| Compound ID |
Compound Name |
Compound Formula |
|
CP0040803
|
N-(2,6-difluorophenyl)-5-[3-[2-[5-ethyl-2-methoxy-4-[4-(4-methylsulfonylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]-2-methoxybenzamide
Show/Hide
|
C44H47F2N9O5S
|
2
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
IC50 < 100 nM
|
|
|
|
CP0040804
|
3-(3-(2-(4-(1,4'-bipiperidin-1'-yl)-2-methoxyphenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H40F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0042282
|
N-(2,6-difluorophenyl)-3-[3-[2-[5-ethyl-2-methoxy-4-[4-(4-methylsulfonylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H45F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0069911
|
N-(2,6-difluorophenyl)-3-[3-[2-[2-methoxy-4-[4-(4-methylsulfonylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H41F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0177146
|
3-(3-(2-(4-(1,4'-bipiperidin-1'-yl)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)benzamide
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|
C40H38F2N8O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0388757
|
N-(2,6-difluorophenyl)-3-[3-[2-[4-[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F2N8O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0461636
|
3-(3-(2-(4-(4-(4-acetylpiperazin-1-yl)piperidin-1-yl)-2-methoxyphenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H41F2N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0475298
|
N-(2,6-difluorophenyl)-3-[3-[2-[2-methoxy-4-(4-pyrrolidin-1-ylpiperidin-1-yl)anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H38F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0509038
|
N-(2,6-difluorophenyl)-3-[3-[2-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H41F2N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845764
|
3-[3-(2-{[4-(1,4'-bipiperidin-l'-yl)-2-methylphenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H40F2N8O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0845773
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(4-thiomorpholinyl)-1-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C40H38F2N8O2S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0845774
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[(9aS)-hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H43F2N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845775
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[1-(2-fluoroethyl)-4-piperidinyl]-1-piperazinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845776
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(cis-4-{4-[2-(methylsulfonyl)-ethyl]-1-piperazinyl}cyclohexyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845777
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{1'-[2-(methylsulfonyl)ethyl]-4,4'-bipiperidin-1-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C45H48F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845778
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2,5-bis(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845779
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(ethyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazin-yl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H47F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845780
|
N-(2,6-difluorophenyl)-3-{3-[2-({4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)-2-[(2,2,2-trifluoroethyl)oxy]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C44H44F5N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845782
|
N-(2,6-difluorophenyl)-5-[3-(2-{[2-(ethyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845783
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[2-(ethyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H43F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845802
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{1'-[2-(methylsulfonyl)ethyl]-4,4'-bipiperidin-1-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845803
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{1'-[2-(methylsulfonyl)ethyl]-1,4'-bipiperidin-4-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845804
|
N-(2,6-difluorophenyl)-3-(3-(2-((2-(methyloxy)-4-(4-(2-(methylsulfonyl)ethyl)-1,4'-bipiperidin-1'-yl)phenyl)amino)-4-pyrimidinyl)imidazo(1,2-a)pyridin-2-yl)benzamide
Show/Hide
|
C44H46F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845805
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-chloro-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C41H39ClF2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845806
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845807
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2,5-bis(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H44F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845810
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-{3-[2-({2-(methyloxy)-4-[2-(4-methyl-1-piperazinyl)ethyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845836
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[3-(1-piperidinyl)propyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C39H37F2N7O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0845845
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C43H45F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845847
|
3-[3-(2-{[4-(1,4'-bipiperidin-l'-yl)-2-(ethyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0845849
|
N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(1-piperidinylmethyl)-1-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0845866
|
N-(2,6-difluorophenyl)-2-[(1-methylethyl)oxy]-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C43H45F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848311
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C40H40F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848316
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[(3R)-3-hydroxy-1-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C36H31F2N7O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0848317
|
N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H37F2N7O4S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0848319
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C43H45F2N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848470
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H44F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848471
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-[4-(l-methylethyl)-1-piperazinyl]-2-(methyloxy)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C39H38F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848472
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-[(1-methylethyl)oxy]benzamide
Show/Hide
|
C43H45F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848486
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[5-methyl-2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H43F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848487
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
|
C44H47F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848526
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-(4-methyl-1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0848527
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-3-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(ethyloxy)benzamide
Show/Hide
|
C44H46F2N8O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0848528
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C42H42F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848529
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H46F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848530
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-(4-hydroxy-1,4'-bipiperidin-1'-yl)-2-(methyloxy)-phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848531
