Brief Information of the Compound and Protein
Compound Name
3-[2-bromo-4-(trifluoromethoxy)phenyl]-N,N-bis(2-methoxyethyl)-5-methyltriazolo[4,5-d]pyrimidin-7-amine
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PubChem ID
CID: 10791657
SID: 15830502
Canonical SMILES
COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(OC(F)(F)F)cc1Br
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Compound Formula C18H20BrF3N6O3
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki = 33.2 nM
   TI
   LI
   LO
   TS