| Compound ID |
Compound Name |
Compound Formula |
|
CP0123177
|
2-(6-(4-chlorophenyl)-2,2-dimethyl-7-phenyl-2,3-dihydro-1H-pyrrolizin-5-yl)acetic acid
Show/Hide
|
C23H22ClNO2
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0514592
|
2-(9-(2-hydroxy-2-methylpropyl)-6-(isopentyloxy)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
Show/Hide
|
C32H30N4O2
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0039500
|
2-(6-(2-cyclopropylethoxy)-9-(2-hydroxy-2-methylpropyl)-1H-phenanthro[9,10-d]imidazol-2-yl)-5-fluoroisophthalonitrile
Show/Hide
|
C32H27FN4O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0371058
|
1-(3-(cyclopropylethynyl)benzyl)-3-isopropyl-1-(3-(phenylethynyl)benzyl)urea
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|
C31H30N2O
|
2
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 160 nM
|
|
|
|
CP0433142
|
5-[5-bromo-2-(2-chloro-6-fluorophenyl)-1H-imidazol-4-yl]-2-(2-phenylethynyl)pyridine
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|
C22H12BrClFN3
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0528794
|
1-[[3-(2-phenylethynyl)phenyl]methyl]-3-propan-2-yl-1-[[3-(2-pyridin-3-ylethynyl)phenyl]methyl]urea
Show/Hide
|
C33H29N3O
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0130091
|
N-(3-chloro-2-methylphenyl)-6-[[2-chloro-6-(trifluoromethyl)benzoyl]amino]-2-(methoxymethyl)-1H-benzimidazole-4-carboxamide
Show/Hide
|
C25H19Cl2F3N4O3
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0419564
|
(4S)-N-[4-(hydroxymethyl)cyclohexyl]-3,3-dimethyl-1-(8-methylquinolin-2-yl)piperidine-4-carboxamide
Show/Hide
|
C25H35N3O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0320229
|
2-(2-chloro-6-fluoroanilino)-1,7,7-trimethyl-N-[4-(trifluoromethyl)phenyl]-8H-furo[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C26H21ClF4N4O2
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0237234
|
(4S)-N-[(1S,3S)-3-(hydroxymethyl)cyclohexyl]-3,3-dimethyl-1-(8-methylquinolin-2-yl)piperidine-4-carboxamide
Show/Hide
|
C25H35N3O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0069222
|
2-(2-chloro-6-fluoroanilino)-1,7,7-trimethyl-N-[3-(trifluoromethyl)phenyl]-8H-furo[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C26H21ClF4N4O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0320230
|
2-(2-chloro-6-fluoroanilino)-N-(2-fluoro-4-methylphenyl)-1,7,7-trimethyl-8H-furo[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C26H23ClF2N4O2
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0563853
|
N-(5-cyclopropyl-2-fluorophenyl)-2-(2,6-dichloroanilino)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C27H23Cl2FN4O2
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0201007
|
4-chloro-2-[[(1S,2S)-2-[[1-[4-(trifluoromethyl)phenyl]piperidine-4-carbonyl]amino]cyclopentyl]methylamino]benzoic acid
Show/Hide
|
C26H29ClF3N3O3
|
1
|
| 1 |
IC50 = 3.5 nM
|
|
|
|
CP0573750
|
5-[2-(2-chloro-6-fluorophenyl)-1H-imidazol-5-yl]-2-[2-(3-chlorophenyl)ethynyl]pyridine
Show/Hide
|
C22H12Cl2FN3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0567264
|
2-(2-chloro-6-fluoroanilino)-1,7,7-trimethyl-N-[5-(trifluoromethyl)pyridin-2-yl]-8H-furo[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H20ClF4N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0470788
|
2-(2,6-dichloroanilino)-7,7-dimethyl-N-phenyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H20Cl2N4O2
|
1
|
| 1 |
IC50 = 4.1 nM
|
|
|
|
CP0104197
|
2-(2,6-dichloroanilino)-7,7-dimethyl-N-[5-(trifluoromethyl)pyridin-2-yl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H18Cl2F3N5O2
|
1
|
| 1 |
IC50 = 4.1 nM
|
|
|
|
CP0523514
|
2-(2-chloro-6-fluoroanilino)-N-(4-cyclohexylphenyl)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C30H30ClFN4O2
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
|
CP0438381
|
2-(2-chloro-6-fluoroanilino)-N-(4-cyclopropylphenyl)-1,7,7-trimethyl-8H-furo[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C28H26ClFN4O2
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
|
CP0349862
|
2-(2,6-dichloroanilino)-7,7-dimethyl-N-[4-(trifluoromethyl)phenyl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H19Cl2F3N4O2
|
1
|
| 1 |
IC50 = 4.4 nM
|
|
|
|
CP0131815
|
N-[[4-chloro-3-[4-oxo-7-[4-(trifluoromethyl)phenyl]-3H-pyrido[4,3-d]pyrimidin-2-yl]phenyl]methyl]-2-methylpropanamide
Show/Hide
|
C25H20ClF3N4O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0181874
|
(4S)-N-[(2S,4S)-2-(hydroxymethyl)oxan-4-yl]-3,3-dimethyl-1-(8-methylquinolin-2-yl)piperidine-4-carboxamide
Show/Hide
|
C24H33N3O3
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0241969
|
2-(2,6-dichloroanilino)-7,7-dimethyl-N-[2-(trifluoromethyl)phenyl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H19Cl2F3N4O2
|
1
|
| 1 |
IC50 = 5.2 nM
|
|
|
|
CP0169344
|
2-(2-chloro-6-fluoroanilino)-N-(5-cyclopropyl-2-fluorophenyl)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C27H23ClF2N4O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0515995
|
2-(2-chloro-6-fluoroanilino)-7,7-dimethyl-N-[2-methyl-4-(trifluoromethyl)phenyl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C26H21ClF4N4O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0566737
|
2-(2-chloro-6-fluoroanilino)-N-[5-(difluoromethyl)-2-fluorophenyl]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H19ClF4N4O2
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0416843
|
2-[(3,5-dichloropyridin-4-yl)amino]-7,7-dimethyl-N-[4-(trifluoromethyl)phenyl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H18Cl2F3N5O2
|
1
|
| 1 |
IC50 = 7.2 nM
|
|
|
|
CP0416839
|
N-(cyclohexylmethyl)-2-[(3,5-dichloropyridin-4-yl)amino]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H27Cl2N5O2
|
1
|
| 1 |
IC50 = 7.8 nM
|
|
|
|
CP0137642
|
2-(2-chloro-6-fluoroanilino)-N-[2-fluoro-5-(trifluoromethyl)phenyl]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H18ClF5N4O2
|
1
|
| 1 |
IC50 = 9.6 nM
|
|
|
|
CP0515996
|
2-(2-chloro-6-fluoroanilino)-N-[2-fluoro-4-(trifluoromethyl)phenyl]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H18ClF5N4O2
|
1
|
| 1 |
IC50 = 9.6 nM
|
|
|
|
CP0476673
|
2-(2-chloro-6-fluoroanilino)-7,7-dimethyl-N-[2-(trifluoromethyl)phenyl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H19ClF4N4O2
|
1
|
| 1 |
IC50 = 9.7 nM
|
|
|
|
CP0250919
|
N-[[4-chloro-3-[4-oxo-7-[4-(trifluoromethyl)phenyl]-3H-quinazolin-2-yl]phenyl]methyl]-2-methylpropanamide
Show/Hide
|
C26H21ClF3N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0097550
|
2-(2-chloro-6-fluoroanilino)-7,7-dimethyl-N-[4-(trifluoromethyl)phenyl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H19ClF4N4O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0069219
|
2-(2-chloro-6-methylanilino)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C26H21ClF4N4O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0360800
|
N-[[4-chloro-3-[4-oxo-7-[4-(trifluoromethyl)phenyl]-3H-pyrido[2,3-d]pyrimidin-2-yl]phenyl]methyl]-2-methylpropanamide
Show/Hide
|
C25H20ClF3N4O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0455231
|
(4S)-N-[(1S,3S)-3-(hydroxymethyl)cyclohexyl]-3,3-dimethyl-1-[4-(trifluoromethyl)phenyl]piperidine-4-carboxamide
Show/Hide
|
C22H31F3N2O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0429932
|
2-(2,6-dichloroanilino)-N-(4-fluorophenyl)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H19Cl2FN4O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0311347
|
2-(2-chloro-6-methylanilino)-7,7-dimethyl-N-[4-(trifluoromethyl)phenyl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C26H22ClF3N4O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0058531
|
2-(difluoromethyl)-5-[(2-methylpropanoylamino)methyl]-N-[5-methyl-4-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]pyridine-3-carboxamide
Show/Hide
|
C23H22F5N5O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0232206
|
2-(2,6-dichloroanilino)-7,7-dimethyl-N-(2,2,3,3,3-pentafluoropropyl)-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C21H17Cl2F5N4O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0416840
|
2-[(3,5-dichloropyridin-4-yl)amino]-N-[2-fluoro-4-(trifluoromethyl)phenyl]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H17Cl2F4N5O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0550327
|
N-cyclohexyl-2-[(3,5-dichloropyridin-4-yl)amino]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C23H25Cl2N5O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0281117
|
2-(6-chloro-9-(3-hydroxy-3-methylbut-1-ynyl)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
Show/Hide
|
C28H17ClN4O
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0069221
|
2-(2-chloro-6-fluoroanilino)-7,7-dimethyl-N-[5-(trifluoromethyl)pyridin-2-yl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H18ClF4N5O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0137651
|
2-(2-chloro-6-fluoroanilino)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H18ClF5N4O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0398666
|
2-(2-chloro-6-fluoroanilino)-N-[3-fluoro-5-(trifluoromethyl)phenyl]-7,8-dihydro-3H-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
|
C23H14ClF5N4O3
|
1
|
| 1 |
IC50 = 14.34 nM
|
|
|
|
CP0561794
|
2-(2,6-dichloroanilino)-N-(2,6-difluorophenyl)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H18Cl2F2N4O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0451763
|
2-(2-chloro-6-fluoroanilino)-N-[4-(2-cyclopropylethynyl)-3-fluorophenyl]-7,8-dihydro-3H-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
|
C27H19ClF2N4O3
|
1
|
| 1 |
IC50 = 16.21 nM
|
|
|
|
CP0071480
|
2-(2-chloro-6-fluoroanilino)-N-[3-fluoro-5-(trifluoromethyl)phenyl]-1-methyl-7,8-dihydro-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H16ClF5N4O3
|
2
|
| 1 |
IC50 = 16.24 nM
|
|
|
| 2 |
IC50 = 1900 nM
|
|
|
|
CP0404220
|
2-(2,6-dichloroanilino)-7-methyl-N-[3-(trifluoromethyl)phenyl]-3H-furo[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H15Cl2F3N4O2
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0507838
|
2-(2-chloro-6-fluoroanilino)-1-methyl-N-[4-(trifluoromethyl)phenyl]-7,8-dihydro-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H17ClF4N4O3
|
1
|
| 1 |
IC50 = 18.53 nM
|
|
|
|
CP0466940
|
N-[5-(4-chlorophenyl)-1H-imidazol-2-yl]-2-(difluoromethyl)-5-[(2-methylpropanoylamino)methyl]benzamide
Show/Hide
|
C22H21ClF2N4O2
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0470789
|
2-(2-chloro-6-fluoroanilino)-N-(3-cyclohexylphenyl)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C30H30ClFN4O2
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0093902
|
2-(2-chlorophenyl)-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C21H13ClN2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0451020
|
2-(2,6-dichloroanilino)-7,7-dimethyl-N-[6-(trifluoromethyl)pyridin-3-yl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H18Cl2F3N5O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0519801
|
2-(2-chloro-6-fluoroanilino)-N-(4-fluorophenyl)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H19ClF2N4O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0433695
|
2-(9-(2-(1H-pyrrol-1-yl)ethoxy)-6-chloro-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
Show/Hide
|
C29H18ClN5O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0115746
|
4-chloro-2-[[(1S,2S)-2-[(1-phenylpiperidine-4-carbonyl)amino]cyclopentyl]methylamino]benzoic acid
Show/Hide
|
C25H30ClN3O3
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0411841
|
N-[[4-chloro-3-[4-oxo-7-[6-(trifluoromethyl)pyridin-3-yl]-3H-quinazolin-2-yl]phenyl]methyl]-2-methylpropanamide
Show/Hide
|
C25H20ClF3N4O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0419567
|
(4S)-3,3-dimethyl-1-(8-methylquinolin-2-yl)-N-[(3S)-oxolan-3-yl]piperidine-4-carboxamide
Show/Hide
|
C22H29N3O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0551485
|
2-(2-chloro-6-fluoroanilino)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-1-methyl-7,8-dihydro-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H16ClF5N4O3
|
1
|
| 1 |
IC50 = 26.69 nM
|
|
|
|
CP0485330
|
2-(6-chloro-9-((1-hydroxycyclopentyl)ethynyl)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
Show/Hide
|
C30H19ClN4O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0394336
|
2-(2-chloro-6-methylanilino)-7,7-dimethyl-N-[5-(trifluoromethyl)pyridin-2-yl]-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H21ClF3N5O2
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0518038
|
2-(2-chloro-6-methylanilino)-N-[3-fluoro-5-(trifluoromethyl)phenyl]-7,8-dihydro-3H-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
