Compound ID |
Compound Name |
Compound Formula |
CP0392201
|
3-(2,4-dibromophenyl)-N-heptan-4-yl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C18H22Br2N6
|
1
|
1 |
Ki = 0.8 nM
|
|
|
CP0283841
|
Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-amine
Show/Hide
|
C24H34N4
|
1
|
1 |
Ki = 0.84 nM
|
|
|
CP0412470
|
9-(2-bromo-4-propan-2-ylphenyl)-N-butyl-N-ethyl-2,8-dimethylpurin-6-amine
Show/Hide
|
C22H30BrN5
|
1
|
1 |
Ki = 0.9 nM
|
|
|
CP0406407
|
9-(2-bromo-4-propan-2-ylphenyl)-N-butyl-N-ethyl-2-methyl-8-(trifluoromethyl)purin-6-amine
Show/Hide
|
C22H27BrF3N5
|
1
|
1 |
Ki = 1.4 nM
|
|
|
CP0497796
|
3-(2-Bromo-4-isopropyl-phenyl)-7-(1-ethyl-pentyloxy)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidine
Show/Hide
|
C21H28BrN5O
|
1
|
1 |
Ki = 1.5 nM
|
|
|
CP0255382
|
Butyl-[2,5-dimethyl-7-(2,4,6-trimethyl-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-ethyl-amine
Show/Hide
|
C23H32N4
|
2
|
1 |
Ki = 1.61 nM
|
|
|
2 |
Ki = 2.7 nM
|
|
|
CP0495062
|
3-(2-Bromo-4-isopropyl-phenyl)-7-(1-ethyl-propoxy)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidine
Show/Hide
|
C19H24BrN5O
|
1
|
1 |
Ki = 1.9 nM
|
|
|
CP0505801
|
3-(2-Bromo-4-isopropyl-phenyl)-7-(1-methoxymethyl-propoxy)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidine
Show/Hide
|
C19H24BrN5O2
|
1
|
1 |
Ki = 1.9 nM
|
|
|
CP0523276
|
Butyl-ethyl-[3-(4-isopropyl-2-methylsulfanyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-b]pyridin-7-yl]-amine
Show/Hide
|
C22H31N5S
|
1
|
1 |
Ki = 2.2 nM
|
|
|
CP0505264
|
(2-Bromo-4-isopropyl-phenyl)-ethyl-[4-methyl-6-(2-nitro-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
|
C22H23BrN4O2
|
1
|
1 |
Ki = 2.4 nM
|
|
|
CP0393666
|
(2-Bromo-4-methylsulfanyl-phenyl)-ethyl-[4-methyl-6-(2-trifluoromethyl-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
|
C21H19BrF3N3S
|
1
|
1 |
Ki = 2.5 nM
|
|
|
CP0514436
|
3-(2-bromo-4-propan-2-ylphenyl)-N-hexan-3-yl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C20H27BrN6
|
1
|
1 |
Ki = 2.8 nM
|
|
|
CP0534479
|
9-(2-Bromo-4-isopropyl-phenyl)-6-(1-ethyl-pentyloxy)-2-methyl-9H-purine
Show/Hide
|
C22H29BrN4O
|
1
|
1 |
Ki = 2.9 nM
|
|
|
CP0514429
|
3-(2-bromo-4,6-dimethoxyphenyl)-N-butyl-N-ethyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C19H25BrN6O2
|
1
|
1 |
Ki = 3 nM
|
|
|
CP0498255
|
(2-Bromo-4-isopropyl-phenyl)-ethyl-[4-methyl-6-(2-trifluoromethyl-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
|
C23H23BrF3N3
|
1
|
1 |
Ki = 3.1 nM
|
|
|
CP0464912
|
3-(2-bromo-4-propan-2-ylphenyl)-N-heptan-3-yl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C21H29BrN6
|
1
|
1 |
Ki = 3.1 nM
|
|
|
CP0449381
|
9-(2-bromo-4,6-dimethoxyphenyl)-N-butyl-N-ethyl-2-methylpurin-6-amine
Show/Hide
|
C20H26BrN5O2
|
1
|
1 |
Ki = 3.5 nM
|
|
|
CP0464919
|
Butyl-[9-(2-chloro-4,6-dimethoxy-phenyl)-2,8-dimethyl-9H-purin-6-yl]-ethyl-amine
Show/Hide
|
C21H28ClN5O2
|
1
|
1 |
Ki = 3.5 nM
|
|
|
CP0498303
|
9-(2-Bromo-4-isopropyl-phenyl)-6-(1-ethyl-propoxy)-2-methyl-9H-purine
Show/Hide
|
C20H25BrN4O
|
1
|
1 |
Ki = 3.5 nM
|
|
|
CP0404383
|
9-(2-bromo-4-propan-2-ylphenyl)-N-heptan-4-yl-2-methylpurin-6-amine
Show/Hide
|
C22H30BrN5
|
1
|
1 |
Ki = 3.6 nM
|
|
|
CP0460914
|
3-(2-bromo-4-propan-2-ylphenyl)-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C20H27BrN6O2
|
1
|
1 |
Ki = 3.7 nM
|
|
|
CP0521967
|
3-(2-bromo-4-propan-2-ylphenyl)-N-butyl-N-ethyl-2,5-dimethylimidazo[4,5-b]pyridin-7-amine
Show/Hide
|
C23H31BrN4
|
1
|
1 |
Ki = 3.9 nM
|
|
|
CP0518074
|
N-heptan-4-yl-5-methyl-3-(2,4,6-trimethylphenyl)triazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C21H30N6
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0417281
|
Allyl-[3-(2-bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-(2-methoxy-ethyl)-amine
Show/Hide
|
C20H25BrN6O
|
1
|
1 |
Ki = 4.3 nM
|
|
|
CP0456877
|
9-(2-bromo-4-propan-2-ylphenyl)-N-butyl-N-ethyl-2-methylpurin-6-amine
Show/Hide
|
C21H28BrN5
|
1
|
1 |
Ki = 4.3 nM
|
|
|
CP0451965
|
9-(2-bromo-4-propan-2-ylphenyl)-N-hexan-3-yl-2-methylpurin-6-amine
Show/Hide
|
C21H28BrN5
|
1
|
1 |
Ki = 4.4 nM
|
|
|
CP0504121
|
Butyl-[3-(2-chloro-4,6-dimethoxy-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-ethyl-amine
Show/Hide
|
C19H25ClN6O2
|
1
|
1 |
Ki = 4.4 nM
|
|
|
CP0418874
|
3-(2-bromo-4-propan-2-ylphenyl)-5-methyl-N-nonan-5-yltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C23H33BrN6
|
1
|
1 |
Ki = 4.5 nM
|
|
|
CP0391424
|
1-(3-Bromo-4-{ethyl-[4-methyl-6-(2-trifluoromethyl-phenyl)-pyrimidin-2-yl]-amino}-phenyl)-ethanone
Show/Hide
|
C22H19BrF3N3O
|
1
|
1 |
Ki = 4.6 nM
|
|
|
CP0446162
|
