| Compound ID |
Compound Name |
Compound Formula |
|
CP0388224
|
4-((1H-Imidazol-4-yl)methyl)-1-(3-(trifluoromethyl)-phenyl)piperidine
Show/Hide
|
C16H18F3N3
|
1
|
| 1 |
EC50 = 0.21 nM
|
|
|
|
CP0110239
|
4-(1H-imidazol-4-ylmethyl)piperidine
Show/Hide
|
C9H15N3
|
1
|
| 1 |
EC50 = 0.67 nM
|
|
|
|
CP0092861
|
2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole
Show/Hide
|
C15H20N2S
|
1
|
| 1 |
EC50 = 0.75 nM
|
|
|
|
CP0400527
|
4-((1H-Imidazol-4-yl)methyl)-1-(4-fluorophenyl)piperidine
Show/Hide
|
C15H18FN3
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0438775
|
4-((1H-Imidazol-4-yl)methyl)-1-(4-(trifluoromethyl)-phenyl)piperidine
Show/Hide
|
C16H18F3N3
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0400521
|
4-((1H-Imidazol-4-yl)methyl)-1-(naphthalen-2-yl)piperidine
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|
C19H21N3
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0418459
|
4-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)-N-methylaniline
Show/Hide
|
C16H22N4
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0428302
|
4-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)-N,N-dimethylaniline
Show/Hide
|
C17H24N4
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0400519
|
4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)piperidine
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|
C16H21N3O
|
1
|
| 1 |
EC50 = 7.6 nM
|
|
|
|
CP0400529
|
4-((1H-Imidazol-4-yl)methyl)-1-(4-nitrophenyl)piperidine
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|
C15H18N4O2
|
1
|
| 1 |
EC50 = 8.8 nM
|
|
|
|
CP0400265
|
4-((1H-Imidazol-4-yl)methyl)-1-(4-isopropylphenyl)piperidine
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|
C18H25N3
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0388225
|
4-((1H-Imidazol-4-yl)methyl)-1-(4-tert-butylphenyl)piperidine
Show/Hide
|
C19H27N3
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0400525
|
4-((1H-Imidazol-4-yl)methyl)-1-phenylpiperidine
Show/Hide
|
C15H19N3
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0400523
|
3-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)pyridine
Show/Hide
|
C14H18N4
|
1
|
| 1 |
EC50 = 177 nM
|
|
|
|
CP0279719
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-2,5-dimethyl-4(3H)-quinazolinone
Show/Hide
|
C25H29N3O2
|
2
|
| 1 |
IC50 = 0.27 nM
|
|
|
| 2 |
Ki = 1.7 nM
|
|
|
|
CP0094412
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methyl-5-(trifluoromethyl)-4(3H)-quinazolinone
Show/Hide
|
C25H26F3N3O2
|
2
|
| 1 |
IC50 = 0.33 nM
|
|
|
| 2 |
Ki = 3.6 nM
|
|
|
|
CP0506284
|
5-Chloro-3-(4-[(1-cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H26ClN3O2
|
1
|
| 1 |
IC50 = 0.34 nM
|
|
|
|
CP0193419
|
6-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)-N-methylnicotinamide
Show/Hide
|
C21H25N3O2
|
2
|
| 1 |
IC50 = 0.55 nM
|
|
|
| 2 |
Ki = 0.1995 nM
|
|
|
|
CP0221898
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-5-fluoro-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H26FN3O2
|
2
|
| 1 |
IC50 = 0.55 nM
|
|
|
| 2 |
Ki = 6.8 nM
|
|
|
|
CP0194592
|
(R)-4-(2-(2-(2-methylpyrrolidin-1-yl)ethyl)benzofuran-5-yl)benzonitrile
Show/Hide
|
C22H22N2O
|
1
|
| 1 |
IC50 = 0.63 nM
|
|
|
|
CP0232075
|
2-Phenyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
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|
C27H27N3O2
|
1
|
| 1 |
IC50 = 0.66 nM
|
|
|
|
CP0202877
|
2-Propyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 0.69 nM
|
|
|
|
CP0372646
|
2-Methyl-3-[4-({3-[(3S)-3-methyl-1-piperidinyl]propyl}oxy)phenyl]-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 0.72 nM
|
|
|
|
CP0533600
|
(4-cyclobutyl-1,4-diazepan-1-yl)-[7-(oxan-4-yl)-7-azaspiro[3.5]nonan-2-yl]methanone
Show/Hide
|
C23H39N3O2
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0305864
|
2-Isopropyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 0.81 nM
|
|
|
|
CP0485614
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-8-fluoro-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H26FN3O2
|
1
|
| 1 |
IC50 = 0.84 nM
|
|
|
|
CP0432409
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-6,7-difluoro-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H25F2N3O2
|
1
|
| 1 |
IC50 = 0.91 nM
|
|
|
|
CP0297753
|
2-Methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-7-(trifluoromethyl)-4(3H)-quinazolinone
Show/Hide
|
C23H24F3N3O2
|
1
|
| 1 |
IC50 = 0.96 nM
|
|
|
|
CP0206060
|
2,5-Dimethyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 0.98 nM
|
|
|
|
CP0206059
|
6-Methoxy-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0387559
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-5-methoxy-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0441445
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-6-fluoro-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H26FN3O2
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0090649
|
2,7-Dimethyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0434956
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-7-fluoro-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H26FN3O2
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0290003
|
5-Chloro-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C22H24ClN3O2
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0305863
|
5-Methoxy-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0434957
|
6-Chloro-3-(4-[(1-cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H26ClN3O2
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0469710
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H27N3O2
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0475040
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-6-methoxy-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0305862
|
8-Fluoro-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C22H24FN3O2
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0497930
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methylpyrido[2,3-d]pyrimidin-4(3H)-one
Show/Hide
|
C23H26N4O2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0218857
|
6-Fluoro-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C22H24FN3O2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0291530
|
2-Ethyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0522483
|
3-(4-{[3-(1-Azepanyl)propyl]oxy}phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0481276
|
(4-cyclohexylpiperazin-1-yl)-[7-(oxan-4-yl)-7-azaspiro[3.5]nonan-2-yl]methanone
Show/Hide
|
C24H41N3O2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0305865
|
2-Methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C22H25N3O2
|
2
|
| 1 |
IC50 = 1.7 nM
|
|
|
| 2 |
IC50 = 3.5 nM
|
|
|
|
CP0485617
|
8-Chloro-3-(4-[(1-cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H26ClN3O2
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0142753
|
2,8-Dimethyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0164197
|
2-Methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-5-(trifluoromethyl)-4(3H)-quinazolinone
Show/Hide
|
C23H24F3N3O2
|
3
|
| 1 |
IC50 = 1.7 nM
|
|
|
| 2 |
Kd = 0.631 nM
|
|
|
| 3 |
Ki = 6.8 nM
|
|
|
|
CP0473254
|
[7-(oxan-4-yl)-7-azaspiro[3.5]nonan-2-yl]-(4-propan-2-ylpiperazin-1-yl)methanone
Show/Hide
|
C21H37N3O2
|
2
|
| 1 |
IC50 = 1.7 nM
|
|
|
| 2 |
Ki = 0.3 nM
|
|
|
|
CP0373082
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methylpyrido[3,4-d]pyrimidin-4(3H)-one
Show/Hide
|
C23H26N4O2
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0399776
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-7-methoxy-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0073728
|
7-Fluoro-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C22H24FN3O2
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0121871
|
(4-cyclobutylpiperazin-1-yl)-[7-(oxan-4-yl)-7-azaspiro[3.5]nonan-2-yl]methanone
Show/Hide
|
C22H37N3O2
|
1
|
| 1 |
IC50 = 1.9 nM
|
|
|
|
CP0510140
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methylpyrido[4,3-d]pyrimidin-4(3H)-one
Show/Hide
|
C23H26N4O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0206057
|
5-Fluoro-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C22H24FN3O2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0313614
|
2-Methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-8-(trifluoromethyl)-4(3H)-quinazolinone
Show/Hide
|
C23H24F3N3O2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0490845
|
2-Methyl-3-[4-({3-[(2S)-2-methyl-1-pyrrolidinyl]propyl}oxy)phenyl]-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0310817
|
7-Methoxy-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0047136
|
(2R)-1-(1H-imidazol-5-yl)propan-2-amine
Show/Hide
|
C6H11N3
|
2
|
| 1 |
IC50 = 2.3 nM
|
|
|
| 2 |
Ki = 1.1 nM
|
|
|
|
CP0422118
|
[8-(benzenesulfonyl)-2,8-diazaspiro[4.5]decan-2-yl]-(4-cyclobutyl-1,4-diazepan-1-yl)methanone
Show/Hide
|
C24H36N4O3S
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
|
CP0387558
|
7-Chloro-3-(4-[(1-cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H26ClN3O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0372875
|
2-Methyl-3-(4-{[3-(1-piperidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0490646
|
3-(4-[(1-Cyclopentyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C25H29N3O2
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0422088
|
[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]-(4-propan-2-ylpiperazin-1-yl)methanone
Show/Hide
|
C20H35N3O2
|
2
|
| 1 |
IC50 = 3.2 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0422092
|
(4-cyclobutyl-1,4-diazepan-1-yl)-(8-propan-2-ylsulfonyl-2,8-diazaspiro[4.5]decan-2-yl)methanone
Show/Hide
|
C21H38N4O3S
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0231381
|
3-(4-{[3-(1-Pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C21H23N3O2
|
1
|
| 1 |
IC50 = 3.5 nM
|
|
|
|
CP0422251
|
(4-cyclobutylpiperazin-1-yl)-[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]methanone
Show/Hide
|
C21H35N3O2
|
2
|
| 1 |
IC50 = 3.6 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0467079
|
[2-(4-cyclobutyl-1,4-diazepane-1-carbonyl)-2,8-diazaspiro[4.5]decan-8-yl]-phenylmethanone
Show/Hide
|
C25H36N4O2
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0296479
|
8-Methoxy-2-methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone trifluoroacetate
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0231995
|
2,6-Dimethyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0422082
|
[2-(4-cyclobutyl-1,4-diazepane-1-carbonyl)-2,9-diazaspiro[4.5]decan-9-yl]-phenylmethanone
Show/Hide
|
C25H36N4O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0373081
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-8-methoxy-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
IC50 = 4.2 nM
|
|
|
|
CP0437940
|
2-Methyl-3-[4-({3-[(2R)-2-methyl-1-pyrrolidinyl]propyl}oxy)phenyl]-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
|
CP0487073
|
(4-cyclobutyl-1,4-diazepan-1-yl)-[9-(oxan-4-yl)-2,9-diazaspiro[4.5]decan-2-yl]methanone
Show/Hide
|
C23H40N4O2
|
1
|
| 1 |
IC50 = 4.4 nM
|
|
|
|
CP0102038
|
2-(1-cyclobutylpiperidin-4-yl)-6-(1-cyclobutylpiperidin-4-yl)oxy-3,4-dihydroisoquinolin-1-one
Show/Hide
|
C27H39N3O2
|
1
|
| 1 |
IC50 = 4.8 nM
|
|
|
|
CP0498998
|
2-Methyl-3-(4-{[3-(3-methyl-1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 5.8 nM
|
|
|
|
CP0458806
|
1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl-[7-(oxan-4-yl)-7-azaspiro[3.5]nonan-2-yl]methanone
Show/Hide
|
C22H37N3O2
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0467077
|
[7-(benzenesulfonyl)-2,7-diazaspiro[4.5]decan-2-yl]-(4-cyclobutyl-1,4-diazepan-1-yl)methanone
Show/Hide
|
C24H36N4O3S
|
1
|
| 1 |
IC50 = 6.5 nM
|
|
|
|
CP0452149
|
4-((1H-Imidazol-4-yl)methyl)-1-(3-isopropylphenyl)piperidine
Show/Hide
|
C18H25N3
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
|
CP0432410
|
