Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-cyclobutyl-7-[5-(1H-pyrazol-5-yl)pyridin-2-yl]oxy-1,2,4,5-tetrahydro-3-benzazepine
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 PubChem ID
CID: 10021441
SID: 15002806
Canonical SMILES
C1CC(C1)N1CCc2ccc(Oc3ccc(cn3)-c3cc[nH]n3)cc2CC1
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Compound Formula C22H24N4O
Compound Structure
Protein Name
 Protein Info 
Histamine H3 receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 0.2512 nM
   TI
   LI
   LO
   TS