3-(2-bromo-4-propan-2-ylphenyl)-N-(cyclopropylmethyl)-N-(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C21H27BrN6O
|
1
|
1 |
Ki = 4.6 nM
|
|
|
CP0375832
|
3-(2-bromo-4-propan-2-ylphenyl)-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-b]pyridin-7-amine
Show/Hide
|
C21H28BrN5O2
|
1
|
1 |
Ki = 4.7 nM
|
|
|
CP0453252
|
N,N-bis(2-methoxyethyl)-5-methyl-3-(2-methylsulfanyl-4-propan-2-ylphenyl)triazolo[4,5-b]pyridin-7-amine
Show/Hide
|
C22H31N5O2S
|
1
|
1 |
Ki = 4.7 nM
|
|
|
CP0540604
|
Benzyl-[3-(2-bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-(2-methoxy-ethyl)-amine
Show/Hide
|
C24H27BrN6O
|
1
|
1 |
Ki = 5 nM
|
|
|
CP0436530
|
9-(2-bromo-4-propan-2-ylphenyl)-N-heptan-3-yl-2-methylpurin-6-amine
Show/Hide
|
C22H30BrN5
|
1
|
1 |
Ki = 5.1 nM
|
|
|
CP0520511
|
Butyl-[9-(2-chloro-4,6-dimethoxy-phenyl)-2-methyl-9H-purin-6-yl]-ethyl-amine
Show/Hide
|
C20H26ClN5O2
|
1
|
1 |
Ki = 5.2 nM
|
|
|
CP0523945
|
3-(2-bromo-4-propan-2-ylphenyl)-5-methyl-N-pentan-3-yltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C19H25BrN6
|
1
|
1 |
Ki = 5.2 nM
|
|
|
CP0521966
|
(1-Ethyl-propyl)-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
Show/Hide
|
C19H26N6
|
1
|
1 |
Ki = 5.7 nM
|
|
|
CP0534991
|
(2,4-Dibromo-phenyl)-ethyl-[4-methyl-6-(2-trifluoromethyl-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
|
C20H16Br2F3N3
|
1
|
1 |
Ki = 5.8 nM
|
|
|
CP0535736
|
2-{2-[(2-Bromo-4-isopropyl-phenyl)-ethyl-amino]-6-methyl-pyrimidin-4-yl}-benzonitrile
Show/Hide
|
C23H23BrN4
|
1
|
1 |
Ki = 5.8 nM
|
|
|
CP0501273
|
9-(2-bromo-4-propan-2-ylphenyl)-N,N-bis(2-methoxyethyl)-2-methylpurin-6-amine
Show/Hide
|
C21H28BrN5O2
|
1
|
1 |
Ki = 5.9 nM
|
|
|
CP0496563
|
9-(2-bromo-4-propan-2-ylphenyl)-N,N-dibutyl-2-methylpurin-6-amine
Show/Hide
|
C23H32BrN5
|
1
|
1 |
Ki = 6.1 nM
|
|
|
CP0523972
|
9-(2-bromo-4-propan-2-ylphenyl)-N,N-bis(2-methoxyethyl)-2,8-dimethylpurin-6-amine
Show/Hide
|
C22H30BrN5O2
|
1
|
1 |
Ki = 6.7 nM
|
|
|
CP0425314
|
3-(2-Bromo-4-isopropyl-phenyl)-7-(2-methoxy-1-methoxymethyl-ethoxy)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidine
Show/Hide
|
C19H24BrN5O3
|
1
|
1 |
Ki = 7.1 nM
|
|
|
CP0447215
|
Bis-(2-methoxy-ethyl)-[2,5,6-trimethyl-7-(2,4,6-trimethyl-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-amine
Show/Hide
|
C24H34N4O2
|
1
|
1 |
Ki = 7.1 nM
|
|
|
CP0475685
|
(1-Methyl-butyl)-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
Show/Hide
|
C19H26N6
|
1
|
1 |
Ki = 7.1 nM
|
|
|
CP0548635
|
3-(2,4-dibromophenyl)-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C17H20Br2N6O2
|
1
|
1 |
Ki = 7.4 nM
|
|
|
CP0534472
|
3-(2-bromo-4-propan-2-ylphenyl)-N-butyl-N-ethyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C20H27BrN6
|
1
|
1 |
Ki = 7.5 nM
|
|
|
CP0523969
|
(1-Ethyl-pentyl)-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
Show/Hide
|
C21H30N6
|
1
|
1 |
Ki = 7.6 nM
|
|
|
CP0493809
|
(2-Bromo-4-isopropyl-phenyl)-ethyl-(4-methyl-6-naphthalen-1-yl-pyrimidin-2-yl)-amine
Show/Hide
|
C26H26BrN3
|
1
|
1 |
Ki = 7.8 nM
|
|
|
CP0402768
|
9-(2-bromo-4-propan-2-ylphenyl)-N-(1-methoxypentan-3-yl)-2-methylpurin-6-amine
Show/Hide
|
C21H28BrN5O
|
1
|
1 |
Ki = 8 nM
|
|
|
CP0431695
|
(4-Biphenyl-2-yl-6-methyl-pyrimidin-2-yl)-(2-bromo-4-isopropyl-phenyl)-ethyl-amine
Show/Hide
|
C28H28BrN3
|
1
|
1 |
Ki = 8.4 nM
|
|
|
CP0506460
|
(2-Bromo-4,6-dimethoxy-phenyl)-ethyl-[4-methyl-6-(2-trifluoromethyl-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
|
C22H21BrF3N3O2
|
1
|
1 |
Ki = 8.6 nM
|
|
|
CP0275845
|
2-N-(2-bromo-4-propan-2-ylphenyl)-2-N-ethyl-6-methyl-4-N,4-N-dipropylpyrimidine-2,4-diamine
Show/Hide
|
C22H33BrN4
|
1
|
1 |
Ki = 9 nM
|
|
|
CP0506558
|
(2-Bromo-4,6-dimethoxy-phenyl)-[4-(2-chloro-phenyl)-6-methyl-pyrimidin-2-yl]-ethyl-amine
Show/Hide
|
C21H21BrClN3O2
|
1
|
1 |
Ki = 9.1 nM
|
|
|
CP0520450
|
9-(2-bromo-4-propan-2-ylphenyl)-N-ethyl-N-(2-methoxyethyl)-2-methylpurin-6-amine
Show/Hide
|
C20H26BrN5O
|
1
|
1 |
Ki = 9.2 nM
|
|
|
CP0535749
|
2-Bromo-N*1*-ethyl-6-methoxy-N*4*,N*4*-dimethyl-N*1*-[4-methyl-6-(2-trifluoromethyl-phenyl)-pyrimidin-2-yl]-benzene-1,4-diamine
Show/Hide
|
C23H24BrF3N4O
|
1
|
1 |
Ki = 9.4 nM
|
|
|
CP0534511
|
9-(2-Bromo-4-isopropyl-phenyl)-6-(1-methoxymethyl-propoxy)-2-methyl-9H-purine
Show/Hide
|
C20H25BrN4O2
|
1
|
1 |
Ki = 9.7 nM
|
|
|
CP0530250
|
3-(2-bromo-4-propan-2-ylphenyl)-N,N-bis(2-methoxyethyl)-2,5-dimethylimidazo[4,5-b]pyridin-7-amine
Show/Hide
|
C23H31BrN4O2
|
1
|
1 |
Ki = 9.8 nM
|
|
|
CP0439194
|
(2-Bromo-4-isopropyl-phenyl)-[4-(2,6-dichloro-phenyl)-6-methyl-pyrimidin-2-yl]-ethyl-amine
Show/Hide
|
C22H22BrCl2N3
|
1
|
1 |
Ki = 10.1 nM
|
|
|
CP0464458
|