3-(4-[(1-Cyclopentyl-4-azepanyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C26H31N3O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0225036
|
[(2S)-6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]-(4-propan-2-ylpiperazin-1-yl)methanone
Show/Hide
|
C20H35N3O2
|
2
|
| 1 |
IC50 = 8.3 nM
|
|
|
| 2 |
Ki = 0.8 nM
|
|
|
|
CP0469125
|
(4-cyclopentylpiperazin-1-yl)-[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]methanone
Show/Hide
|
C22H37N3O2
|
2
|
| 1 |
IC50 = 8.8 nM
|
|
|
| 2 |
Ki = 1.4 nM
|
|
|
|
CP0434955
|
2-methyl-3-[4-(4-pyrrolidin-1-ylcyclohexyl)oxyphenyl]quinazolin-4-one
Show/Hide
|
C25H29N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0468526
|
3-(4-[(1-Cyclobutyl-4-azepanyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C25H29N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0437715
|
3-(4-{[3-(1-Azocanyl)propyl]oxy}phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C25H31N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0422090
|
(6-cyclohexyl-6-azaspiro[2.5]octan-2-yl)-(4-cyclohexylpiperazin-1-yl)methanone
Show/Hide
|
C24H41N3O
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
Ki = 19 nM
|
|
|
|
CP0522482
|
2-Methyl-3-(4-{[3-(2-methyl-1-piperidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0566246
|
(4-cyclobutylpiperazin-1-yl)-(7-methylsulfonyl-7-azaspiro[3.5]nonan-2-yl)methanone
Show/Hide
|
C18H31N3O3S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0119048
|
1-(3-(3-(4-chlorophenyl)propoxy)propyl)piperidine
Show/Hide
|
C17H26ClNO
|
4
|
| 1 |
IC50 = 12 nM
|
|
|
| 2 |
Ki = 2.4 nM
|
|
|
| 3 |
Ki = 2.512 nM
|
|
|
| 4 |
Ki = 30 nM
|
|
|
|
CP0487028
|
(7-benzoyl-7-azaspiro[3.5]nonan-2-yl)-(4-propan-2-yl-1,4-diazepan-1-yl)methanone
Show/Hide
|
C24H35N3O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0555257
|
(4-cyclohexylpiperazin-1-yl)-[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]methanone
Show/Hide
|
C23H39N3O2
|
2
|
| 1 |
IC50 = 12 nM
|
|
|
| 2 |
Ki = 26 nM
|
|
|
|
CP0487070
|
[2-(4-cyclobutylpiperazine-1-carbonyl)-2,8-diazaspiro[4.5]decan-8-yl]-phenylmethanone
Show/Hide
|
C24H34N4O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0417400
|
3-(4-[(1-Isopropyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0522566
|
3-(4-[(1-Cyclobutyl-4-piperidinyl)oxy]phenyl)-2-methylpyrido[3,2-d]pyrimidin-4(3H)-one
Show/Hide
|
C23H26N4O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0422253
|
[7-(oxan-4-yl)-7-azaspiro[3.5]nonan-2-yl]-(4-propan-2-yl-1,4-diazepan-1-yl)methanone
Show/Hide
|
C22H39N3O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0102037
|
6-(1-propan-2-ylpiperidin-4-yl)oxy-2-(1-propan-2-ylpyrrolidin-3-yl)-3,4-dihydroisoquinolin-1-one
Show/Hide
|
C24H37N3O2
|
1
|
| 1 |
IC50 = 14.3 nM
|
|
|
|
CP0422250
|
(4-cyclohexylpiperazin-1-yl)-[6-(2-phenylethyl)-6-azaspiro[2.5]octan-2-yl]methanone
Show/Hide
|
C26H39N3O
|
2
|
| 1 |
IC50 = 16 nM
|
|
|
| 2 |
Ki = 21 nM
|
|
|
|
CP0555258
|
(4-cyclobutyl-1,4-diazepan-1-yl)-[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]methanone
Show/Hide
|
C22H37N3O2
|
2
|
| 1 |
IC50 = 17 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0478595
|
[2-(4-cyclobutyl-1,4-diazepane-1-carbonyl)-2,9-diazaspiro[5.5]undecan-9-yl]-phenylmethanone
Show/Hide
|
C26H38N4O2
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0467078
|
(4-cyclopropylpiperazin-1-yl)-[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]methanone
Show/Hide
|
C20H33N3O2
|
2
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
Ki = 11 nM
|
|
|
|
CP0487074
|
(4-cyclohexylpiperazin-1-yl)-(6-propan-2-yl-6-azaspiro[2.5]octan-2-yl)methanone
Show/Hide
|
C21H37N3O
|
2
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
Ki = 47 nM
|
|
|
|
CP0437941
|
3-[4-({3-[(2R,5R)-2,5-Dimethyl-1-pyrrolidinyl]propyl}oxy)phenyl]-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0165491
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-morpholin-4-ylacetamide;dihydrochloride
Show/Hide
|
C21H33Cl2N3O3
|
2
|
| 1 |
IC50 = 20 nM
|
|
|
| 2 |
Ki = 8.73 nM
|
|
|
|
CP0471261
|
[8-(benzenesulfonyl)-2,8-diazaspiro[4.5]decan-2-yl]-(4-cyclobutylpiperazin-1-yl)methanone
Show/Hide
|
C23H34N4O3S
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0474653
|
2-Methyl-3-(4-{[3-(4-methyl-1-piperidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0499008
|
3-(4-{[3-(3,5-Dimethyl-1-piperidinyl)propyl]oxy}phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C25H31N3O2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0489305
|
[8-(oxan-4-yl)-2,8-diazaspiro[4.5]decan-2-yl]-(4-propan-2-ylpiperazin-1-yl)methanone
Show/Hide
|
C21H38N4O2
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0498997
|
3-(4-{[3-(Diethylamino)propyl]oxy}phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0387557
|
3-(4-[(1-Cyclopentyl-3-pyrrolidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H27N3O2
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0474756
|
2-Methyl-3-[4-({3-[(3R)-3-methyl-1-piperidinyl]propyl}oxy)phenyl]-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0387556
|
3-(4-[(1-Cyclohexyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C26H31N3O2
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0478593
|
(7-benzoyl-7-azaspiro[3.5]nonan-2-yl)-(4-cyclobutylpiperazin-1-yl)methanone
Show/Hide
|
C24H33N3O2
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0526157
|
3-(4-[(1-Ethyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C22H25N3O2
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0441444
|
2-Methyl-3-(4-[(1-propyl-4-piperidinyl)oxy]phenyl)-4(3H)-quinazolinone
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0422084
|
(4-cyclobutylpiperazin-1-yl)-(7-phenyl-7-azaspiro[3.5]nonan-2-yl)methanone
Show/Hide
|
C23H33N3O
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0533599
|
(6-cyclobutyl-6-azaspiro[2.5]octan-2-yl)-[4-(oxan-4-yl)piperazin-1-yl]methanone
Show/Hide
|
C21H35N3O2
|
2
|
| 1 |
IC50 = 66 nM
|
|
|
| 2 |
Ki = 67 nM
|
|
|
|
CP0487029
|
(4-cycloheptylpiperazin-1-yl)-[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]methanone
Show/Hide
|
C24H41N3O2
|
2
|
| 1 |
IC50 = 74 nM
|
|
|
| 2 |
Ki = 65 nM
|
|
|
|
CP0450897
|
1-naphthalen-1-yl-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C24H27N3O4S
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0478594
|
(4-cyclohexylpiperazin-1-yl)-(6-pyridin-4-yl-6-azaspiro[2.5]octan-2-yl)methanone
Show/Hide
|
C23H34N4O
|
2
|
| 1 |
IC50 = 83 nM
|
|
|
| 2 |
Ki = 55 nM
|
|
|
|
CP0489300
|
[(2R)-6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]-(4-propan-2-ylpiperazin-1-yl)methanone
Show/Hide
|
C20H35N3O2
|
2
|
| 1 |
IC50 = 87 nM
|
|
|
| 2 |
Ki = 16 nM
|
|
|
|
CP0400970
|
3-(4-[(1-Butyl-4-piperidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C24H29N3O2
|
1
|
| 1 |
IC50 = 91 nM
|
|
|
|
CP0373079
|
3-(4-[(1-Cyclobutyl-3-pyrrolidinyl)oxy]phenyl)-2-methyl-4(3H)-quinazolinone
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
IC50 = 103 nM
|
|
|
|
CP0513749
|
4-(3-piperidin-1-ylpropoxy)benzenesulfonamide
Show/Hide
|
C14H22N2O3S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0487072
|
[9-(oxan-4-yl)-2,9-diazaspiro[4.5]decan-2-yl]-(4-propan-2-ylpiperazin-1-yl)methanone
Show/Hide
|
C21H38N4O2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0567009
|
[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]-(4-pyridin-4-ylpiperazin-1-yl)methanone
Show/Hide
|
C22H32N4O2
|
2
|
| 1 |
IC50 = 140 nM
|
|
|
| 2 |
Ki = 8.4 nM
|
|
|
|
CP0044460
|
N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
Show/Hide
|
C15H24N4S
|
4
|
| 1 |
IC50 = 140 nM
|
|
|
| 2 |
Ki = 6.5 nM
|
|
|
| 3 |
Ki = 60 nM
|
|
|
| 4 |
Ki = 602.56 nM
|
|
|
|
CP0433491
|
1-phenyl-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C20H25N3O4S
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0392107
|
US8748435, 39
Show/Hide
|
C27H39N5
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0467379
|
4-(3-pyrrolidin-1-ylpropoxy)benzenesulfonamide
Show/Hide
|
C13H20N2O3S
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0181076
|
4-(1-cyclopentylpiperidin-4-yl)oxy-N-(1-propan-2-ylpyrrolidin-3-yl)benzamide
Show/Hide
|
C24H37N3O2
|
1
|
| 1 |
IC50 = 273.9 nM
|
|
|
|
CP0389075
|
2-ethyl-6,8-dimethyl-3-[[4-[(E)-3-(4-propan-2-ylpiperazin-1-yl)prop-1-enyl]phenyl]methyl]imidazo[1,2-b]pyridazine
Show/Hide
|
C27H37N5
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0428245
|
1-(4-methylphenyl)-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C21H27N3O4S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0430661
|
1-(4-acetylphenyl)-3-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C23H29N3O5S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0045343
|
4-(1-propan-2-ylpiperidin-4-yl)oxy-N-(1-propan-2-ylpyrrolidin-3-yl)benzamide
Show/Hide
|
C22H35N3O2
|
1
|
| 1 |
IC50 = 323.8 nM
|
|
|
|
CP0910622
|
CAMIZESTRANT
Show/Hide
|
C24H28F4N6
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0414587
|
(8-benzoyl-2,8-diazaspiro[4.5]decan-2-yl)-(1-cyclobutylpiperidin-4-yl)methanone
Show/Hide
|
C25H35N3O2
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0388226
|
4-((1H-Imidazol-4-yl)methyl)-1-(biphenyl-4-yl)piperidine
Show/Hide
|
C21H23N3
|
1
|
| 1 |
IC50 = 347 nM
|
|
|
|
CP0489302
|
6-azaspiro[2.5]octan-2-yl-(4-cyclohexylpiperazin-1-yl)methanone
Show/Hide
|
C18H31N3O
|
2
|
| 1 |
IC50 = 360 nM
|
|
|
| 2 |
Ki = 439 nM
|
|
|
|
CP0430662
|
4-(4-piperidin-1-ylbutoxy)benzenesulfonamide
Show/Hide
|
C15H24N2O3S
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0446950
|
1-(4-acetylphenyl)-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C22H27N3O5S
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0494645
|
1-(4-methylphenyl)-3-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C22H29N3O4S
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0521447
|
4-(3-morpholin-4-ylpropoxy)benzenesulfonamide
Show/Hide
|
C13H20N2O4S
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0305594
|
N-[1-(2-methylpropyl)pyrrolidin-3-yl]-4-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
Show/Hide
|
C23H37N3O2
|
1
|
| 1 |
IC50 = 458.7 nM
|
|
|
|
CP0430660
|
1-benzhydryl-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C27H31N3O4S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0433489
|
1-[4-(dimethylamino)phenyl]-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C22H30N4O4S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0521446
|
1-benzhydryl-3-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C28H33N3O4S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0467380
|
4-(4-pyrrolidin-1-ylbutoxy)benzenesulfonamide
Show/Hide
|
C14H22N2O3S
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0522565
|
2-Methyl-3-(4-[(1-methyl-4-piperidinyl)oxy]phenyl)-4(3H)-quinazolinone
Show/Hide
|
C21H23N3O2
|
1
|
| 1 |
IC50 = 740 nM
|
|
|
|
CP0538065
|
2-methyl-3-[4-(4-pyrrolidin-1-ylcyclohexyl)oxyphenyl]quinazolin-4-one
Show/Hide
|
C25H29N3O2
|
1
|
| 1 |
IC50 = 813 nM
|
|
|
|
CP0446948
|
1-phenyl-3-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
|
C21H27N3O4S
|
1
|
| 1 |
IC50 = 830 nM
|
|
|
|
CP0404255
|
2-ethyl-5,7-dimethyl-3-[[4-[(E)-3-(4-propan-2-ylpiperazin-1-yl)prop-1-enyl]phenyl]methyl]pyrazolo[1,5-a]pyrimidine
Show/Hide
|
C27H37N5
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0381038
|
[7-(oxan-4-yl)-2,7-diazaspiro[3.5]nonan-2-yl]-(4-propan-2-ylpiperazin-1-yl)methanone
Show/Hide
|
C20H36N4O2
|
2
|
| 1 |
IC50 = 900 nM
|
|
|
| 2 |
Ki = 97 nM
|
|
|
|
CP0314508
|
US8748435, 40
Show/Hide
|
C27H37N5
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0422089
|
(4-methylpiperazin-1-yl)-[6-(oxan-4-yl)-6-azaspiro[2.5]octan-2-yl]methanone
Show/Hide
|
C18H31N3O2
|
2
|
| 1 |
IC50 = 1100 nM
|
|
|
| 2 |
Ki = 1300 nM
|
|
|
|
CP0428900
|
1-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonyl-3-propan-2-ylurea
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C18H29N3O4S
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1
