Brief Information of the Compound and Protein
Compound Name
3-(2-Bromo-4-isopropyl-phenyl)-7-(2-methoxy-1-methoxymethyl-ethoxy)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidine
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PubChem ID
CID: 10503714
SID: 15528717
Canonical SMILES
COCC(COC)Oc1nc(C)nc2n(nnc12)-c1ccc(cc1Br)C(C)C
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Compound Formula C19H24BrN5O3
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki = 7.1 nM
   TI
   LI
   LO
   TS