3-chloro-N-[[3-[2-[2-[2-[2-[2-[4-[[(7S)-7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]methyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]pyridin-4-yl]phenyl]methyl]-N-[4-(methylamino)cyclohexyl]-1-benzothiophene-2-carboxamide

CHEMBL4877645

3-chloro-N-[[3-[2-[2-[2-[2-[2-[4-[2-[2-[(7S)-7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]pyridin-4-yl]phenyl]methyl]-N-[4-(methylamino)cyclohexyl]-1-benzothiophene-2-carboxamide

3-chloro-N-[4-(methylamino)cyclohexyl]-N-[(3-pyridin-4-ylphenyl)methyl]-1-benzothiophene-2-carboxamide

CHEMBL4875874

3-chloro-N-[[3-[2-[2-[2-[2-[2-[2-[2-[4-[2-[2-[2-[2-[2-[2-[2-[2-[(7R)-7-[(3S,8S,9S,10R,13R,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]pyridin-4-yl]phenyl]methyl]-N-[4-(methylamino)cyclohexyl]-1-benzothiophene-2-carboxamide

CHEMBL4850805

CHEMBL4855383

CHEMBL4865069

3-chloro-N-[[3-[2-[2-[2-[2-[2-[2-[2-[4-[2-[2-[2-[2-[2-[2-[2-[(7R)-7-[(3S,8S,9S,10R,13R,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]pyridin-4-yl]phenyl]methyl]-N-[4-(methylamino)cyclohexyl]-1-benzothiophene-2-carboxamide

CHEMBL4846477

3-chloro-N-[[3-[2-[2-[2-[2-[2-[4-(2-hydroxyethoxymethyl)triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]pyridin-4-yl]phenyl]methyl]-N-[4-(methylamino)cyclohexyl]-1-benzothiophene-2-carboxamide

(3S,8S,9S,10R,13S,14S)-17-[2-hydroxy-8-[2-[[1-[2-[2-[2-(2-hydroxyethoxy)ethoxy]ethoxy]ethyl]triazol-4-yl]methoxy]ethoxy]octan-2-yl]-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3-ol

7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octane-1,7-diol

(R)-(3-methyl-4-(1-(4-(trifluoromethyl)phenyl)pyrido[3,4-d]pyridazin-4-yl)piperazin-1-yl)(phenyl)methanone

N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-4-phenoxy-2-(trifluoromethyl)benzamide

LY-2940680

(R)-(3-methyl-4-(1-phenylpyrido[3,4-d]pyridazin-4-yl)piperazin-1-yl)(phenyl)methanone

(5S)-1-[(4-azidophenyl)methyl]-3-(4-chlorophenyl)-5-methylimidazolidine-2,4-dione

4-fluoro-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)naphthalen-1-yl)piperidin-4-yl)-2-(trifluoromethyl)benzamide

2-chloro-N-(4-chloro-3-(pyridin-2-yl)phenyl)-4-(methylsulfonyl)benzamide

N-(2-methylcyclohexyl)-1-[5-[5-[[(5-methylpyridin-2-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

2-chloro-N-[4-[4-phenyl-5-(trifluoromethyl)-1,3-oxazol-2-yl]phenyl]benzamide

N-(2-methylcyclohexyl)-1-[5-[5-[(pyridin-2-ylamino)methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)-4-[2-[2-[2-[2-[2-[2-[4-[2-[7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylsulfonyl]benzamide

2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)-4-[2-[2-[2-[2-[2-[4-[2-[7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethylsulfonyl]benzamide

2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)-4-[2-[2-[2-[2-[4-[2-[7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethylsulfonyl]benzamide

2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)-4-[2-[2-[2-[2-[2-[2-[4-[2-[2-[2-[2-[7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxy]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylsulfonyl]benzamide

2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)-4-[2-[2-[2-[2-[2-[2-[4-[2-[2-[7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylsulfonyl]benzamide

2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)-4-[2-[2-[2-[4-[2-[7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethylsulfonyl]benzamide

2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)-4-[2-[2-[2-[2-[2-[2-[4-[2-[2-[2-[2-[2-[2-[7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylsulfonyl]benzamide

2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)-4-[2-[2-[2-[2-[2-[2-[4-[2-[2-[2-[2-[2-[2-[2-[2-[7-hydroxy-7-[(3S,8S,9S,10R,13S,14S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]octoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylsulfonyl]benzamide

(4-(4-phenylphthalazin-1-yl)piperazin-1-yl)(thiophen-2-yl)methanone

2-chloro-N-[4-(4-phenylpyridin-2-yl)phenyl]benzamide

(5S)-1-[(4-azidophenyl)methyl]-5-methyl-3-(4-prop-2-ynoxyphenyl)imidazolidine-2,4-dione

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-3-chlorobenzamide

N-(2-methylcyclohexyl)-1-[5-[5-[(5-methylpyridin-2-yl)oxymethyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

1-[5-[5-[(4-methylanilino)methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]-N-(2-methylcyclohexyl)piperidine-4-carboxamide