3-(2-bromo-4-propan-2-ylphenyl)-N-(1,3-dimethoxypropan-2-yl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C19H25BrN6O2
|
1
|
1 |
Ki = 10.3 nM
|
|
|
CP0464248
|
3-(2-bromo-4-propan-2-ylphenyl)-N-ethyl-N-(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C19H25BrN6O
|
1
|
1 |
Ki = 10.5 nM
|
|
|
CP0538772
|
3-[2-bromo-4-(dimethylamino)phenyl]-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C19H26BrN7O2
|
1
|
1 |
Ki = 10.5 nM
|
|
|
CP0464434
|
3-(2-bromo-4-methylsulfanylphenyl)-N-butyl-N-ethyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C18H23BrN6S
|
1
|
1 |
Ki = 10.6 nM
|
|
|
CP0384052
|
(2-Bromo-4-isopropyl-phenyl)-ethyl-[4-methyl-6-(2,4,6-trimethyl-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
|
C25H30BrN3
|
1
|
1 |
Ki = 11.2 nM
|
|
|
CP0480633
|
3-(2-bromo-4-propan-2-ylphenyl)-N-(1-methoxybutan-2-yl)-N,5-dimethyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C20H27BrN6O
|
1
|
1 |
Ki = 11.2 nM
|
|
|
CP0465378
|
9-(2-bromo-4-propan-2-ylphenyl)-N,N-diethyl-2-methylpurin-6-amine
Show/Hide
|
C19H24BrN5
|
1
|
1 |
Ki = 12.4 nM
|
|
|
CP0491796
|
(2-Bromo-4-isopropyl-phenyl)-[4-(2-chloro-phenyl)-6-methyl-pyrimidin-2-yl]-ethyl-amine
Show/Hide
|
C22H23BrClN3
|
1
|
1 |
Ki = 13.5 nM
|
|
|
CP0526916
|
(2-Bromo-4,6-dimethoxy-phenyl)-ethyl-(4-methyl-6-phenyl-pyrimidin-2-yl)-amine
Show/Hide
|
C21H22BrN3O2
|
1
|
1 |
Ki = 13.9 nM
|
|
|
CP0451964
|
N,N-bis(2-methoxyethyl)-5-methyl-3-(2-methylsulfanyl-4-propan-2-ylphenyl)triazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C21H30N6O2S
|
1
|
1 |
Ki = 15.3 nM
|
|
|
CP0497797
|
Butyl-[3-(4-dimethylamino-2-trifluoromethyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-ethyl-amine
Show/Hide
|
C20H26F3N7
|
1
|
1 |
Ki = 15.4 nM
|
|
|
CP0391398
|
(2-Bromo-4-isopropyl-phenyl)-ethyl-[4-methyl-6-(3-trifluoromethyl-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
|
C23H23BrF3N3
|
1
|
1 |
Ki = 17.4 nM
|
|
|
CP0504147
|
(2-Bromo-4-isopropyl-phenyl)-ethyl-(4-methyl-6-o-tolyl-pyrimidin-2-yl)-amine
Show/Hide
|
C23H26BrN3
|
1
|
1 |
Ki = 18.4 nM
|
|
|
CP0507622
|
2-[3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino]-butyric acid methyl ester
Show/Hide
|
C19H23BrN6O2
|
1
|
1 |
Ki = 19.4 nM
|
|
|
CP0436358
|
Butyl-[3-(2,4-dibromo-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-ethyl-amine
Show/Hide
|
C17H20Br2N6
|
1
|
1 |
Ki = 20.4 nM
|
|
|
CP0496753
|
(2-Bromo-4-methanesulfonyl-phenyl)-ethyl-[4-methyl-6-(2-trifluoromethyl-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
|
C21H19BrF3N3O2S
|
1
|
1 |
Ki = 20.6 nM
|
|
|
CP0375831
|
Bis-(2-methoxy-ethyl)-[2-methyl-9-(2,4,6-trimethyl-phenyl)-9H-purin-6-yl]-amine
Show/Hide
|
C21H29N5O2
|
1
|
1 |
Ki = 20.7 nM
|
|
|
CP0475653
|
N-ethyl-N-(2-methoxyethyl)-5-methyl-3-(2,4,6-trimethylphenyl)triazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C19H26N6O
|
1
|
1 |
Ki = 20.7 nM
|
|
|
CP0458723
|
3-(2-chloro-4,6-dimethoxyphenyl)-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
|
C19H25ClN6O4
|
1
|
1 |
Ki = 21 nM
|
|
|
CP0452019
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3-(2-bromo-4-propan-2-ylphenyl)-N-(1,3-dimethoxypropan-2-yl)-N,5-dimethyltriazolo[4,5-d]pyrimidin-7-amine
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C20H27BrN6O2
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1
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1 |
Ki = 21.3 nM
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CP0503290
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Butyl-[8-butyl-9-(2-chloro-4,6-dimethoxy-phenyl)-2-methyl-9H-purin-6-yl]-ethyl-amine
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C24H34ClN5O2
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1
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1 |
Ki = 22 nM
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CP0427044
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(2-Bromo-4-isopropyl-phenyl)-ethyl-[4-(2-fluoro-phenyl)-6-methyl-pyrimidin-2-yl]-amine
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C22H23BrFN3
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1
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1 |
Ki = 23.4 nM
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CP0460890
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3-[4-(dimethylamino)-2-(trifluoromethyl)phenyl]-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C20H26F3N7O2
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1
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1 |
Ki = 23.5 nM
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CP0412485