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[1'-(2-fluoroethyl)-4,4'-bipiperidin-1-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H43F3N8O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0848532
|
N-(2,6-difluorophenyl)-3-[3-(2-{[5-methyl-2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C40H39F2N7O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848534
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
|
C43H46F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856490
|
3-{3-[2-({4-(1,4'-bipiperidin-1'-yl)-2-[(1-methylethyl)oxy]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C43H44F2N8O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0856492
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-8-methylimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0856495
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-[(9aS)-hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C38H34F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856497
|
N-(2,6-difluorophenyl)-3-(7-fluoro-3-(2-((2-(methyloxy)-4-(4-(4-(methylsulfonyl)-1-piperazinyl)-1-piperidinyl)phenyl)amino)-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C41H40F3N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856498
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-fluoroimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C42H41F3N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856500
|
N-(2,6-difluorophenyl)-5-{3-[2-({5-methyl-2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
|
C39H38F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856509
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-2-propylphenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C43H45F2N7O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856510
|
N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C41H42F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0856511
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3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-8-fluoroimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C41H39F3N8O2
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1
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| 1 |
IC50 = 100 nM
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CP0856513
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]hexahydro-1H-1,4-diazepin-1-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H44F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0857311
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C40H40F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0857313
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0857314
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C45H49F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0857315
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
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C43H45F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0857317
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[3-(1-piperidinyl)propyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C40H39F2N7O3
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1
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| 1 |
IC50 < 100 nM
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CP0857318
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N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[3-(4-methyl-1-piperazinyl)propyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C39H38F2N8O2
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1
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| 1 |
IC50 = 100 nM
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CP0857321
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N-(2,6-difluorophenyl)-3-(3-{2-[(5-methyl-2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C40H39F2N7O4S
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1
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| 1 |
IC50 < 100 nM
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CP0857322
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-[3-(2-{[2-(methyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C39H38F2N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0857323
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N-(2,6-difluorophenyl)-3-[8-fluoro-3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C42H41F4N9O2
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1
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| 1 |
IC50 = 100 nM
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CP0857324
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
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C46H51F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0857326
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C44H47F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0857327
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0857328
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N-(2,6-difluorophenyl)-2-((1-methylethyl)oxy)-5-(3-(2-((2-(methyloxy)-4-(4-(4-(methylsulfonyl)-1-piperazinyl)-1-piperidinyl)phenyl)amino)-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C44H47F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0861201
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N-(2,6-difluorophenyl)-5-[3-(2-{[4-{(3S)-3-(1-methylethyl)-4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
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C42H44F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0861239
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-[1'-(2-fluoroethyl)-1,4'-bipiperidin-4-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C43H43F3N8O2
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1
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| 1 |
IC50 < 100 nM
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CP0861240
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N-(2,6-difluorophenyl)-5-[3-(2-{[4-[(9aS)-hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)-benzamide
Show/Hide
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C39H36F2N8O4
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1
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| 1 |
IC50 < 100 nM
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CP0861241
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C40H39F2N7O4S
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1
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| 1 |
IC50 < 100 nM
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CP0861242
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C40H40F2N8O4S
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1
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| 1 |
IC50 < 100 nM
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CP0863036
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N-(2,6-difluorophenyL)-3-[8-methyl-3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C44H47F2N9O4S
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1
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| 1 |
IC50 = 100 nM
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CP0863042
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[1-(2-fluoroethyl)-4-piperidinyl]-1-piperazinyl]phenyl)amino}-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C43H44F3N9O2
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1
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| 1 |
IC50 < 100 nM
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CP0866109
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N-(2,6-difluorophenyl)-5-(7-fluoro-3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C40H38F3N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0866111
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C38H36F2N8O4S
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1