N-(2-methylcyclohexyl)-1-[5-[5-[[(6-methylpyridin-3-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

N-(2-methylcyclohexyl)-1-[5-[5-[2-(5-methylpyridin-2-yl)ethyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

(5S)-3-(4-azidophenyl)-1-benzyl-5-methylimidazolidine-2,4-dione

(5S)-1-benzyl-3-(4-chlorophenyl)-5-methylimidazolidine-2,4-dione

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]benzamide

N-(4-fluoro-2-(trifluoromethyl)benzyl)-N-methyl-1-(4-(1-methyl-1Hpyrazol-5-yl)phthalazin-1-yl)piperidin-4-amine

N-(2-methylcyclohexyl)-1-[5-[5-[(pyridin-3-ylamino)methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

N-[[5-fluoro-6-(2-methylpyridin-4-yl)pyridin-3-yl]methyl]-9H-carbazole-2-carboxamide

N-(2-methylcyclohexyl)-1-[5-[5-[[(6-methylpyridazin-3-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

(5S)-3-(4-chlorophenyl)-5-methyl-1-(2-phenylethyl)imidazolidine-2,4-dione

N-[6-[6-chloro-5-[[cyano(phenyl)methyl]amino]pyridin-3-yl]-1,3-benzothiazol-2-yl]acetamide

N-[6-[6-chloro-5-[(4-fluorophenyl)sulfonylamino]pyridin-3-yl]-1,3-benzothiazol-2-yl]acetamide

3-chloro-N-[2-chloro-5-[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]pyridin-3-yl]benzamide

N-[2-chloro-5-[2-(cyclopropylmethylamino)-1,3-benzothiazol-6-yl]pyridin-3-yl]benzamide

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-4-fluorobenzamide

N-(2-methylcyclohexyl)-1-[5-[5-[[(5-methylpyrimidin-2-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

3-chloro-N-[2-chloro-5-[2-(cyclopropylmethylamino)-1,3-benzothiazol-6-yl]pyridin-3-yl]benzamide

N-[2-chloro-5-[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]pyridin-3-yl]benzamide

N-(3-methylpyridin-4-yl)-1-[5-[5-[[(5-methylpyridin-2-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-4-nitrobenzamide

N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-4-phenoxybenzamide

N-(3-methylpyridin-2-yl)-1-[5-[5-[[(5-methylpyridin-2-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

N-(2-methylcyclohexyl)-1-[5-[2-[[(5-methylpyridin-2-yl)amino]methyl]phenyl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

(5S)-3-(4-chlorophenyl)-1-(cyclohexylmethyl)-5-methylimidazolidine-2,4-dione

N-(2-methylcyclohexyl)-1-[5-[5-[[(5-methylpyrazin-2-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

N-(2-methylpyridin-3-yl)-1-[5-[5-[[(5-methylpyridin-2-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

(5S)-3-(4-chlorophenyl)-5-methyl-1-phenylimidazolidine-2,4-dione

N-(4-methylpyridin-3-yl)-1-[5-[5-[[(5-methylpyridin-2-yl)amino]methyl]pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-4-methylbenzamide

(4-(methyl(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)carbamoyl)phenyl)boronic acid

N-[6-[5-(benzylamino)-6-chloropyridin-3-yl]-1,3-benzothiazol-2-yl]acetamide

1-((2-(3-chlorophenyl)-5-methyloxazol-4-yl)methyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)piperidine-4-carboxamide

N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)benzamide

benzyl 3-(3-(3,4-difluorobenzyl)-2-oxotetrahydropyrimidin-1(2H)-yl)phenylcarbamate

N-[[5-cyano-6-(2-methylpyridin-4-yl)pyridin-3-yl]methyl]-9H-carbazole-2-carboxamide

4-(dimethylamino)-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)benzamide

(5S)-1-benzyl-5-methyl-3-(2,3,4,5,6-pentafluorophenyl)imidazolidine-2,4-dione

4-fluoro-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)benzamide

4-(benzyloxy)-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)benzamide

N-(2-methylcyclohexyl)-1-[5-[1-methyl-5-[[(5-methylpyridin-2-yl)amino]methyl]pyrazol-4-yl]-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

4-amino-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)benzamide

N-(6-(4-(2-hydroxybenzyl)piperazin-1-yl)pyridin-3-yl)-2-(trifluoromethyl)benzamide

4-(methyl(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)carbamoyl)benzenesulfonic acid

4-formyl-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)benzamide

6-(2-methyl-2,3-dihydroindole-1-carbonyl)-2-[3-oxo-3-(4-phenylpiperazin-1-yl)propyl]pyridazin-3-one

4-[2-[2-[2-[2-[2-(2-azidoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethylsulfonyl]-2-chloro-N-(4-chloro-3-pyridin-2-ylphenyl)benzamide

N1-methyl-N1-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)terephthalamide

N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-4-sulfamoylbenzamide

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-2-phenylacetamide

N-[[5-methoxy-6-(2-methylpyridin-4-yl)pyridin-3-yl]methyl]-9H-carbazole-2-carboxamide