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9-(2-chloro-4,6-dimethoxyphenyl)-N-(2-methoxyethyl)-N-(3-methoxypropyl)-2-methylpurin-6-amine
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C21H28ClN5O4
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1
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1 |
Ki = 23.8 nM
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CP0505262
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(2-Bromo-4-isopropyl-phenyl)-[4-(2-bromo-phenyl)-6-methyl-pyrimidin-2-yl]-ethyl-amine
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C22H23Br2N3
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1
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1 |
Ki = 24 nM
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CP0412475
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Bis-(2-methoxy-ethyl)-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
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C20H28N6O2
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1
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1 |
Ki = 24.1 nM
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CP0497931
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(2-Bromo-4-isopropyl-6-methyl-phenyl)-ethyl-[4-methyl-6-(2,4,6-trimethyl-pyridin-3-yl)-pyrimidin-2-yl]-amine
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C25H31BrN4
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1
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1 |
Ki = 24.9 nM
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CP0449838
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Butyl-ethyl-[2-methyl-9-(2,4,6-trimethyl-phenyl)-9H-purin-6-yl]-amine
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C21H29N5
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1
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1 |
Ki = 25 nM
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CP0404382
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3-(2-bromo-4-propan-2-ylphenyl)-N,N-diethyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C18H23BrN6
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1
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1 |
Ki = 25.3 nM
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CP0418548
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2-[3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino]-butan-1-ol
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C18H23BrN6O
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1
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1 |
Ki = 25.3 nM
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CP0465280
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2-[2,5,6-Trimethyl-7-(2,4,6-trimethyl-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino]-butan-1-ol
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C22H30N4O
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1
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1 |
Ki = 27.3 nM
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CP0500974
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Butyl-ethyl-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
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C20H28N6
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1
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1 |
Ki = 27.5 nM
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CP0507650
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(1-Methoxymethyl-2-phenyl-ethyl)-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
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C24H28N6O
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1
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1 |
Ki = 27.7 nM
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CP0404223
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3-(2-bromo-4,6-dimethoxyphenyl)-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C19H25BrN6O4
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1
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1 |
Ki = 28.3 nM
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CP0538236
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Butyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-amine
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C22H30N4
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1
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1 |
Ki = 29 nM
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CP0518081
