-(4-bromophenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C14H9BrN2OS2
|
1
|
| 1 |
IC50 = 1690 nM
|
|
|
|
CP0845046
|
(E,Z)-5-((2-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)thiazol-5-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C15H9N3O3S2
|
1
|
| 1 |
IC50 = 1720 nM
|
|
|
|
CP0852233
|
(E,Z)-5-((7-(1-oxo-1,3-dihydroisobenzofuran-5-yl)quinolin-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C21H13N3O3S
|
1
|
| 1 |
IC50 = 1720 nM
|
|
|
|
CP0389688
|
2,4,6-trifluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H16F3N3O3S2
|
1
|
| 1 |
IC50 = 1760 nM
|
|
|
|
CP0899758
|
(E,Z)-5-(4-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)benzylidene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C18H12N2O3S
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0509433
|
2-methyl-6-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C17H13N3O2S2
|
1
|
| 1 |
IC50 = 1890 nM
|
|
|
|
CP0570147
|
2,4-difluoro-N-[2-fluoro-5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H16F3N3O3S2
|
1
|
| 1 |
IC50 = 1990 nM
|
|
|
|
CP0854428
|
(E,Z)-5-((6-(1-oxo-1,3-dihydroisobenzofuran-5-yl)pyridin-3-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C17H11N3O3S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0389683
|
2-fluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18FN3O3S2
|
1
|
| 1 |
IC50 = 2030 nM
|
|
|
|
CP0888455
|
(E,Z)-5-(3-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)benzylidene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C18H12N2O3S
|
1
|
| 1 |
IC50 = 2110 nM
|
|
|
|
CP0489137
|
3-bromo-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18BrN3O3S2
|
1
|
| 1 |
IC50 = 2110 nM
|
|
|
|
CP0574869
|
N-(2,4-difluorophenyl)-5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridine-3-sulfonamide
Show/Hide
|
C24H17F2N3O3S2
|
1
|
| 1 |
IC50 = 2240 nM
|
|
|
|
CP0873207
|
(E,Z)-5-((5-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)benzo[b]thiophen-3-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C20H12N2O3S2
|
1
|
| 1 |
IC50 = 2270 nM
|
|
|
|
CP0390632
|
N-[2-methoxy-5-[5-(6-methyl-7-oxo-5H-pyrrolo[3,4-b]pyridin-3-yl)thiophen-2-yl]pyridin-3-yl]-2-nitrobenzenesulfonamide
Show/Hide
|
C24H19N5O6S2
|
1
|
| 1 |
IC50 = 2300 nM
|
|
|
|
CP0395656
|
2-methyl-6-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3,4-dihydroisoquinolin-1-one
Show/Hide
|
C18H15N3O2S2
|
1
|
| 1 |
IC50 = 2330 nM
|
|
|
|
CP0415167
|
(Z)-1-((5-Methoxybenzofuran-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H13NO4S
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0489136
|
3-chloro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18ClN3O3S2
|
1
|
| 1 |
IC50 = 2420 nM
|
|
|
|
CP0457362
|
N-(2,3-dihydroxypropyl)-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C18H17N3O4S2
|
1
|
| 1 |
IC50 = 2440 nM
|
|
|
|
CP0867641
|
(E,Z)-5-((5-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)-1Hpyrrol-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C16H11N3O3S
|
1
|
| 1 |
IC50 = 2450 nM
|
|
|
|
CP0461972
|
CHEMBL3103898
Show/Hide
|
C20H14N4O2S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0916490
|
(E,Z)-5-((3-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)isothiazol-4-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C15H9N3O3S2
|
1
|
| 1 |
IC50 = 2540 nM
|
|
|
|
CP0451673
|
5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-2,3-dihydroisoindol-1-one
Show/Hide
|
C16H11N3O2S2
|
1
|
| 1 |
IC50 = 2550 nM
|
|
|
|
CP0899567
|
(E,Z)-6-(2-((2-Oxo-5-thioxoimidazolidin-4-ylidene)methyl)quinolin-6-yl)-3,4-dihydroisoquinolin-1(2H)-one
Show/Hide
|
C22H16N4O2S
|
1
|
| 1 |
IC50 = 2550 nM
|
|
|
|
CP0523545
|
3-methoxy-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C25H21N3O4S2
|
1
|
| 1 |
IC50 = 2560 nM
|
|
|
|
CP0567558
|
N-(2-amino-2-oxoethyl)-2-hydroxy-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C21H16N2O5S
|
1
|
| 1 |
IC50 = 2650 nM
|
|
|
|
CP0410627
|
2-bromo-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18BrN3O3S2
|
1
|
| 1 |
IC50 = 2660 nM
|
|
|
|
CP0373423
|
(Z)-6-Methyl-1-((5-methylfuran-2-yl)methylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C14H11NO3S
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0390175
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-4-nitrobenzenesulfonamide
Show/Hide
|
C24H18N4O5S2
|
1
|
| 1 |
IC50 = 2740 nM
|
|
|
|
CP0510724
|
(5E)-2-amino-1-methyl-5-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]imidazol-4-one
Show/Hide
|
C17H13N3O3S
|
1
|
| 1 |
IC50 = 2750 nM
|
|
|
|
CP0451996
|
1-amino-3-[4-(2-hydroxyethoxy)phenyl]pyrido[1,2-a]benzimidazole-2,4-dicarbonitrile
Show/Hide
|
C21H15N5O2
|
1
|
| 1 |
IC50 = 2870 nM
|
|
|
|
CP0488975
|
2,4-dibromo-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H17Br2N3O3S2
|
1
|
| 1 |
IC50 = 2870 nM
|
|
|
|
CP0570158
|
methyl 2-[[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]sulfamoyl]benzoate
Show/Hide
|
C26H21N3O5S2
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0573896
|
3-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C19H13NO3S
|
1
|
| 1 |
IC50 = 2970 nM
|
|
|
|
CP0434773
|
(Z)-1-((7-Methoxybenzofuran-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H13NO4S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0478190
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)benzamide
Show/Hide
|
C20H12N6O
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0466973
|
5-[5-[(Z)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-3-yl]-2,3-dihydroisoindol-1-one
Show/Hide
|
C16H11N3O2S2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0444284
|
methyl 2-methyl-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzoate
Show/Hide
|
C17H14N2O3S2
|
1
|
| 1 |
IC50 = 3030 nM
|
|
|
|
CP0461282
|
[4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]phenyl]methyl acetate
Show/Hide
|
C17H14N2O3S2
|
1
|
| 1 |
IC50 = 3040 nM
|
|
|
|
CP0574877
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-4-(1,3-oxazol-5-yl)benzenesulfonamide
Show/Hide
|
C27H20N4O4S2
|
1
|
| 1 |
IC50 = 3050 nM
|
|
|
|
CP0473568
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-(2-hydroxyethyl)benzamide
Show/Hide
|
C22H16N6O2
|
1
|
| 1 |
IC50 = 3080 nM
|
|
|
|
CP0432665
|
(5E)-5-[[5-[4-chloro-3-(trifluoromethyl)phenyl]thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C15H8ClF3N2OS2
|
1
|
| 1 |
IC50 = 3090 nM
|
|
|
|
CP0517437
|
(Z)-1-((6-Methoxy-1H-indol-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H14N2O3S
|
1
|
| 1 |
IC50 = 3100 nM
|
|
|
|
CP0511320
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-ethylbenzamide
Show/Hide
|
C22H16N6O
|
1
|
| 1 |
IC50 = 3160 nM
|
|
|
|
CP0517537
|
5-[5-(1,3-oxazol-5-yl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
|
C15H9NO3S
|
1
|
| 1 |
IC50 = 3180 nM
|
|
|
|
CP0347285
|
2,3-dimethyl-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
|
C18H15N3O2S2
|
1
|
| 1 |
IC50 = 3210 nM
|
|
|
|
CP0460753
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-(2,3-dihydroxypropyl)benzamide
Show/Hide
|
C23H18N6O3
|
1
|
| 1 |
IC50 = 3240 nM
|
|
|
|
CP0444041
|
2-hydroxy-N-(2-hydroxyethyl)-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C21H17NO5S
|
1
|
| 1 |
IC50 = 3310 nM
|
|
|
|
CP0519082
|
2,4-difluoro-N-[2-methoxy-5-[5-(6-methyl-7-oxo-5H-pyrrolo[3,4-b]pyridin-3-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18F2N4O4S2
|
1
|
| 1 |
IC50 = 3340 nM
|
|
|
|
CP0462386
|
(Z)-6-Methyl-1-((5-phenylthiophen-2-yl)methylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C19H13NO2S2
|
1
|
| 1 |
IC50 = 3400 nM
|
|
|
|
CP0379767
|
5-[3-[(Z)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]phenyl]-2,3-dihydroisoindol-1-one
Show/Hide
|
C18H13N3O2S
|
1
|
| 1 |
IC50 = 3440 nM
|
|
|
|
CP0465073
|
2-[4-(1-amino-2,4-dicyano-7,8-dimethylpyrido[1,2-a]benzimidazol-3-yl)phenoxy]acetamide
Show/Hide
|
C23H18N6O2
|
1
|
| 1 |
IC50 = 3530 nM
|
|
|
|
CP0485657
|
2,4-difluoro-N-[2-methoxy-5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C25H19F2N3O4S2
|
1
|
| 1 |
IC50 = 3560 nM
|
|
|
|
CP0395664
|
N-(2-hydroxyethyl)-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C17H15N3O3S2
