All Bioactivity

Brief Information of the Cell Line and Protein

Cell Line ID: CL000016 , IMR-32

Cell Line Info

Synonyms	IMR 32 IMR32 Institute for Medical Research-32 GM03320 GM3320C GM03320D AG03320 AG3320
Category	Cancer cell line
Organism	Homo sapiens (Human)
Cellosaurus ID	CVCL_0346

Protein ID: PT01588 , Corticotropin-releasing factor receptor 1

Protein Info

Gene Name	CRHR1
Organism	Homo sapiens, Human
Protein Classification	Membrane receptor
Uniprot ID	P34998

Table of Molecular Bioactivities Related to the Cell Line and Protein

Cell Line ID: CL000016

Cell Line Info

Protein ID: PT01588

Protein Info

Compound ID	Compound Name	Compound Formula
CP0036466 Compound Info	Pyrazolo[1,5-a]-1,3,5-triazine, 12-35 Show/Hide	C19H23ClFN5O	1
1	IC50 = 1.2 nM Bioactivity Info	TI LI LO TS
CP0858280 Compound Info	(3S,6S,9S,12S,15S,18S,21S,24S,27S,30S,33S,36S,39S,42S,45S,48S,51S,54S,57S,60S,63S,66S,69S,72S,75S,78S,81S,84S,87S,90S,93S,96S)-15-((1H-imidazol-5-yl)methyl)-3-amino-96-((S)-1-amino-1-oxopropan-2-ylcarbamoyl)-78-(2-amino-2-oxoethyl)-54,66-bis(3-amino-3-oxopropyl)-45-(4-aminobutyl)-12-benzyl-27,36,51,57,63,93-hexakis(2-carboxyethyl)-24,81-bis(3-guanidinopropyl)-9-((R)-1-hydroxyethyl)-6,18,21,33,75,84,87,90-octaisobutyl-42,48,60,69,72-pentamethyl-30,39-bis(2-(methylthio)ethyl)-4,7,10,13,16,19,22,25,28,31,34,37,40,43,46,49,52,55,58,61,64,67,70,73,76,79,82,85,88,91,94-hentriacontaoxo-5,8,11,14,17,20,23,26,29,32,35,38,41,44,47,50,53,56,59,62,65,68,71,74,77,80,83,86,89,92,95-hentriacontaazanonanonacontane-1,99-dioic acid Show/Hide	C166H274N46O53S2	1
1	IC50 = 2 nM Bioactivity Info	TI LI LO TS
CP0073001 Compound Info	Pyrazolo[1,5-a]-1,3,5-triazine, 12-16 Show/Hide	C20H27N5O2	1
1	IC50 = 3.4 nM Bioactivity Info	TI LI LO TS
CP0116903 Compound Info	3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dimethyl-N,N-dipropylpyrazolo[1,5-a]pyrimidin-7-amine Show/Hide	C22H32N6	4
1	IC50 = 4 nM Bioactivity Info	TI LI LO TS
2	Ki = 3 nM Bioactivity Info	TI LI LO TS
3	Ki = 5 nM Bioactivity Info	TI LI LO TS
4	Ki = 8.3 nM Bioactivity Info	TI LI LO TS
CP0089343 Compound Info	Pyrazolo[1,5-a]-1,3,5-triazine, 12-3 Show/Hide	C21H29N5O3	1
1	IC50 = 4.7 nM Bioactivity Info	TI LI LO TS
CP0388820 Compound Info	N-butyl-3-[4-(ethoxymethyl)-2,6-dimethoxyphenyl]-6-methoxy-N-(oxan-4-yl)pyrazolo[5,1-b][1,3]thiazol-7-amine Show/Hide	C26H37N3O5S	1
1	IC50 = 7.1 nM Bioactivity Info	TI LI LO TS
CP0072999 Compound Info	Pyrazolo[1,5-a]-1,3,5-triazine, 12-33 Show/Hide	C22H31N5O3	1
1	IC50 = 15.2 nM Bioactivity Info	TI LI LO TS
CP0042279 Compound Info	3-methoxy-5-[2-methoxy-4-(trifluoromethoxy)phenyl]-6-methyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H24F3N3O3	2
1	IC50 = 93 nM Bioactivity Info	TI LI LO TS
2	Ki = 1 nM Bioactivity Info	TI LI LO TS
CP0549511 Compound Info	3-(4-chloro-2-morpholinothiazol-5-yl)-2,6-dimethyl-8-(pentan-3-yl)imidazo[1,2-b]pyridazine Show/Hide	C20H26ClN5OS	1
1	Ki = 0.2 nM Bioactivity Info	TI LI LO TS
CP0510311 Compound Info	8-(2,4-dichlorophenyl)-2-methyl-N,N-dipropylquinolin-4-amine Show/Hide	C22H24Cl2N2	1
1	Ki = 0.9 nM Bioactivity Info	TI LI LO TS
CP0510775 Compound Info	1,5-dimethyl-N,N-dipropyl-3-(2,4,6-trimethylphenyl)pyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C22H31N5	1
1	Ki = 1 nM Bioactivity Info	TI LI LO TS
CP0520733 Compound Info	5-(2-chloro-4-methoxyphenyl)-3-ethyl-6-methoxy-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H26ClN3O2	1
1	Ki = 1.1 nM Bioactivity Info	TI LI LO TS
CP0512533 Compound Info	3-methoxy-5-[2-methoxy-4-(trifluoromethyl)phenyl]-6-methyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H24F3N3O2	1
1	Ki = 1.3 nM Bioactivity Info	TI LI LO TS
CP0499122 Compound Info	5-[2-chloro-4-(difluoromethoxy)phenyl]-6-ethyl-3-methoxy-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H24ClF2N3O2	1
1	Ki = 1.4 nM Bioactivity Info	TI LI LO TS
CP0524564 Compound Info	6-ethyl-5-(2-ethyl-4-methoxyphenyl)-3-methoxy-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H31N3O2	1
1	Ki = 1.9 nM Bioactivity Info	TI LI LO TS
CP0392281 Compound Info	Butyl-[3-(2,4-dichloro-phenyl)-2,5-dimethyl-2H-pyrazolo[4,3-d]pyrimidin-7-yl]-ethyl-amine Show/Hide	C19H23Cl2N5	1
