Brief Information of the Compound and Protein
Compound Name
[2-(4-cyclobutyl-1,4-diazepane-1-carbonyl)-2,9-diazaspiro[5.5]undecan-9-yl]-phenylmethanone
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PubChem ID
CID: 76314725
Canonical SMILES
O=C(N1CCCC2(CCN(CC2)C(=O)c2ccccc2)C1)N1CCCN(CC1)C1CCC1
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Compound Formula C26H38N4O2
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 18 nM
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