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9-(2-bromo-4,6-dimethoxyphenyl)-N,N-bis(2-methoxyethyl)-2-methylpurin-6-amine
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C20H26BrN5O4
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1
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1 |
Ki = 31.3 nM
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CP0521965
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3-(2-bromo-4-propan-2-ylphenyl)-N,N-dibutyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C22H31BrN6
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1
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1 |
Ki = 32.5 nM
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CP0401225
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3-[2-bromo-4-(trifluoromethoxy)phenyl]-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C18H20BrF3N6O3
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1
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1 |
Ki = 33.2 nM
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CP0487365
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1-{3-Bromo-4-[7-(butyl-ethyl-amino)-5-methyl-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]-phenyl}-ethanone
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C19H23BrN6O
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1
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1 |
Ki = 33.7 nM
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CP0418545
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3-(2-bromo-4-propan-2-ylphenyl)-N-(1-methoxy-3-phenylpropan-2-yl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C24H27BrN6O
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1
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1 |
Ki = 36.7 nM
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CP0406378
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2-N-[3-(2-bromo-4-propan-2-ylphenyl)-5-methyltriazolo[4,5-d]pyrimidin-7-yl]-1-N,1-N-dimethylpentane-1,2-diamine
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C21H30BrN7
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1
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1 |
Ki = 38.7 nM
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CP0488141
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3-(2-Bromo-4-isopropyl-phenyl)-7-(2-ethoxy-1-ethoxymethyl-ethoxy)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidine
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C21H28BrN5O3
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1
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1 |
Ki = 39.7 nM
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CP0496609
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3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-7-piperidin-1-yl-3H-[1,2,3]triazolo[4,5-d]pyrimidine
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C19H23BrN6
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1
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1 |
Ki = 46 nM
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CP0545049
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3-[2-bromo-6-(dimethylamino)-4-methoxyphenyl]-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C20H28BrN7O3
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1
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1 |
Ki = 48.2 nM
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CP0485169
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3-(2-bromo-4-propan-2-ylphenyl)-N-(2-methoxyethyl)-5-methyl-N-(pyridin-3-ylmethyl)triazolo[4,5-d]pyrimidin-7-amine
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C23H26BrN7O
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1
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1 |
Ki = 48.5 nM
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CP0449366
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(2-Bromo-4,6-dimethoxy-phenyl)-ethyl-[4-(2-methoxy-phenyl)-6-methyl-pyrimidin-2-yl]-amine
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C22H24BrN3O3
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1
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1 |
Ki = 54.8 nM
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CP0404463
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(1-Methoxymethyl-propyl)-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
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C19H26N6O
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1
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1 |