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0392364 Compound Info	3-(2,4-dichlorophenyl)-2,5-dimethyl-N,N-dipropylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C19H23Cl2N5	1
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0459482 Compound Info	N-(1,3-dimethoxypropan-2-yl)-8-(4-methoxy-2-methylphenyl)-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-4-amine Show/Hide	C20H27N5O3	1
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0478377 Compound Info	2-(4-chloro-2,6-dimethoxyphenyl)-4-methoxy-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C20H28ClN3O3	1
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0906425 Compound Info	4-(2-chloro-4-methoxy-5-methylphenyl)-N-((S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl)-5-methyl-N-(prop-2-ynyl)thiazol-2-amine hydrochloride Show/Hide	C27H29Cl2FN2OS	1
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0503181 Compound Info	6-ethyl-3-methoxy-5-[4-methoxy-2-(trifluoromethyl)phenyl]-N-pentan-3-ylpyrazin-2-amine Show/Hide	C20H26F3N3O2	1
1	Ki = 2.2 nM Bioactivity Info	TI LI LO TS
CP0505632 Compound Info	5-[2-chloro-4-(difluoromethoxy)phenyl]-3-ethyl-6-methoxy-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H24ClF2N3O2	1
1	Ki = 2.5 nM Bioactivity Info	TI LI LO TS
CP0255382 Compound Info	Butyl-[2,5-dimethyl-7-(2,4,6-trimethyl-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-ethyl-amine Show/Hide	C23H32N4	2
1	Ki = 2.7 nM Bioactivity Info	TI LI LO TS
2	Ki = 3 nM Bioactivity Info	TI LI LO TS
CP0497031 Compound Info	3-(2,4-dichlorophenyl)-N-ethyl-2,5-dimethyl-N-propylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C18H21Cl2N5	1
1	Ki = 3 nM Bioactivity Info	TI LI LO TS
CP0502148 Compound Info	2,5-dimethyl-N,N-dipropyl-3-(2,4,6-trimethylphenyl)pyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C22H31N5	1
1	Ki = 3 nM Bioactivity Info	TI LI LO TS
CP0527710 Compound Info	2-ethyl-5-methyl-N,N-dipropyl-3-(2,4,6-trimethylphenyl)pyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C23H33N5	1
1	Ki = 3 nM Bioactivity Info	TI LI LO TS
CP0530824 Compound Info	3-(2,4-dichlorophenyl)-N,N-bis(2-methoxyethyl)-2,5-dimethylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C19H23Cl2N5O2	1
1	Ki = 3 nM Bioactivity Info	TI LI LO TS
CP0486865 Compound Info	(5-{[(4-Chloro-benzyl)-(3,3,3-trifluoro-propyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C21H15Cl4F6N3S	1
1	Ki = 3.2 nM Bioactivity Info	TI LI LO TS
CP0377337 Compound Info	(5-{[(3-Fluoro-benzyl)-(3,3,3-trifluoro-propyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C21H15Cl3F7N3S	1
1	Ki = 3.7 nM Bioactivity Info	TI LI LO TS
CP0387701 Compound Info	5-(2,4-dichlorophenyl)-N-(dicyclopropylmethyl)-3,6-diethylpyrazin-2-amine Show/Hide	C21H25Cl2N3	1
1	Ki = 3.7 nM Bioactivity Info	TI LI LO TS
CP0490259 Compound Info	3-(4-chloro-2-methylphenyl)-2,5-dimethyl-N,N-dipropylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C20H26ClN5	1
1	Ki = 4 nM Bioactivity Info	TI LI LO TS
CP0548513 Compound Info	5-Dipropylamino-3,6-diethyl-2-(2-methoxy-4,6-dimethyl-phenyl)-3H-pyrimidin-4-one Show/Hide	C23H35N3O2	1
1	Ki = 4 nM Bioactivity Info	TI LI LO TS
CP0425058 Compound Info	3,6-diethyl-5-[4-methoxy-2-(trifluoromethoxy)phenyl]-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H28F3N3O2	1
1	Ki = 4.1 nM Bioactivity Info	TI LI LO TS
CP0425060 Compound Info	5-(2,4-dichlorophenyl)-3,6-diethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H25Cl2N3	1
1	Ki = 4.1 nM Bioactivity Info	TI LI LO TS
CP0524570 Compound Info	3,6-diethyl-5-(2-methoxy-4-propan-2-yloxyphenyl)-N-pentan-3-ylpyrazin-2-amine Show/Hide	C23H35N3O2	1
1	Ki = 4.2 nM Bioactivity Info	TI LI LO TS
CP0520734 Compound Info	5-(2,4-dichlorophenyl)-3-methoxy-6-methyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C17H21Cl2N3O	1
1	Ki = 4.3 nM Bioactivity Info	TI LI LO TS
CP0424468 Compound Info	6-ethyl-3-methoxy-5-[2-methoxy-4-(trifluoromethyl)phenyl]-N-pentan-3-ylpyrazin-2-amine Show/Hide	C20H26F3N3O2	1
1	Ki = 4.4 nM Bioactivity Info	TI LI LO TS