|
C24H17ClF4N4O3
|
1
|
| 1 |
IC50 = 27.82 nM
|
|
|
|
CP0470787
|
2-(2-chloro-6-fluoroanilino)-N-(5-chloropyridin-2-yl)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C23H18Cl2FN5O2
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0401000
|
(4S)-1-(8-chloroquinolin-2-yl)-N-[4-(hydroxymethyl)cyclohexyl]-3,3-dimethylpiperidine-4-carboxamide
Show/Hide
|
C24H32ClN3O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0137643
|
2-(2-chloro-6-methylanilino)-N-[2-fluoro-5-(trifluoromethyl)phenyl]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
|
C26H21ClF4N4O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0377490
|
2-(2-chloro-6-fluoroanilino)-N-(4,4-dimethylcyclohexyl)-1-methyl-7,8-dihydro-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
|
C25H28ClFN4O3
|
1
|
| 1 |
IC50 = 30.62 nM
|
|
|
|
CP0156847
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2-(2-chloro-6-fluorophenyl)-7-phenyl-3,5-dihydroimidazo[4,5-c]quinolin-4-one
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C22H13ClFN3O
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1
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| 1 |
IC50 = 33 nM
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CP0483610
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N-[[6-(difluoromethyl)-5-[4-oxo-7-[4-(trifluoromethyl)phenyl]-3H-quinazolin-2-yl]pyridin-3-yl]methyl]-2-methylpropanamide
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C26H21F5N4O2
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1
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| 1 |
IC50 = 33 nM
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CP0346754
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2-(2-chloro-6-fluoroanilino)-N-[6-(difluoromethyl)pyridin-3-yl]-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
Show/Hide
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C24H19ClF3N5O2
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1
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| 1 |
IC50 = 33 nM
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CP0433711
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2-(6-chloro-9-(2-hydroxypropan-2-yl)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
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C26H17ClN4O
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1
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| 1 |
IC50 = 34 nM
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CP0446032
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2-(2-chloro-6-fluoroanilino)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-7,8-dihydro-3H-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
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C23H14ClF5N4O3
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1
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| 1 |
IC50 = 35.07 nM
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CP0497717
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N-[5-(4-chlorophenyl)-1H-imidazol-2-yl]-2-(difluoromethyl)-5-[(2-methylpropanoylamino)methyl]pyridine-3-carboxamide
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C21H20ClF2N5O2
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1
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| 1 |
IC50 = 37 nM
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CP0439310
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2-(6-chloro-9-(3-cyanopropoxy)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
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C27H16ClN5O
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1
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| 1 |
IC50 = 38 nM
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CP0377491
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2-(2-chloro-6-fluoroanilino)-N-[4-(trifluoromethyl)phenyl]-7,8-dihydro-3H-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
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C23H15ClF4N4O3
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1
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| 1 |
IC50 = 38.39 nM
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CP0406677
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N-[4-(4-chlorophenyl)-5-methyl-1H-imidazol-2-yl]-2-(difluoromethyl)-5-[(2-methylpropanoylamino)methyl]pyridine-3-carboxamide
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C22H22ClF2N5O2
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1
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| 1 |
IC50 = 39 nM
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CP0416838
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N-cyclohexyl-2-[(3,5-dichloropyridin-4-yl)amino]-7-methyl-3H-furo[3,2-e]benzimidazole-5-carboxamide
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C22H21Cl2N5O2
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1
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| 1 |
IC50 = 39 nM
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CP0508484
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2-(2-chloro-6-fluoroanilino)-N-[3-(trifluoromethyl)phenyl]-7,8-dihydro-3H-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
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C23H15ClF4N4O3
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1
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| 1 |
IC50 = 41.38 nM
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CP0507834
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2-(2-chloro-6-fluoroanilino)-1-methyl-N-[3-(trifluoromethyl)phenyl]-7,8-dihydro-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
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C24H17ClF4N4O3
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1
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| 1 |
IC50 = 42.65 nM
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CP0398668
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2-(2-chloro-6-fluoroanilino)-N-[3-(trifluoromethyl)phenyl]-3H-imidazo[4,5-f]quinoline-5-carboxamide
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C24H14ClF4N5O
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1
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| 1 |
IC50 = 43.1 nM
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CP0485328
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2-(6-chloro-9-(4-(methylsulfonyl)phenyl)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
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C30H17ClN4O2S
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1
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| 1 |
IC50 = 45 nM
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CP0511703
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N-(cyclopropylmethyl)-2-(2,6-dichloroanilino)-7,7-dimethyl-3,8-dihydrofuro[3,2-e]benzimidazole-5-carboxamide
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C22H22Cl2N4O2
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1
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| 1 |
IC50 = 47 nM
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CP0377489
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2-(2-chloro-6-fluoroanilino)-N-[3-fluoro-5-(trifluoromethyl)phenyl]-6,7-dimethoxy-1-methylbenzimidazole-5-carboxamide
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C24H18ClF5N4O3
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1
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| 1 |
IC50 = 47.38 nM
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CP0446033
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2-(2-chloro-6-fluoroanilino)-N-[4-(2-cyclopropylethynyl)-3-fluorophenyl]-1-methyl-7,8-dihydro-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
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C28H21ClF2N4O3
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1
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| 1 |
IC50 = 51.13 nM
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CP0454687
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2-(2-chloro-6-fluoroanilino)-1-ethyl-N-[3-fluoro-5-(trifluoromethyl)phenyl]-7,8-dihydro-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
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C25H18ClF5N4O3
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1
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| 1 |
IC50 = 54.69 nM
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CP0047355
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2-(6-chloro-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
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C23H11ClN4
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3
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| 1 |
IC50 = 56 nM
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| 2 |
IC50 = 76 nM
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| 3 |
IC50 = 420 nM
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CP0430972
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2-(6-chloro-9-(pyridin-3-ylethynyl)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
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C30H14ClN5
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1
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| 1 |
IC50 = 57 nM
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CP0498613
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2-(6-chloro-9-(3-methoxyprop-1-ynyl)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
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C27H15ClN4O
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1
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| 1 |
IC50 = 60 nM
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CP0443667
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N-(9-ethylcarbazol-3-yl)-2-(trifluoromethyl)benzamide
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C22H17F3N2O
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1
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| 1 |
IC50 = 60 nM
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CP0474564
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7-bromo-2-(2-chlorophenyl)-4-methoxy-3H-imidazo[4,5-c]quinoline
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C17H11BrClN3O
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1
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| 1 |
IC50 = 60 nM
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CP0398667
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2-(2-chloro-6-fluoroanilino)-N-(4,4-dimethylcyclohexyl)-7,8-dihydro-3H-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
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C24H26ClFN4O3
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1
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| 1 |
IC50 = 64.3 nM
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CP0454686
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2-(2-chloro-6-fluoroanilino)-1-methyl-N-[4-(trifluoromethyl)cyclohexyl]-7,8-dihydro-[1,4]dioxino[2,3-e]benzimidazole-5-carboxamide
Show/Hide
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C24H23ClF4N4O3
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1
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| 1 |
IC50 = 65 nM
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CP0413896
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2,3-dihydro-1H-inden-5-yl N-anilino-N-(4-methoxyphenyl)sulfonylcarbamate
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C23H22N2O5S
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1
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| 1 |
IC50 = 70 nM
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CP0140129
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(4S)-3,3-dimethyl-1-(8-methylquinolin-2-yl)-N-[(3S)-oxan-3-yl]piperidine-4-carboxamide
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C23H31N3O2
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1
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| 1 |
IC50 = 72 nM
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CP0433697
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2-(6-chloro-9-(pyridin-4-ylethynyl)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
