Brief Information of the Compound and Protein
Compound Name
2-N-(2-bromo-4-propan-2-ylphenyl)-2-N-ethyl-6-methyl-4-N,4-N-dipropylpyrimidine-2,4-diamine
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PubChem ID
CID: 10717634
SID: 15752811
Canonical SMILES
CCCN(CCC)c1cc(C)nc(n1)N(CC)c1ccc(cc1Br)C(C)C
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Compound Formula C22H33BrN4
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki = 9 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 9 nM