CP0425057 Compound Info	3,6-diethyl-5-[4-methoxy-2-(trifluoromethyl)phenyl]-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H28F3N3O	1
1	Ki = 4.4 nM Bioactivity Info	TI LI LO TS
CP0503465 Compound Info	5-[2-chloro-4-(difluoromethoxy)phenyl]-3-methoxy-6-methyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C18H22ClF2N3O2	1
1	Ki = 4.6 nM Bioactivity Info	TI LI LO TS
CP0409652 Compound Info	(5-{[(4-Fluoro-benzyl)-(3,3,3-trifluoro-propyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C21H15Cl3F7N3S	1
1	Ki = 4.8 nM Bioactivity Info	TI LI LO TS
CP0528803 Compound Info	N-(cyclopropylmethyl)-1-(2-methoxy-4,6-dimethylphenyl)-3-methyl-N-propylisoquinolin-4-amine Show/Hide	C26H32N2O	1
1	Ki = 5 nM Bioactivity Info	TI LI LO TS
CP0482059 Compound Info	3,6-diethyl-5-[2-methoxy-4-(trifluoromethyl)phenyl]-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H28F3N3O	1
1	Ki = 5.6 nM Bioactivity Info	TI LI LO TS
CP0501775 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-(2-phenylethyl)propan-1-amine Show/Hide	C29H32ClN5	1
1	Ki = 5.9 nM Bioactivity Info	TI LI LO TS
CP0502938 Compound Info	5-(2,4-dichlorophenyl)-6-ethyl-3-methoxy-N-pentan-3-ylpyrazin-2-amine Show/Hide	C18H23Cl2N3O	1
1	Ki = 5.9 nM Bioactivity Info	TI LI LO TS
CP0504885 Compound Info	5-(2-chloro-4-ethoxyphenyl)-3-methoxy-6-methyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H26ClN3O2	1
1	Ki = 5.9 nM Bioactivity Info	TI LI LO TS
CP0505456 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-(cyclobutylmethyl)propan-1-amine Show/Hide	C26H32ClN5	1
1	Ki = 6 nM Bioactivity Info	TI LI LO TS
CP0453236 Compound Info	1-(2-methoxy-4,6-dimethylphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C25H32N2O	1
1	Ki = 6 nM Bioactivity Info	TI LI LO TS
CP0453239 Compound Info	4-methoxy-2-(2-methoxy-4,6-bis(trifluoromethyl)phenyl)-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C21H25F6N3O2	1
1	Ki = 6 nM Bioactivity Info	TI LI LO TS
CP0436476 Compound Info	(5-{[Benzyl-(3,3,3-trifluoro-propyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C21H16Cl3F6N3S	1
1	Ki = 6.1 nM Bioactivity Info	TI LI LO TS
CP0390086 Compound Info	3-ethyl-6-methoxy-5-[2-methoxy-4-(trifluoromethoxy)phenyl]-N-pentan-3-ylpyrazin-2-amine Show/Hide	C20H26F3N3O3	1
1	Ki = 6.1 nM Bioactivity Info	TI LI LO TS
CP0408026 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-ethyl-2-phenylethanamine Show/Hide	C28H30ClN5	1
1	Ki = 6.4 nM Bioactivity Info	TI LI LO TS
CP0546296 Compound Info	N,N-bis(cyclopropylmethyl)-1-(2-methoxy-4,6-dimethylphenyl)-3-methylisoquinolin-4-amine Show/Hide	C27H32N2O	1
1	Ki = 7 nM Bioactivity Info	TI LI LO TS
CP0470742 Compound Info	5-Dipropylamino-6-ethyl-2-(2-methoxy-4,6-dimethyl-phenyl)-3-methyl-3H-pyrimidin-4-one Show/Hide	C22H33N3O2	1
1	Ki = 7 nM Bioactivity Info	TI LI LO TS
CP0528742 Compound Info	3,6-diethyl-5-[2-methoxy-4-(trifluoromethoxy)phenyl]-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H28F3N3O2	1
1	Ki = 7.2 nM Bioactivity Info	TI LI LO TS
CP0387702 Compound Info	5-(2,4-dimethoxyphenyl)-3,6-diethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H31N3O2	1
1	Ki = 7.3 nM Bioactivity Info	TI LI LO TS
CP0524569 Compound Info	5-[4-(dimethylamino)-6-methylpyridin-3-yl]-3,6-diethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H33N5	1
1	Ki = 7.6 nM Bioactivity Info	TI LI LO TS
CP0510943 Compound Info	N-ethyl-N-[[4-methyl-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-2-phenylethanamine Show/Hide	C29H33N5	1
1	Ki = 7.8 nM Bioactivity Info	TI LI LO TS
CP0494007 Compound Info	5-(4-ethoxy-2-methoxyphenyl)-3,6-diethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C22H33N3O2	1
1	Ki = 7.8 nM Bioactivity Info	TI LI LO TS
CP0471135 Compound Info	1-(2,4-bis(2,2-difluoroethyl)-6-methoxyphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C27H32F4N2O	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0447409 Compound Info	N-(cyclopropylmethyl)-2,2,2-trifluoro-N-[[2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl]methyl]ethanamine Show/Hide	C23H28F6N4	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0486464 Compound Info	4-methoxy-2-(2-methoxy-4,6-dimethylphenyl)-6-methyl-5-(pentan-3-yloxy)pyrimidine Show/Hide	C20H28N2O3	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0503466 Compound Info	5-(2,4-dichlorophenyl)-3-ethyl-6-methoxy-N-pentan-3-ylpyrazin-2-amine Show/Hide	C18H23Cl2N3O	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0501777 Compound Info	N-(cyclobutylmethyl)-N-[[4-methyl-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]propan-1-amine Show/Hide	C27H35N5	1