Ki = 59.4 nM
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CP0404163
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2-[[3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-(2-methoxy-ethyl)-amino]-ethanol
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C19H25BrN6O2
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1
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1 |
Ki = 64 nM
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CP0392207
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Butyl-ethyl-[5-methyl-3-(2,4,6-trimethyl-pyridin-3-yl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
Show/Hide
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C19H27N7
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1
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1 |
Ki = 65 nM
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CP0520230
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3-(2-bromo-4-propan-2-ylphenyl)-N-(2-methoxyethyl)-N-(3-methoxypropyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C21H29BrN6O2
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1
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1 |
Ki = 66.9 nM
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CP0466832
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3-(2-bromo-4-propan-2-ylphenyl)-N-butyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C18H23BrN6
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1
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1 |
Ki = 69.6 nM
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CP0457312
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(2-Bromo-4-isopropyl-phenyl)-[4-(2-dimethylamino-phenyl)-6-methyl-pyrimidin-2-yl]-ethyl-amine
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C24H29BrN4
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1
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1 |
Ki = 78.2 nM
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CP0504667
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Butyl-ethyl-[3-(4-isopropyl-2-methanesulfonyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-b]pyridin-7-yl]-amine
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C22H31N5O2S
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1
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1 |
Ki = 83 nM
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CP0467100
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(4-Biphenyl-3-yl-6-methyl-pyrimidin-2-yl)-(2-bromo-4-isopropyl-phenyl)-ethyl-amine
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C28H28BrN3
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1
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1 |
Ki = 84.6 nM
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CP0449837
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3-(2-bromo-4-methylsulfonylphenyl)-N-butyl-N-ethyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C18H23BrN6O2S
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1
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1 |
Ki = 100 nM
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CP0399751
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(2-Bromo-4-isopropyl-phenyl)-ethyl-(4-methyl-6-phenyl-pyrimidin-2-yl)-amine
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C22H24BrN3
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1
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1 |
Ki = 109 nM
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CP0428654
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3-(2-bromo-4-propan-2-ylphenyl)-N-cyclopentyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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C19H23BrN6
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1
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1 |
Ki = 120 nM
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CP0525456
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3-(2-bromo-4-propan-2-ylphenyl)-N-(1,3-dimethoxypropan-2-yl)-N-ethyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
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C21H29BrN6O2
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1
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1 |
Ki = 123 nM
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CP0441415
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Butyl-[9-(2-chloro-4,6-dimethoxy-phenyl)-2-methyl-8-phenyl-9H-purin-6-yl]-ethyl-amine
