Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-[(8R,9S,13S,14S,15R)-13-methyl-3-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-15-yl]acetamide
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 PubChem ID
CID: 155556196
Canonical SMILES
C[C@@H]1CCCN1CCCOc1ccc2[C@H]3CC[C@@]4(C)[C@@H]([C@@H](CC4=O)NC(C)=O)[C@@H]3CCc2c1
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Compound Formula C28H40N2O3
Compound Structure
Protein Name
 Protein Info 
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 10 nM
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