| Compound ID |
Compound Name |
Compound Formula |
|
CP0095953
|
ENZALUTAMIDE
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|
C21H16F4N4O2S
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0570758
|
N-(4-cyanophenyl)-2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]acetamide
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|
C20H12F3N5O
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0273406
|
2-[1-(3-chloro-4-cyanophenyl)pyrazol-3-yl]-N-(6-fluoropyridin-3-yl)acetamide
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|
C17H11ClFN5O
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0578085
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(4-nitrophenyl)acetamide
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|
C19H12F3N5O3
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0355222
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(4-fluorophenyl)acetamide
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|
C19H12F4N4O
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0260233
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(6-fluoropyridin-3-yl)acetamide
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|
C18H11F4N5O
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0577151
|
2-[1-(3-chloro-4-cyanophenyl)pyrazol-3-yl]-N-(5-fluoropyridin-2-yl)acetamide
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|
C17H11ClFN5O
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0495153
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(3,4-difluorophenyl)acetamide
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|
C19H11F5N4O
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0570982
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]-4-methylpyrazol-3-yl]methyl]-4-fluorobenzamide
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|
C20H14F4N4O
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0571986
|
2-[1-(3-chloro-4-cyanophenyl)pyrazol-3-yl]-N-(4-fluorophenyl)acetamide
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|
C18H12ClFN4O
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0578068
|
4-cyano-N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]benzamide
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|
C20H12F3N5O
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0546216
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(5-fluoropyridin-2-yl)acetamide
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|
C18H11F4N5O
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0578345
|
N-(4-fluorophenyl)-2-[1-[4-nitro-3-(trifluoromethyl)phenyl]pyrazol-3-yl]acetamide
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|
C18H12F4N4O3
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0578070
|
N-(6-fluoropyridin-3-yl)-2-[1-[4-nitro-3-(trifluoromethyl)phenyl]pyrazol-3-yl]acetamide
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|
C17H11F4N5O3
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0578342
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]-4-methylpyrazol-3-yl]methyl]-4-nitrobenzamide
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|
C20H14F3N5O3
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
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CP0579454
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-4-fluorobenzamide
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|
C19H12F4N4O
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0578754
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-6-fluoropyridine-3-carboxamide
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|
C18H11F4N5O
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0545341
|
4-chloro-N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]benzamide
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|
C19H12ClF3N4O
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
|
CP0571980
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-4-nitrobenzamide
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|
C19H12F3N5O3
|
1
|
| 1 |
IC50 = 1850 nM
|
|
|
|
CP0495154
|
N-(5-fluoropyridin-2-yl)-2-[1-[4-nitro-3-(trifluoromethyl)phenyl]pyrazol-3-yl]acetamide
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|
C17H11F4N5O3
|
1
|
| 1 |
IC50 = 2570 nM
|
|
|
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CP0579456
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(4-methylphenyl)acetamide
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|
C20H15F3N4O
|
1
|
| 1 |
IC50 = 4530 nM
|
|
|
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CP0568513
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-5-fluoropyridine-2-carboxamide
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|
C18H11F4N5O
|
1
|
| 1 |
IC50 = 5820 nM
|
|
|
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CP0571985
|
N-(3-cyano-4-fluorophenyl)-2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]acetamide
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|
C20H11F4N5O
|
1
|
| 1 |
IC50 = 6340 nM
|
|
|
|
CP0578751
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(4-methoxyphenyl)acetamide
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|
C20H15F3N4O2
|
1
|
| 1 |
IC50 = 9200 nM
|
|
|
|
CP0546209
|
4-cyano-N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]-4-methylpyrazol-3-yl]methyl]benzamide
Show/Hide
|
C21H14F3N5O
|
1
|
| 1 |
IC50 = 14900 nM
|
|
|
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CP0578084
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]-4-(trifluoromethyl)pyrazol-3-yl]methyl]-4-fluorobenzamide
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|
C20H11F7N4O
|
1
|
| 1 |
IC50 = 16240 nM
|
|
|
|
CP0495151
|
N-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-4-fluorobenzamide
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|
C18H10F4N4O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0495152
|
N-[3-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]propyl]-4-fluorobenzamide
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|
C21H16F4N4O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0545342
|
4-N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-2-fluoro-1-N-methylbenzene-1,4-dicarboxamide
Show/Hide
|
C21H15F4N5O2
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0545343
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-pyridin-4-ylacetamide
Show/Hide
|
C18H12F3N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0569872
|
1-[4-cyano-3-(trifluoromethyl)phenyl]-N-(6-fluoropyridin-3-yl)pyrazole-3-carboxamide
Show/Hide
|
C17H9F4N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0570757
|
1-[4-cyano-3-(trifluoromethyl)phenyl]-N-(5-fluoropyridin-2-yl)pyrazole-3-carboxamide
Show/Hide
|
C17H9F4N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0570981
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-4-fluorobenzenesulfonamide
Show/Hide
|
C18H12F4N4O2S
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0571979
|
1-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-3-(4-fluorophenyl)urea
Show/Hide
|
C19H13F4N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0571981
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C20H12F6N4O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0571982
|
4-cyano-N-[2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]ethyl]benzamide
Show/Hide
|
C21H14F3N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0571983
|
1-[4-cyano-3-(trifluoromethyl)phenyl]-N-(4-fluorophenyl)pyrazole-3-carboxamide
Show/Hide
|
C18H10F4N4O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0571984
|
N-(4-cyanophenyl)-1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazole-3-carboxamide
Show/Hide
|
C19H10F3N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0573463
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]-4-phenylpyrazol-3-yl]methyl]-4-fluorobenzamide
Show/Hide
|
C25H16F4N4O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0575239
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-4-(2-hydroxypropan-2-yl)benzamide
Show/Hide
|
C22H19F3N4O2
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0575240
|
N-[[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]-5-(1-hydroxyethyl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C18H15F3N6O2
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0575241
|
4-cyano-N-[3-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]propyl]benzamide
Show/Hide
|
C22H16F3N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0578069
|
N-[2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]ethyl]-4-fluorobenzamide
Show/Hide
|
C20H14F4N4O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0578341
|
1-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-3-(4-fluorophenyl)urea
Show/Hide
|
C18H11F4N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
|
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CP0578343
|
N-[2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]ethyl]-4-nitrobenzamide
Show/Hide
|
C20H14F3N5O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
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CP0578344
|
N-[3-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]propyl]-4-nitrobenzamide
Show/Hide
|
C21H16F3N5O3
|
1
|
| 1 |
IC50 > 25000 nM
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CP0579455
|
1-[4-cyano-3-(trifluoromethyl)phenyl]-N-pyridin-4-ylpyrazole-3-carboxamide
Show/Hide
|
C17H10F3N5O
|
1
|
| 1 |
IC50 > 25000 nM
|
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|