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C26H30ClN5O2
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1
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1 |
Ki = 133 nM
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CP0503509
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3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-7-pyrrolidin-1-yl-3H-[1,2,3]triazolo[4,5-d]pyrimidine
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C18H21BrN6
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1
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1 |
Ki = 194 nM
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CP0485170
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3-(2-bromo-4-propan-2-ylphenyl)-N-(1-methoxy-2-methylpropan-2-yl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
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C19H25BrN6O
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1
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1 |
Ki = 195 nM
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CP0397986
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2,5,6-Trimethyl-4-morpholin-4-yl-7-(2,4,6-trimethyl-phenyl)-7H-pyrrolo[2,3-d]pyrimidine
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C22H28N4O
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1
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1 |
Ki = 201 nM
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CP0507722
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3-(2-bromo-4-propan-2-ylphenyl)-N,N-bis(2-methoxyethyl)triazolo[4,5-d]pyrimidin-7-amine
Show/Hide
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C19H25BrN6O2
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1
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1 |
Ki = 203 nM
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CP0510026
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9-(2-bromo-4-propan-2-ylphenyl)-N-(2-methoxyethyl)-2-methylpurin-6-amine
Show/Hide
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C18H22BrN5O
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1
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1 |
Ki = 210 nM
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CP0415377
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(2-Bromo-4,6-dimethoxy-phenyl)-ethyl-(4-methyl-6-pyridin-2-yl-pyrimidin-2-yl)-amine
Show/Hide
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C20H21BrN4O2
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1
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1 |
Ki = 222 nM
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CP0493482
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(2-Bromo-4,6-dimethoxy-phenyl)-ethyl-(4-methyl-6-pyridin-3-yl-pyrimidin-2-yl)-amine
Show/Hide
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C20H21BrN4O2
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1
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1 |
Ki = 229 nM
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CP0506121
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2-[3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino]-pentanoic acid dimethylamide
Show/Hide
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C21H28BrN7O
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1
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1 |
Ki = 235 nM
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CP0425313
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3-(2-bromo-4-propan-2-ylphenyl)-N-(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
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C17H21BrN6O
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1
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1 |
Ki = 242 nM
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CP0403837
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3-(2-bromo-4-propan-2-ylphenyl)-N-butyl-N-ethyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
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C19H25BrN6
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1
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1 |
Ki = 287 nM
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CP0490336
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3-(2-bromo-4-propan-2-ylphenyl)-N-(3-methoxypropyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
Show/Hide
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C18H23BrN6O
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1
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1 |