1	Ki = 8.2 nM Bioactivity Info	TI LI LO TS
CP0535079 Compound Info	8-(2-chloro-4,6-dimethyl-phenyl)-2-methyl-3-(3-phenyl-pyrrolidin-1-ylmethyl)-8H-1,3a,7,8-tetraaza-cyclopenta[a]indene Show/Hide	C28H28ClN5	1
1	Ki = 8.4 nM Bioactivity Info	TI LI LO TS
CP0473579 Compound Info	5-(2,4-dichlorophenyl)-3,6-dimethoxy-N-pentan-3-ylpyrazin-2-amine Show/Hide	C17H21Cl2N3O2	1
1	Ki = 8.4 nM Bioactivity Info	TI LI LO TS
CP0275883 Compound Info	5-[[cyclopropylmethyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C18H19Cl3F3N3S	1
1	Ki = 8.6 nM Bioactivity Info	TI LI LO TS
CP0499391 Compound Info	5-(2,4-dichlorophenyl)-3-ethyl-6-methyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C18H23Cl2N3	1
1	Ki = 8.6 nM Bioactivity Info	TI LI LO TS
CP0501739 Compound Info	3-ethyl-1-(2-methoxy-4,6-dimethylphenyl)-N,N-dipropylisoquinolin-4-amine Show/Hide	C26H34N2O	1
1	Ki = 9 nM Bioactivity Info	TI LI LO TS
CP0423071 Compound Info	2-(4-(difluoromethyl)-2,6-dimethoxyphenyl)-4-methoxy-6-methyl-5-(pentan-3-yloxy)pyrimidine Show/Hide	C20H26F2N2O4	1
1	Ki = 9 nM Bioactivity Info	TI LI LO TS
CP0486463 Compound Info	2-(4-chloro-2,6-dimethoxyphenyl)-4-methoxy-6-methyl-5-(pentan-3-yloxy)pyrimidine Show/Hide	C19H25ClN2O4	1
1	Ki = 9 nM Bioactivity Info	TI LI LO TS
CP0453362 Compound Info	3-(2,4-dimethoxyphenyl)-2,5-dimethyl-N,N-dipropylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C21H29N5O2	1
1	Ki = 10 nM Bioactivity Info	TI LI LO TS
CP0509484 Compound Info	5-methyl-N,N,2-tripropyl-3-(2,4,6-trimethylphenyl)pyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C24H35N5	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0409481 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-(cyclopropylmethyl)propan-1-amine Show/Hide	C25H30ClN5	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0428071 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-prop-2-enylpropan-1-amine Show/Hide	C24H28ClN5	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0541689 Compound Info	(5-{[(4-Chloro-benzyl)-propyl-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C21H18Cl4F3N3S	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0535442 Compound Info	3,6-diethyl-N-((1R,2S)-2-(2-fluoroethoxy)-2,3-dihydro-1H-inden-1-yl)-5-(4-methylpyridin-2-yloxy)pyrazin-2-amine Show/Hide	C25H29FN4O2	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0714287 Compound Info	N-(Cyclopropylmethyl)-7-[2,6-dimethoxy-4-(methoxymethyl)phenyl]-2-ethyl-N-[(tetrahydro-2H-pyran-4-yl)methyl]pyrazolo[1,5-a]pyridin-3-amine 4-methylbenzenesulfonate Show/Hide	C36H47N3O7S	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0524568 Compound Info	5-(2,6-dimethoxypyridin-3-yl)-3,6-diethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C20H30N4O2	1
1	Ki = 11.6 nM Bioactivity Info	TI LI LO TS
CP0512524 Compound Info	5-(2,4-dichlorophenyl)-6-ethyl-3-iodo-N-pentan-3-ylpyrazin-2-amine Show/Hide	C17H20Cl2IN3	1
1	Ki = 12 nM Bioactivity Info	TI LI LO TS
CP0447410 Compound Info	N-(cyclopropylmethyl)-2,2,3,3,3-pentafluoro-N-[[2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl]methyl]propan-1-amine Show/Hide	C24H28F8N4	1
1	Ki = 14 nM Bioactivity Info	TI LI LO TS
CP0505634 Compound Info	5-(2,4-dichlorophenyl)-6-methoxy-3-methyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C17H21Cl2N3O	1
1	Ki = 14.4 nM Bioactivity Info	TI LI LO TS
CP0507713 Compound Info	1-ethyl-5-methyl-N,N-dipropyl-3-(2,4,6-trimethylphenyl)pyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C23H33N5	1
1	Ki = 15 nM Bioactivity Info	TI LI LO TS
CP0412639 Compound Info	N-(cyclopropylmethyl)-N-[[4-methyl-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]propan-1-amine Show/Hide	C26H33N5	1
