Brief Information of the Compound and Protein
Compound Name
2,5,6-Trimethyl-4-morpholin-4-yl-7-(2,4,6-trimethyl-phenyl)-7H-pyrrolo[2,3-d]pyrimidine
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PubChem ID
CID: 10761294
SID: 15798752
Canonical SMILES
Cc1c(C)c2c(nc(C)nc2n1-c1c(C)cc(C)cc1C)N1CCOCC1
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Compound Formula C22H28N4O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki = 201 nM
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