|
1
|
| 1 |
IC50 = 3640 nM
|
|
|
|
CP0390176
|
4-fluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-3-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H17F4N3O3S2
|
1
|
| 1 |
IC50 = 3750 nM
|
|
|
|
CP0415166
|
(Z)-1-[(4-Methoxy-1-benzothien-3-yl)methylene]-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridine-3(1H)-one
Show/Hide
|
C18H13NO3S2
|
1
|
| 1 |
IC50 = 3800 nM
|
|
|
|
CP0509291
|
1,3-dimethyl-5-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]-1,3-diazinane-2,4,6-trione
Show/Hide
|
C19H14N2O5S
|
1
|
| 1 |
IC50 = 3960 nM
|
|
|
|
CP0434769
|
(Z)-6-Methyl-1-((5-phenylfuran-2-yl)methylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C19H13NO3S
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0574871
|
2-chloro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18ClN3O3S2
|
1
|
| 1 |
IC50 = 4010 nM
|
|
|
|
CP0492091
|
(Z)-1-((1H-Indol-7-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C17H12N2O2S
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0574905
|
N-[2-fluoro-5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]pyridine-2-sulfonamide
Show/Hide
|
C23H17FN4O3S2
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0459881
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-(3-hydroxypropyl)benzamide
Show/Hide
|
C23H18N6O2
|
1
|
| 1 |
IC50 = 4180 nM
|
|
|
|
CP0373422
|
(Z)-6-Methyl-1-((1-methyl-1H-indol-3-yl)methylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H14N2O2S
|
1
|
| 1 |
IC50 = 4300 nM
|
|
|
|
CP0519083
|
2,4-difluoro-N-[5-[5-(6-methyl-7-oxo-5H-pyrrolo[3,4-b]pyridin-3-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C23H16F2N4O3S2
|
1
|
| 1 |
IC50 = 4300 nM
|
|
|
|
CP0444283
|
N-(3-hydroxypropyl)-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C18H17N3O3S2
|
1
|
| 1 |
IC50 = 4350 nM
|
|
|
|
CP0526214
|
(Z)-1-(Furan-2-ylmethylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C13H9NO3S
|
1
|
| 1 |
IC50 = 4400 nM
|
|
|
|
CP0433059
|
5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-2-propan-2-yl-3H-isoindol-1-one
Show/Hide
|
C19H17N3O2S2
|
1
|
| 1 |
IC50 = 4420 nM
|
|
|
|
CP0446936
|
N-methyl-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C16H13N3O2S2
|
1
|
| 1 |
IC50 = 4530 nM
|
|
|
|
CP0531248
|
5-(5-pyridin-4-ylthiophen-2-yl)-3H-2-benzofuran-1-one
Show/Hide
|
C17H11NO2S
|
1
|
| 1 |
IC50 = 4530 nM
|
|
|
|
CP0483799
|
2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-methylacetamide
Show/Hide
|
C22H16N6O2
|
1
|
| 1 |
IC50 = 4560 nM
|
|
|
|
CP0460349
|
(5E)-5-[[5-(3,4-difluorophenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C14H8F2N2OS2
|
1
|
| 1 |
IC50 = 4590 nM
|
|
|
|
CP0415165
|
(Z)-1-((5-Methoxy-1H-indol-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H14N2O3S
|
1
|
| 1 |
IC50 = 4600 nM
|
|
|
|
CP0415168
|
(Z)-1-(Benzo[b]thiophen-2-ylmethylene)-6-methylfuro[3,4-c]pyridine-3,4(1H,5H)-dione
Show/Hide
|
C17H11NO3S
|
1
|
| 1 |
IC50 = 4600 nM
|
|
|
|
CP0433060
|
(5E)-2-sulfanylidene-5-[[5-[4-(trifluoromethyl)phenyl]thiophen-2-yl]methylidene]imidazolidin-4-one
Show/Hide
|
C15H9F3N2OS2
|
1
|
| 1 |
IC50 = 4660 nM
|
|
|
|
CP0422977
|
(Z)-1-((6-Methoxybenzo[b]thiophen-3-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H13NO3S2
|
1
|
| 1 |
IC50 = 4700 nM
|
|
|
|
CP0563990
|
2,4-difluoro-N-[4-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-2-yl]benzenesulfonamide
Show/Hide
|
C24H17F2N3O3S2
|
1
|
| 1 |
IC50 = 4700 nM
|
|
|
|
CP0460346
|
2-methyl-7-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3,4-dihydroisoquinolin-1-one
Show/Hide
|
C18H15N3O2S2
|
1
|
| 1 |
IC50 = 4760 nM
|
|
|
|
CP0420587
|
3-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzenesulfonamide
Show/Hide
|
C18H13NO4S2
|
1
|
| 1 |
IC50 = 4850 nM
|
|
|
|
CP0526218
|
(Z)-6-Methyl-1-((5-phenylthiophen-2-yl)methylene)furo[3,4-c]pyridine-3,4(1H,5H)-dione
Show/Hide
|
C19H13NO3S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0570156
|
4-iodo-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18IN3O3S2
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0422974
|
(Z)-1-((6-(Benzyloxy)-5-methoxybenzofuran-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C25H19NO5S
|
1
|
| 1 |
IC50 = 5100 nM
|
|
|
|
CP0422976
|
(Z)-1-((5-Methoxybenzo[b]thiophen-3-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H13NO3S2
|
1
|
| 1 |
IC50 = 5100 nM
|
|
|
|
CP0524698
|
2-[4-[2-cyano-2-(5,6-dimethyl-1H-benzimidazol-2-yl)ethenyl]phenoxy]acetamide
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 = 5140 nM
|
|
|
|
CP0563991
|
4-cyano-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C25H18N4O3S2
|
1
|
| 1 |
IC50 = 5170 nM
|
|
|
|
CP0460248
|
2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]acetamide
Show/Hide
|
C21H14N6O2
|
1
|
| 1 |
IC50 = 5190 nM
|
|
|
|
CP0459880
|
2-[4-(1-amino-2,4-dicyano-6,7-dimethylpyrido[1,2-a]benzimidazol-3-yl)phenoxy]acetamide
Show/Hide
|
C23H18N6O2
|
1
|
| 1 |
IC50 = 5210 nM
|
|
|
|
CP0493921
|
(5E)-5-[[5-(4-chlorophenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C14H9ClN2OS2
|
1
|
| 1 |
IC50 = 5220 nM
|
|
|
|
CP0899585
|
5-((5-(3-Acetyl-1-methyl-1H-indol-5-yl)thiophen-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C19H15N3O2S2
|
1
|
| 1 |
IC50 = 5300 nM
|
|
|
|
CP0571107
|
4-chloro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18ClN3O3S2
|
1
|
| 1 |
IC50 = 5390 nM
|
|
|
|
CP0526221
|
(Z)-1-((6-Methoxybenzo[b]thiophen-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H13NO3S2
|
1
|
| 1 |
IC50 = 5400 nM
|
|
|
|
CP0523546
|
4-fluoro-2-methyl-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C25H20FN3O3S2
|
1
|
| 1 |
IC50 = 5530 nM
|
|
|
|
CP0449149
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-(2-hydroxypropyl)benzamide
Show/Hide
|
C23H18N6O2
|
1
|
| 1 |
IC50 = 5550 nM
|
|
|
|
CP0509432
|
5-[4-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]phenyl]-2,3-dihydroisoindol-1-one
Show/Hide
|
C18H13N3O2S
|
1
|
| 1 |
IC50 = 5550 nM
|
|
|
|
CP0538988
|
(5E)-2-sulfanylidene-5-[[5-[3-(trifluoromethyl)phenyl]thiophen-2-yl]methylidene]imidazolidin-4-one
Show/Hide
|
C15H9F3N2OS2
|
1
|
| 1 |
IC50 = 5660 nM
|
|
|
|
CP0487332
|
2-[4-(1-amino-6-chloro-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]acetamide
Show/Hide
|
C21H13ClN6O2
|
1
|
| 1 |
IC50 = 5670 nM
|
|
|
|
CP0576317
|
2,4-difluoro-N-[5-[5-(7-oxo-5,6-dihydropyrrolo[3,4-b]pyridin-3-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C22H14F2N4O3S2
|
1
|
| 1 |
IC50 = 5730 nM
|
|
|
|
CP0563989
|
2,4-difluoro-N-[3-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]phenyl]benzenesulfonamide
Show/Hide
|
C25H18F2N2O3S2
|
1
|
| 1 |
IC50 = 5740 nM
|
|
|
|
CP0545022
|
2-amino-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzoic acid
Show/Hide
|
C19H13NO4S
|
1
|
| 1 |
IC50 = 5840 nM
|
|
|
|
CP0573800
|
5-[5-(3-hydroxyphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
|
C18H12O3S
|
1
|
| 1 |
IC50 = 5890 nM
|
|
|
|
CP0559159
|
4-[5-(1-oxo-2,3-dihydroisoindol-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C19H14N2O2S
|
1
|
| 1 |
IC50 = 6040 nM
|
|
|
|
CP0573797
|
N-tert-butyl-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzenesulfonamide
Show/Hide
|
C22H21NO4S2
|
1
|
| 1 |
IC50 = 6090 nM
|
|
|
|
CP0878664
|
(E,Z)-5-((5-(1-oxo-1,3-dihydroisobenzofuran-5-yl)furan-2-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C16H10N2O4S
|
1
|
| 1 |
IC50 = 6200 nM
|
|
|
|
CP0420588
|
5-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
|
C20H12O4S
|
1
|
| 1 |
IC50 = 6240 nM
|
|
|
|
CP0572526
|
4-methoxy-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C25H21N3O4S2
|
1
|
| 1 |
IC50 = 6270 nM
|
|
|
|
CP0467696
|
(Z)-1-((5-Fluoro-6-methoxy-1H-indol-3-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H13FN2O3S
|
1
|
| 1 |
IC50 = 6300 nM
|
|
|
|
CP0465043
|
5-(1-oxo-3H-2-benzofuran-5-yl)thiophene-2-carbaldehyde
Show/Hide
|
C13H8O3S
|
1
|
| 1 |
IC50 = 6310 nM
|
|
|
|
CP0451677
|
N-(2-hydroxypropyl)-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C18H17N3O3S2
|
1
|
| 1 |
IC50 = 6500 nM
|
|
|
|
CP0485661
