Brief Information of the Compound and Protein
Compound Name
(2-Bromo-4-isopropyl-6-methyl-phenyl)-ethyl-[4-methyl-6-(2,4,6-trimethyl-pyridin-3-yl)-pyrimidin-2-yl]-amine
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PubChem ID
CID: 44266439
Canonical SMILES
CCN(c1nc(C)cc(n1)-c1c(C)cc(C)nc1C)c1c(C)cc(cc1Br)C(C)C
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Compound Formula C25H31BrN4
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki = 24.9 nM
   TI
   LI
   LO
   TS