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| 1 |
IC50 < 100 nM
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CP0866112
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N-(2,6-difluorophenyl)-3-{3-[2-({5-methyl-2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C37H34F2N8O4S
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1
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| 1 |
IC50 < 100 nM
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CP0866113
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N-(2,6-difluorophenyl)-3-(3-(2-((5-methyl-2-(methyloxy)-4-(4-(2-(methylsulfonyl)ethyl)-1-piperidinyl)phenyl)amino)-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C40H39F2N7O4S
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1
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| 1 |
IC50 < 100 nM
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CP0866114
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C37H34F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0866115
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C41H42F2N8O4
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1
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| 1 |
IC50 < 100 nM
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CP0866958
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N-(2,6-difluorophenyl)-3-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N9O4S
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1
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| 1 |
IC50 < 100 nM
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CP0866960
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3-[3-(2-{[4-(4-{bis[2-(methyloxy)ethyl]amino}-1-piperidinyl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C42H44F2N8O4
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1
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| 1 |
IC50 < 100 nM
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CP0866983
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N-(2,6-difluorophenyl)-3-[3-(2-{[5-methyl-2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C44H47F2N9O4S
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1
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| 1 |
IC50 < 100 nM
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CP0866984
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3-[3-(2-{[4-{4-[4-(2,2-difluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(ethyloxy)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C43H43F4N9O2
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1
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| 1 |
IC50 < 100 nM
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CP0866985
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[4-(3,3,3-trifluoropropyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C44H44F5N9O2
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1
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| 1 |
IC50 = 100 nM
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CP0866986
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N-(2,6-difluorophenyl)-5-[3-(2-{[4-(4-hydroxy-1-piperidinyl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
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C37H33F2N7O4
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1
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| 1 |
IC50 < 100 nM
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CP0866988
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N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C40H40F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0866989
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C41H42F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0866990
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C39H38F2N8O4S
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1
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| 1 |
IC50 < 100 nM
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CP0866991
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N-(2,6-difluorophenyl)-3-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C39H38F2N8O4S
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1
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| 1 |
IC50 < 100 nM
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CP0866992
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N-(2,6-difluorophenyl)-3-(3-(2-((2-(ethyloxy)-4-(4-(1-methylethyl)-1-piperazinyl)phenyl)amino)-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C39H38F2N8O2
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1
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| 1 |
IC50 < 100 nM
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CP0866994
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N-(2,6-difluorophenyl)-3-(8-fluoro-3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C41H40F3N9O4S
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1
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| 1 |
IC50 = 100 nM
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CP0866995
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N-(2,6-difluorophenyl)-3-[7-fluoro-3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C42H41F4N9O2
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1
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| 1 |
IC50 = 100 nM
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CP0866996
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5-(3-{2-[(5-chloro-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
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C39H37ClF2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0866997
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N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C42H43F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0867011
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5-(3-(2-(4-(1,4'-bipiperidin-1'-yl)-2-methoxyphenylamino)pyrimidin-4-yl)-7-methoxyimidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)-2-methoxybenzamide
Show/Hide
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C43H44F2N8O4
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1
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| 1 |
IC50 < 100 nM
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CP0867154
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H44F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0867164
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3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(propyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyri-din-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C43H44F2N8O2
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1
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| 1 |
IC50 = 100 nM
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CP0867165
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N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C43H45F2N9O4S
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1
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| 1 |
IC50 < 100 nM
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CP0867166
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3-[3-(2-{[5-chloro-4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C42H41ClF3N9O2
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1
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| 1 |
IC50 < 100 nM
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CP0869257
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-[3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)-ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo-[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C44H47F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0869420
