General Information of the Compound
Compound ID
CP0379998
Compound Name
2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanylacetic acid
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Structure
Formula
C15H10Cl2N4O2S2
Molecular Weight
413.311
Canonical SMILES
OC(=O)CSc1nc(Cl)cc(Nc2nc(cs2)-c2ccc(Cl)cc2)n1
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InChI
InChI=1S/C15H10Cl2N4O2S2/c16-9-3-1-8(2-4-9)10-6-24-14(18-10)20-12-5-11(17)19-15(21-12)25-7-13(22)23/h1-6H,7H2,(H,22,23)(H,18,19,20,21)
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InChIKey
ICVVXTDMPDJJEV-UHFFFAOYSA-N
Physicochemical Property
logP
4.8272
Rotatable Bonds
6
Heavy Atom Count
25
Polar Areas
88
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
25

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 72734878
ChEMBL ID
CHEMBL3091496
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01242, Polyunsaturated fatty acid 5-lipoxygenase
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000831 PMNL Homo sapiens (Human)  1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
Protein ID: PT02025, Prostaglandin E synthase
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549 Homo sapiens (Human)  1
1
IC50 = 2300 nM
   TI
   LI
   LO
   TS