Show/Hide
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C30H14ClN5
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1
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| 1 |
IC50 = 75 nM
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CP0419568
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(4S)-3,3-dimethyl-N-[(2R)-3-methylbutan-2-yl]-1-(8-methylquinolin-2-yl)piperidine-4-carboxamide
Show/Hide
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C23H33N3O
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1
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| 1 |
IC50 = 89 nM
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CP0477246
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2-(difluoromethyl)-N-[5-methyl-4-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]-5-[(propanoylamino)methyl]pyridine-3-carboxamide
Show/Hide
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C22H20F5N5O2
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1
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| 1 |
IC50 = 98 nM
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CP0433694
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2-(6-chloro-9-(methylsulfonyl)-1H-phenanthro[9,10-d]imidazol-2-yl)isophthalonitrile
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C24H13ClN4O2S
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1
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| 1 |
IC50 = 110 nM
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CP0428919
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N-[[6-(difluoromethyl)-5-[4-oxo-7-[4-(trifluoromethyl)phenyl]-3H-pyrido[4,3-d]pyrimidin-2-yl]pyridin-3-yl]methyl]-2-methylpropanamide
Show/Hide
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C25H20F5N5O2
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1
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| 1 |
IC50 = 111 nM
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CP0446108
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CHEMBL3956753
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C24H24ClF3N4O3
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1
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| 1 |
IC50 = 128.6 nM
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CP0546399
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(4-phenylmethoxyphenyl) N-(3-chloroanilino)-N-(4-chlorophenyl)sulfonylcarbamate
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C26H20Cl2N2O5S
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1
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| 1 |
IC50 = 150 nM
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CP0517462
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2-(2-chloro-6-fluoroanilino)-1-methyl-N-[3-(trifluoromethyl)phenyl]imidazo[4,5-f]quinoline-5-carboxamide
Show/Hide
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C25H16ClF4N5O
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1
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| 1 |
IC50 = 153.2 nM
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CP0546401
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(4-phenylmethoxyphenyl) N-benzyl-N-(4-chlorophenyl)sulfonylcarbamate
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C27H22ClNO5S
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2
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| 1 |
IC50 = 160 nM
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| 2 |
IC50 = 2000 nM
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CP0018449
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2-chloro-N-[3-[(2-chlorophenyl)methyl]-4-oxo-2-propylquinazolin-6-yl]benzamide
Show/Hide
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C25H21Cl2N3O2
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1
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| 1 |
IC50 = 180 nM
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CP0019782
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2-chloro-N-[3-[[4-(4-chlorophenyl)phenyl]methyl]-4-oxo-2-propylquinazolin-6-yl]benzamide
Show/Hide
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C31H25Cl2N3O2
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1
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| 1 |
IC50 = 180 nM
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CP0257285
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2-bromo-5-[(2,2-dimethylpropanoylamino)methyl]-N-(1H-imidazol-2-yl)benzamide
Show/Hide
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C16H19BrN4O2
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2
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| 1 |
IC50 = 180 nM
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| 2 |
IC50 = 284 nM
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CP0546400
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(4-phenylmethoxyphenyl) N-anilino-N-(4-chlorophenyl)sulfonylcarbamate
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C26H21ClN2O5S
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2
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| 1 |
IC50 = 190 nM
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| 2 |
IC50 = 250 nM
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CP0255649
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5-hydroxy-1H-benzo[g]indole-3-carboxylate, 11f
Show/Hide
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C22H18BrNO3
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1
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| 1 |
IC50 = 200 nM
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CP0062008
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CHEBI:3962
Show/Hide
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C21H20O6
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2
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| 1 |
IC50 = 200 nM
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| 2 |
IC50 = 220 nM
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CP0303348
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1-(3-((4-chlorophenyl)ethynyl)benzyl)-3-isopropyl-1-(3-(pyridin-3-ylethynyl)benzyl)urea
Show/Hide
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C33H28ClN3O
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1
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| 1 |
IC50 = 240 nM
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CP0546402
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1-benzyl-1-(4-chlorophenyl)sulfonyl-3-[4-(4-phenylbutoxy)phenyl]urea
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C30H29ClN2O4S
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2
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| 1 |
IC50 = 240 nM
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| 2 |
IC50 = 1000 nM
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CP0477692
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2-[4,4-dimethyl-7-[2-[2-(trifluoromethoxy)phenyl]ethynyl]-3H-chromeno[3,4-d]imidazol-2-yl]benzene-1,3-dicarbonitrile
Show/Hide
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C29H17F3N4O2
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1
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| 1 |
IC50 = 266.7 nM
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CP0433710
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2-(6-bromo-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazol-9-yl)propan-2-ol
Show/Hide
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C24H17BrClFN2O
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1
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| 1 |
IC50 = 280 nM
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CP0458560
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2-[4,4-dimethyl-7-[2-[2-(trifluoromethyl)phenyl]ethynyl]-3H-chromeno[3,4-d]imidazol-2-yl]benzene-1,3-dicarbonitrile
Show/Hide
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C29H17F3N4O
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1
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| 1 |
IC50 = 297.6 nM
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CP0458856
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2-[4-chloro-6-[[4-(3,4-dichlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C21H21Cl3N4O2S2
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1
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| 1 |
IC50 = 300 nM
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CP0473898
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1-(6-bromo-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazol-9-yl)ethanone
Show/Hide
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C23H13BrClFN2O
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1
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| 1 |
IC50 = 330 nM
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CP0322260
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3-isopropyl-1-(3-(pyridin-3-ylethynyl)benzyl)-1-(3-((4-(trifluoromethyl)phenyl)ethynyl)benzyl)urea
Show/Hide
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C34H28F3N3O
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1
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| 1 |
IC50 = 330 nM
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CP0371059
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1-(3-((4-chlorophenyl)ethynyl)benzyl)-3-isopropyl-1-(3-(pyridin-4-ylethynyl)benzyl)urea
Show/Hide
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C33H28ClN3O
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1
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| 1 |
IC50 = 340 nM
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CP0288197
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3-isopropyl-1-(3-(phenylethynyl)benzyl)-1-((5-(phenylethynyl)pyridin-3-yl)methyl)urea
Show/Hide
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C33H29N3O
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1
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| 1 |
IC50 = 360 nM
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CP0401161
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7-bromo-2-(2-methylphenyl)-3H-imidazo[4,5-c]quinoline
Show/Hide
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C17H12BrN3
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1
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| 1 |
IC50 = 395 nM
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CP0147938
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2-[4-chloro-6-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C25H25ClN4O2S2
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1
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| 1 |
IC50 = 400 nM
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CP0415361
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2-[4-chloro-6-[[4-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C25H29ClN4O2S2
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1
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| 1 |
IC50 = 400 nM
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CP0484518
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2-[4-chloro-6-[[4-[4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C22H22ClF3N4O2S2
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1
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| 1 |
IC50 = 400 nM
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CP0489861
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2-[4-chloro-6-[[4-(2,4-dichlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C21H21Cl3N4O2S2
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1
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| 1 |
IC50 = 400 nM
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CP0063083
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(2S)-2-[(3R,5R,9R,10R,13S,14S,17S)-3-acetyloxy-4,4,10,13,14-pentamethyl-2,3,5,6,9,11,12,15,16,17-decahydro-1H-cyclopenta[a]phenanthren-17-yl]-6-methylhept-5-enoic acid
Show/Hide
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C32H50O4
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1
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| 1 |
IC50 = 400 nM
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CP0308443