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| 1 |
IC50 = 1330 nM
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CP0444058
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1-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonyl-3-[4-(trifluoromethyl)phenyl]urea
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C22H26F3N3O4S
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1
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| 1 |
IC50 = 1740 nM
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CP0437712
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1-(2,5-dichlorophenyl)-3-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonylurea
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C21H25Cl2N3O4S
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1
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| 1 |
IC50 = 2570 nM
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CP0411514
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4-[3-[4-[(2-ethyl-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]phenyl]propyl]-1-propan-2-ylpiperidin-4-ol
Show/Hide
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C28H40N4O
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1
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| 1 |
IC50 = 2600 nM
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CP0428897
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1-phenyl-3-[4-(4-piperidin-1-ylbutoxy)phenyl]sulfonylurea
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C22H29N3O4S
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1
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| 1 |
IC50 = 4850 nM
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CP0430657
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1-cyclohexyl-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
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C20H31N3O4S
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1
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| 1 |
IC50 = 6060 nM
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CP0450452
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4-(2-pyrrolidin-1-ylethoxy)benzenesulfonamide
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C12H18N2O3S
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1
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| 1 |
IC50 = 7060 nM
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CP0494646
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1-(2,5-dichlorophenyl)-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
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C20H23Cl2N3O4S
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1
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| 1 |
IC50 = 8310 nM
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CP0467405
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1-[4-(4-piperidin-1-ylbutoxy)phenyl]sulfonyl-3-[4-(trifluoromethyl)phenyl]urea
Show/Hide
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C23H28F3N3O4S
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1
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| 1 |
IC50 = 10000 nM
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CP0474050
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1-phenyl-3-[4-(2-piperidin-1-ylethoxy)phenyl]sulfonylurea
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C20H25N3O4S
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1
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| 1 |
IC50 = 10000 nM
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CP0522900
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4-(2-piperidin-1-ylethoxy)benzenesulfonamide
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C13H20N2O3S
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1
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| 1 |
IC50 = 10000 nM
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CP0428904
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1-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonyl-3-[2-(trifluoromethyl)phenyl]urea
Show/Hide
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C22H26F3N3O4S
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1
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| 1 |
IC50 = 10400 nM
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CP0428898
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1-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonyl-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
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C21H24F3N3O4S
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1
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| 1 |
IC50 = 11800 nM
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CP0444062
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1-(2,5-dichlorophenyl)-3-[4-(4-piperidin-1-ylbutoxy)phenyl]sulfonylurea
Show/Hide
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C22H27Cl2N3O4S
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1
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| 1 |
IC50 = 13200 nM
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CP0428433
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1-propan-2-yl-3-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
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C17H27N3O4S
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1
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| 1 |
IC50 = 13400 nM
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CP0489103
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1-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]sulfonyl-3-[4-(trifluoromethyl)phenyl]urea
Show/Hide
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C21H24F3N3O4S
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1
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| 1 |
IC50 = 16500 nM
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CP0437709
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1-[4-(2-piperidin-1-ylethoxy)phenyl]sulfonyl-3-propan-2-ylurea
Show/Hide
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C17H27N3O4S
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1
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| 1 |
IC50 = 16600 nM
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CP0437703
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1-(2,5-dichlorophenyl)-3-[4-(4-pyrrolidin-1-ylbutoxy)phenyl]sulfonylurea
Show/Hide
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C21H25Cl2N3O4S
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1
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| 1 |
IC50 = 17500 nM
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CP0389786
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1-phenyl-3-[4-(4-pyrrolidin-1-ylbutoxy)phenyl]sulfonylurea
Show/Hide
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C21H27N3O4S
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1
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| 1 |
IC50 = 18000 nM
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CP0430659
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1-[4-(4-piperidin-1-ylbutoxy)phenyl]sulfonyl-3-propan-2-ylurea
Show/Hide
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C19H31N3O4S
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1
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| 1 |
IC50 = 18500 nM
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CP0430658
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1-propan-2-yl-3-[4-(4-pyrrolidin-1-ylbutoxy)phenyl]sulfonylurea
Show/Hide
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C18H29N3O4S
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1
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| 1 |
IC50 = 19600 nM
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CP0428899
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1-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonyl-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
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C22H26F3N3O4S
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1
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| 1 |
IC50 = 20900 nM
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CP0459321
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1-[4-(4-pyrrolidin-1-ylbutoxy)phenyl]sulfonyl-3-[4-(trifluoromethyl)phenyl]urea
Show/Hide
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C22H26F3N3O4S
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1
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| 1 |
IC50 = 22600 nM
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CP0437704
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1-(4-methoxyphenyl)-3-[4-(3-piperidin-1-ylpropoxy)phenyl]sulfonylurea
Show/Hide
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C22H29N3O5S
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1
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| 1 |
IC50 = 29800 nM
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CP0481427
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1-cyclohexyl-3-[4-(4-pyrrolidin-1-ylbutoxy)phenyl]sulfonylurea
Show/Hide
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C21H33N3O4S
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1
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| 1 |
IC50 = 29900 nM
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CP0389066
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4-[3-[4-[(2-ethyl-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]phenyl]propyl]piperidin-4-ol
Show/Hide
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C25H34N4O
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1
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| 1 |
IC50 > 30000 nM
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CP0392108
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3-[4-[(2-ethyl-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]phenyl]-1-piperazin-1-ylpropan-1-one
Show/Hide
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C24H31N5O
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1
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| 1 |
IC50 > 30000 nM
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CP0392109
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US8748435, 35
Show/Hide
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C24H28N6O
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1
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| 1 |
IC50 > 30000 nM
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CP0408534
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(2R)-3-[4-[(E)-3-[4-[(2-ethyl-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]phenyl]prop-2-enyl]piperazin-1-yl]propane-1,2-diol
Show/Hide
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C27H37N5O2
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1
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| 1 |
IC50 > 30000 nM
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CP0411513
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4-[(E)-3-[4-[(2-ethyl-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]phenyl]prop-2-enyl]piperazin-2-one
Show/Hide
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C24H29N5O
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1
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| 1 |
IC50 > 30000 nM
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CP0541187
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1-[(E)-3-[4-[(2-ethyl-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)methyl]phenyl]prop-2-enyl]piperazin-2-one
