| Compound ID |
Compound Name |
Compound Formula |
|
CP0361108
|
2-[4-[3-[(1S)-1-pyrazolo[1,5-a]pyridin-5-ylethyl]triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol
Show/Hide
|
C18H17N9O
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0378506
|
3-[(1S)-1-imidazo[1,2-a]pyridin-6-ylethyl]-5-(1-methylpyrazol-4-yl)triazolo[4,5-b]pyrazine
Show/Hide
|
C17H15N9
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0088790
|
5-(1-methylpyrazol-4-yl)-3-(2H-pyrazolo[3,4-b]pyridin-3-ylmethyl)triazolo[4,5-b]pyrazine
Show/Hide
|
C15H12N10
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0334867
|
6-[[5-(1-methylpyrazol-4-yl)triazolo[4,5-b]pyrazin-3-yl]methyl]quinoline
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|
C18H14N8
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0318467
|
2-[4-[3-(pyrazolo[1,5-a]pyridin-5-ylmethyl)triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol
Show/Hide
|
C17H15N9O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0361106
|
3-(imidazo[1,2-a]pyridin-6-ylmethyl)-5-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]triazolo[4,5-b]pyrazine
Show/Hide
|
C17H12F3N9
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0318468
|
3-(2H-pyrazolo[3,4-b]pyridin-3-ylmethyl)-5-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]triazolo[4,5-b]pyrazine
Show/Hide
|
C16H11F3N10
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0318465
|
2-[4-[3-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol
Show/Hide
|
C17H15N9O
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0361107
|
3-(pyrazolo[1,5-a]pyridin-5-ylmethyl)-5-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]triazolo[4,5-b]pyrazine
Show/Hide
|
C17H12F3N9
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0365548
|
3-(imidazo[1,2-a]pyridin-6-ylmethyl)-5-(1-methylpyrazol-4-yl)triazolo[4,5-b]pyrazine
Show/Hide
|
C16H13N9
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0116106
|
5-(4-fluorophenyl)-3-(2H-pyrazolo[3,4-b]pyridin-3-ylmethyl)triazolo[4,5-b]pyrazine
Show/Hide
|
C17H11FN8
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0303786
|
5-(4-fluorophenyl)-3-(imidazo[1,2-a]pyridin-6-ylmethyl)triazolo[4,5-b]pyrazine
Show/Hide
|
C18H12FN7
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0361103
|
5-[[5-(1-methylpyrazol-4-yl)triazolo[4,5-b]pyrazin-3-yl]methyl]-1H-thieno[3,2-c]pyrazole
Show/Hide
|
C14H11N9S
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0303785
|
5-(1-methylpyrazol-4-yl)-3-(pyrazolo[1,5-a]pyridin-5-ylmethyl)triazolo[4,5-b]pyrazine
Show/Hide
|
C16H13N9
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0352623
|
2-[4-[3-(2H-pyrazolo[3,4-b]pyridin-3-ylmethyl)triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol
Show/Hide
|
C16H14N10O
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0481631
|
5-[3-(imidazo[1,2-a]pyridin-6-ylmethyl)triazolo[4,5-b]pyrazin-5-yl]pyridine-2-carbonitrile
Show/Hide
|
C18H11N9
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0271717
|
2-[4-[3-[(1R)-1-pyrazolo[1,5-a]pyridin-5-ylethyl]triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol
Show/Hide
|
C18H17N9O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0481630
|
5-[3-(2H-pyrazolo[3,4-b]pyridin-3-ylmethyl)triazolo[4,5-b]pyrazin-5-yl]pyridine-2-carbonitrile
Show/Hide
|
C17H10N10
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0318469
|
3-[(1R)-1-imidazo[1,2-a]pyridin-6-ylethyl]-5-(1-methylpyrazol-4-yl)triazolo[4,5-b]pyrazine
Show/Hide
|
C17H15N9
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0494304
|
2-[4-[3-(imidazo[1,2-a]pyridin-6-ylmethyl)triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol
Show/Hide
|
C17H15N9O
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0318466
|
2-[[5-(1-methylpyrazol-4-yl)triazolo[4,5-b]pyrazin-3-yl]methyl]thieno[3,2-c]pyridine
Show/Hide
|
C16H12N8S
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0052888
|
3-(imidazo[1,2-b]pyridazin-6-ylmethyl)-5-(1-methylpyrazol-4-yl)triazolo[4,5-b]pyrazine
Show/Hide
|
C15H12N10
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0155931
|
6-[[6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methyl]quinoline
Show/Hide
|
C19H15N7
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0261572
|
5-(1-methylpyrazol-4-yl)-3-([1,2,4]triazolo[1,5-a]pyridin-6-ylmethyl)triazolo[4,5-b]pyrazine
Show/Hide
|
C15H12N10
|
1
|
| 1 |
IC50 = 77 nM
|
|
|
|
CP0433290
|
6-[[5-(1-methylpyrazol-4-yl)imidazo[4,5-b]pyrazin-3-yl]methyl]quinoline
Show/Hide
|
C19H15N7
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