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C41H42F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0870269
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N-(2,6-difluorophenyl)-3-(3-(2-(3-(1-methyl-1H-pyrazol-4-yl)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C34H24F2N8O
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1
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| 1 |
IC50 = 100 nM
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CP0870972
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C42H43F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0870973
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N-(2,6-difluorophenyl)-5-(7-fluoro-3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C41H40F3N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0870974
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C41H41F2N7O4S
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1
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| 1 |
IC50 < 100 nM
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CP0870978
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[2-(methyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C40H40F2N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0870979
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0870980
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(ethyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C43H45F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0870981
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C43H45F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0870983
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C41H41F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0871077
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5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-fluoro-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
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C42H41F3N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0871078
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C40H40F2N8O4
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1
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| 1 |
IC50 < 100 nM
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CP0873426
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3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-fluoro-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C41H39F3N8O2
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1
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| 1 |
IC50 < 100 nM
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CP0873427
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N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[1-(2-methylpropyl)-4-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C40H39F2N7O2
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1
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| 1 |
IC50 < 100 nM
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CP0873428
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-[(3S)-3-hydroxyl-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C36H31F2N7O3
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1
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| 1 |
IC50 = 100 nM
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CP0873429
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N-(2,6-difluorophenyl)-5-[3-(2-{[4-[1-(2-fluoroethyl)-4-piperidinyl]-2-(methyloxy)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
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C39H36F3N7O3
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1
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| 1 |
IC50 < 100 nM
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CP0873430
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C43H45F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0873431
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3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C42H42F2N8O3
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1
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| 1 |
IC50 = 100 nM
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CP0873433
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-[4-(hexahydro-1H-azepin-1-yl)-1-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C42H42F2N8O2
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1
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| 1 |
IC50 < 100 nM
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CP0873434
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N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(trifluoromethyl)-1,4'-bipiperidin-1'-yl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C42H39F5N8O2
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1
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| 1 |
IC50 = 100 nM
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CP0873436
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-[4-(4-ethyl-1-piperazinyl)-1-piperidinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C42H43F2N9O2
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1
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| 1 |
IC50 < 100 nM
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CP0873438
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0873679
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C38H36F2N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0873683
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-3-oxo-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C42H40F3N9O3
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1
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| 1 |
IC50 < 100 nM
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CP0873684
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N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C39H37F2N7O2
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1
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| 1 |
IC50 < 100 nM
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CP0873685
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N-(2,6-difluorophenyl)-3-{3-[2-({2-(ethyloxy)-4-[2-(4-methyl-1-piperazinyl)ethyl]-phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C37H34F2N8O2
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1
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| 1 |
IC50 < 100 nM
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CP0882930
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-[3-(2-{[2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C40H39F2N7O3
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1
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| 1 |
IC50 < 100 nM
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CP0882931
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N-(2,6-difluorophenyl)-5-[3-(2-{[2-(ethyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
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C41H41F2N7O3
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1
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| 1 |
IC50 < 100 nM
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CP0883053
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3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(4-chloro-2-fluorophenyl)benzamide
Show/Hide
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C41H40ClFN8O2
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1
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| 1 |
IC50 = 100 nM
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CP0883055
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[1-(2-methylpropyl)-4-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C41H41F2N7O3