Show/Hide
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C24H29N5O
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1
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| 1 |
IC50 > 30000 nM
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CP0526162
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1-cyclohexyl-3-[4-(2-piperidin-1-ylethoxy)phenyl]sulfonylurea
Show/Hide
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C20H31N3O4S
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1
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| 1 |
IC50 = 53800 nM
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CP0428432
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ethyl 1-[2-[4-(phenylcarbamoylsulfamoyl)phenoxy]ethyl]piperidine-4-carboxylate
Show/Hide
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C23H29N3O6S
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1
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| 1 |
IC50 = 77900 nM
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CP0467382
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1-[4-(2-piperidin-1-ylethoxy)phenyl]sulfonyl-3-[4-(trifluoromethyl)phenyl]urea
Show/Hide
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C21H24F3N3O4S
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1
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| 1 |
IC50 = 82000 nM
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CP0437707
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1-phenyl-3-[4-(2-pyrrolidin-1-ylethoxy)phenyl]sulfonylurea
Show/Hide
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C19H23N3O4S
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1
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| 1 |
IC50 = 88600 nM
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CP0450319
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ethyl 1-[3-[4-(phenylcarbamoylsulfamoyl)phenoxy]propyl]piperidine-4-carboxylate
Show/Hide
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C24H31N3O6S
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1
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| 1 |
IC50 = 91100 nM
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CP0415739
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1-(2,5-dichlorophenyl)-3-[4-(2-piperidin-1-ylethoxy)phenyl]sulfonylurea
Show/Hide
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C20H23Cl2N3O4S
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1
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| 1 |
IC50 = 93600 nM
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CP0506283
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2-Methyl-3-[4-(4-piperidinyloxy)phenyl]-4(3H)-quinazolinone
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C20H21N3O2
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1
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| 1 |
IC50 > 1000 nM
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CP0391159
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N-[(3S)-1-[[4-(3-piperidin-1-ylpropoxy)phenyl]methyl]pyrrolidin-3-yl]-1,3-benzodioxole-5-carboxamide
Show/Hide
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C27H35N3O4
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1
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| 1 |
Ki = 0.02512 nM
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CP0551646
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1-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]azetidin-2-one
Show/Hide
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C22H25N3O2
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1
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| 1 |
Ki = 0.07943 nM
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CP0085130
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1-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]pyrrolidin-2-one
Show/Hide
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C23H27N3O2
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1
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| 1 |
Ki = 0.1 nM
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CP0429802
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1-[5-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-2-yl]ethanone
Show/Hide
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C21H24N2O2
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1
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| 1 |
Ki = 0.1 nM
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CP0493724
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1-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]-3-methylimidazolidin-2-one
Show/Hide
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C23H28N4O2
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1
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| 1 |
Ki = 0.1 nM
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CP0386243
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6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-N-propan-2-ylpyridine-3-carboxamide
Show/Hide
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C23H29N3O2
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1
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| 1 |
Ki = 0.1259 nM
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CP0515215
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1-[6-[(3-cyclopentyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]pyrrolidin-2-one
Show/Hide
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C24H29N3O2
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1
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| 1 |
Ki = 0.1259 nM
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CP0429785
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3-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]-1,3-oxazolidin-2-one
Show/Hide
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C22H25N3O3
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1
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| 1 |
Ki = 0.1585 nM
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CP0429787
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2-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]-5-methyl-1,3,4-oxadiazole
Show/Hide
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C22H24N4O2
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1
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| 1 |
Ki = 0.1585 nM
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CP0159421
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5-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)-N-methylpyrazine-2-carboxamide
Show/Hide
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C20H24N4O2
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1
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| 1 |
Ki = 0.1995 nM
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CP0429784
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(4R)-1-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]-4-hydroxypyrrolidin-2-one
Show/Hide
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C23H27N3O3
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1
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| 1 |
Ki = 0.1995 nM
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CP0471632
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N-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]acetamide
Show/Hide
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C21H25N3O2
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1
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| 1 |
Ki = 0.1995 nM
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CP0515219
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6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-2-methylpyridine-3-carbonitrile
Show/Hide
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C21H23N3O
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1
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| 1 |
Ki = 0.1995 nM
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CP0350525
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3-cyclobutyl-7-phenylmethoxy-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
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C21H25NO
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1
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| 1 |
Ki = 0.2512 nM
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CP0489799
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[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]-pyrrolidin-1-ylmethanone
Show/Hide
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C24H29N3O2
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1
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| 1 |
Ki = 0.2512 nM
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CP0501081
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3-cyclobutyl-7-[5-(1H-pyrazol-5-yl)pyridin-2-yl]oxy-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
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C22H24N4O
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1
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| 1 |
Ki = 0.2512 nM
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CP0098027
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2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide
Show/Hide
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C6H10N4S
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1
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| 1 |
Ki = 0.3 nM
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CP0429783
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1-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]piperidin-2-one
Show/Hide
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C24H29N3O2
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1
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| 1 |
Ki = 0.3162 nM
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CP0515216
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1-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]-5-methylpyrrolidin-2-one
Show/Hide
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C24H29N3O2
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1
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| 1 |
Ki = 0.3162 nM
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CP0853422
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3-cyclobutyl-7-(piperidin-4-yloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
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C19H28N2O
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1
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| 1 |
Ki = 0.3162 nM
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CP0347336
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6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxymethyl]-1-methylquinolin-2-one
Show/Hide
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C25H28N2O2
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1
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| 1 |
Ki = 0.3981 nM
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CP0403939
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4-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-N-methylbenzamide
Show/Hide
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C22H26N2O2
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1
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| 1 |
Ki = 0.5012 nM
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CP0429786