1	Ki = 15 nM Bioactivity Info	TI LI LO TS
CP0428070 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-(2-cyclopropylethyl)propan-1-amine Show/Hide	C26H32ClN5	1
1	Ki = 15 nM Bioactivity Info	TI LI LO TS
CP0542177 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-propylpropan-1-amine Show/Hide	C24H30ClN5	1
1	Ki = 15 nM Bioactivity Info	TI LI LO TS
CP0500372 Compound Info	2-(2,4-Dichloro-phenyl)-5-dipropylamino-3-ethyl-6-methyl-3H-pyrimidin-4-one Show/Hide	C19H25Cl2N3O	1
1	Ki = 15 nM Bioactivity Info	TI LI LO TS
CP0497735 Compound Info	4-methoxy-2-(2-methoxy-4,6-dimethylphenyl)-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C21H31N3O2	1
1	Ki = 15 nM Bioactivity Info	TI LI LO TS
CP0497699 Compound Info	3-(2,4-dichlorophenyl)-2,5-dimethyl-N-pentan-3-ylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C18H21Cl2N5	1
1	Ki = 16 nM Bioactivity Info	TI LI LO TS
CP0917196 Compound Info	[5-Methyl-3-(2,4,6-trimethyl-phenyl)-1H-pyrazolo[4,3-d]pyrimidin-7-yl]-dipropyl-amine Show/Hide	C21H29N5	1
1	Ki = 16 nM Bioactivity Info	TI LI LO TS
CP0495634 Compound Info	N-(cyclopropylmethyl)-N-[[4-(trifluoromethyl)-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]propan-1-amine Show/Hide	C26H30F3N5	1
1	Ki = 16 nM Bioactivity Info	TI LI LO TS
CP0462294 Compound Info	4-ethoxy-2-(2-methoxy-4,6-dimethylphenyl)-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C22H33N3O2	1
1	Ki = 16 nM Bioactivity Info	TI LI LO TS
CP0530826 Compound Info	N-cyclopentyl-3-(2,4-dichlorophenyl)-2,5-dimethylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C18H19Cl2N5	1
1	Ki = 17 nM Bioactivity Info	TI LI LO TS
CP0427894 Compound Info	N-(cyclobutylmethyl)-N-[[4-ethyl-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]propan-1-amine Show/Hide	C28H37N5	1
1	Ki = 17 nM Bioactivity Info	TI LI LO TS
CP0486733 Compound Info	1-(4-(difluoromethoxy)-2-methoxyphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C24H28F2N2O2	1
1	Ki = 17 nM Bioactivity Info	TI LI LO TS
CP0498423 Compound Info	5-(2,4-dimethoxypyrimidin-5-yl)-3,6-diethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H29N5O2	1
1	Ki = 17.2 nM Bioactivity Info	TI LI LO TS
CP0542176 Compound Info	N-butyl-N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]butan-1-amine Show/Hide	C26H34ClN5	1
1	Ki = 18 nM Bioactivity Info	TI LI LO TS
CP0400293 Compound Info	N,N-bis(prop-2-enyl)-2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C23H27F3N4O	1
1	Ki = 19 nM Bioactivity Info	TI LI LO TS
CP0521841 Compound Info	N-(cyclopropylmethyl)-5-(2,4-dichlorophenyl)-3,6-diethyl-N-propylpyrazin-2-amine Show/Hide	C21H27Cl2N3	1
1	Ki = 19.2 nM Bioactivity Info	TI LI LO TS
CP0535721 Compound Info	3-(2,6-dichlorophenyl)-2,5-dimethyl-N,N-dipropylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C19H23Cl2N5	1
1	Ki = 20 nM Bioactivity Info	TI LI LO TS
CP0541075 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-(cyclobutylmethyl)ethanamine Show/Hide	C25H30ClN5	1
1	Ki = 20 nM Bioactivity Info	TI LI LO TS
CP0526998 Compound Info	1-(4-chloro-2-methylphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C23H27ClN2	1
1	Ki = 21 nM Bioactivity Info	TI LI LO TS
CP0458943 Compound Info	5-Dipropylamino-3-ethyl-2-(2-methoxy-4,6-dimethyl-phenyl)-6-methyl-3H-pyrimidin-4-one Show/Hide	C22H33N3O2	1
1	Ki = 21 nM Bioactivity Info	TI LI LO TS
CP0522008 Compound Info	N-(cyclobutylmethyl)-N-[[2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl]methyl]propan-1-amine Show/Hide	C25H35F3N4	1
1	Ki = 21 nM Bioactivity Info	TI LI LO TS
CP0444900 Compound Info	3,6-diethyl-N-((1R,2S)-2-isopropoxy-2,3-dihydro-1H-inden-1-yl)-5-(4-methylpyridin-2-yloxy)pyrazin-2-amine Show/Hide	C26H32N4O2	1
1	Ki = 22 nM Bioactivity Info	TI LI LO TS
CP0535437 Compound Info	5-(4,6-dimethylpyridin-2-yloxy)-N-((1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6-diethylpyrazin-2-amine Show/Hide	C26H32N4O2	1
1	Ki = 22 nM Bioactivity Info	TI LI LO TS
CP0511880 Compound Info	4-ethyl-6-methoxy-2-(2-methoxy-4,6-dimethylphenyl)-N,N-dipropylpyrimidin-5-amine Show/Hide	C22H33N3O2	1
1	Ki = 22 nM Bioactivity Info	TI LI LO TS