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-2-nitrobenzenesulfonamide
Show/Hide
|
C24H18N4O5S2
|
1
|
| 1 |
IC50 = 6650 nM
|
|
|
|
CP0395665
|
(5E)-5-[[5-(4-fluorophenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C14H9FN2OS2
|
1
|
| 1 |
IC50 = 6690 nM
|
|
|
|
CP0526220
|
(Z)-1-((4-Methoxybenzofuran-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H13NO4S
|
1
|
| 1 |
IC50 = 6700 nM
|
|
|
|
CP0494120
|
2-[4-[2-(4-chloro-1H-benzimidazol-2-yl)-2-cyanoethenyl]phenoxy]acetamide
Show/Hide
|
C18H13ClN4O2
|
1
|
| 1 |
IC50 = 6720 nM
|
|
|
|
CP0563992
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-2-methylsulfonylbenzenesulfonamide
Show/Hide
|
C25H21N3O5S3
|
1
|
| 1 |
IC50 = 6800 nM
|
|
|
|
CP0461926
|
(3Z)-3-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]pyrrolidin-2-one
Show/Hide
|
C17H13NO3S
|
1
|
| 1 |
IC50 = 6810 nM
|
|
|
|
CP0465071
|
2-[4-(1-amino-2,4-dicyano-6-methylpyrido[1,2-a]benzimidazol-3-yl)phenoxy]acetamide
Show/Hide
|
C22H16N6O2
|
1
|
| 1 |
IC50 = 6870 nM
|
|
|
|
CP0395065
|
4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzonitrile
Show/Hide
|
C19H11NO2S
|
1
|
| 1 |
IC50 = 6870 nM
|
|
|
|
CP0465072
|
2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N,N-dimethylacetamide
Show/Hide
|
C23H18N6O2
|
1
|
| 1 |
IC50 = 6890 nM
|
|
|
|
CP0510457
|
N,N-dimethyl-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C17H15N3O2S2
|
1
|
| 1 |
IC50 = 6930 nM
|
|
|
|
CP0461925
|
(3Z)-3-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]pyrrolidine-2,5-dione
Show/Hide
|
C17H11NO4S
|
1
|
| 1 |
IC50 = 6970 nM
|
|
|
|
CP0389686
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-5-(1,2-oxazol-5-yl)thiophene-2-sulfonamide
Show/Hide
|
C25H18N4O4S3
|
1
|
| 1 |
IC50 = 7100 nM
|
|
|
|
CP0469265
|
N-(3-amino-3-oxopropyl)-2-hydroxy-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C22H18N2O5S
|
1
|
| 1 |
IC50 = 7120 nM
|
|
|
|
CP0486784
|
(5E)-5-[[5-(3-chlorophenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C14H9ClN2OS2
|
1
|
| 1 |
IC50 = 7190 nM
|
|
|
|
CP0422967
|
(Z)-6-Methyl-1-((5-methylthiophen-2-yl)methylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C14H11NO2S2
|
1
|
| 1 |
IC50 = 7200 nM
|
|
|
|
CP0435013
|
(Z)-1-((6-Methoxybenzofuran-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C18H13NO4S
|
1
|
| 1 |
IC50 = 7200 nM
|
|
|
|
CP0919191
|
(E,Z)-5-((2-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)oxazol-5-yl)methylene)-2-thioxoimidazolidin-4-one
Show/Hide
|
C15H9N3O4S
|
1
|
| 1 |
IC50 = 7280 nM
|
|
|
|
CP0460247
|
2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-ethylacetamide
Show/Hide
|
C23H18N6O2
|
1
|
| 1 |
IC50 = 7440 nM
|
|
|
|
CP0508285
|
2-[4-(1-amino-2,4-dicyano-6-methoxypyrido[1,2-a]benzimidazol-3-yl)phenoxy]acetamide
Show/Hide
|
C22H16N6O3
|
1
|
| 1 |
IC50 = 7490 nM
|
|
|
|
CP0373421
|
(Z)-1-((5-Bromobenzo[b]thiophen-3-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C17H10BrNO2S2
|
1
|
| 1 |
IC50 = 7500 nM
|
|
|
|
CP0510458
|
N-[4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]phenyl]methanesulfonamide
Show/Hide
|
C15H13N3O3S3
|
1
|
| 1 |
IC50 = 7700 nM
|
|
|
|
CP0486783
|
(5E)-5-[[5-(4-hydroxyphenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C14H10N2O2S2
|
1
|
| 1 |
IC50 = 7720 nM
|
|
|
|
CP0489139
|
methyl 3-[[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]sulfamoyl]benzoate
Show/Hide
|
C26H21N3O5S2
|
1
|
| 1 |
IC50 = 7770 nM
|
|
|
|
CP0493920
|
N-(3-morpholin-4-ylpropyl)-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
|
C22H24N4O3S2
|
1
|
| 1 |
IC50 = 8130 nM
|
|
|
|
CP0563994
|
3-chloro-4-methyl-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C25H20ClN3O3S2
|
1
|
| 1 |
IC50 = 8140 nM
|
|
|
|
CP0389685
|
methyl 4-[[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]sulfamoyl]benzoate
Show/Hide
|
C26H21N3O5S2
|
1
|
| 1 |
IC50 = 8160 nM
|
|
|
|
CP0387522
|
(Z)-1-(Benzofuran-2-ylmethylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C17H11NO3S
|
1
|
| 1 |
IC50 = 8200 nM
|
|
|
|
CP0494119
|
2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-(2-hydroxyethyl)acetamide
Show/Hide
|
C23H18N6O3
|
1
|
| 1 |
IC50 = 8250 nM
|
|
|
|
CP0390171
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H19N3O3S2
|
1
|
| 1 |
IC50 = 8460 nM
|
|
|
|
CP0454985
|
(Z)-1-(Benzo[b]thiophen-3-ylmethylene)-6-methylfuro[3,4-c]pyridine-3,4(1H,5H)-dione
Show/Hide
|
C17H11NO3S
|
1
|
| 1 |
IC50 = 8500 nM
|
|
|
|
CP0462384
|
(Z)-6-Methyl-1-(thiophen-2-ylmethylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C13H9NO2S2
|
1
|
| 1 |
IC50 = 8600 nM
|
|
|
|
CP0574872
|
4-bromo-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18BrN3O3S2
|
1
|
| 1 |
IC50 = 8770 nM
|
|
|
|
CP0563988
|
3-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]-N-pyridin-2-ylbenzenesulfonamide
Show/Hide
|
C24H19N3O3S2
|
1
|
| 1 |
IC50 = 8920 nM
|
|
|
|
CP0525379
|
5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-2-(3-pyrrolidin-1-ylpropyl)-3H-isoindol-1-one
Show/Hide
|
C23H24N4O2S2
|
1
|
| 1 |
IC50 = 8930 nM
|
|
|
|
CP0485659
|
2-cyano-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C25H18N4O3S2
|
1
|
| 1 |
IC50 = 9170 nM
|
|
|
|
CP0573039
|
5-[5-(4-methoxyphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
|
C19H14O3S
|
1
|
| 1 |
IC50 = 9360 nM
|
|
|
|
CP0462392
|
(Z)-1-(Benzo[b]thiophen-2-ylmethylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
|
C17H11NO2S2
|
1
|
| 1 |
IC50 = 9500 nM
|
|
|
|
CP0541350
|
4-fluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C24H18FN3O3S2
|
1
|
| 1 |
IC50 = 9650 nM
|
|
|
|
CP0460348
|
3-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzonitrile
Show/Hide
|
C15H9N3OS2
|
1
|
| 1 |
IC50 = 9680 nM
|
|
|
|
CP0541349
|
2-methoxy-5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]-N-pyridin-2-ylbenzenesulfonamide
Show/Hide
|
C25H21N3O4S2
|
1
|
| 1 |
IC50 = 9680 nM
|
|
|
|
CP0440709
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-(2-morpholin-4-ylethyl)benzamide
Show/Hide
|
C26H23N7O2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0487336
|
2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-(2-pyridin-4-ylethyl)acetamide
Show/Hide
|
C28H21N7O2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0496471
|
(5E)-5-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
Show/Hide
|
C16H9NO3S3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0446937
|
(5E)-5-[(5-pyridin-4-ylthiophen-2-yl)methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C13H9N3OS2
|
1
|
| 1 |
IC50 = 10060 nM
|
|
|
|
CP0452005
|
4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-(2-pyridin-4-ylethyl)benzamide
Show/Hide
|
C27H19N7O
|
1
|
| 1 |
IC50 = 10500 nM
|
|
|
|
CP0406159
|
N-methyl-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
|
C20H15NO3S
|
1
|
| 1 |
IC50 = 10700 nM
|
|
|
|
CP0432666
|
(5E)-5-[[5-(3-fluorophenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C14H9FN2OS2
|
1
|
| 1 |
IC50 = 10770 nM
|
|
|
|
CP0567557
|
ethyl 4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzoate
Show/Hide
|
C21H16O4S
|
1
|
| 1 |
IC50 = 10970 nM
|
|
|
|
CP0489141
|
4-methyl-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-1,3-thiazole-5-sulfonamide
Show/Hide
|
C22H18N4O3S3
|
1
|
| 1 |
IC50 = 11600 nM
|
|
|
|
CP0486782
|
5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-2-(3-piperidin-1-ylpropyl)-3H-isoindol-1-one
Show/Hide
|
C24H26N4O2S2
|
1
|
| 1 |
IC50 = 11780 nM
|
|
|
|
CP0429810
|
5-[5-(4-aminophenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
|
C18H13NO2S
|
1
|
| 1 |
IC50 = 11820 nM
|
|
|
|
CP0563995
|
N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]thiophene-3-sulfonamide
Show/Hide
|
C22H17N3O3S3
|
1
|
| 1 |
IC50 = 12500 nM
|
|
|
|
CP0420615
|
2-hydroxy-N-(2-morpholin-4-ylethyl)-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
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C25H24N2O5S
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1
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| 1 |
IC50 = 12750 nM
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CP0458474