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3-cyclobutyl-7-(5-pyrazol-1-ylpyridin-2-yl)oxy-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
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C22H24N4O
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1
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| 1 |
Ki = 0.5012 nM
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CP0433011
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5-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-N-methylpyridine-2-carboxamide
Show/Hide
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C21H25N3O2
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1
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| 1 |
Ki = 0.5012 nM
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CP0458899
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4-[6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridin-3-yl]-3,5-dimethyl-1,2-oxazole
Show/Hide
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C24H27N3O2
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1
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| 1 |
Ki = 0.5012 nM
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CP0476544
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6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]pyridine-3-carboxamide
Show/Hide
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C20H23N3O2
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1
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| 1 |
Ki = 0.5012 nM
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CP0876139
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6-(3-cyclopentyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)-N-methylnicotinamide
Show/Hide
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C22H27N3O2
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1
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| 1 |
Ki = 0.5012 nM
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CP0347352
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3-cyclobutyl-7-(piperidin-4-ylmethoxy)-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
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C20H30N2O
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1
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| 1 |
Ki = 0.5012 nM
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CP0391158
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3-(cyclopropylmethyl)-7-(3-piperidin-1-ylpropoxy)-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
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C22H34N2O
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1
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| 1 |
Ki = 0.5012 nM
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CP0391160
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3-(oxolan-2-ylmethyl)-7-(3-piperidin-1-ylpropoxy)-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
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C23H36N2O2
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1
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| 1 |
Ki = 0.5012 nM
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CP0941894
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(4-chlorophenyl)(4-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)piperidin-1-yl)methanone
Show/Hide
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C26H31ClN2O2
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1
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| 1 |
Ki = 0.5012 nM
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CP0477402
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1-[3-[[(8R,9S,13S,14S,17S)-13-methyl-17-pyrrolidin-1-yl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-3-yl]oxy]propyl]pyrrolidine
Show/Hide
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C29H44N2O
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1
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| 1 |
Ki = 0.6 nM
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CP0515217
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5-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-N-ethylpyridine-2-carboxamide
Show/Hide
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C22H27N3O2
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1
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| 1 |
Ki = 0.631 nM
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CP0515218
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6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-N-ethyl-N-methylpyridine-3-carboxamide
Show/Hide
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C23H29N3O2
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1
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| 1 |
Ki = 0.631 nM
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CP0874333
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3-cyclobutyl-7-(pyridin-2-yloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C19H22N2O
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1
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| 1 |
Ki = 0.7943 nM
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CP0075842
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3-cyclobutyl-7-(1-methylsulfonylpiperidin-4-yl)oxy-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
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C20H30N2O3S
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1
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| 1 |
Ki = 0.7943 nM
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CP0138243
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3-cyclopentyl-7-phenylmethoxy-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
|
C22H27NO
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1
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| 1 |
Ki = 0.7943 nM
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CP0525012
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3-(cyclopropylmethyl)-7-(2-piperidin-1-ylethoxy)-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
|
C21H32N2O
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1
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| 1 |
Ki = 0.7943 nM
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CP0572682
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N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-(trifluoromethyl)phenyl]-2-(4-propan-2-yl-1,4-diazepan-1-yl)acetamide
Show/Hide
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C26H39F3N4O2
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1
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| 1 |
Ki = 0.96 nM
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CP0433012
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[4-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]piperidin-1-yl]-morpholin-4-ylmethanone
Show/Hide
|
C24H35N3O3
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1
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| 1 |
Ki = 1 nM
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CP0535377
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ethyl 4-[2-[4-(1-cyclobutylpiperidin-4-yl)oxyanilino]-2-oxoethyl]piperazine-1-carboxylate;dihydrochloride
Show/Hide
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C24H38Cl2N4O4
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1
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| 1 |
Ki = 1.07 nM
|
|
|
|
CP0344770
|
1-{4-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-phenyl}-ethanone
Show/Hide
|
C13H14N2OS
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0578986
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-pyrrolidin-1-ylacetamide;dihydrochloride
Show/Hide
|
C21H33Cl2N3O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0536455
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-[2-(hydroxymethyl)pyrrolidin-1-yl]acetamide;dihydrochloride
Show/Hide
|
C22H35Cl2N3O3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0386242
|
6-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]-N-methylpyridazine-3-carboxamide
Show/Hide
|
C20H24N4O2
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0877794
|
3-cyclobutyl-7-(pyrazin-2-yloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C18H21N3O
|
1
|
| 1 |
Ki = 1.585 nM
|
|
|
|
CP0108364
|
[4-[(3-cyclobutyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)oxy]piperidin-1-yl]-(5-methyl-1,2-oxazol-3-yl)methanone
Show/Hide
|
C24H31N3O3
|
1
|
| 1 |
Ki = 1.585 nM
|
|
|
|
CP0239657
|
cyclopropyl-[4-(3-piperidin-1-ylpropoxy)phenyl]methanone
Show/Hide
|
C18H25NO2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0555211
|
2-(4-cyclobutyl-1,4-diazepan-1-yl)-N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-(trifluoromethyl)phenyl]acetamide
Show/Hide
|
C27H39F3N4O2
|
1
|
| 1 |
Ki = 1.61 nM
|
|
|
|
CP0541086
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-methylphenyl]-2-pyrrolidin-1-ylacetamide;dihydrochloride
Show/Hide
|
C22H35Cl2N3O2
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0524655
|
[(8S,9S,13S,14S,17S)-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl]-pyrrolidin-1-ylmethanone
Show/Hide
|
C31H46N2O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0358724
|
4-(4-Phenyl-butyl)-1H-imidazole
Show/Hide
|
C13H16N2
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0041493
|
Clobenpropit
Show/Hide
|
C14H17ClN4S
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0476236
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-methylphenyl]-2-[(2R)-2-methylpyrrolidin-1-yl]acetamide
Show/Hide
|
C23H35N3O2
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0553762
|
4-(1-cyclopentylpiperidin-4-yl)oxy-N-(2-pyrrolidin-1-ylethyl)benzamide
Show/Hide
|
C23H35N3O2
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0213459
|
3-(1H-imidazol-4-yl)propylphenylmethyl ether
Show/Hide
|
C13H16N2O
|
2
|
| 1 |
Ki = 2.512 nM
|
|
|
| 2 |
Ki = 2.7 nM
|
|
|
|
CP0877795
|
3-cyclobutyl-7-(pyrimidin-2-yloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C18H21N3O
|
1
|
| 1 |
Ki = 2.512 nM
|
|
|
|
CP0936806
|
3-cyclobutyl-7-(pyridin-3-yloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 2.512 nM
|
|
|
|
CP0391163
|
7-(1-propan-2-ylpiperidin-4-yl)oxy-2,3,4,5-tetrahydro-1H-3-benzazepine
Show/Hide
|
C18H28N2O
|
1
|
| 1 |
Ki = 2.512 nM
|
|
|
|
CP0727267
|
6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline
Show/Hide
|
C17H26N2O
|
1
|
| 1 |
Ki = 2.512 nM
|
|
|
|
CP0476234
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-[(2R)-2-methylpyrrolidin-1-yl]acetamide
Show/Hide
|
C22H33N3O2
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0572681
|
2-(azepan-1-yl)-N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]acetamide;(2R,3R)-2,3-dihydroxybutanedioic acid
Show/Hide
|
C27H41N3O8
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0438629
|
4-(1-cyclobutylpiperidin-4-yl)oxy-N-(2-morpholin-4-ylethyl)benzamide
Show/Hide
|
C22H33N3O3
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0476233
|
4-(1-cyclobutylpiperidin-4-yl)oxy-N-(2-pyrrolidin-1-ylethyl)benzamide
Show/Hide
|
C22H33N3O2
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0477403
|
(8R,9S,13S,14R,15S)-N-ethyl-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C29H42N2O3
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0479001
|
1-(3-(3-phenylpropoxy)propyl)piperidine
Show/Hide
|
C17H27NO
|
1
|
| 1 |
Ki = 3.162 nM
|
|
|
|
CP0908416
|
3-cyclobutyl-7-phenoxy-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 3.162 nM
|
|
|
|
CP0555206
|
4-(1-cyclobutylpiperidin-4-yl)oxy-N-(2-piperidin-1-ylethyl)benzamide;(2R,3R)-2,3-dihydroxybutanedioic acid
Show/Hide
|
C27H41N3O8
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0535375