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(2S)-2-[(3R,5R,10S,13S,14S,17S)-3-acetyloxy-4,4,10,13,14-pentamethyl-2,3,5,6,7,11,12,15,16,17-decahydro-1H-cyclopenta[a]phenanthren-17-yl]-6-methylhept-5-enoic acid
Show/Hide
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C32H50O4
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1
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| 1 |
IC50 = 400 nM
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CP0385952
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Arzanol
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C22H26O7
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1
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| 1 |
IC50 = 400 nM
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CP0055252
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4-(2,4-dihydroxy-6-pentylbenzoyl)oxy-2-hydroxy-6-pentylbenzoic acid
Show/Hide
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C24H30O7
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1
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| 1 |
IC50 = 400 nM
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CP0039011
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3,8-Dihydroxy-11-oxo-1-(2-oxo-heptyl)-6-pentyl-11H-dibenzo[b,e][1,4]dioxepine-7-carboxylic acid
Show/Hide
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C26H30O8
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1
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| 1 |
IC50 = 430 nM
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CP0433709
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2-(6-bromo-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazol-9-yl)-1,1,1,3,3,3-hexafluoropropan-2-ol
Show/Hide
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C24H11BrClF7N2O
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1
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| 1 |
IC50 = 450 nM
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CP0402842
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2-(2-chloro-6-fluorophenyl)-7-[2-[2-fluoro-5-(trifluoromethyl)phenyl]ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazole
Show/Hide
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C27H16ClF5N2O
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1
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| 1 |
IC50 = 461 nM
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CP0358106
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1-(3-((4-chlorophenyl)ethynyl)benzyl)-3-isopropyl-1-(3-(pyridin-2-ylethynyl)benzyl)urea
Show/Hide
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C33H28ClN3O
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1
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| 1 |
IC50 = 480 nM
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CP0047353
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1-((5-(cyclopentylethynyl)pyridin-3-yl)methyl)-3-isopropyl-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
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C32H33N3O
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1
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| 1 |
IC50 = 490 nM
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CP0282713
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1-((5-(cyclopropylethynyl)pyridin-3-yl)methyl)-3-isopropyl-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
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C30H29N3O
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1
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| 1 |
IC50 = 490 nM
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CP0379997
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2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyl-2-naphthalen-1-ylacetic acid
Show/Hide
|
C25H16Cl2N4O2S2
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1
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| 1 |
IC50 = 500 nM
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CP0429185
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2-[4-chloro-6-[[4-(4-phenylphenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C27H27ClN4O2S2
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1
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| 1 |
IC50 = 500 nM
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CP0147392
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2-(trifluoromethyl)-N-[3-[[5-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]benzamide
Show/Hide
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C21H13F6N3O2
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1
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| 1 |
IC50 = 500 nM
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CP0376546
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ethyl 2-(3-fluoroanilino)-5-hydroxy-1H-benzo[g]indole-3-carboxylate
Show/Hide
|
C21H17FN2O3
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1
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| 1 |
IC50 = 500 nM
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CP0461622
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7-bromo-2-(2-bromophenyl)-3H-imidazo[4,5-c]quinoline
Show/Hide
|
C16H9Br2N3
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1
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| 1 |
IC50 = 506 nM
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CP0042594
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1-[5-chloro-6-(4-chlorophenyl)-1,3-benzoxazol-2-yl]-N-[(1S,3S)-3-(hydroxymethyl)cyclohexyl]piperidine-4-carboxamide
Show/Hide
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C26H29Cl2N3O3
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1
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| 1 |
IC50 = 520 nM
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CP0573749
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15-fluoro-4-[2-(trifluoromethyl)phenyl]-3,5,10-triazatetracyclo[11.4.0.02,6.07,12]heptadeca-1(13),2(6),4,7(12),8,14,16-heptaen-11-one
Show/Hide
|
C21H11F4N3O
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1
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| 1 |
IC50 = 560 nM
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CP0560277
|
2-(2-chloro-6-fluorophenyl)-4,4-dimethyl-7-[2-[2-(trifluoromethoxy)phenyl]ethynyl]-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C27H17ClF4N2O2
|
1
|
| 1 |
IC50 = 578 nM
|
|
|
|
CP0484519
|
(2R)-2-[4-chloro-6-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C25H25ClN4O2S2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0515606
|
(2S)-2-[4-chloro-6-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C25H25ClN4O2S2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0525471
|
2-[4-chloro-6-[(4,5-diphenyl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C27H27ClN4O2S2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0003494
|
US9187397, 1 (curcumin)
Show/Hide
|
C21H20O6
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0034689
|
5-hydroxy-1H-benzo[g]indole-3-carboxylate, 11h
Show/Hide
|
C23H21NO4
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0039780
|
5-hydroxy-1H-benzo[g]indole-3-carboxylate, 11a
Show/Hide
|
C22H18ClNO3
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0578592
|
1-benzyl-1-(4-chlorophenyl)sulfonyl-3-(4-phenylmethoxyphenyl)urea
Show/Hide
|
C27H23ClN2O4S
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0458567
|
2-(2-chloro-6-fluorophenyl)-4,4-dimethyl-7-[3-(trifluoromethyl)phenyl]-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C25H17ClF4N2O
|
1
|
| 1 |
IC50 = 616.1 nM
|
|
|
|
CP0458563
|
2-(2-chloro-6-fluorophenyl)-7-[2-[2-fluoro-6-(trifluoromethyl)phenyl]ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C27H16ClF5N2O
|
1
|
| 1 |
IC50 = 691.5 nM
|
|
|
|
CP0457603
|
2-(2-chloro-6-fluorophenyl)-4,4-dimethyl-7-[2-[2-(trifluoromethyl)phenyl]ethynyl]-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C27H17ClF4N2O
|
1
|
| 1 |
IC50 = 692.6 nM
|
|
|
|
CP0384537
|
2-[4-chloro-6-[(5-methyl-4-phenyl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C22H25ClN4O2S2
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0415500
|
2-[4-chloro-6-[[4-(4-methylphenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C22H25ClN4O2S2
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0474289
|
2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H22Cl2N4O2S2
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0891746
|
4-(5-iodo-4-((4-nitro-2-(trifluoromethyl)phenoxy)methyl)-1H-1,2,3-triazol-1-yl)-2-(trifluoromethyl)benzonitrile
Show/Hide
|
C18H8F6IN5O3
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0475961
|
2-(2-chloro-6-fluorophenyl)-7-[2-[5-fluoro-2-(trifluoromethyl)phenyl]ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C27H16ClF5N2O
|
1
|
| 1 |
IC50 = 705.7 nM
|
|
|
|
CP0485329
|
6-chloro-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C21H11Cl2FN2
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0428619
|
5-(acetamidomethyl)-2-(difluoromethyl)-N-[5-methyl-4-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]pyridine-3-carboxamide
Show/Hide
|
C21H18F5N5O2
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0447418
|
6-bromo-2-(2-chloro-6-fluorophenyl)-9-methoxy-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C22H13BrClFN2O
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0400356
|
2-[4-chloro-6-[(4-phenyl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H23ClN4O2S2
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0557492
|
2-[4-[[4-(4-bromophenyl)-1,3-thiazol-2-yl]amino]-6-chloropyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H22BrClN4O2S2
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0957424
|
3-((3-acetyl-2,4,6-trihydroxy-5-(3-methylbut-2-enyl)phenyl)(phenyl)methyl)-6-ethyl-4-hydroxy-5-methyl-2H-pyran-2-one
Show/Hide
|
C28H30O7
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0457604
|
2-[7-[2-[2-fluoro-6-(trifluoromethyl)phenyl]ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazol-2-yl]benzene-1,3-dicarbonitrile
Show/Hide
|
C29H16F4N4O
|
1
|
| 1 |
IC50 = 835.9 nM
|
|
|
|
CP0407239
|
2-(2-chloro-6-fluorophenyl)-7-[2-(5-chloro-2-fluorophenyl)ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C26H16Cl2F2N2O
|
1
|
| 1 |
IC50 = 838.7 nM
|
|
|
|
CP0407243
|
2-(2-chloro-6-fluorophenyl)-4,4-dimethyl-7-[3-(trifluoromethoxy)phenyl]-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C25H17ClF4N2O2
|
1
|
| 1 |
IC50 = 839.7 nM
|
|
|
|
CP0122189
|
2-chloro-5-[(2,2-dimethylpropanoylamino)methyl]-N-(1H-imidazol-2-yl)benzamide
Show/Hide
|
C16H19ClN4O2
|
1
|
| 1 |
IC50 = 870 nM
|
|
|
|
CP0245203
|
2-(4-(biphenyl-4-ylmethylamino)-6-chloropyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C29H22ClN3O2S
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
|
CP0057487
|
2-(4-chloro-6-(3,5-di-tert-butylphenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C30H32ClN3O2S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0403610
|
2-[4-[[4-(1-adamantyl)-1,3-thiazol-2-yl]amino]-6-chloropyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C25H33ClN4O2S2
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0086628
|
(1R,3aS,5aR,5bR,7aR,8R,9S,11aR,11bR,13aR,13bR)-9-acetyloxy-3a-(hydroxymethyl)-5a,5b,8,11a-tetramethyl-1-prop-1-en-2-yl-1,2,3,4,5,6,7,7a,9,10,11,11b,12,13,13a,13b-hexadecahydrocyclopenta[a]chrysene-8-carboxylic acid
Show/Hide
|
C32H50O5
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0168476
|
Beta-elemonic acid
Show/Hide
|
C30H46O3
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0376540
|
7-bromo-2-(3-chlorophenyl)-3H-imidazo[4,5-c]quinoline
Show/Hide
|
C16H9BrClN3
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0322588
|
1-benzyl-3-isopropyl-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
|
C26H26N2O
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0520385
|
(1E,6E)-1-(4-hydroxy-3-methoxyphenyl)-7-[3-methoxy-4-(3-methylbut-2-enoxy)phenyl]hepta-1,6-diene-3,5-dione
Show/Hide
|
C26H28O6
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0058057
|
2-(4-chloro-6-(4-phenoxyphenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C28H20ClN3O3S
|
1
|
| 1 |
IC50 = 940 nM
|
|
|
|
CP0289445
|
2-(4-(biphenyl-4-ylamino)-6-chloropyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C28H20ClN3O2S
|