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(5E)-5-[(5-pyridin-3-ylthiophen-2-yl)methylidene]-2-sulfanylideneimidazolidin-4-one
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C13H9N3OS2
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1
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| 1 |
IC50 = 12890 nM
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CP0574876
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3-chloro-2-fluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
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C24H17ClFN3O3S2
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1
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| 1 |
IC50 = 13000 nM
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CP0434774
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(Z)-1-((5-Methoxybenzo[b]thiophen-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C18H13NO3S2
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1
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| 1 |
IC50 = 13100 nM
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CP0449217
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2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-propan-2-ylacetamide
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C24H20N6O2
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1
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| 1 |
IC50 = 13200 nM
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CP0509428
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(5E)-5-[[5-(4-methylsulfonylphenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
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C15H12N2O3S3
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1
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| 1 |
IC50 = 13800 nM
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CP0390173
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3,4-dimethoxy-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
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C26H23N3O5S2
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1
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| 1 |
IC50 = 13800 nM
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CP0465930
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2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-propylacetamide
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C24H20N6O2
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1
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| 1 |
IC50 = 13900 nM
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CP0452696
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5-[5-(3-aminophenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
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C18H13NO2S
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1
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| 1 |
IC50 = 13970 nM
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CP0537959
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N-[5-[5-[2-(2,3-dihydroxypropyl)-1-oxo-3H-isoindol-5-yl]thiophen-2-yl]pyridin-3-yl]-2,4-difluorobenzenesulfonamide
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C26H21F2N3O5S2
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1
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| 1 |
IC50 = 14200 nM
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CP0452699
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2-amino-N-(2-morpholin-4-ylethyl)-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
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C25H25N3O4S
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1
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| 1 |
IC50 = 14710 nM
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CP0571109
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2-methoxy-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
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C25H21N3O4S2
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1
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| 1 |
IC50 = 14800 nM
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CP0570155
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2,4-dichloro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
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C24H17Cl2N3O3S2
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1
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| 1 |
IC50 = 15000 nM
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CP0481073
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N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]pyridine-3-sulfonamide
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C23H18N4O3S2
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1
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| 1 |
IC50 = 15100 nM
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CP0503199
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(3Z)-3-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]piperidin-2-one
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C18H15NO3S
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1
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| 1 |
IC50 = 15200 nM
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CP0389684
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N-[4-methyl-3-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]phenyl]pyridine-2-sulfonamide
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C25H21N3O3S2
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1
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| 1 |
IC50 = 15400 nM
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CP0489135
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2,4-difluoro-N-methyl-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
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C25H19F2N3O3S2
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1
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| 1 |
IC50 = 16100 nM
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CP0574727
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2,4-difluoro-N-[5-[5-[2-(2-morpholin-4-ylethyl)-1-oxo-3H-isoindol-5-yl]thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
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C29H26F2N4O4S2
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1
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| 1 |
IC50 = 17000 nM
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CP0574873
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N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-2-(trifluoromethoxy)benzenesulfonamide
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C25H18F3N3O4S2
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1
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| 1 |
IC50 = 17700 nM
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CP0390172
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3,4-difluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
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C24H17F2N3O3S2
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1
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| 1 |
IC50 = 18600 nM
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CP0572527
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4-(3,5-dimethylpyrazol-1-yl)-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
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C29H25N5O3S2
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1
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| 1 |
IC50 = 19100 nM
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CP0410669
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ethyl 4-[[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]sulfamoyl]benzoate
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C27H23N3O5S2