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-methylphenyl]-2-piperidin-1-ylacetamide;dihydrochloride
Show/Hide
|
C23H37Cl2N3O2
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0559952
|
N-[4-(1-cyclopentylpiperidin-4-yl)oxyphenyl]-2-pyrrolidin-1-ylacetamide
Show/Hide
|
C22H33N3O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0559953
|
2-piperidin-1-yl-N-[4-(1-propan-2-ylpiperidin-4-yl)oxyphenyl]acetamide;dihydrochloride
Show/Hide
|
C21H35Cl2N3O2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0407304
|
7-(3-piperidin-1-ylpropoxy)-2,3,4,5-tetrahydro-1H-3-benzazepine
Show/Hide
|
C18H28N2O
|
1
|
| 1 |
Ki = 3.981 nM
|
|
|
|
CP0476237
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-[2-(hydroxymethyl)morpholin-4-yl]acetamide
Show/Hide
|
C22H33N3O4
|
1
|
| 1 |
Ki = 4.05 nM
|
|
|
|
CP0553763
|
N-[4-(1-cyclopentylpiperidin-4-yl)oxyphenyl]-2-piperidin-1-ylacetamide;dihydrochloride
Show/Hide
|
C23H37Cl2N3O2
|
1
|
| 1 |
Ki = 4.1 nM
|
|
|
|
CP0433666
|
((S)-2-Methyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C12H21N3O2
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
|
CP0549194
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-piperidin-1-ylacetamide;dihydrochloride
Show/Hide
|
C22H35Cl2N3O2
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0555120
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-N-methyl-2-morpholin-4-ylacetamide
Show/Hide
|
C22H33N3O3
|
1
|
| 1 |
Ki = 4.89 nM
|
|
|
|
CP0562330
|
(8R,9S,13R,14R,15S)-N-(cyclobutylmethyl)-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C32H48N2O2
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0077617
|
(1R,2S,5S,6S,9R,12S,13R,16S)-N,N,6,7,13-pentamethyl-7-azapentacyclo[10.8.0.0^{2,9}.0^{5,9}.0^{13,18}]icos-18-en-16-amine
Show/Hide
|
C24H40N2
|
1
|
| 1 |
Ki = 5.012 nM
|
|
|
|
CP0928455
|
7-(benzyloxy)-3-cyclopropyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 5.012 nM
|
|
|
|
CP0438631
|
2-(4-acetylpiperazin-1-yl)-N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]acetamide
Show/Hide
|
C23H34N4O3
|
1
|
| 1 |
Ki = 5.39 nM
|
|
|
|
CP0374615
|
4-[3-(4,4-Dimethyl-pentyloxy)-propyl]-1H-imidazole;C2H2O4
Show/Hide
|
C13H24N2O
|
1
|
| 1 |
Ki = 5.4 nM
|
|
|
|
CP0375886
|
3-(1H-imidazol-5-yl)propyl N-[1-(1-methylcyclopropyl)ethyl]carbamate
Show/Hide
|
C13H21N3O2
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0549193
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-(dimethylamino)acetamide
Show/Hide
|
C19H29N3O2
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0553765
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-(4-hydroxypiperidin-1-yl)acetamide;dihydrochloride
Show/Hide
|
C22H35Cl2N3O3
|
1
|
| 1 |
Ki = 6.4 nM
|
|
|
|
CP0404504
|
3-(1H-imidazol-5-yl)propyl N-[(2R)-3,3-dimethylbutan-2-yl]carbamate
Show/Hide
|
C13H23N3O2
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0403651
|
3-(1H-imidazol-5-yl)propyl N-(dicyclopropylmethyl)carbamate
Show/Hide
|
C14H21N3O2
|
1
|
| 1 |
Ki = 8.2 nM
|
|
|
|
CP0430405
|
(2-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C13H23N3O2
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
|
CP0484773
|
2-morpholin-4-yl-N-[4-(1-propan-2-ylpiperidin-4-yl)oxyphenyl]acetamide;dihydrochloride
Show/Hide
|
C20H33Cl2N3O3
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
|
CP0849831
|
1-(5-(4-(tert-Pentyl)phenoxy)pentyl)piperidine hydrogen oxalate
Show/Hide
|
C23H37NO5
|
1
|
| 1 |
Ki = 8.8 nM
|
|
|
|
CP0354477
|
(8R,9S,13R,14R,15S)-N-(cyclopropylmethyl)-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C31H46N2O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0421579
|
1-[3-[[(8R,9S,13S,14S,17S)-13-methyl-17-pyrrolidin-1-yl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-3-yl]oxy]propyl]pyrrolidin-2-one
Show/Hide
|
C29H42N2O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0421580
|
(8R,9S,13R,14R,15S)-N-ethyl-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C29H44N2O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0562331
|
(8R,9S,13S,14R,15S,17S)-N-ethyl-17-methoxy-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C30H46N2O3
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0553764
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-(1,1-dioxo-1,4-thiazinan-4-yl)acetamide;dihydrochloride
Show/Hide
|
C21H33Cl2N3O4S
|
1
|
| 1 |
Ki = 9.17 nM
|
|
|
|
CP0572679
|
N-(2-piperidin-1-ylethyl)-4-(1-propan-2-ylpiperidin-4-yl)oxybenzamide
Show/Hide
|
C22H35N3O2
|
1
|
| 1 |
Ki = 9.5 nM
|
|
|
|
CP0537953
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-pyridin-4-ylacetamide;(2R,3R)-2,3-dihydroxybutanedioic acid
Show/Hide
|
C26H33N3O8
|
1
|
| 1 |
Ki = 9.51 nM
|
|
|
|
CP0539789
|
3-(1H-imidazol-5-yl)propyl N-[(1R)-1-cyclohexylethyl]carbamate
Show/Hide
|
C15H25N3O2
|
1
|
| 1 |
Ki = 9.7 nM
|
|
|
|
CP0271224
|
3-(cyclopropylmethyl)-7-phenylmethoxy-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
|
C21H25NO
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0407360
|
3-phenyl-7-(3-piperidin-1-ylpropoxy)-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
|
C24H32N2O
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0914164
|
7-(benzyloxy)-3-cyclohexyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C23H29NO
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0554024
|
N-[(8R,9S,13S,14S,15R)-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-15-yl]acetamide
Show/Hide
|
C28H40N2O3
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0572680
|
4-(1-propan-2-ylpiperidin-4-yl)oxy-N-(2-pyrrolidin-1-ylethyl)benzamide
Show/Hide
|
C21H33N3O2
|
1
|
| 1 |
Ki = 10.4 nM
|
|
|
|
CP0578987
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-N-ethyl-2-morpholin-4-ylacetamide
Show/Hide
|
C23H35N3O3
|
1
|
| 1 |
Ki = 10.8 nM
|
|
|
|
CP0430455
|
4-[3-(3,3-Dimethyl-butoxy)-propyl]-1H-imidazole
Show/Hide
|
C12H22N2O
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0483327
|
7-nitro-N-(5-(piperidin-1-yl)pentyl)benzo[c][1,2,5]oxadiazol-4-amine
Show/Hide
|
C16H23N5O3
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0538124
|
N-[4-(1-cyclopentylpiperidin-4-yl)oxyphenyl]-2-(4-fluoropiperidin-1-yl)acetamide;dihydrochloride
Show/Hide
|
C23H36Cl2FN3O2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0438630
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-(diethylamino)acetamide
Show/Hide
|
C21H33N3O2
|
1
|
| 1 |
Ki = 11.7 nM
|
|
|
|
CP0428877
|
((R)-sec-Butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C11H19N3O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0087269
|
(3-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C13H23N3O2
|
2
|
| 1 |
Ki = 13 nM
|
|
|
| 2 |
Ki = 128.82 nM
|
|
|
|
CP0430872
|
3-(1H-imidazol-4-yl)propyl 4-methylpentylcarbamate
Show/Hide
|
C13H23N3O2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0227869
|
3-methyl-1-[5-[4-(2-methylbutan-2-yl)phenoxy]pentyl]piperidine;oxalic acid
Show/Hide
|
C24H39NO5
|
1
|
| 1 |
Ki = 13.6 nM
|
|
|
|
CP0448548
|
3-(1H-imidazol-5-yl)propyl N-[(2S)-3,3-dimethylbutan-2-yl]carbamate
Show/Hide
|
C13H23N3O2
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0460830
|
4-[3-(5,5-Dimethyl-hexyloxy)-propyl]-1H-imidazole;0.8C2H2O4
Show/Hide
|
C14H26N2O
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0931008
|
3-(1H-imidazol-4-yl)propyl pent-4-enylcarbamate hydrogenmalate
Show/Hide
|
C16H23N3O6
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0535376
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-(trifluoromethyl)phenyl]-2-piperidin-1-ylacetamide
Show/Hide
|
C23H32F3N3O2
|
1
|
| 1 |
Ki = 14.8 nM
|
|
|
|
CP0484774
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-fluorophenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C21H30FN3O3
|
1
|
| 1 |
Ki = 14.9 nM
|
|
|
|
CP0471724
|
((R)-1-Methyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C12H21N3O2
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0438632
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-pyridin-3-ylacetamide
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
Ki = 15.8 nM
|
|
|
|
CP0215922
|
1-(7-(3-(piperidin-1-yl)propoxy)-1,2,4,5-tetrahydrobenzo[d]azepin-3-yl)ethanone
Show/Hide
|
C20H30N2O2
|
1
|
| 1 |
Ki = 15.85 nM
|
|
|
|
CP0875499
|
5-(3-(piperidin-1-yl)propoxy)indoline
Show/Hide
|
C16H24N2O
|
1
|
| 1 |
Ki = 15.85 nM
|
|
|
|
CP0375904
|
(1-Cyclohexyl-ethyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester;C2H2O4
Show/Hide
|
C15H25N3O2
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0847652
|
3-(1H-imidazol-4-yl)propyl 2-cyclopropylethylcarbamate maleate
Show/Hide
|
C16H23N3O6
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0184940
|
1-{4-[3-(1H-Imidazol-4-yl)-propylsulfanyl]-phenyl}-ethanone
Show/Hide
|
C14H16N2OS
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0347219
|
1-{4-[4-(1H-Imidazol-4-yl)-butoxy]-phenyl}-ethanone
Show/Hide
|
C15H18N2O2
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0470022
|
((R)-1-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C13H23N3O2
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0951378
|
7-(benzyloxy)-3-isopropyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C20H25NO
|
1
|
| 1 |
Ki = 19.95 nM
|
|
|
|
CP0409399
|
(1-Cyclopropyl-ethyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester;C2H2O4
Show/Hide
|
C12H19N3O2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0878923
|
(E)-3-(1H-Imidazol-4-yl)propyl3,7-dimethylocta-2,6-dienylcarbamate hydrogenmaleate
Show/Hide
|
C21H31N3O6
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0433665
|
(1-Methyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C12H21N3O2
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0563403
|
(8R,9S,13S,14R,15S)-N-ethyl-13-methyl-3-[3-[(2S)-2-methylpyrrolidin-1-yl]propoxy]-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C29H42N2O3
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0906501
|
1-(5-(4-(tert-Pentyl)phenoxy)pentyl)azepane hydrogen oxalate
Show/Hide
|
C24H39NO5
|
1
|
| 1 |
Ki = 21.4 nM
|
|
|
|
CP0484775
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-methylphenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C22H33N3O3
|
1
|
| 1 |
Ki = 22.1 nM
|
|
|
|
CP0802154
|
4-Methyl-1-(5-(4-(tert-pentyl)phenoxy)pentyl)piperidine hydrogen oxalate
Show/Hide
|
C24H39NO5
|
1
|
| 1 |
Ki = 23.4 nM
|
|
|
|
CP0431945
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-(4,4-difluoropiperidin-1-yl)acetamide
Show/Hide
|
C22H31F2N3O2
|
1
|
| 1 |
Ki = 23.6 nM
|
|
|
|
CP0919479
|
(E)-3-(1H-Imidazol-4-yl)propylhex-2-enylcarbamatehydrogen maleate
Show/Hide
|
C17H25N3O6
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0895071
|
3-(1H-Imidazol-4-yl)propyl2-cyclohexylethylcarbamate hydrogenmaleate
Show/Hide
|
C19H29N3O6
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0853424
|
7-(benzyloxy)-3-isobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C21H27NO
|
1
|
| 1 |
Ki = 25.12 nM
|
|
|
|
CP0895069
|
(E)-3-(1H-Imidazol-4-yl)propylhex-3-enylcarbamatehydrogenmaleate
Show/Hide
|
C17H25N3O6
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0895070
|
3-(1H-Imidazol-4-yl)propyl2-cyclohexenylethylcarbamate hydrogenmaleate
Show/Hide
|
C19H27N3O6
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0577153
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-(trifluoromethyl)phenyl]-2-pyrrolidin-1-ylacetamide;dihydrochloride
Show/Hide
|
C22H32Cl2F3N3O2
|
1
|
| 1 |
Ki = 26.9 nM
|
|
|
|
CP0445198
|
4-(3-Phenoxy-propyl)-1H-imidazole with (0.95M)oxalic acid
Show/Hide
|
C12H14N2O
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0847651
|
(Z)-3-(1H-Imidazol-4-yl)propylpent-2-enylcarbamate hydrogenmaleate
Show/Hide
|
C16H23N3O6
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0924100
|
(E)-3-(1H-Imidazol-4-yl)propylpent-2-enylcarbamate hydrogenmaleate
Show/Hide
|
C16H23N3O6
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0879276
|