1
|
| 1 |
IC50 = 940 nM
|
|
|
|
CP0471667
|
2-[2-[5-[2-(2-chloro-6-fluorophenyl)-1H-imidazol-5-yl]pyridin-2-yl]ethynyl]-1,3-thiazole
Show/Hide
|
C19H10ClFN4S
|
1
|
| 1 |
IC50 = 940 nM
|
|
|
|
CP0407240
|
2-[4,4-dimethyl-7-(2-phenylethynyl)-3H-chromeno[3,4-d]imidazol-2-yl]benzene-1,3-dicarbonitrile
Show/Hide
|
C28H18N4O
|
1
|
| 1 |
IC50 = 984 nM
|
|
|
|
CP0322589
|
1-benzyl-3-isopropyl-1-(3-((4-(trifluoromethyl)phenyl)ethynyl)benzyl)urea
Show/Hide
|
C27H25F3N2O
|
1
|
| 1 |
IC50 = 990 nM
|
|
|
|
CP0433708
|
6,9-dibromo-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C21H10Br2ClFN2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0086625
|
3-[(1S,2S,4aR,4bS,6aR,9R,10S,10aR,12aR)-1,4a,4b,6a,9,10-hexamethyl-12-oxo-2-propan-2-yl-3,4,5,6,7,8,9,10,10a,12a-decahydro-2H-chrysen-1-yl]propanoic acid
Show/Hide
|
C30H48O3
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0852794
|
3-((3-acetyl-2,4,6-trihydroxy-5-(3-methylbut-2-enyl)phenyl)(phenyl)methyl)-4-hydroxy-6-methyl-2H-pyran-2-one
Show/Hide
|
C26H26O7
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0957425
|
Hyperforin
Show/Hide
|
C35H52O4
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0541343
|
1-[3-[1-(3-acetyl-2,4,6-trihydroxyphenyl)-3-methylbutyl]-2,4,6-trihydroxyphenyl]ethanone
Show/Hide
|
C21H24O8
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0466937
|
(1E,6E)-1-[4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-3-methoxyphenyl]-7-(4-hydroxy-3-methoxyphenyl)hepta-1,6-diene-3,5-dione
Show/Hide
|
C31H36O6
|
1
|
| 1 |
IC50 = 1020 nM
|
|
|
|
CP0433696
|
6-bromo-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C21H11BrClFN2
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0439311
|
2-(2-chloro-6-fluorophenyl)-6,9-dimethyl-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C23H16ClFN2
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0224818
|
CHEBI:10274
Show/Hide
|
C30H48O3
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0327846
|
1-[5-[1-[3-acetyl-2,6-dihydroxy-4-methoxy-5-(3-methylbut-2-enyl)phenyl]-3-methylbutyl]-4,6-dihydroxy-2-(2-hydroxypropan-2-yl)-2,3-dihydro-1-benzofuran-7-yl]ethanone
Show/Hide
|
C32H42O9
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0327847
|
CHEBI:2440
Show/Hide
|
C32H42O8
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0534837
|
1-[3-[1-[3-acetyl-2,6-dihydroxy-4-methoxy-5-(3-methylbut-2-enyl)phenyl]-3-methylbutyl]-2,4,6-trihydroxy-5-[(2S)-2-hydroxy-3-methylbut-3-enyl]phenyl]ethanone
Show/Hide
|
C32H42O9
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0190508
|
4-[2,4-dihydroxy-6-(2-oxoheptyl)benzoyl]oxy-2-hydroxy-6-pentylbenzoic acid
Show/Hide
|
C26H32O8
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
|
CP0458556
|
2-[7-[2-[2-chloro-5-(trifluoromethyl)phenyl]ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazol-2-yl]benzene-1,3-dicarbonitrile
Show/Hide
|
C29H16ClF3N4O
|
1
|
| 1 |
IC50 = 1196 nM
|
|
|
|
CP0400697
|
2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanylhexanoic acid
Show/Hide
|
C19H18Cl2N4O2S2
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0092232
|
(2S)-2-[(3S,5R,10S,13S,14S,17S)-3-hydroxy-4,4,10,13,14-pentamethyl-2,3,5,6,7,11,12,15,16,17-decahydro-1H-cyclopenta[a]phenanthren-17-yl]-6-methylhept-5-enoic acid
Show/Hide
|
C30H48O3
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0327845
|
1-[6-[1-(8-acetyl-5,7-dihydroxy-2,2-dimethylchromen-6-yl)-3-methylbutyl]-5,7-dihydroxy-2,2-dimethylchromen-8-yl]ethanone
Show/Hide
|
C31H36O8
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0406679
|
2-chloro-5-[(2,2-dimethylbutanoylamino)methyl]-N-(1H-imidazol-2-yl)benzamide
Show/Hide
|
C17H21ClN4O2
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
|
CP0520419
|
sodium;3-[1-[(4-chlorophenyl)methyl]-5-(3-fluoro-4-phenylphenyl)-3-methylindol-2-yl]-2,2-dimethylpropanoate
Show/Hide
|
C33H28ClFNNaO2
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
|
CP0477689
|
2-(2-chloro-6-fluorophenyl)-7-[2-[4-fluoro-3-(trifluoromethyl)phenyl]ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C27H16ClF5N2O
|
1
|
| 1 |
IC50 = 1252 nM
|
|
|
|
CP0287373
|
1-benzyl-3-isopropyl-1-(3-((3-methoxyphenyl)ethynyl)benzyl)urea
Show/Hide
|
C27H28N2O2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0384541
|
2-[4-[[4-(4-bromophenyl)-5-methyl-1,3-thiazol-2-yl]amino]-6-chloropyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C22H24BrClN4O2S2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0525472
|
2-[4-chloro-6-[[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C22H25ClN4O3S2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0288232
|
N-[4-chloro-3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-2-(trifluoromethyl)benzamide
Show/Hide
|
C22H14ClF3N2O2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0467503
|
2-[5-(4-bromophenyl)-1H-imidazol-2-yl]benzonitrile
Show/Hide
|
C16H10BrN3
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0247541
|
Acrofolione A
Show/Hide
|
C32H42O9
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0384539
|
2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanylbutanoic acid
Show/Hide
|
C17H14Cl2N4O2S2
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0557493
|
2-[4-chloro-6-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanylbutanoic acid
Show/Hide
|
C21H17ClN4O2S2
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0388951
|
5-[4-(benzenesulfonyl)phenyl]-2-(2-chloro-6-fluorophenyl)-1H-imidazole
Show/Hide
|
C21H14ClFN2O2S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0489202
|
2-(2-chloro-6-fluorophenyl)-7-[2-(2,5-dichlorophenyl)ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C26H16Cl3FN2O
|
1
|
| 1 |
IC50 = 1416 nM
|
|
|
|
CP0058056
|
2-(4-chloro-6-(4-cyclohexylphenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C28H26ClN3O2S
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
|
CP0058121
|
2-(4-(4-benzylphenylamino)-6-chloropyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C29H22ClN3O2S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0229013
|
(1E,4E)-1,5-bis[4-hydroxy-3-methoxy-5-(3-methylbut-2-enyl)phenyl]penta-1,4-dien-3-one
Show/Hide
|
C29H34O5
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0461960
|
7-bromo-2-(3-methylphenyl)-3H-imidazo[4,5-c]quinoline
Show/Hide
|
C17H12BrN3
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0058122
|
2-(4-(9H-fluoren-2-ylamino)-6-chloropyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C29H20ClN3O2S
|
1
|
| 1 |
IC50 = 1550 nM
|
|
|
|
CP0230609
|
2-(4-(Biphenyl-4-ylamino)-6-chloropyrimidine-2-ylthio)octanoic acid
Show/Hide
|
C24H26ClN3O2S
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0230611
|
(R)-2-(4-Chloro-6-(4'-cyanobiphenyl-4-ylamino)pyrimidin-2-ylthio)octanoic acid
Show/Hide
|
C25H25ClN4O2S
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0258508
|
1-benzyl-2-cyano-3-isopropyl-1-(3-(phenylethynyl)benzyl)guanidine
Show/Hide
|
C27H26N4
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1
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| 1 |
IC50 = 1600 nM
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CP0303350
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1-benzyl-3-(pentan-3-yl)-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
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C28H30N2O
|
1
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| 1 |
IC50 = 1600 nM
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CP0240937
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2-(4-chloro-6-(4'-cyanobiphenyl-4-ylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
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C29H19ClN4O2S
|
1
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| 1 |
IC50 = 1600 nM
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CP0384532
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2-[4-chloro-6-[[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C21H21ClF2N4O2S2
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1
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| 1 |
IC50 = 1600 nM
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CP0230610
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2-(4-Chloro-6-(4'-cyanobiphenyl-4-ylamino)pyrimidin-2-ylthio)octanoic acid
Show/Hide
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C25H25ClN4O2S
|
1
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| 1 |
IC50 = 1700 nM
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CP0557490
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2-[4-chloro-6-[(5-ethyl-4-phenyl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C23H27ClN4O2S2
|
1
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| 1 |
IC50 = 1700 nM
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CP0557491
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2-[4-chloro-6-[(4-naphthalen-1-yl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C25H25ClN4O2S2
|
1
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| 1 |
IC50 = 1700 nM
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CP0166358
|
1H-benzo[g]indole-3-carboxylate, 19
Show/Hide
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C24H22ClNO5
|
1
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| 1 |
IC50 = 1700 nM
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CP0322259
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1-benzyl-1-(biphenyl-3-ylmethyl)-3-isopropylurea
Show/Hide
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C24H26N2O
|
2
|
| 1 |
IC50 = 1700 nM
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| 2 |
IC50 = 11900 nM
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CP0267329
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1-benzyl-3-isopropyl-1-(3-((3-(trifluoromethyl)phenyl)ethynyl)benzyl)urea
Show/Hide
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C27H25F3N2O
|
1
|
| 1 |
IC50 = 1800 nM
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CP0379172
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2-[4-chloro-6-[[4-(2,4-difluorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C21H21ClF2N4O2S2
|
1
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| 1 |
IC50 = 1800 nM
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CP0085429
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2-(4-(biphenyl-3-ylamino)-6-chloropyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
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C28H20ClN3O2S
|
1
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| 1 |
IC50 = 1900 nM
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CP0245202
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2-(4-chloro-6-(naphthalen-2-ylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
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C26H18ClN3O2S
|
1
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| 1 |
IC50 = 1900 nM
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CP0379171
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2-[4-chloro-6-[(7-methoxy-4,5-dihydrobenzo[e][1,3]benzothiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C24H27ClN4O3S2
|
1
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| 1 |
IC50 = 1900 nM
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CP0460796
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1-[8-[1-[3-acetyl-2,6-dihydroxy-4-methoxy-5-(3-methylbut-2-enyl)phenyl]-3-methylbutyl]-3,5,7-trihydroxy-2,2-dimethyl-3,4-dihydrochromen-6-yl]ethanone
Show/Hide
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C32H42O9
|
1
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| 1 |
IC50 = 1900 nM
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CP0373928
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6-bromo-2-(2-chloro-6-fluorophenyl)-9-isopropyl-1H-phenanthro[9,10-d]imidazole
Show/Hide
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C24H17BrClFN2
|
1
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| 1 |
IC50 = 2000 nM
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CP0272303
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1-benzyl-1-(3-((4-chlorophenyl)ethynyl)benzyl)-3-isopropylurea
Show/Hide
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C26H25ClN2O
|
1
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| 1 |
IC50 = 2000 nM
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CP0039355
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3-(1-(4-chlorobenzyl)-3-(tert-butylthio)-5-isopropyl-1H-indol-2-yl)-2,2-dimethylpropanoic acid