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1
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| 1 |
IC50 = 19400 nM
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CP0373417
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(Z)-1-(4-Methoxybenzylidene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C16H15NO3S
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1
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| 1 |
IC50 > 20000 nM
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CP0373418
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(Z)-6-Methyl-1-(thiophen-3-ylmethylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C13H9NO2S2
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1
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| 1 |
IC50 > 20000 nM
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CP0373420
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(Z)-6-Methyl-1-((1-methyl-1H-indol-2-yl)methylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C18H14N2O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0415164
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(Z)-1-(4-(Dimethylamino)benzylidene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C17H16N2O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0422968
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(Z)-1-((1H-Pyrrol-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C13H10N2O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0422969
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(Z)-1-((1H-Imidazol-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C12H9N3O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0422970
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(Z)-6-Methyl-1-((1-methyl-1H-pyrrol-2-yl)methylene)-4-thioxo-a4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C14H12N2O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0422972
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(Z)-6-Methyl-1-((5-phenylthiophen-2-yl)methylene)-4-thioxo-4,5-dihydro-1H-pyrrolo[3,4-c]pyridin-3(2H)-one
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C19H14N2OS2
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1
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| 1 |
IC50 > 20000 nM
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CP0422973
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(Z)-6-Methyl-1-((5-phenylthiophen-2-yl)methylene)-1H-pyrrolo[3,4-c]pyridine-3,4(2H,5H)-dione
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C19H14N2O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0434770
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(Z)-1-(4-Chlorobenzylidene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C15H10ClNO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0434771
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(Z)-6-Methyl-1-(4-methylbenzylidene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C16H13NO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0434772
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(Z)-6-Methyl-1-((5-methylfuran-2-yl)methylene)-1H-pyrrolo[3,4-c]pyridine-3,4(2H,5H)-dione
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C14H12N2O3
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1
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| 1 |
IC50 > 20000 nM
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CP0434775
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(Z)-1-((6-(Benzyloxy)-5-methoxy-1H-indol-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C25H20N2O4S
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1
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| 1 |
IC50 > 20000 nM
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CP0434776
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(Z)-1-((5-(Benzyloxy)-1H-indol-2-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C24H18N2O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0435010
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(Z)-1-Benzylidene-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C15H11NO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0462388
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(Z)-1-(Biphenyl-4-ylmethylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
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C21H15NO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0462390
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(Z)-1-((1H-Pyrrol-2-yl)methylene)-6-methylfuro[3,4-c]pyridine-3,4(1H,5H)-dione
Show/Hide
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C13H10N2O3
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1
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| 1 |
IC50 > 20000 nM
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CP0463792
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(Z)-1-((1H-Indol-3-yl)methylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C17H12N2O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0466766
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(Z)-1-(Furan-3-ylmethylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C13H9NO3S
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1
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| 1 |
IC50 > 20000 nM
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CP0493463
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(Z)-6-Methyl-1-((1-methyl-1H-indol-3-yl)methylene)furo[3,4-c]pyridine-3,4(1H,5H)-dione
Show/Hide
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C18H14N2O3
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1
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| 1 |
IC50 > 20000 nM
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CP0502281
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(Z)-1-(4-Fluorobenzylidene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C15H10FNO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0512414
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(Z)-6-Methyl-4-thioxo-1-(4-(trifluoromethoxy)benzylidene)-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C16H10F3NO3S
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1
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| 1 |
IC50 > 20000 nM
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CP0517436
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(Z)-6-Methyl-1-(4-(methylthio)benzylidene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C16H13NO2S2
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1
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| 1 |
IC50 > 20000 nM
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CP0517438
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(Z)-1-(Benzo[b]thiophen-3-ylmethylene)-6-methyl-4-thioxo-4,5-dihydro-1H-pyrrolo[3,4-c]pyridin-3(2H)-one
Show/Hide
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C17H12N2OS2
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1
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| 1 |
IC50 > 20000 nM
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CP0526215
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(Z)-6-Methyl-4-thioxo-1-(4-(trifluoromethyl)benzylidene)-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C16H10F3NO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0526216
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(Z)-N-(4-((6-Methyl-3-oxo-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-1(3H)-ylidene)methyl)phenyl)acetamide
Show/Hide
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C17H14N2O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0526217
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(Z)-6-Methyl-1-((5-methylfuran-2-yl)methylene)furo[3,4-c]pyridine-3,4(1H,5H)-dione
Show/Hide
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C14H11NO4
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1
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| 1 |