CP0445055 Compound Info	1-cyclopropyl-N-(cyclopropylmethyl)-N-[[4-methyl-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]methanamine Show/Hide	C27H33N5	1
1	Ki = 23 nM Bioactivity Info	TI LI LO TS
CP0538249 Compound Info	5-[[cyclopropylmethyl(ethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C17H17Cl3F3N3S	1
1	Ki = 23 nM Bioactivity Info	TI LI LO TS
CP0507975 Compound Info	3,6-diethyl-5-(2-methoxy-4-methylphenyl)-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H31N3O	1
1	Ki = 23.7 nM Bioactivity Info	TI LI LO TS
CP0439694 Compound Info	3-(2,4-dichlorophenyl)-2,5-dimethyl-N-propylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C16H17Cl2N5	1
1	Ki = 24 nM Bioactivity Info	TI LI LO TS
CP0439049 Compound Info	7-(2,4-Dichloro-6-methyl-phenyl)-2-ethyl-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-(2,2,2-trifluoro-ethyl)-amide Show/Hide	C21H23Cl2F3N4O	1
1	Ki = 24 nM Bioactivity Info	TI LI LO TS
CP0542035 Compound Info	Butyl-[3-(2,4-dichloro-phenyl)-2,5-dimethyl-2H-pyrazolo[4,3-d]pyrimidin-7-yl]-amine Show/Hide	C17H19Cl2N5	1
1	Ki = 25 nM Bioactivity Info	TI LI LO TS
CP0390943 Compound Info	(5-{[(4-Fluoro-benzyl)-propyl-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C21H18Cl3F4N3S	1
1	Ki = 25 nM Bioactivity Info	TI LI LO TS
CP0510942 Compound Info	N-[[4-methyl-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-prop-2-enylprop-2-en-1-amine Show/Hide	C25H29N5	1
1	Ki = 26 nM Bioactivity Info	TI LI LO TS
CP0492022 Compound Info	5-[[bis(cyclopropylmethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C19H19Cl3F3N3S	1
1	Ki = 26 nM Bioactivity Info	TI LI LO TS
CP0528804 Compound Info	1-(4-methoxy-2,6-dimethylphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C25H32N2O	1
1	Ki = 26 nM Bioactivity Info	TI LI LO TS
CP0487179 Compound Info	7-(2-Bromo-4,6-dimethyl-phenyl)-2-ethyl-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-(2,2,2-trifluoro-ethyl)-amide Show/Hide	C22H26BrF3N4O	1
1	Ki = 26 nM Bioactivity Info	TI LI LO TS
CP0498422 Compound Info	N,N-bis(cyclopropylmethyl)-5-(2,4-dichlorophenyl)-3,6-diethylpyrazin-2-amine Show/Hide	C22H27Cl2N3	1
1	Ki = 26 nM Bioactivity Info	TI LI LO TS
CP0390412 Compound Info	N-(cyclobutylmethyl)-2,2,2-trifluoro-N-[[2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl]methyl]ethanamine Show/Hide	C24H30F6N4	1
1	Ki = 27 nM Bioactivity Info	TI LI LO TS
CP0507997 Compound Info	5-(2,4-dichlorophenyl)-3,6-dimethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C17H21Cl2N3	1
1	Ki = 27 nM Bioactivity Info	TI LI LO TS
CP0445056 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-prop-2-enylprop-2-en-1-amine Show/Hide	C24H26ClN5	1
1	Ki = 28 nM Bioactivity Info	TI LI LO TS
CP0525326 Compound Info	N-benzyl-N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]propan-1-amine Show/Hide	C28H30ClN5	1
1	Ki = 28 nM Bioactivity Info	TI LI LO TS
CP0390912 Compound Info	5-[[2-phenylethyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C22H21Cl3F3N3S	1
1	Ki = 28 nM Bioactivity Info	TI LI LO TS
CP0535380 Compound Info	1-(4-methoxy-2-methylphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C24H30N2O	1
1	Ki = 28 nM Bioactivity Info	TI LI LO TS
CP0464736 Compound Info	3-(2,4-dichlorophenyl)-N-ethyl-N-hexyl-2,5-dimethylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C21H27Cl2N5	1
1	Ki = 29 nM Bioactivity Info	TI LI LO TS
CP0464660 Compound Info	3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-((1R,2S)-2-propoxy-2,3-dihydro-1H-inden-1-yl)pyrazin-2-amine Show/Hide	C26H32N4O2	1
1	Ki = 30 nM Bioactivity Info	TI LI LO TS
CP0559998 Compound Info	1-(2,4-dimethyl-6-(2-morpholinoethoxy)phenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C30H41N3O2	1
1	Ki = 30 nM Bioactivity Info	TI LI LO TS
CP0390413 Compound Info	N-(cyclopropylmethyl)-N-[[2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl]methyl]ethanamine Show/Hide	C23H31F3N4	1
1	Ki = 31 nM Bioactivity Info	TI LI LO TS
CP0546295 Compound Info	1-(2-(2-(4-(dipropylamino)-3-methylisoquinolin-1-yl)-3,5-dimethylphenoxy)ethyl)piperidin-3-ol Show/Hide	C31H43N3O2	1
1	Ki = 32 nM Bioactivity Info	TI LI LO TS