Show/Hide
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C27H34ClNO2S
|
4
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| 1 |
IC50 = 2000 nM
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| 2 |
IC50 = 2100 nM
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| 3 |
IC50 = 2400 nM
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| 4 |
IC50 = 2500 nM
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CP0388808
|
(1E,6E)-1,7-bis[4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-3-methoxyphenyl]-4,4-bis[(2E)-3,7-dimethylocta-2,6-dienyl]hepta-1,6-diene-3,5-dione
Show/Hide
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C61H84O6
|
1
|
| 1 |
IC50 = 2000 nM
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CP0406735
|
(1E,6E)-1,7-bis[3-methoxy-4-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]phenyl]hepta-1,6-diene-3,5-dione
Show/Hide
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C51H68O6
|
1
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| 1 |
IC50 = 2000 nM
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CP0424961
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(1E,6E)-1,7-bis[3-methoxy-4-(3-methylbut-2-enoxy)phenyl]-4,4-bis(3-methylbut-2-enyl)hepta-1,6-diene-3,5-dione
Show/Hide
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C41H52O6
|
1
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| 1 |
IC50 = 2000 nM
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CP0433338
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(1E,6E)-1,7-bis[3-methoxy-4-(3-methylbut-2-enoxy)phenyl]-4-(3-methylbut-2-enyl)hepta-1,6-diene-3,5-dione
Show/Hide
|
C36H44O6
|
1
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| 1 |
IC50 = 2000 nM
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CP0478456
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(1E,6E)-1,7-bis[3-methoxy-4-(3-methylbut-2-enoxy)phenyl]hepta-1,6-diene-3,5-dione
Show/Hide
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C31H36O6
|
1
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| 1 |
IC50 = 2000 nM
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CP0478457
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(1E,6E)-1,7-bis[4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-3-methoxyphenyl]-4-[(2E)-3,7-dimethylocta-2,6-dienyl]hepta-1,6-diene-3,5-dione
Show/Hide
|
C51H68O6
|
1
|
| 1 |
IC50 = 2000 nM
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CP0478458
|
(1E,6E)-1-(4-hydroxy-3-methoxyphenyl)-7-[3-methoxy-4-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]phenyl]hepta-1,6-diene-3,5-dione
Show/Hide
|
C36H44O6
|
1
|
| 1 |
IC50 = 2000 nM
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CP0573901
|
(1E,6E)-1,7-bis[4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-3-methoxyphenyl]hepta-1,6-diene-3,5-dione
Show/Hide
|
C41H52O6
|
1
|
| 1 |
IC50 = 2000 nM
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CP0036076
|
2-(4-Chloro-6-(5-methoxy-2-methylbiphenyl-4-ylamino)pyrimidin-2-ylthio)octanoic acid
Show/Hide
|
C26H30ClN3O3S
|
1
|
| 1 |
IC50 = 2100 nM
|
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CP0289702
|
(S)-2-(4-Chloro-6-(4'-cyanobiphenyl-4-ylamino)pyrimidin-2-ylthio)octanoic acid
Show/Hide
|
C25H25ClN4O2S
|
1
|
| 1 |
IC50 = 2100 nM
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CP0456801
|
butyl (2R,3R)-5-[(E)-3-butoxy-3-oxoprop-1-enyl]-2-(3,4-dihydroxyphenyl)-7-hydroxy-2,3-dihydro-1-benzofuran-3-carboxylate
Show/Hide
|
C26H30O8
|
1
|
| 1 |
IC50 = 2100 nM
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CP0397162
|
2-(2-(2-chloro-6-fluorophenyl)-6-(2-hydroxypropan-2-yl)-1H-phenanthro[9,10-d]imidazol-9-yl)-1,1,1,3,3,3-hexafluoropropan-2-ol
Show/Hide
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C27H18ClF7N2O2
|
1
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| 1 |
IC50 = 2300 nM
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CP0379998
|
2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanylacetic acid
Show/Hide
|
C15H10Cl2N4O2S2
|
1
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| 1 |
IC50 = 2300 nM
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CP0477688
|
2-[7-[2-(2,5-dichlorophenyl)ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazol-2-yl]benzene-1,3-dicarbonitrile
Show/Hide
|
C28H16Cl2N4O
|
1
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| 1 |
IC50 = 2320 nM
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CP0272304
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1-benzyl-3-cyclobutyl-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
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C27H26N2O
|
1
|
| 1 |
IC50 = 2400 nM
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CP0376538
|
4-(3-chlorophenyl)-15-fluoro-3,5,10-triazatetracyclo[11.4.0.02,6.07,12]heptadeca-1(13),2(6),4,7(12),8,14,16-heptaen-11-one
Show/Hide
|
C20H11ClFN3O
|
1
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| 1 |
IC50 = 2500 nM
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CP0336681
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2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole
Show/Hide
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C21H12ClFN2
|
1
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| 1 |
IC50 = 2600 nM
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CP0371060
|
1-benzyl-3-isopropyl-1-(3-(phenylethynyl)benzyl)thiourea
Show/Hide
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C26H26N2S
|
1
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| 1 |
IC50 = 2700 nM
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CP0548779
|
1-[6-[1-[3-acetyl-2,6-dihydroxy-4-methoxy-5-(3-methylbut-2-enyl)phenyl]-3-methylbutyl]-3,5,7-trihydroxy-2,2-dimethyl-3,4-dihydrochromen-8-yl]ethanone
Show/Hide
|
C32H42O9
|
1
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| 1 |
IC50 = 2700 nM
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CP0081203
|
2-chloro-N-(1H-imidazol-2-yl)-5-[(2-methylpropanoylamino)methyl]benzamide
Show/Hide
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C15H17ClN4O2
|
1
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| 1 |
IC50 = 2770 nM
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CP0470398
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2-phenylethyl (2S,3S)-2-(3,4-dihydroxyphenyl)-7-hydroxy-5-[(E)-3-oxo-3-(2-phenylethoxy)prop-1-enyl]-2,3-dihydro-1-benzofuran-3-carboxylate
Show/Hide
|
C34H30O8
|
1
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| 1 |
IC50 = 2800 nM
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CP0458565
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2-(2-chloro-6-fluorophenyl)-7-[2-[4-chloro-2-(trifluoromethyl)phenyl]ethynyl]-4,4-dimethyl-3H-chromeno[3,4-d]imidazole
Show/Hide
|
C27H16Cl2F4N2O
|
1
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| 1 |
IC50 = 2828 nM
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CP0303349
|
1-benzyl-1-(3-(phenylethynyl)benzyl)-3-propylurea
Show/Hide
|
C26H26N2O
|
1
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| 1 |
IC50 = 2900 nM
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CP0388385
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7-bromo-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C21H11BrClFN2
|
1
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| 1 |
IC50 = 3000 nM
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CP0218628
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3-isopropyl-1-(3-methylbenzyl)-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
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C27H28N2O
|
1
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| 1 |
IC50 = 3000 nM
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CP0036905
|
(3R,4R,4aR,6aR,6bS,8aR,11R,12S,12aR,14aR,14bS)-3-hydroxy-4,6a,6b,8a,11,12,14b-heptamethyl-14-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,14,14a,14b-icosahydropicene-4-carboxylic acid
Show/Hide
|
C30H46O4
|
1
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| 1 |
IC50 = 3000 nM
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CP0096636
|
Acetyl-Beta-Boswellic Acid
Show/Hide
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C32H50O4
|
1
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| 1 |
IC50 = 3000 nM
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CP0168524
|
(3R,4R,4aR,6aR,6bS,8aR,11R,12S,12aR,14aR,14bS)-3-acetoxy-4,6a,6b,8a,11,12,14b-heptamethyl-14-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,14,14a,14b-icosahydropicene-4-carboxylic acid
Show/Hide
|
C32H48O5
|
1
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| 1 |
IC50 = 3000 nM
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CP0183411
|
(2S)-2-[(3R,5R,9R,10R,13S,14S,17S)-3-hydroxy-4,4,10,13,14-pentamethyl-2,3,5,6,9,11,12,15,16,17-decahydro-1H-cyclopenta[a]phenanthren-17-yl]-6-methylhept-5-enoic acid
Show/Hide
|
C30H48O3
|
1
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| 1 |
IC50 = 3000 nM
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CP0406678
|
2-(difluoromethyl)-N-(1H-imidazol-2-yl)-5-[(2-methylpropanoylamino)methyl]benzamide
Show/Hide
|
C16H18F2N4O2
|
1
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| 1 |
IC50 = 3150 nM
|
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CP0532338
|
5-[(2,2-dimethylpropanoylamino)methyl]-N-(1H-imidazol-2-yl)-2-(trifluoromethyl)benzamide
Show/Hide
|
C17H19F3N4O2
|
1
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| 1 |
IC50 = 3230 nM
|
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CP0557085
|
2-(difluoromethyl)-5-[(2,2-dimethylpropanoylamino)methyl]-N-(1H-imidazol-2-yl)benzamide
Show/Hide
|
C17H20F2N4O2
|
1
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| 1 |
IC50 = 3250 nM
|
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CP0075614
|
1-[3-[(2E)-3,7-dimethylocta-2,6-dienyl]-2,4,6-trihydroxyphenyl]ethanone
Show/Hide
|
C18H24O4
|
1
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| 1 |
IC50 = 3500 nM
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CP0371056
|
3-isopropyl-1-(3-methoxybenzyl)-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
|
C27H28N2O2
|
1
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| 1 |
IC50 = 3600 nM
|
|
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CP0448176
|
ethyl (2R,3R)-2-(3,4-dihydroxyphenyl)-5-[(E)-3-ethoxy-3-oxoprop-1-enyl]-7-hydroxy-2,3-dihydro-1-benzofuran-3-carboxylate
Show/Hide
|
C22H22O8
|
1
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| 1 |
IC50 = 3600 nM
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CP0371055
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1-benzyl-1-(3-((3-chlorophenyl)ethynyl)benzyl)-3-isopropylurea
Show/Hide
|
C26H25ClN2O
|
1
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| 1 |
IC50 = 3700 nM
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CP0371057
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1-(biphenyl-3-ylmethyl)-3-isopropyl-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
|
C32H30N2O
|
1
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| 1 |
IC50 = 3700 nM
|
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CP0492135
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1-benzyl-3-(cyclopropylmethyl)-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
|
C27H26N2O
|
1
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| 1 |
IC50 = 3700 nM
|
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CP0443666
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2-(4-bromophenyl)-5-(2-chloro-6-fluorophenyl)-1H-imidazole
Show/Hide
|
C15H9BrClFN2
|
1
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| 1 |
IC50 = 3700 nM
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CP0045837
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2-chloro-N-[(5Z)-5-[(3-ethoxy-4-hydroxyphenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]benzamide
Show/Hide
|
C19H15ClN2O4S2
|
1
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| 1 |
IC50 = 3800 nM
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CP0282712
|
3-isopropyl-1-(3-(phenylethynyl)benzyl)-1-(3-(trifluoromethyl)benzyl)urea
Show/Hide
|
C27H25F3N2O
|
1
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| 1 |
IC50 = 4100 nM
|
|
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CP0501854
|
1-benzyl-3-isopropyl-1-(3-((4-methoxyphenyl)ethynyl)benzyl)urea