IC50 > 20000 nM
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CP0526219
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(Z)-6-Methyl-1-((5-phenylthiophen-3-yl)methylene)-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C19H13NO2S2
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1
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| 1 |
IC50 > 20000 nM
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CP0526222
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(Z)-1-(Benzofuran-3-ylmethylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one
Show/Hide
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C17H11NO3S
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1
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| 1 |
IC50 > 20000 nM
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CP0478521
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4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-(2-piperidin-1-ylethyl)benzamide
Show/Hide
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C27H25N7O
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1
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| 1 |
IC50 > 20000 nM
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CP0486221
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2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-(3-hydroxypropyl)acetamide
Show/Hide
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C24H20N6O3
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1
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| 1 |
IC50 > 20000 nM
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CP0486222
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2-[4-[2-cyano-2-(4,5-dimethyl-1H-benzimidazol-2-yl)ethenyl]phenoxy]acetamide
Show/Hide
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C20H18N4O2
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1
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| 1 |
IC50 > 20000 nM
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CP0487334
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3-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenyl]-N-methylpropanamide
Show/Hide
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C23H18N6O
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1
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| 1 |
IC50 > 20000 nM
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CP0487335
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2-[4-[2-cyano-2-(4-methoxy-1H-benzimidazol-2-yl)ethenyl]phenoxy]acetamide
Show/Hide
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C19H16N4O3
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1
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| 1 |
IC50 > 20000 nM
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CP0494121
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2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-(2,3-dihydroxypropyl)acetamide
Show/Hide
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C24H20N6O4
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1
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| 1 |
IC50 > 20000 nM
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CP0494122
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4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N-[2-(dimethylamino)ethyl]benzamide
Show/Hide
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C24H21N7O
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1
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| 1 |
IC50 > 20000 nM
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CP0504772
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3-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenyl]-N,N-dimethylpropanamide
Show/Hide
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C24H20N6O
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1
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| 1 |
IC50 > 20000 nM
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CP0505296
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4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)-N,N-dimethylbenzamide
Show/Hide
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C22H16N6O
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1
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| 1 |
IC50 > 20000 nM
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CP0505298
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2-[4-[2-cyano-2-(4-methyl-1H-benzimidazol-2-yl)ethenyl]phenoxy]acetamide
Show/Hide
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C19H16N4O2
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1
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| 1 |
IC50 > 20000 nM
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CP0524699
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2-[4-(1-amino-2,4-dicyanopyrido[1,2-a]benzimidazol-3-yl)phenoxy]-N-(2-hydroxypropyl)acetamide
Show/Hide
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C24H20N6O3
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1
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| 1 |
IC50 > 20000 nM
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CP0524700
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2-[4-[2-(1H-benzimidazol-2-yl)-2-cyanoethenyl]phenoxy]acetamide
Show/Hide
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C18H14N4O2
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1
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| 1 |
IC50 > 20000 nM
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CP0393026
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5-thiophen-2-yl-3H-2-benzofuran-1-one
Show/Hide
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C12H8O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0399058
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5-(5-acetylthiophen-2-yl)-3H-2-benzofuran-1-one
Show/Hide
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C14H10O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0463114
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methyl 2-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]acetate
Show/Hide
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C15H12O4S
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1
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| 1 |
IC50 > 20000 nM
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CP0497356
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2-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]acetic acid
Show/Hide
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C14H10O4S
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1
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| 1 |
IC50 > 20000 nM
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CP0500872
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(3Z)-1-[(4-methoxyphenyl)methyl]-3-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]pyrrolidin-2-one
Show/Hide
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C25H21NO4S
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1
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| 1 |
IC50 > 20000 nM
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CP0504070
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(3Z)-1-benzyl-3-[[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]methylidene]pyrrolidin-2-one
Show/Hide
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C24H19NO3S
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1
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| 1 |
IC50 > 20000 nM
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CP0852232
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(E,Z)-5-(2-(1-Oxo-1,3-dihydroisobenzofuran-5-yl)benzylidene)-2-thioxoimidazolidin-4-one
Show/Hide
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C18H12N2O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0897906