CP0520355 Compound Info	N-(cyclopropylmethyl)-N-[[2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl]methyl]propan-1-amine Show/Hide	C24H33F3N4	1
1	Ki = 32 nM Bioactivity Info	TI LI LO TS
CP0486467 Compound Info	4-chloro-2-(2-methoxy-4,6-dimethylphenyl)-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C20H28ClN3O	1
1	Ki = 33 nM Bioactivity Info	TI LI LO TS
CP0493324 Compound Info	N-[(1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C25H30N4O2	1
1	Ki = 35 nM Bioactivity Info	TI LI LO TS
CP0522329 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-(cyclopropylmethyl)ethanamine Show/Hide	C24H28ClN5	1
1	Ki = 36 nM Bioactivity Info	TI LI LO TS
CP0541074 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-ethylbutan-1-amine Show/Hide	C24H30ClN5	1
1	Ki = 36 nM Bioactivity Info	TI LI LO TS
CP0530477 Compound Info	1-(2-ethyl-4-methoxyphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C25H32N2O	1
1	Ki = 36 nM Bioactivity Info	TI LI LO TS
CP0436475 Compound Info	(5-{[(4-Methoxy-benzyl)-propyl-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C22H21Cl3F3N3OS	1
1	Ki = 37 nM Bioactivity Info	TI LI LO TS
CP0498134 Compound Info	3-(2,4-dichlorophenyl)-2,5-dimethyl-N-pentylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C18H21Cl2N5	1
1	Ki = 38 nM Bioactivity Info	TI LI LO TS
CP0495079 Compound Info	5-[[benzyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C21H19Cl3F3N3S	1
1	Ki = 38 nM Bioactivity Info	TI LI LO TS
CP0467998 Compound Info	2-(2,4-Dimethoxy-phenyl)-5-dipropylamino-3-ethyl-6-methyl-3H-pyrimidin-4-one Show/Hide	C21H31N3O3	1
1	Ki = 38 nM Bioactivity Info	TI LI LO TS
CP0447411 Compound Info	2,2,2-trifluoro-N-((8-mesityl-2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-3-yl)methyl)-N-phenethylethanamine Show/Hide	C27H30F6N4	1
1	Ki = 38 nM Bioactivity Info	TI LI LO TS
CP0449173 Compound Info	5-Dipropylamino-3-(2-fluoro-ethyl)-2-(2-methoxy-4,6-dimethyl-phenyl)-6-methyl-3H-pyrimidin-4-one Show/Hide	C22H32FN3O2	1
1	Ki = 39 nM Bioactivity Info	TI LI LO TS
CP0542179 Compound Info	N-[[4-methyl-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-prop-2-enylpropan-1-amine Show/Hide	C25H31N5	1
1	Ki = 41 nM Bioactivity Info	TI LI LO TS
CP0552932 Compound Info	1-(2-(2-(4-(dipropylamino)-3-methylisoquinolin-1-yl)-3,5-dimethylphenoxy)ethyl)piperidin-4-ol Show/Hide	C31H43N3O2	1
1	Ki = 41 nM Bioactivity Info	TI LI LO TS
CP0497245 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-(2,2,2-trifluoro-ethyl)-amide Show/Hide	C23H29F3N4O	1
1	Ki = 41 nM Bioactivity Info	TI LI LO TS
CP0502903 Compound Info	7-(2-Chloro-4,6-dimethyl-phenyl)-2-ethyl-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-(2,2,2-trifluoro-ethyl)-amide Show/Hide	C22H26ClF3N4O	1
1	Ki = 41 nM Bioactivity Info	TI LI LO TS
CP0441732 Compound Info	(5-{[(2-Fluoro-benzyl)-propyl-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C21H18Cl3F4N3S	1
1	Ki = 42 nM Bioactivity Info	TI LI LO TS
CP0552930 Compound Info	1-(2,4-dimethoxyphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C24H30N2O2	1
1	Ki = 42 nM Bioactivity Info	TI LI LO TS
CP0432784 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-propyl-amide Show/Hide	C24H34N4O	1
1	Ki = 42 nM Bioactivity Info	TI LI LO TS
CP0541076 Compound Info	(2-cyclopropyl-ethyl)-[2-methyl-8-(2,4,6-trimethyl-phenyl)-8H-1,3a,7,8-tetraaza-cyclopenta[a]inden-3-ylmethyl]-propyl-amine Show/Hide	C27H35N5	1
1	Ki = 43 nM Bioactivity Info	TI LI LO TS
CP0409244 Compound Info	(5-{[Cyclopropylmethyl-(2,2,2-trifluoro-ethyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C17H14Cl3F6N3S	1
1	Ki = 43 nM Bioactivity Info	TI LI LO TS
CP0431528 Compound Info	(5-{[Cyclopropylmethyl-(3,3,3-trifluoro-propyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C18H16Cl3F6N3S	1
1	Ki = 46 nM Bioactivity Info	TI LI LO TS
CP0507998 Compound Info	2-(2,4-dichlorophenyl)-3,6-diethyl-5-pentan-3-yloxypyrazine Show/Hide	C19H24Cl2N2O	1
1	Ki = 46 nM Bioactivity Info	TI LI LO TS
CP0463203 Compound Info	5-Dipropylamino-3-isopropyl-2-(2-methoxy-4,6-dimethyl-phenyl)-6-methyl-3H-pyrimidin-4-one Show/Hide	C23H35N3O2	1
1	Ki = 47 nM Bioactivity Info	TI LI LO TS