Show/Hide
|
C27H28N2O2
|
1
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| 1 |
IC50 = 4200 nM
|
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CP0110880
|
1-[6-[1-[3-acetyl-2,6-dihydroxy-4-methoxy-5-(3-methylbut-2-enyl)phenyl]-3-methylbutyl]-5,7-dihydroxy-2,2-dimethylchromen-8-yl]ethanone
Show/Hide
|
C32H40O8
|
1
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| 1 |
IC50 = 4200 nM
|
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CP0498614
|
5-chloro-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C21H11Cl2FN2
|
1
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| 1 |
IC50 = 4300 nM
|
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CP0353529
|
N-[3-[[benzyl(propan-2-ylcarbamoyl)amino]methyl]phenyl]benzamide
Show/Hide
|
C25H27N3O2
|
1
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| 1 |
IC50 = 4300 nM
|
|
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CP0388950
|
N-[(E)-[5-[(2-chlorophenyl)methyl]-2-hydroxyphenyl]methylideneamino]-2-methoxybenzamide
Show/Hide
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C22H19ClN2O3
|
1
|
| 1 |
IC50 = 4500 nM
|
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CP0452174
|
(4R)-N-[(1S,3S)-3-(hydroxymethyl)cyclohexyl]-3,3-dimethyl-1-[4-(trifluoromethyl)phenyl]piperidine-4-carboxamide
Show/Hide
|
C22H31F3N2O2
|
1
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| 1 |
IC50 = 4500 nM
|
|
|
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CP0499719
|
5-[(2,2-dimethylpropanoylamino)methyl]-N-(1H-imidazol-2-yl)-2-methylbenzamide
Show/Hide
|
C17H22N4O2
|
1
|
| 1 |
IC50 = 4620 nM
|
|
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CP0485327
|
4-bromo-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole
Show/Hide
|
C21H11BrClFN2
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
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CP0400354
|
2-[4-chloro-6-[[4-(4-nitrophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H22ClN5O4S2
|
1
|
| 1 |
IC50 = 5000 nM
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CP0130812
|
(3R,4R,4aR,6aR,6bS,8aR,11R,12S,12aR,14aR,14bR)-3-hydroxy-4,6a,6b,8a,11,12,14b-heptamethyl-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,14,14a,14b-icosahydropicene-4-carboxylic acid
Show/Hide
|
C30H48O3
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
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CP0011912
|
CARNOSIC ACID
Show/Hide
|
C20H28O4
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
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CP0315351
|
(1R,8S,10S)-3,4-dihydroxy-11,11-dimethyl-5-propan-2-yl-16-oxatetracyclo[6.6.2.01,10.02,7]hexadeca-2,4,6-trien-15-one
Show/Hide
|
C20H26O4
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
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CP0266724
|
2-(4-chloro-6-(2,3-dimethylphenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C24H20ClN3O2S
|
1
|
| 1 |
IC50 = 5100 nM
|
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|
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CP0267779
|
2-(4-chloro-6-(4-chlorophenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C22H15Cl2N3O2S
|
1
|
| 1 |
IC50 = 5100 nM
|
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CP0353533
|
1-benzyl-3-cyclopropyl-1-(3-(phenylethynyl)benzyl)urea
Show/Hide
|
C26H24N2O
|
1
|
| 1 |
IC50 = 5200 nM
|
|
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CP0481575
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1-[3-[1-[3-acetyl-5-[(2E)-3,7-dimethylocta-2,6-dienyl]-2,4,6-trihydroxyphenyl]-3-methylbutyl]-5-[(2Z)-3,7-dimethylocta-2,6-dienyl]-2,4,6-trihydroxyphenyl]ethanone
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C41H56O8
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1
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| 1 |
IC50 = 5340 nM
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CP0230612
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ethyl 2-[4-chloro-6-(quinolin-6-ylamino)pyrimidin-2-yl]sulfanyloctanoate
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C23H27ClN4O2S
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1
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| 1 |
IC50 = 5600 nM
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CP0225016
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2-(4-chloro-6-(3,4-dimethylphenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
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C24H20ClN3O2S
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1
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| 1 |
IC50 = 5700 nM
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CP0248135
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2-(4-(Biphenyl-4-ylmethylamino)-6-chloropyrimidin-2-ylthio)octanoic acid
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C25H28ClN3O2S
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1
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| 1 |
IC50 = 6000 nM
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CP0261620
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2-(4-chloro-6-(3-phenylpropylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
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C25H22ClN3O2S
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1
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| 1 |
IC50 = 6100 nM
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CP0566570
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(4-methylphenyl) N-anilino-N-(4-methylphenyl)sulfonylcarbamate
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C21H20N2O4S
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1
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| 1 |
IC50 = 6100 nM
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CP0375712
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(4-phenoxyphenyl) N-anilino-N-(4-methoxyphenyl)sulfonylcarbamate
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C26H22N2O6S
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1
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| 1 |
IC50 = 6600 nM
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CP0373942
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5-bromo-2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole
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C21H11BrClFN2
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1
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| 1 |
IC50 = 7400 nM
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CP0086626
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(1R,3aR,5aR,5bR,7aR,8R,9S,11aR,11bR,13aR,13bR)-9-hydroxy-3a,5a,5b,8,11a-pentamethyl-1-prop-1-en-2-yl-1,2,3,4,5,6,7,7a,9,10,11,11b,12,13,13a,13b-hexadecahydrocyclopenta[a]chrysene-8-carboxylic acid
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C30H48O3
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1
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| 1 |
IC50 = 8500 nM
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CP0256149
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methyl (2R,3R)-2-(3,4-dihydroxyphenyl)-7-hydroxy-5-[(E)-3-methoxy-3-oxoprop-1-enyl]-2,3-dihydro-1-benzofuran-3-carboxylate
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C20H18O8
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1
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| 1 |
IC50 = 8500 nM
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CP0303347
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1-benzyl-3-isopropyl-1-(3-phenoxybenzyl)urea
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C24H26N2O2
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1
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| 1 |
IC50 = 8600 nM
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CP0115322
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(1E,6E)-1,7-bis(3-fluoro-4-hydroxy-5-methoxyphenyl)hepta-1,6-diene-3,5-dione
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C21H18F2O6
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1
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| 1 |
IC50 = 8700 nM
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CP0428630
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2-chloro-N-(1H-imidazol-2-yl)-4-methyl-5-[(2-methylpropanoylamino)methyl]benzamide
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C16H19ClN4O2
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1
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| 1 |
IC50 = 8850 nM
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CP0520420
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2-(difluoromethyl)-N-(1H-imidazol-2-yl)-5-[[[(2S)-2-methylbutanoyl]amino]methyl]benzamide
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C17H20F2N4O2
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1
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| 1 |
IC50 = 8860 nM
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CP0166357
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5-hydroxy-1H-benzo[g]indole-3-carboxylate, 11k
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C21H16ClNO3
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1
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| 1 |
IC50 = 9200 nM
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CP0086627
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(1R,3aR,5aR,5bR,7aR,8R,9S,11aR,11bR,13aR,13bR)-9-acetyloxy-3a,5a,5b,8,11a-pentamethyl-1-prop-1-en-2-yl-1,2,3,4,5,6,7,7a,9,10,11,11b,12,13,13a,13b-hexadecahydrocyclopenta[a]chrysene-8-carboxylic acid
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C32H50O4
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1
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| 1 |
IC50 = 10000 nM
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CP0086648
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3-[(1S,2S,4aR,4bS,6aR,9R,10S,10aR,12aR)-1,4a,4b,6a,9,10-hexamethyl-2-prop-1-en-2-yl-2,3,4,5,6,7,8,9,10,10a,12,12a-dodecahydrochrysen-1-yl]propanoic acid
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C30H48O2
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1
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| 1 |
IC50 > 10000 nM
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CP0213396
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3-[(1S,2S,4aR,4bS,6aR,10aR,12aR)-1,4a,4b,6a,9,9-hexamethyl-2-propan-2-yl-3,4,5,6,7,8,10,10a,12,12a-decahydro-2H-chrysen-1-yl]propanoic acid
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C30H50O2
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1
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| 1 |
IC50 > 10000 nM
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CP0224322
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3-[(1S,2S,4aR,4bS,6aR,9R,10S,10aR,12aR)-1,4a,4b,6a,9,10-hexamethyl-2-propan-2-yl-2,3,4,5,6,7,8,9,10,10a,12,12a-dodecahydrochrysen-1-yl]propanoic acid
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C30H50O2
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1
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| 1 |
IC50 > 10000 nM
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CP0474365
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4-[2-[[2-(1-carboxyheptylsulfanyl)-6-chloropyrimidin-4-yl]amino]-1,3-thiazol-4-yl]benzoic acid
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C22H23ClN4O4S2
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1
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| 1 |
IC50 > 10000 nM
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CP0017229
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4-tert-butyl-15-fluoro-3,5,10-triazatetracyclo[11.4.0.0^{2,6}.0^{7,12}]heptadeca-1(13),2(6),3,7(12),8,14,16-heptaen-11-one
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C18H16FN3O
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1
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| 1 |
IC50 > 10000 nM
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CP0410813
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3-benzyl-1-phenyl-1-[[3-(2-phenylethynyl)phenyl]methyl]urea
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C29H24N2O
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1
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| 1 |