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(E,Z)-1-Oxo-N-(3-(5-oxo-2-thioxoimidazolidin-4-ylidene)propyl)-1,3-dihydroisobenzofuran-5-carboxamide
Show/Hide
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C15H13N3O4S
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1
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| 1 |
IC50 > 20000 nM
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CP0395667
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(5E)-5-[(5-phenylthiophen-2-yl)methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
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C14H10N2OS2
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1
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| 1 |
IC50 > 20000 nM
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CP0432664
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N-(2-morpholin-4-ylethyl)-4-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]benzamide
Show/Hide
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C21H22N4O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0433101
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2-[3-(dimethylamino)propyl]-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
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C21H22N4O2S2
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1
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| 1 |
IC50 > 20000 nM
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CP0436025
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(5E)-5-[[5-(2-chlorophenyl)thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
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C14H9ClN2OS2
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1
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| 1 |
IC50 > 20000 nM
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CP0436031
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(5E)-5-[[5-[4-(morpholine-4-carbonyl)phenyl]thiophen-2-yl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
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C19H17N3O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0486781
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2-[3-(4-methylpiperazin-1-yl)propyl]-5-[5-[(E)-(5-oxo-2-sulfanylideneimidazolidin-4-ylidene)methyl]thiophen-2-yl]-3H-isoindol-1-one
Show/Hide
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C24H27N5O2S2
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1
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| 1 |
IC50 > 20000 nM
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CP0390427
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5-[5-(4-methylsulfonylphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C19H14O4S2
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1
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| 1 |
IC50 > 20000 nM
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CP0406157
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5-(5-phenylthiophen-2-yl)-3H-2-benzofuran-1-one
Show/Hide
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C18H12O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0406158
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5-[5-(3-methylphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C19H14O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0420611
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5-[5-(2-chlorophenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C18H11ClO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0420612
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5-[5-(3-methoxyphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C19H14O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0420614
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4-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]benzamide
Show/Hide
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C20H16N2O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0444040
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5-[5-[4-(4-methylpiperazine-1-carbonyl)phenyl]thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C24H22N2O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0452698
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N-[2-(dimethylamino)ethyl]-2-hydroxy-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
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C23H22N2O4S
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1
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| 1 |
IC50 > 20000 nM
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CP0452700
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2-amino-N-[2-(dimethylamino)ethyl]-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
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C23H23N3O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0455636
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5-[5-(2-methylphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C19H14O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0469263
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3-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzonitrile
Show/Hide
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C19H11NO2S
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1
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| 1 |
IC50 = 20000 nM
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CP0469264
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ethyl 2-hydroxy-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzoate
Show/Hide
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C21H16O5S
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1
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| 1 |
IC50 > 20000 nM
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CP0473440
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5-[5-(4-methylsulfanylphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C19H14O2S2
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1
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| 1 |
IC50 > 20000 nM
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CP0531348
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5-[5-(4-hydroxyphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C18H12O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0545020
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5-[5-(4-methylphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C19H14O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0545021
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5-[5-(3-chlorophenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C18H11ClO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0559158
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5-[5-(4-chlorophenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C18H11ClO2S
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1
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| 1 |
IC50 > 20000 nM
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CP0567555
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N,N-dimethyl-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
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C21H17NO3S
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1
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| 1 |
IC50 > 20000 nM
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CP0567556
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N-[3-(dimethylamino)propyl]-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
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C24H24N2O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0573040
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2-hydroxy-N-(2-hydroxypropyl)-4-[5-(1-oxo-3H-2-benzofuran-5-yl)thiophen-2-yl]benzamide
Show/Hide
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C22H19NO5S
