Brief Information of the Compound and Protein
Compound Name
N,N-bis(2-methoxyethyl)-5-methyl-3-(2-methylsulfanyl-4-propan-2-ylphenyl)triazolo[4,5-d]pyrimidin-7-amine
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PubChem ID
CID: 10717531
SID: 15752713
Canonical SMILES
COCCN(CCOC)c1nc(C)nc2n(nnc12)-c1ccc(cc1SC)C(C)C
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Compound Formula C21H30N6O2S
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki = 15.3 nM
   TI
   LI
   LO
   TS