IC50 > 10000 nM
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CP0410814
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15-fluoro-4-(4-methoxyphenyl)-3,5,10-triazatetracyclo[11.4.0.02,6.07,12]heptadeca-1(13),2(6),4,7(12),8,14,16-heptaen-11-one
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C21H14FN3O2
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1
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| 1 |
IC50 > 10000 nM
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CP0542704
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9-fluoro-2-phenyl-3,6-dihydro-1,3,6-triaza-cyclopenta[l]phenanthren-7-one
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C20H12FN3O
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1
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| 1 |
IC50 > 10000 nM
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CP0573748
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1-benzyl-3-phenyl-1-(3-(phenylethynyl)benzyl)urea
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C29H24N2O
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1
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| 1 |
IC50 > 10000 nM
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CP0248013
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(4-phenylmethoxyphenyl) N-anilino-N-(4-methoxyphenyl)sulfonylcarbamate
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C27H24N2O6S
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1
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| 1 |
IC50 > 10000 nM
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CP0407703
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(4-phenylmethoxyphenyl) N-anilino-N-(4-tert-butylphenyl)sulfonylcarbamate
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C30H30N2O5S
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1
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| 1 |
IC50 > 10000 nM
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CP0413895
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(2-methoxyphenyl) N-anilino-N-(4-methylphenyl)sulfonylcarbamate
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C21H20N2O5S
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1
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| 1 |
IC50 > 10000 nM
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CP0425045
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phenyl N-anilino-N-(benzenesulfonyl)carbamate
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C19H16N2O4S
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1
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| 1 |
IC50 > 10000 nM
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CP0425435
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(4-ethylphenyl) N-anilino-N-(4-methoxyphenyl)sulfonylcarbamate
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C22H22N2O5S
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1
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| 1 |
IC50 > 10000 nM
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CP0468615
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(4-phenylmethoxyphenyl) N-anilino-N-(4-methylphenyl)sulfonylcarbamate
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C27H24N2O5S
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1
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| 1 |
IC50 > 10000 nM
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CP0553935
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(4-ethoxyphenyl) N-anilino-N-(4-methoxyphenyl)sulfonylcarbamate
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C22H22N2O6S
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1
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| 1 |
IC50 > 10000 nM
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CP0532339
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2-chloro-4-fluoro-N-(1H-imidazol-2-yl)-5-[(2-methylpropanoylamino)methyl]benzamide
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C15H16ClFN4O2
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1
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| 1 |
IC50 > 10000 nM
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CP0551224
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(4R)-1-(8-chloroquinolin-2-yl)-N-[4-(hydroxymethyl)cyclohexyl]-3,3-dimethylpiperidine-4-carboxamide
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C24H32ClN3O2
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1
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| 1 |
IC50 > 10000 nM
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CP0247540
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1-[3-[1-[3-acetyl-2,4,6-trihydroxy-5-(3-methylbut-2-enyl)phenyl]-3-methylbutyl]-2,4,6-trihydroxy-5-(3-methylbut-2-enyl)phenyl]ethanone
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C31H40O8
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1
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| 1 |
IC50 > 10000 nM
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CP0365175
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1-[5-[1-(7-acetyl-4,6-dihydroxy-2-prop-1-en-2-yl-2,3-dihydro-1-benzofuran-5-yl)-3-methylbutyl]-4,6-dihydroxy-2-prop-1-en-2-yl-2,3-dihydro-1-benzofuran-7-yl]ethanone
Show/Hide
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C31H36O8
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1
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| 1 |
IC50 > 10000 nM
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CP0541344
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1-[2,4,6-trihydroxy-3-(3-methylbut-2-enyl)phenyl]ethanone
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C13H16O4
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1
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| 1 |
IC50 > 10000 nM
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CP0272297
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3-isopropyl-1-(2-methoxybenzyl)-1-(3-(phenylethynyl)benzyl)urea
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C27H28N2O2
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1
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| 1 |
IC50 = 10600 nM
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CP0161385
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1-benzyl-1-(3-(benzyloxy)benzyl)-3-isopropylurea
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C25H28N2O2
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1
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| 1 |
IC50 = 11900 nM
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CP0037112
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2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidin-2-yl}sulfanyl)octanoic acid
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C20H26ClN3O2S
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1
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| 1 |
IC50 = 12000 nM
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CP0288255
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3-isopropyl-1-(4-methoxybenzyl)-1-(3-(phenylethynyl)benzyl)urea
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C27H28N2O2
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1
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| 1 |
IC50 = 14800 nM
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CP0508345
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1-benzyl-3-isopropyl-1-(3-(phenylethynyl)benzyl)guanidine
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C26H27N3
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1
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| 1 |
IC50 = 17000 nM
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CP0045344
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4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol-3-ylmethyl)-3-methoxy-N-o-tolylsulfonylbenzamide
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C31H33N3O6S
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1
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| 1 |
IC50 = 18100 nM
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CP0292244
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tert-butyl N-[N-benzyl-N-[[3-(2-phenylethynyl)phenyl]methyl]-N'-propan-2-ylcarbamimidoyl]carbamate
Show/Hide
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C31H35N3O2
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1
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| 1 |
IC50 = 27000 nM
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CP0266725
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2-(4-(3,5-bis(2,2,2-trifluoroethoxy)phenylamino)-6-chloropyrimidin-2-ylthio)octanoic acid
Show/Hide
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C22H24ClF6N3O4S
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1
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| 1 |
IC50 >= 30000 nM
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CP0484691
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5-(4-bromophenyl)-3-(2-chloro-6-fluorophenyl)-1,2,4-oxadiazole
Show/Hide
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C14H7BrClFN2O
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1
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| 1 |
IC50 > 30000 nM
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CP0855335
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2-(trifluoromethyl)-4-(4-((4-(trifluoromethyl)phenoxy)methyl)-1H-1,2,3-triazol-1-yl)benzonitrile
Show/Hide
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C18H10F6N4O
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1
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| 1 |
IC50 > 30000 nM
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CP0855799
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4-((4-nitro-2-(trifluoromethyl)phenoxy)methyl)-1-(3-(trifluoromethyl)phenyl)-1H-1,2,3-triazole
Show/Hide
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C17H10F6N4O3
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1
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| 1 |
IC50 > 30000 nM
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CP0855800
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4-(4-((4-nitro-2-(trifluoromethyl)phenoxy)methyl)-1H-1,2,3-triazol-1-yl)-2-(trifluoromethyl)benzonitrile
Show/Hide
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C18H9F6N5O3
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1
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| 1 |
IC50 > 30000 nM
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CP0896937
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2-(trifluoromethyl)-4-(4-((3-(trifluoromethyl)phenoxy)methyl)-1H-1,2,3-triazol-1-yl)benzonitrile
Show/Hide
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C18H10F6N4O
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1
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| 1 |
IC50 > 30000 nM
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CP0430971
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1,1'-(2-(2-chloro-6-fluorophenyl)-1H-phenanthro[9,10-d]imidazole-6,9-diyl)diethanone
Show/Hide
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C25H16ClFN2O2
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1
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| 1 |
IC50 > 50000 nM
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CP0353531
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1-[[3-(benzenesulfonamido)phenyl]methyl]-1-benzyl-3-propan-2-ylurea
Show/Hide
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C24H27N3O3S
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1
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| 1 |
IC50 > 50000 nM
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CP0446106
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2-(2-chloro-6-fluoroanilino)-N-[3-fluoro-5-(trifluoromethyl)phenyl]-6,7-dihydroxy-1-methylbenzimidazole-5-carboxamide
Show/Hide
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C22H14ClF5N4O3
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1
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| 1 |
IC50 > 8000 nM
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