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1
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| 1 |
IC50 > 20000 nM
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CP0573799
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5-[5-(2-methoxyphenyl)thiophen-2-yl]-3H-2-benzofuran-1-one
Show/Hide
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C19H14O3S
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1
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| 1 |
IC50 > 20000 nM
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CP0389687
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2,4-difluoro-N-[4-methyl-3-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]phenyl]benzenesulfonamide
Show/Hide
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C26H20F2N2O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0390174
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N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
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C25H18F3N3O4S2
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1
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| 1 |
IC50 > 20000 nM
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CP0410668
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3-cyano-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
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C25H18N4O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0481074
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N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-4-methylsulfonylbenzenesulfonamide
Show/Hide
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C25H21N3O5S3
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1
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| 1 |
IC50 > 20000 nM
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CP0485663
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N-[4-fluoro-3-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]phenyl]pyridine-2-sulfonamide
Show/Hide
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C24H18FN3O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0489134
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4-methyl-3-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]-N-pyridin-2-ylbenzenesulfonamide
Show/Hide
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C25H21N3O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0489140
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2-chloro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
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C25H17ClF3N3O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0523547
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3-bromo-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-5-(trifluoromethyl)benzenesulfonamide
Show/Hide
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C25H17BrF3N3O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0563997
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N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-3,5-bis(trifluoromethyl)benzenesulfonamide
Show/Hide
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C26H17F6N3O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0570146
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N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
Show/Hide
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C26H21N3O5S2
|
1
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| 1 |
IC50 > 20000 nM
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CP0570153
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2,4-difluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-2-yl]benzenesulfonamide
Show/Hide
|
C24H17F2N3O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0570154
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3-fluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
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C24H18FN3O3S2
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1
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| 1 |
IC50 = 20000 nM
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CP0574867
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N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]-2-(trifluoromethoxy)phenyl]pyridine-2-sulfonamide
Show/Hide
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C25H18F3N3O4S2
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1
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| 1 |
IC50 > 20000 nM
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CP0574868
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2,4-difluoro-N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]benzamide
Show/Hide
|
C25H17F2N3O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0574875
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N-[5-[5-(2-methyl-1-oxo-3H-isoindol-5-yl)thiophen-2-yl]pyridin-3-yl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H18F3N3O3S2
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1
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| 1 |
IC50 > 20000 nM
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|
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CP0390631
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N-[5-[5-(6-methyl-7-oxo-5H-pyrrolo[3,4-b]pyridin-3-yl)thiophen-2-yl]pyridin-3-yl]-3-(trifluoromethyl)benzenesulfonamide
Show/Hide
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C24H17F3N4O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0396988
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2,4-difluoro-N-[5-[5-[2-[2-(4-methylpiperazin-1-yl)ethyl]-1-oxo-3H-isoindol-5-yl]thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
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C30H29F2N5O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0440951
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2,4-difluoro-N-[5-[5-(5-oxo-6,7-dihydropyrrolo[3,4-b]pyridin-3-yl)thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
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C22H14F2N4O3S2
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1
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| 1 |
IC50 > 20000 nM
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CP0444730
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2,4-difluoro-N-[5-[5-[2-(3-hydroxypropyl)-1-oxo-3H-isoindol-5-yl]thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
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C26H21F2N3O4S2
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1
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| 1 |
IC50 > 20000 nM
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CP0537960
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N-[5-[5-[2-[2-(dimethylamino)ethyl]-1-oxo-3H-isoindol-5-yl]thiophen-2-yl]pyridin-3-yl]-2,4-difluorobenzenesulfonamide
Show/Hide
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C27H24F2N4O3S2
|
1
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| 1 |
IC50 > 20000 nM
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CP0551204
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2,4-difluoro-N-[5-[5-[1-oxo-2-(2-piperidin-1-ylethyl)-3H-isoindol-5-yl]thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
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C30H28F2N4O3S2
|
1
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| 1 |
IC50 > 20000 nM
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CP0553249
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2,4-difluoro-N-[5-[5-[1-oxo-2-(2-pyrrolidin-1-ylethyl)-3H-isoindol-5-yl]thiophen-2-yl]pyridin-3-yl]benzenesulfonamide
Show/Hide
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C29H26F2N4O3S2
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1
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| 1 |
IC50 > 20000 nM
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