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1
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| 1 |
IC50 < 100 nM
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CP0883056
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[4-[4-(1-methylethyl)-1-piperazinyl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C40H40F2N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0883073
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoro-ethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-8-methylimidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C43H44F3N9O2
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1
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| 1 |
IC50 < 100 nM
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CP0883074
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)-ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C45H49F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0883075
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N-(2,6-difluorophenyl)-5-[3-(2-{[4-{4-[(9aS)-hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
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C44H45F2N9O4
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1
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| 1 |
IC50 < 100 nM
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CP0888258
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C39H38F2N8O4
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1
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| 1 |
IC50 < 100 nM
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CP0888352
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N-(2,6-difluorophenyl)-3-[8-fluoro-3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C43H44F3N9O4S
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1
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| 1 |
IC50 = 100 nM
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CP0888354
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N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-[(1-methylethyl)oxy]benzamide
Show/Hide
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C44H47F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0888370
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N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-[(1-methylethyl)oxy]benzamide
Show/Hide
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C43H46F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0888393
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5-(3-(2-(4-(1,4'-bipiperidin-1'-yl)-2-methoxyphenylamino)pyrimidin-4-yl)-7-methylimidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)-2-methoxybenzamide
Show/Hide
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C43H44F2N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0888395
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3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-propylphenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C43H44F2N8O
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1
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| 1 |
IC50 = 100 nM
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CP0894025
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N-(2,6-difluorophenyl)-3-(8-methyl-3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N9O4S
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1
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| 1 |
IC50 = 100 nM
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CP0894026
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-[(3S)-3-hydroxy-1,4'-bipiperidin-1'-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C41H40F2N8O3
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1
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| 1 |
IC50 = 100 nM
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CP0895685
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N-(2,6-difluorophenyl)-3-(3-(2-(2-methyl-4-(1-(2-(methylsulfonyl)ethyl)piperidin-4-yloxy)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C39H37F2N7O4S
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1
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| 1 |
IC50 = 100 nM
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CP0895686
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[(1S,4S)-5-(2-fluoroethyl)-2,5-diazabicyclo-[2.2.1]hept-2-yl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C43H42F3N9O2
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1
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| 1 |
IC50 < 100 nM
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CP0895687
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1,4'-bipiperidin-1'-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C45H48F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0895688
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C43H44F3N9O2
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1
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| 1 |
IC50 < 100 nM
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CP0895690
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N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C38H36F2N8O2
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1
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| 1 |
IC50 < 100 nM
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CP0895691
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N-(2,6-difluorophenyl)-5-[7-fluoro-3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
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C43H43F4N9O3
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1
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| 1 |
IC50 < 100 nM
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CP0895692
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
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C45H49F2N9O5S
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1
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| 1 |
IC50 < 100 nM
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CP0895693
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(ethyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N9O4S
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1
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| 1 |
IC50 < 100 nM
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CP0899488
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C41H41F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0899726
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C40H39F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0899730
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5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
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C42H42F2N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0899732
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N-(2,6-difluorophenyl)-3-(3-{2-[(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-2-propylphenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C41H41F2N7O3S
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1
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| 1 |
IC50 = 100 nM
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CP0901852
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C39H37F2N7O4S
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1
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| 1 |
IC50 < 100 nM
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CP0901853
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C41H41F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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CP0902860