Pitolisant hydrochloride
Show/Hide
|
C17H27Cl2NO
|
1
|
| 1 |
Ki = 27.6 nM
|
|
|
|
CP0447780
|
(1-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C13H23N3O2
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0572683
|
N-[4-(1-cyclopentylpiperidin-4-yl)oxyphenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C22H33N3O3
|
1
|
| 1 |
Ki = 29.91 nM
|
|
|
|
CP0439083
|
(R,S)-3-(1H-imidazol-4-yl)propyl 5-methylhexan-2-ylcarbamate
Show/Hide
|
C14H25N3O2
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0564473
|
(8R,9S,13S,14R,15R)-13-methyl-3-[3-[(2S)-2-methylpyrrolidin-1-yl]propoxy]-15-(pyrrolidine-1-carbonyl)-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one
Show/Hide
|
C31H44N2O3
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0445521
|
2-(6-(piperidin-1-yl)hexyl)-2H-isoindole-1-carbonitrile
Show/Hide
|
C20H27N3
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0502463
|
2-(5-(piperidin-1-yl)pentyl)-2H-isoindole-1-carbonitrile
Show/Hide
|
C19H25N3
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0439081
|
((S)-sec-Butyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C11H19N3O2
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0482476
|
3-methyl-1-[6-[4-(2-methylbutan-2-yl)phenoxy]hexyl]piperidine;oxalic acid
Show/Hide
|
C25H41NO5
|
1
|
| 1 |
Ki = 33.8 nM
|
|
|
|
CP0567244
|
(8R,9S,13S,14R,15R)-N,N-diethyl-13-methyl-3-[3-[(2S)-2-methylpyrrolidin-1-yl]propoxy]-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C31H46N2O3
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0552470
|
3-methyl-1-[7-[4-(2-methylbutan-2-yl)phenoxy]heptyl]piperidine;oxalic acid
Show/Hide
|
C26H43NO5
|
1
|
| 1 |
Ki = 36.6 nM
|
|
|
|
CP0931000
|
(S)(1-Cyclohexyl-ethyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester
Show/Hide
|
C19H31N3O7
|
1
|
| 1 |
Ki = 37 nM
|
|
|
|
CP0430406
|
(R,S)-3-(1H-imidazol-4-yl)propyl 2-ethylhexylcarbamate
Show/Hide
|
C15H27N3O2
|
1
|
| 1 |
Ki = 37 nM
|
|
|
|
CP0801652
|
1-(3-(4-tert-pentylphenoxy)propyl)piperidine
Show/Hide
|
C19H31NO
|
1
|
| 1 |
Ki = 37 nM
|
|
|
|
CP0214392
|
5-{3-[(4-iodophenyl)methoxy]propyl}-1H-imidazole
Show/Hide
|
C13H15IN2O
|
1
|
| 1 |
Ki = 41 nM
|
|
|
|
CP0430403
|
((R)-1-Methyl-hexyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C14H25N3O2
|
1
|
| 1 |
Ki = 41 nM
|
|
|
|
CP0963911
|
1-(6-(4-(tert-Pentyl)phenoxy)hexyl)azepane hydrogen oxalate
Show/Hide
|
C25H41NO5
|
1
|
| 1 |
Ki = 41.2 nM
|
|
|
|
CP0227935
|
1-{4-[2-(1H-Imidazol-4-yl)-ethoxy]-phenyl}-ethanone
Show/Hide
|
C13H14N2O2
|
1
|
| 1 |
Ki = 42 nM
|
|
|
|
CP0532300
|
((S)-1-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C13H23N3O2
|
1
|
| 1 |
Ki = 42 nM
|
|
|
|
CP0554025
|
(8R,9S,13S,14R,15R)-N-ethyl-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C29H42N2O3
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0099745
|
4-[3-(4-cyclopropanecarbonylphenoxy)propyl]-1H-imidazole
Show/Hide
|
C16H18N2O2
|
2
|
| 1 |
Ki = 46 nM
|
|
|
| 2 |
Ki = 63.1 nM
|
|
|
|
CP0899159
|
1-(6-(4-(tert-Pentyl)phenoxy)hexyl)piperidine hydrogen oxalate
Show/Hide
|
C24H39NO5
|
1
|
| 1 |
Ki = 46.5 nM
|
|
|
|
CP0040043
|
4-[3-(4-Methoxy-phenoxy)-propyl]-1H-imidazole; compound with but-2-enedioic acid(0.25M H2O)
Show/Hide
|
C13H16N2O2
|
1
|
| 1 |
Ki = 47 nM
|
|
|
|
CP0428876
|
3-(1H-imidazol-5-yl)propyl N-butan-2-ylcarbamate
Show/Hide
|
C11H19N3O2
|
1
|
| 1 |
Ki = 49 nM
|
|
|
|
CP0470024
|
(1-Methyl-hexyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C14H25N3O2
|
1
|
| 1 |
Ki = 52 nM
|
|
|
|
CP0919185
|
(E/Z)-3-(1H-Imidazol-4-yl)propylbut-2-enylcarbamate hydrogenmaleate
Show/Hide
|
C15H21N3O6
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0847653
|
3-(1H-Imidazol-4-yl)propylbut-3-enylcarbamate hydrogenmaleate
Show/Hide
|
C15H21N3O6
|
1
|
| 1 |
Ki = 55 nM
|
|
|
|
CP0926379
|
1-(7-(4-(tert-Pentyl)phenoxy)heptyl)piperidine hydrogen oxalate
Show/Hide
|
C25H41NO5
|
1
|
| 1 |
Ki = 55 nM
|
|
|
|
CP0544373
|
6-chloro-2-[5-(3-methylpiperidin-1-yl)pentoxy]xanthen-9-one
Show/Hide
|
C24H28ClNO3
|
1
|
| 1 |
Ki = 56 nM
|
|
|
|
CP0892861
|
4-Methyl-1-(6-(4-(tert-pentyl)phenoxy)hexyl)piperidine hydrogen oxalate
Show/Hide
|
C25H41NO5
|
1
|
| 1 |
Ki = 60.5 nM
|
|
|
|
CP0575030
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-3-fluorophenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C21H30FN3O3
|
1
|
| 1 |
Ki = 62.04 nM
|
|
|
|
CP0482199
|
1-[3-[4-(2-methylbutan-2-yl)phenoxy]propyl]pyrrolidine
Show/Hide
|
C18H29NO
|
1
|
| 1 |
Ki = 63 nM
|
|
|
|
CP0968907
|
4-Methyl-1-(7-(4-(tert-pentyl)phenoxy)heptyl)piperidine hydrogen oxalate
Show/Hide
|
C26H43NO5
|
1
|
| 1 |
Ki = 64.4 nM
|
|
|
|
CP0421634
|
((S)-1-Methyl-hexyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C14H25N3O2
|
1
|
| 1 |
Ki = 74 nM
|
|
|
|
CP0430404
|
(R,S)-3-(1H-imidazol-4-yl)propyl 6-methylheptan-2-ylcarbamate
Show/Hide
|
C15H27N3O2
|
1
|
| 1 |
Ki = 75 nM
|
|
|
|
CP0438633
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-(trifluoromethyl)phenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C22H30F3N3O3
|
1
|
| 1 |
Ki = 75.8 nM
|
|
|
|
CP0505126
|
(1-tert-Butyl-2,2-dimethyl-propyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester;C2H2O4
Show/Hide
|
C16H29N3O2
|
1
|
| 1 |
Ki = 77 nM
|
|
|
|
CP0266723
|
cyclopropyl-[4-[3-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]propoxy]phenyl]methanone
Show/Hide
|
C26H32N2O2
|
1
|
| 1 |
Ki = 83 nM
|
|
|
|
CP0847654
|
3-(1H-Imidazol-4-yl)propyl2-cyclohexylpropylcarbamate hydrogenmaleate
Show/Hide
|
C20H31N3O6
|
1
|
| 1 |
Ki = 86 nM
|
|
|
|
CP0451654
|
2-[5-(azepan-1-yl)pentoxy]-6-chloroxanthen-9-one
Show/Hide
|
C24H28ClNO3
|
1
|
| 1 |
Ki = 86 nM
|
|
|
|
CP0041994
|
1-{4-[3-(1H-Imidazol-4-yl)-propoxy]-phenyl}-ethanone
Show/Hide
|
C14H16N2O2
|
1
|
| 1 |
Ki = 87 nM
|
|
|
|
CP0535378
|
N-[4-(1-cyclobutylpiperidin-4-yl)oxy-2-methoxyphenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C22H33N3O4
|
1
|
| 1 |
Ki = 90.75 nM
|
|
|
|
CP0433664
|
(1-Methyl-heptyl)-carbamic acid 3-(1H-imidazol-4-yl)-propyl ester; compound with (E)-but-2-enedioic acid
Show/Hide
|
C15H27N3O2
|
1
|
| 1 |
Ki = 91 nM
|
|
|
|
CP0451653
|
2-[6-(4-methylpiperidin-1-yl)hexoxy]xanthen-9-one
Show/Hide
|
C25H31NO3
|
1
|
| 1 |
Ki = 97 nM
|
|
|
|
CP0418911
|
1-[3-(4-tert-Butylphenoxy)propyl]-4-piperidino-piperidine
Show/Hide
|
C23H38N2O
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0856505
|
N,N-dimethyl-3-(2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)propan-1-amine
Show/Hide
|
C15H24N2O
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0928454
|
4-(3-(2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)propyl)morpholine
Show/Hide
|
C17H26N2O2
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0458017
|
3-methyl-1-[3-[4-(2-methylbutan-2-yl)phenoxy]propyl]piperidine
Show/Hide
|
C20H33NO
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0549658
|
2-[6-(3-methylpiperidin-1-yl)hexoxy]xanthen-9-one
Show/Hide
|
C25H31NO3
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0549660
|
2-[5-(azepan-1-yl)pentoxy]-7-chloroxanthen-9-one
Show/Hide
|
C24H28ClNO3
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0471260
|
(6-benzyl-6-azaspiro[2.5]octan-2-yl)-(4-cyclohexylpiperazin-1-yl)methanone
Show/Hide
|
C25H37N3O
|
1
|
| 1 |
Ki = 103 nM
|
|
|
|
CP0553767
|
N-[4-[2-[(2R)-2-methylpyrrolidin-1-yl]ethyl]phenyl]-2-morpholin-4-ylacetamide;dihydrochloride
Show/Hide
|
C19H31Cl2N3O2
|
1
|
| 1 |
Ki = 107.6 nM
|
|
|
|
CP0451650
|
2-[5-(4-methylpiperidin-1-yl)pentoxy]xanthen-9-one
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0537955
|
2-morpholin-4-yl-N-[4-(pyrrolidin-1-ylmethyl)phenyl]acetamide
Show/Hide
|
C17H25N3O2
|
1
|
| 1 |
Ki = 114.5 nM
|
|
|
|
CP0448484
|
4-[3-(1,3,3-Trimethyl-butoxy)-propyl]-1H-imidazole;0.85C2H2O4
Show/Hide
|
C13H24N2O
|
1
|
| 1 |
Ki = 119 nM
|
|
|
|
CP0470186
|
3-methyl-1-[8-[4-(2-methylbutan-2-yl)phenoxy]octyl]piperidine;oxalic acid
Show/Hide
|
C27H45NO5
|
1
|
| 1 |
Ki = 120.7 nM
|
|
|
|
CP0851793
|
1-(7-(4-(tert-Pentyl)phenoxy)heptyl)azepane hydrogen oxalate
Show/Hide
|
C26H43NO5
|
1
|
| 1 |
Ki = 128.3 nM
|
|
|
|
CP0447842
|
1-[2-(3-Methoxyphenoxy)ethyl]-4-piperidino-piperidine
Show/Hide
|
C19H30N2O2
|
1
|
| 1 |
Ki = 132 nM
|
|
|
|
CP0387044
|
2,6-dimethyl-1-[3-[4-(2-methylbutan-2-yl)phenoxy]propyl]piperidine
Show/Hide
|
C21H35NO
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0549499
|
2-chloro-7-[5-(4-methylpiperidin-1-yl)pentoxy]xanthen-9-one
Show/Hide
|
C24H28ClNO3
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0199147
|
3-(1H-imidazol-4-yl)propyl pent-4-enylcarbamate hydrogenmalate
Show/Hide
|
C12H19N3O2
|
1
|
| 1 |
Ki = 141.25 nM
|
|
|
|
CP0489500
|
4-methyl-1-[3-[4-(2-methylbutan-2-yl)phenoxy]propyl]piperidine
Show/Hide
|
C20H33NO
|
1
|
| 1 |
Ki = 147 nM
|
|
|
|
CP0140472
|
2-chloro-7-[5-(3-methylpiperidin-1-yl)pentoxy]xanthen-9-one
Show/Hide
|
C24H28ClNO3
|
1
|
| 1 |
Ki = 148 nM
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CP0424613
|
2-chloro-7-(5-piperidin-1-ylpentoxy)xanthen-9-one
Show/Hide
|
C23H26ClNO3
|
1
|
| 1 |
Ki = 150 nM
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CP0424615
|
2-[5-(3-methylpiperidin-1-yl)pentoxy]xanthen-9-one
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 156 nM
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CP0882245
|
7-(2-(piperidin-1-yl)ethoxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C17H26N2O
|
1
|
| 1 |
Ki = 158.49 nM
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CP0547832
|
1-[2-(3-Trifluoromethylphenoxy)ethyl]-4-piperidinopiperidine
Show/Hide
|
C19H27F3N2O
|
1
|
| 1 |
Ki = 164 nM
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CP0479000
|
1-[3-(4-Chlorophenoxy)propyl]-4-piperidino-piperidine
Show/Hide
|
C19H29ClN2O
|
1
|
| 1 |
Ki = 165 nM
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CP0336668
|
3-(1H-imidazol-4-yl)propyl 2-cyclopropylethylcarbamate maleate
Show/Hide
|
C12H19N3O2
|
1
|
| 1 |
Ki = 169.82 nM
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CP0445520
|
7-nitro-N-(4-(piperidin-1-yl)butyl)benzo[c][1,2,5]oxadiazol-4-amine
Show/Hide
|
C15H21N5O3
|
1
|
| 1 |
Ki = 170 nM
|
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CP0140449
|
2-[5-(azepan-1-yl)pentoxy]xanthen-9-one
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 170 nM
|
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CP0549661
|
2-(5-piperidin-1-ylpentoxy)xanthen-9-one
Show/Hide
|
C23H27NO3
|
1
|
| 1 |
Ki = 172 nM
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CP0521176
|
1-[2-(4-Chlorophenoxy)ethyl]-4-piperidino-piperidine
Show/Hide
|
C18H27ClN2O
|
1
|
| 1 |
Ki = 176 nM
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CP0462320
|
2-(4-(piperidin-1-yl)butyl)-2H-isoindole-1-carbonitrile
Show/Hide
|
C18H23N3
|
1
|
| 1 |
Ki = 178 nM
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CP0950523
|
1-(8-(4-(tert-Pentyl)phenoxy)octyl)azepane hydrogen oxalate
Show/Hide
|
C27H45NO5
|
1
|
| 1 |
Ki = 182.5 nM
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CP0919184
|
3-(1H-Imidazol-4-yl)propyl2-cyclohexylbutylcarbamate hydrogenmaleate
Show/Hide
|
C21H33N3O6
|
1
|
| 1 |
Ki = 194 nM
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CP0421382
|
6-chloro-2-(6-piperidin-1-ylhexoxy)xanthen-9-one
Show/Hide
|
C24H28ClNO3
|
1
|
| 1 |
Ki = 203 nM
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CP0508347
|
N-[3-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C21H31N3O3
|
1
|
| 1 |
Ki = 212.1 nM
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CP0390674
|
1-(benzenesulfonyl)-4-(1-cyclobutylpiperidin-4-yl)-2,3-dihydroindole
Show/Hide
|
C23H28N2O2S
|
1
|
| 1 |
Ki = 214 nM
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CP0571703
|
(8R,9S,13S,14R,15S)-N-ethyl-3-[3-[(3R)-3-fluoropyrrolidin-1-yl]propoxy]-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C28H39FN2O3
|
1
|
| 1 |
Ki = 230 nM
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CP0563405
