Brief Information of the Compound and Protein
Compound Name
Bis-(2-methoxy-ethyl)-[2-methyl-9-(2,4,6-trimethyl-phenyl)-9H-purin-6-yl]-amine
    Show/Hide
PubChem ID
CID: 10500190
SID: 15525167
Canonical SMILES
COCCN(CCOC)c1nc(C)nc2n(cnc12)-c1c(C)cc(C)cc1C
    Show/Hide
Compound Formula C21H29N5O2
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
>
Corticotropin releasing factor receptor
>
Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki = 20.7 nM
   TI
   LI
   LO
   TS