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3-[3-(2-{[5-chloro-2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-benzamide
Show/Hide
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C43H44ClF2N9O4S
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1
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| 1 |
IC50 < 100 nM
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CP0904970
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N-(2,6-difluorophenyl)-3-[3-(2-{[2-(ethyloxy)-4-(1-propyl-4-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C40H39F2N7O2
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1
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| 1 |
IC50 < 100 nM
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CP0904973
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N-(2,6-difluorophenyl)-5-(3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)-amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C35H31F2N7O3
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1
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| 1 |
IC50 = 100 nM
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CP0904975
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-(4-hydroxy-1-piperidinyl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C36H31F2N7O3
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1
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| 1 |
IC50 = 100 nM
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CP0904979
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N-(2,6-difluorophenyl)-3-(3-{2-[(5-methyl-2-(methyloxy)-4-{4-[2-(methyloxy)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C39H38F2N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0904980
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N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C41H42F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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CP0912085
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N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(trans-4-{4-[2-(methylsulfonyl)-ethyl]-1-piperazinyl}cyclohexyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C44H46F2N8O4S
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1
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| 1 |
IC50 = 100 nM
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CP0912086
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-{3-[2-({2-(methyloxy)-4-[3-(4-methyl-1-piperazinyl)propyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C40H40F2N8O3
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1
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| 1 |
IC50 < 100 nM
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CP0912113
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3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-methylimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C42H42F2N8O2
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1
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| 1 |
IC50 = 100 nM
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CP0912114
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N-(2,6-difluorophenyl)-3-[3-(2-{[2-(methyloxy)-4-(4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}-1-piperidinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C43H45F2N9O4S
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1
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| 1 |
IC50 < 100 nM
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|
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CP0912117
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-5-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C43H44F3N9O2
|
1
|
| 1 |
IC50 < 100 nM
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|
|
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CP0913017
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N-(2,6-difluorophenyl)-3-(3-(2-(2-methoxy-4-(4-(4-methyl-1,4-diazepan-1-yl)piperidin-1-yl)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N9O2
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1
|
| 1 |
IC50 = 100 nM
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|
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CP0913020
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N-(2,6-difluorophenyl)-3-[3-(2-{[2-(ethyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C39H38F2N8O2
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1
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| 1 |
IC50 < 100 nM
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|
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CP0913021
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl]-2-propylphenyl)amino}-4-pyrimidinyl}imidazo[1,2a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N7O4S
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1
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| 1 |
IC50 < 100 nM
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|
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CP0913022
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N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C40H39F2N7O5S
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1
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| 1 |
IC50 < 100 nM
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|
|
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CP0913023
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-ethyl-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(ethyloxy)benzamide
Show/Hide
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C42H44F2N8O5S
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1
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| 1 |
IC50 < 100 nM
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|
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CP0913162
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5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
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C43H44F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
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|
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CP0913163
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3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-fluoroimidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
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C41H39F3N8O2
|
1
|
| 1 |
IC50 < 100 nM
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|
|
|
CP0913164
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N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-5-methyl-4-{4-[2-(methylsulfonyl)ethyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}-7-fluoroimidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C42H42F3N7O5S
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1
|
| 1 |
IC50 < 100 nM
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|
|
|
CP0913166
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-{3-[2-({2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C38H36F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
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|
|
|
CP0913167
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N-(2,6-difluorophenyl)-3-(3-{2-[(2-(methyloxy)-4-{4-[(4-methyl-1-piperazinyl)methyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
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C42H43F2N9O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0919429
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N-(2,6-difluorophenyl)-5-(3-{2-[(5-methyl-2-(methyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C41H41F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
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CP0919430