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(8R,9S,13S,14R,15R)-N-ethyl-13-methyl-3-[4-[(2S)-2-methylpyrrolidin-1-yl]butoxy]-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C30H44N2O3
|
1
|
| 1 |
Ki = 234 nM
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CP0521175
|
1-[2-(3-Chlorophenoxy)ethyl]-4-piperidino-piperidine
Show/Hide
|
C18H27ClN2O
|
1
|
| 1 |
Ki = 235 nM
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CP0190362
|
2-[6-(azepan-1-yl)hexoxy]-7-chloroxanthen-9-one
Show/Hide
|
C25H30ClNO3
|
1
|
| 1 |
Ki = 238 nM
|
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CP0375971
|
(E)-3-(1H-Imidazol-4-yl)propylhex-2-enylcarbamatehydrogen maleate
Show/Hide
|
C13H21N3O2
|
1
|
| 1 |
Ki = 239.88 nM
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CP0418909
|
4-Propyl-1-[3-(phenylpropoxy)propyl]piperidine
Show/Hide
|
C20H33NO
|
1
|
| 1 |
Ki = 249 nM
|
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CP0397244
|
3-(1H-Imidazol-4-yl)propyl2-cyclohexylethylcarbamate hydrogenmaleate
Show/Hide
|
C15H25N3O2
|
1
|
| 1 |
Ki = 251.19 nM
|
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CP0087268
|
(E)-3-(1H-Imidazol-4-yl)propylhex-3-enylcarbamatehydrogenmaleate
Show/Hide
|
C13H21N3O2
|
1
|
| 1 |
Ki = 257.04 nM
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CP0578866
|
(8R,9S,13S,14R,15R)-N-ethyl-13-methyl-3-[2-[(2S)-2-methylpyrrolidin-1-yl]ethoxy]-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C28H40N2O3
|
1
|
| 1 |
Ki = 260 nM
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CP0503477
|
4-Butyl-1-[3-(phenylpropoxy)propyl]piperidine
Show/Hide
|
C21H35NO
|
1
|
| 1 |
Ki = 274 nM
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CP0462058
|
1-(benzenesulfonyl)-5-(4-ethylpiperazin-1-yl)-2,3-dihydroindole
Show/Hide
|
C20H25N3O2S
|
1
|
| 1 |
Ki = 280 nM
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CP0549657
|
2-chloro-7-(6-piperidin-1-ylhexoxy)xanthen-9-one
Show/Hide
|
C24H28ClNO3
|
1
|
| 1 |
Ki = 282 nM
|
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CP0446519
|
2-(benzenesulfonyl)-5-(4-ethylpiperazin-1-yl)-1,3-dihydroisoindole
Show/Hide
|
C20H25N3O2S
|
1
|
| 1 |
Ki = 294 nM
|
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CP0310269
|
1-[3-[4-(2-methylbutan-2-yl)phenoxy]propyl]azepane
Show/Hide
|
C20H33NO
|
1
|
| 1 |
Ki = 298 nM
|
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|
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CP0415471
|
1-(benzenesulfonyl)-5-(1-methylpiperidin-4-yl)-2,3-dihydroindole
Show/Hide
|
C20H24N2O2S
|
1
|
| 1 |
Ki = 299 nM
|
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CP0493315
|
1-[2-(4-Methylphenoxy)ethyl]-4-piperidino-piperidine
Show/Hide
|
C19H30N2O
|
1
|
| 1 |
Ki = 300 nM
|
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CP0473664
|
2-(benzenesulfonyl)-5-(1-ethylpiperidin-4-yl)-1,3-dihydroisoindole
Show/Hide
|
C21H26N2O2S
|
1
|
| 1 |
Ki = 302 nM
|
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CP0965250
|
4-Methyl-1-(8-(4-(tert-pentyl)phenoxy)octyl)piperidine hydrogen oxalate
Show/Hide
|
C27H45NO5
|
1
|
| 1 |
Ki = 308.1 nM
|
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CP0882244
|
7-(benzyloxy)-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C18H21NO
|
1
|
| 1 |
Ki = 316.23 nM
|
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|
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CP0462049
|
1-(benzenesulfonyl)-4-(1-ethylpiperidin-4-yl)-2,3-dihydroindole
Show/Hide
|
C21H26N2O2S
|
1
|
| 1 |
Ki = 317 nM
|
|
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CP0866459
|
1-(8-(4-(tert-Pentyl)phenoxy)octyl)piperidine hydrogen oxalate
Show/Hide
|
C26H43NO5
|
1
|
| 1 |
Ki = 325.9 nM
|
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CP0418910
|
4-Benzyl-1-[3-phenylpropoxy)propyl]piperidine
Show/Hide
|
C24H33NO
|
1
|
| 1 |
Ki = 326 nM
|
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|
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CP0462080
|
1-(benzenesulfonyl)-4-(4-ethylpiperazin-1-yl)-2,3-dihydroindole
Show/Hide
|
C20H25N3O2S
|
1
|
| 1 |
Ki = 344 nM
|
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CP0515965
|
2-(3-(piperidin-1-yl)propyl)-2H-isoindole-1-carbonitrile
Show/Hide
|
C17H21N3
|
1
|
| 1 |
Ki = 351 nM
|
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|
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CP0503478
|
2-[3-(3-phenylpropoxy)propyl]decahydroisoquinoline
Show/Hide
|
C21H33NO
|
1
|
| 1 |
Ki = 393 nM
|
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|
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CP0482468
|
2-(benzenesulfonyl)-5-(4-cyclobutylpiperazin-1-yl)-1,3-dihydroisoindole
Show/Hide
|
C22H27N3O2S
|
1
|
| 1 |
Ki = 395 nM
|
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CP0199146
|
3-(1H-imidazol-5-yl)propyl N-[2-(4-chlorophenyl)ethyl]carbamate
Show/Hide
|
C15H18ClN3O2
|
1
|
| 1 |
Ki = 426.58 nM
|
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CP0532216
|
2-chloro-7-[6-(3-methylpiperidin-1-yl)hexoxy]xanthen-9-one
Show/Hide
|
C25H30ClNO3
|
1
|
| 1 |
Ki = 436 nM
|
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|
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CP0443963
|
2-methyl-1-[3-[4-(2-methylbutan-2-yl)phenoxy]propyl]piperidine
Show/Hide
|
C20H33NO
|
1
|
| 1 |
Ki = 437 nM
|
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|
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CP0462051
|
1-(benzenesulfonyl)-5-(1-ethylpiperidin-4-yl)-2,3-dihydroindole
Show/Hide
|
C21H26N2O2S
|
1
|
| 1 |
Ki = 448 nM
|
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CP0549662
|
6-chloro-2-[5-(4-methylpiperidin-1-yl)pentoxy]xanthen-9-one
Show/Hide
|
C24H28ClNO3
|
1
|
| 1 |
Ki = 448 nM
|
|
|
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CP0190361
|
2-chloro-7-[6-(4-methylpiperidin-1-yl)hexoxy]xanthen-9-one
Show/Hide
|
C25H30ClNO3
|
1
|
| 1 |
Ki = 465 nM
|
|
|
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CP0546225
|
2-[6-(azepan-1-yl)hexoxy]xanthen-9-one
Show/Hide
|
C25H31NO3
|
1
|
| 1 |
Ki = 496 nM
|
|
|
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CP0544375
|
6-chloro-2-[6-(4-methylpiperidin-1-yl)hexoxy]xanthen-9-one
Show/Hide
|
C25H30ClNO3
|
1
|
| 1 |
Ki = 520 nM
|
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|
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CP0578865
|
(8R,9S,13S,14R,15S)-N-ethyl-3-[3-(4-fluoropiperidin-1-yl)propoxy]-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C29H41FN2O3
|
1
|
| 1 |
Ki = 530 nM
|
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CP0484777
|
N-[4-(4-cyclobutylpiperazin-1-yl)phenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C20H30N4O2
|
1
|
| 1 |
Ki = 532.1 nM
|
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CP0538963
|
3-(1H-Imidazol-4-yl)propylbut-3-enylcarbamate hydrogenmaleate
Show/Hide
|
C11H17N3O2
|
1
|
| 1 |
Ki = 549.54 nM
|
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CP0428175
|
2-[3-(3-Phenylpropoxy)propyl]-1,2,3,4-tetrahydro-isoquinoline
Show/Hide
|
C21H27NO
|
1
|
| 1 |
Ki = 560 nM
|
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CP0410826
|
1-(benzenesulfonyl)-4-(4-cyclobutylpiperazin-1-yl)-2,3-dihydroindole
Show/Hide
|
C22H27N3O2S
|
1
|
| 1 |
Ki = 580 nM
|
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CP0555647
|
2-[6-(azepan-1-yl)hexoxy]-6-chloroxanthen-9-one
Show/Hide
|
C25H30ClNO3
|
1
|
| 1 |
Ki = 602 nM
|
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CP0238502
|
1-[(E)-3-phenylprop-2-enyl]-4-[3-(3-phenylpropoxy)propyl]piperazine
Show/Hide
|
C25H34N2O
|
1
|
| 1 |
Ki = 690 nM
|
|
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CP0087267
|
3-(1H-imidazol-5-yl)propyl N-[2-(2-chlorophenoxy)ethyl]carbamate
Show/Hide
|
C15H18ClN3O3
|
1
|
| 1 |
Ki = 707.95 nM
|
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CP0443965
|
3,5-dimethyl-1-[3-[4-(2-methylbutan-2-yl)phenoxy]propyl]piperidine
Show/Hide
|
C21H35NO
|
1
|
| 1 |
Ki = 753 nM
|
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|
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CP0454159
|
3-(1H-Imidazol-4-yl)propyl2-cyclohexylpropylcarbamate hydrogenmaleate
Show/Hide
|
C16H27N3O2
|
1
|
| 1 |
Ki = 851.14 nM
|
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CP0537954
|
2-[(2R)-2-methylpyrrolidin-1-yl]-N-[4-(morpholin-4-ylmethyl)phenyl]acetamide
Show/Hide
|
C18H27N3O2
|
1
|
| 1 |
Ki = 915 nM
|
|
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CP0375970
|
3-(1H-imidazol-5-yl)propyl N-(4-phenoxybutyl)carbamate
Show/Hide
|
C17H23N3O3
|
1
|
| 1 |
Ki = 1047.13 nM
|
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CP0424614
|
2-(6-piperidin-1-ylhexoxy)xanthen-9-one
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 1060 nM
|
|
|
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CP0140446
|
6-chloro-2-[6-(3-methylpiperidin-1-yl)hexoxy]xanthen-9-one
Show/Hide
|
C25H30ClNO3
|
1
|
| 1 |
Ki = 1105 nM
|
|
|
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CP0397243
|
3-(1H-imidazol-5-yl)propyl N-(3-phenoxypropyl)carbamate
Show/Hide
|
C16H21N3O3
|
1
|
| 1 |
Ki = 1288.25 nM
|
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CP0562332
|
(8R,9S,13S,14R,15S)-3-[3-(4,4-difluoropiperidin-1-yl)propoxy]-N-ethyl-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-15-carboxamide
Show/Hide
|
C29H40F2N2O3
|
1
|
| 1 |
Ki = 1371 nM
|
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CP0484776
|
2-[(2R)-2-methylpyrrolidin-1-yl]-N-(4-morpholin-4-ylphenyl)acetamide
Show/Hide
|
C17H25N3O2
|
1
|
| 1 |
Ki = 1455 nM
|
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CP0469126
|
(4-cyclohexylpiperazin-1-yl)-(6-phenyl-6-azaspiro[2.5]octan-2-yl)methanone
Show/Hide
|
C24H35N3O
|
1
|
| 1 |
Ki = 1670 nM
|
|
|
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CP0195311
|
3-(1H-Imidazol-4-yl)propyl2-cyclohexylbutylcarbamate hydrogenmaleate
Show/Hide
|
C17H29N3O2
|
1
|
| 1 |
Ki = 1949.84 nM
|
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CP0555212
|
N-[4-[[(2R)-2-methylpyrrolidin-1-yl]methyl]phenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C18H27N3O2
|
1
|
| 1 |
Ki = 3572 nM
|
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CP0503479
|
1-[3-(3-Methoxyphenoxy)propyl]-4-piperidino-piperidine
Show/Hide
|
C20H32N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0853421
|
7-(benzyloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C17H19NO
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0861726
|
1-(3-(2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)propyl)piperidin-4-ol
Show/Hide
|
C18H28N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0535379
|
2-morpholin-4-yl-N-(4-piperidin-4-yloxyphenyl)acetamide
Show/Hide
|
C17H25N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0536456
|
N-[2-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-2-morpholin-4-ylacetamide
Show/Hide
|
C21H31N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0928456
|
7-(3-(4,4-difluoropiperidin-1-yl)propoxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C18H26F2N2O
|
1
|
| 1 |
Ki > 398.11 nM
|
|
|
|
CP0853423
|
3-benzyl-7-(benzyloxy)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C24H25NO
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0458018
|
3,3-dimethyl-1-[3-[4-(2-methylbutan-2-yl)phenoxy]propyl]piperidine
Show/Hide
|
C21H35NO
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0119044
|
(2-chlorophenyl)-[4-[3-(cyclobutylmethoxy)propyl]piperazin-1-yl]methanone
Show/Hide
|
C19H27ClN2O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0119047
|
1-(2-ethoxyphenyl)-4-[3-(3-phenylpropoxy)propyl]piperazine
Show/Hide
|
C24H34N2O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0167935
|
1-benzyl-4-[3-(3-phenylpropoxy)propyl]piperazine
Show/Hide
|
C23H32N2O
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