(5S)-1-benzyl-3-(4-chlorophenyl)-5-methyl-2-sulfanylideneimidazolidin-4-one

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-2-chlorobenzamide

(4S)-3-benzyl-1-(4-chlorophenyl)-4-methylimidazolidin-2-one

1-(2-(3,4-dimethylphenyl)pyrazolo[1,5-a]pyrazin-4-yl)-N-(1-phenylethyl)piperidine-4-carboxamide

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-3-fluorobenzamide

(5S)-3-(4-chlorophenyl)-5-methyl-1-[(2,3,4,5,6-pentafluorophenyl)methyl]imidazolidine-2,4-dione

(5S)-1-benzyl-3-cyclohexyl-5-methylimidazolidine-2,4-dione

(5S)-1-benzyl-3-[(4-chlorophenyl)methyl]-5-methylimidazolidine-2,4-dione

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-2-fluorobenzamide

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]cyclopropanecarboxamide

N-[5-(2-acetamido-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-4-chlorobenzamide

N-[2-(1,3-benzothiazol-2-ylamino)-2-oxoethyl]-3-(4-methoxyphenyl)-4-oxophthalazine-1-carboxamide

N-(5-chloro-2-methoxyphenyl)-4-[3-[(3-fluorophenyl)methoxy]-6-oxopyridazin-1-yl]benzamide

N-[2-[2-(5-methoxy-1H-indol-3-yl)ethylcarbamoyl]phenyl]-1,2-benzothiazole-3-carboxamide

2-fluoro-5-(4-(2-fluorophenyl)piperazin-1-ylsulfonyl)-N-(4-isopropylphenyl)benzamide

10-{3-[4-(2-Fluoro-phenyl)-piperazine-1-carbonyl]-phenyl}-6-methoxy-9-methyl-8-oxa-10,12-diaza-tricyclo[7.3.1.0(2,7)]trideca-2(7),3,5-trien-11-one

N-cyclohexyl-5-methyl-4-oxo-3-(2-oxo-2-(3-(trifluoromethyl)phenylamino)ethyl)-3,4-dihydrothieno[2,3-d]pyrimidine-6-carboxamide

4-fluoro-N-(2-(2-(4-fluorophenyl)quinazolin-4-ylamino)ethyl)-2-methoxybenzenesulfonamide

N-benzyl-4-cyano-N-(3-(2-(3-methylbenzylamino)-2-oxoethyl)phenyl)benzamide

N-((5-(2-(benzo[d]thiazol-2-ylamino)-2-oxoethylthio)-4-phenyl-4H-1,2,4-triazol-3-yl)methyl)thiophene-2-carboxamide

2-(7-(3,4-dimethylphenyl)-8-oxo-7,8-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-3-ylthio)-N-o-tolylbutanamide

1-(4-fluorophenyl)-3-(1-(5-(trifluoromethyl)pyridin-2-yl)piperidin-4-ylamino)pyrrolidine-2,5-dione

7-(4-(2-(4-chlorophenyl)acetylcarbamothioyl)piperazin-1-yl)-1-ethyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid

2-chloro-N-(2-(2-(3-chloro-4-methylphenylamino)-2-oxoethylthio)benzo[d]thiazol-6-yl)benzamide

N-benzyl-4-(1-(2-(methyl(phenyl)amino)-2-oxoethyl)-2,4-dioxo-1,2-dihydrothieno[3,2-d]pyrimidin-3(4H)-yl)butanamide

2-((2-chloro-4-fluorobenzylsulfonyl)methyl)-N-(2-(4-methylpiperidin-1-yl)propyl)-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide

(4-(methyl(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)carbamoyl)phenyl)glycine

N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-4-(methylsulfonyl)benzamide

Methyl 4-(methyl(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)carbamoyl)benzoate

N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-4-(2-oxoethyl)benzamide

4-(methyl(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)carbamoyl)benzoic acid

N-(2-methylcyclohexyl)-1-[5-(2-methylpyrazol-3-yl)-1,3,4-thiadiazol-2-yl]piperidine-4-carboxamide

1-[5-(3,5-dimethylpyrazol-1-yl)-1,3,4-thiadiazol-2-yl]-N-(2-methylcyclohexyl)piperidine-4-carboxamide

4-fluoro-N-methyl-N-[1-[5-(2-methylpyrazol-3-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-yl]-2-(trifluoromethyl)benzamide

2-[5-[(2R)-4-(5-benzyl-1,3,4-thiadiazol-2-yl)-2-methylpiperazin-1-yl]pyrazin-2-yl]propan-2-ol

1-[5-[5-(hydroxymethyl)pyrazol-1-yl]-1,3,4-thiadiazol-2-yl]-N-(2-methylcyclohexyl)piperidine-4-carboxamide

N-(2-methylcyclohexyl)-1-(5-pyrazol-1-yl-1,3,4-thiadiazol-2-yl)piperidine-4-carboxamide

N-(1-(4-chlorophthalazin-1-yl)piperidin-4-yl)-4-fluoro-N-methyl-2-(trifluoromethyl)benzamide