Ki = 291 nM
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CP0380797
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(2-Bromo-4-isopropyl-phenyl)-ethyl-[4-methyl-6-(2-methylamino-phenyl)-pyrimidin-2-yl]-amine
Show/Hide
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C23H27BrN4
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1
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1 |
Ki = 369 nM
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CP0507692
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Bis-(2-methoxy-ethyl)-[5-methyl-3-(2,4,6-trimethyl-pyridin-3-yl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
Show/Hide
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C19H27N7O2
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1
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1 |
Ki = 416 nM
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CP0496102
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N,N-bis(2-methoxyethyl)-5-methyl-3-(2-methylsulfonyl-4-propan-2-ylphenyl)triazolo[4,5-b]pyridin-7-amine
Show/Hide
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C22H31N5O4S
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1
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1 |
Ki = 476 nM
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CP0448217
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(2-Bromo-4-isopropyl-phenyl)-ethyl-{4-methyl-6-[2-(1H-tetrazol-5-yl)-phenyl]-pyrimidin-2-yl}-amine
Show/Hide
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C23H24BrN7
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1
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1 |
Ki = 662 nM
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CP0397964
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N,N-bis(2-methoxyethyl)-5-methyl-3-(2-methylsulfonyl-4-propan-2-ylphenyl)triazolo[4,5-d]pyrimidin-7-amine
Show/Hide
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C21H30N6O4S
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1
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1 |
Ki = 1026 nM
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CP0520231
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(2-Methoxy-ethyl)-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
Show/Hide
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C17H22N6O
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1
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1 |
Ki = 1204 nM
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CP0440125
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4-(2-aminophenyl)-N-(2-bromo-4-propan-2-ylphenyl)-N-ethyl-6-methylpyrimidin-2-amine
Show/Hide
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C22H25BrN4
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1
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1 |
Ki = 2359 nM
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CP0453061
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N'-[9-(2-bromo-4-propan-2-ylphenyl)-2-methylpurin-6-yl]-N'-ethyl-N,N-dimethylethane-1,2-diamine
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C21H29BrN6
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1
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1 |
Ki = 2665 nM
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CP0518326
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2-[[3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-(2-hydroxy-ethyl)-amino]-ethanol
Show/Hide
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C18H23BrN6O2
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1
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1 |
Ki = 3460 nM
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CP0502426
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2-{2-[(2-Bromo-4-isopropyl-phenyl)-ethyl-amino]-6-methyl-pyrimidin-4-yl}-benzoic acid
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C23H24BrN3O2
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1
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1 |
Ki = 3536 nM
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CP0402107
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N,N-bis(2-methoxyethyl)-5-methyl-3-(4-propan-2-ylphenyl)triazolo[4,5-d]pyrimidin-7-amine
Show/Hide
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C20H28N6O2
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1
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1 |
Ki = 3918 nM
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