Brief Information of the Compound and Protein
Compound Name
(1-Methoxymethyl-2-phenyl-ethyl)-[5-methyl-3-(2,4,6-trimethyl-phenyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-amine
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PubChem ID
CID: 10764399
SID: 15801949
Canonical SMILES
COCC(Cc1ccccc1)Nc1nc(C)nc2n(nnc12)-c1c(C)cc(C)cc1C
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Compound Formula C24H28N6O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki = 27.7 nM
   TI
   LI
   LO
   TS