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N-(2,6-difluorophenyl)-5-(7-fluoro-3-{2-[(2-(methyloxy)-4-{4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
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C42H42F3N9O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0919431
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N-(2,6-difluorophenyl)-3-{3-[2-({2-(methyloxy)-4-[4-(methylsulfonyl)-1-piperazinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C36H32F2N8O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0920901
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N-(2,6-difluorophenyl)-2-(ethyloxy)-5-{3-[2-({2-(methyloxy)-4-[1-(2-methylpropyl)-4-piperidinyl]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
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C42H43F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921734
|
N-(2,6-difluorophenyl)-5-{3-[2-({2-(ethyloxy)-4-[4-(1-methylethyl)-1-piperazinyl]phenyl}-amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
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C40H40F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921735
|
N-(2,6-difluorophenyl)-5-(3-{2-[(2-(ethyloxy)-4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-2-(methyloxy)benzamide
Show/Hide
|
C41H41F2N7O5S
|
1
|
| 1 |
IC50 < 100 nM
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|
|
|
CP0921758
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,4-difluorophenyl)benzamide
Show/Hide
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C41H40F2N8O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0921759
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-(4-hydroxy-1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
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C42H42F2N8O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0923165
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N-(2,6-difluorophenyl)-3-[3-(2-{[4-(4-fluoro-1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
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C41H39F3N8O2
|
1
|
| 1 |
IC50 = 100 nM
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|
|
|
CP0924036
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-[3-(2-{[2-(ethyloxy)-4-(4-propyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C41H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0926153
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2-chloro-4-fluorophenyl)benzamide
Show/Hide
|
C41H40ClFN8O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0926162
|
N-(2,6-difluorophenyl)-2-(ethyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1,4'-bipiperidin-1'-yl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C46H50F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0926163
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-5-chloro-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C42H41ClF2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0928839
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidinyl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C43H44F3N9O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0928846
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-ethylphenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0928847
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-[1'-(2-fluoroethyl)-4,4'-bipiperidin-1-yl]-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C44H45F3N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0929056
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-(ethyloxy)-4-(4-{1-[2-(methylsulfonyl)ethyl]-4-piperidinyl}-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C44H47F2N9O4S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0929069
|
5-(3-{2-[(5-chloro-2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)-N-(2,6-difluorophenyl)-2-(ethyloxy)benzamide
Show/Hide
|
C41H41ClF2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0944904
|
N-(2,6-difluorophenyl)-2-(methyloxy)-5-(3-{2-[(2-(methyloxy)-4-{4-[2-(methylsulfonyl)ethyl]-1-piperazinyl}phenyl)amino]-4-pyrimidinyl}imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C39H38F2N8O5S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0946200
|
N-(2,6-difluorophenyl)-5-[3-(2-{[5-methyl-2-(methyloxy)-4-(1-propyl-4-piperidinyl)phenyl]-amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C41H41F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0946229
|
N-(2,6-difluorophenyl)-2-isopropoxy-5-{3-[2-({2-methoxy-4-[2-(4-methylpiperazin-1-yl)ethyl]phenyl}amino)pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl}benzamide
Show/Hide
|
C41H42F2N8O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0952419
|
N-(2,4-difluorophenyl)-3-[3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C35H31F2N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0848469
|
3-{3-[2-({4-(1,4'-bipiperidin-1'-yl)-2-[(2-methylpropyl)oxy]phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C44H46F2N8O2
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0848489
|
N-(2,6-difluorophenyl)-3-(3-(2-(2-methyl-4-(1-methylpiperidin-4-yloxy)phenylamino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)benzamide
Show/Hide
|
C37H33F2N7O2
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0848538
|
N-(2,6-difluorophenyl)-3-[3-(2-{[2-methyl-4-(4-piperidinyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C36H31F2N7O2
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0848539
|
N-(2,3-difluorophenyl)-3-[3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C35H31F2N7O3
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0856496
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{4-[4-(2-fluoroethyl)-1-piperazinyl]-1-piperidin}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C43H41F6N9O2
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0857319
|
N-(2,6-difluorophenyl)-5-{3-[2-({2-(ethyloxy)-4-[2-(4-methyl-1-piperazinyl)ethyl]-phenyl}amino)-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl}-2-(methyloxy)benzamide
Show/Hide
|
C38H36F2N8O3
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0866116
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)-7-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H39F5N8O2
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0866959
|
N-(2,6-difluorophenyl)-3-[3-{2-[(3-{[2-(dimethylamino)ethyl]oxy}phenyl)amino]-4-pyrimidinyl}-7-(methyloxy)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C35H31F2N7O3
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0873432
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-(2-methylpropyl)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C44H46F2N8O
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0888394
|
N-(2,6-difluorophenyl)-3-[3-(2-{[4-{5-[(dimethylamino)methyl]-1,3,4-oxadiazol-2-yl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]benzamide
Show/Hide
|
C36H29F2N9O3
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0895724
|
N-(2,6-difluorophenyl)-5-(3-(2-(3-(2-(dimethylamino)ethoxy)phenylamino)pyrimidin-4-yl)-7-methylimidazo[1,2-a]pyridin-2-yl)-2-methoxybenzamide
Show/Hide
|
C36H33F2N7O3
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0913168
|
5-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-3-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)-2-(methyloxy)benzamide
Show/Hide
|
C43H44F2N8O3
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0921733
|
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-3-methyl-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
Show/Hide
|
C42H42F2N8O2
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0923164
|
N-(2,6-difluorophenyl)-5-[3-(2-{[4-{5-[(dimethylamino)methyl]-1,3,4-oxadiazol-2-yl}-2-(methyloxy)phenyl]amino}-4-pyrimidinyl)imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide
Show/Hide
|
C37H31F2N9O4
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