CP0535371 Compound Info	3-(2-benzyl-pyrrolidin-1-ylmethyl)-8-(2-chloro-4,6-dimethyl-phenyl)-2-methyl-8H-1,3a,7,8-tetraaza-cyclopenta[a]indene Show/Hide	C29H30ClN5	1
1	Ki = 48 nM Bioactivity Info	TI LI LO TS
CP0447412 Compound Info	N-prop-2-enyl-N-[[2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl]methyl]propan-1-amine Show/Hide	C23H31F3N4	1
1	Ki = 48 nM Bioactivity Info	TI LI LO TS
CP0486739 Compound Info	1-(2-methoxy-4,6-dimethylphenyl)-N,N-dipropylisoquinolin-4-amine Show/Hide	C24H30N2O	1
1	Ki = 49 nM Bioactivity Info	TI LI LO TS
CP0535372 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-2-cyclopropyl-N-ethylethanamine Show/Hide	C25H30ClN5	1
1	Ki = 50 nM Bioactivity Info	TI LI LO TS
CP0440476 Compound Info	(5-{[Phenethyl-(2,2,2-trifluoro-ethyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C21H16Cl3F6N3S	1
1	Ki = 50 nM Bioactivity Info	TI LI LO TS
CP0467790 Compound Info	3,6-diethyl-N-((1R,2S)-2-(2-fluoroethoxy)-2,3-dihydro-1H-inden-1-yl)-5-(6-methylpyrimidin-4-yloxy)pyrazin-2-amine Show/Hide	C24H28FN5O2	1
1	Ki = 51 nM Bioactivity Info	TI LI LO TS
CP0440858 Compound Info	N-[(1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(4-ethylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C26H32N4O2	1
1	Ki = 53 nM Bioactivity Info	TI LI LO TS
CP0399346 Compound Info	2-(2-methoxy-4,6-dimethylphenyl)-4-methyl-6-propoxy-N,N-dipropylpyrimidin-5-amine Show/Hide	C23H35N3O2	1
1	Ki = 53 nM Bioactivity Info	TI LI LO TS
CP0524565 Compound Info	5-(2,4-dichlorophenyl)-6-ethyl-3-methyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C18H23Cl2N3	1
1	Ki = 54 nM Bioactivity Info	TI LI LO TS
CP0409251 Compound Info	(5-Diallylaminomethyl-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C17H15Cl3F3N3S	1
1	Ki = 57 nM Bioactivity Info	TI LI LO TS
CP0440856 Compound Info	5-(4,6-dimethylpyridin-2-yloxy)-3,6-diethyl-N-((1R,2S)-2-propoxy-2,3-dihydro-1H-inden-1-yl)pyrazin-2-amine Show/Hide	C27H34N4O2	1
1	Ki = 58 nM Bioactivity Info	TI LI LO TS
CP0510696 Compound Info	3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-(1-phenylpropyl)pyrazin-2-amine Show/Hide	C23H28N4O	1
1	Ki = 59 nM Bioactivity Info	TI LI LO TS
CP0505501 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid propyl-(2,2,2-trifluoro-ethyl)-amide Show/Hide	C22H29F3N4O	1
1	Ki = 61 nM Bioactivity Info	TI LI LO TS
CP0503691 Compound Info	5-methyl-N,N,1-tripropyl-3-(2,4,6-trimethylphenyl)pyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C24H35N5	1
1	Ki = 62 nM Bioactivity Info	TI LI LO TS
CP0432917 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-(2,2,3,3,3-pentafluoro-propyl)-amide Show/Hide	C24H29F5N4O	1
1	Ki = 63 nM Bioactivity Info	TI LI LO TS
CP0522009 Compound Info	3,3,3-trifluoro-N-((8-mesityl-2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-3-yl)methyl)-N-propylpropan-1-amine Show/Hide	C23H30F6N4	1
1	Ki = 63 nM Bioactivity Info	TI LI LO TS
CP0535439 Compound Info	N-[(1R,2S)-2-cyclopentyloxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C28H34N4O2	1
1	Ki = 67 nM Bioactivity Info	TI LI LO TS
CP0471532 Compound Info	N-(2-phenylethyl)-N-[[2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-3-yl]methyl]propan-1-amine Show/Hide	C28H35F3N4	1
1	Ki = 67 nM Bioactivity Info	TI LI LO TS
CP0497308 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid bis-cyclopropylmethyl-amide Show/Hide	C25H34N4O	1
1	Ki = 68 nM Bioactivity Info	TI LI LO TS
CP0482057 Compound Info	2-(2,4-dichlorophenyl)-3,6-diethyl-5-(2-ethylbutyl)pyrazine Show/Hide	C20H26Cl2N2	1
1	Ki = 68 nM Bioactivity Info	TI LI LO TS
CP0503468 Compound Info	3-chloro-5-(2,4-dichlorophenyl)-6-ethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C17H20Cl3N3	1
1	Ki = 71 nM Bioactivity Info	TI LI LO TS
CP0535832 Compound Info	5-Dipropylamino-3-ethyl-6-methyl-2-(2,4,6-trimethyl-phenyl)-3H-pyrimidin-4-one Show/Hide	C22H33N3O	1
1	Ki = 72 nM Bioactivity Info	TI LI LO TS
CP0483225 Compound Info	5-[[cyclobutylmethyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C19H21Cl3F3N3S	1
1	Ki = 73 nM Bioactivity Info	TI LI LO TS
CP0469269 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-(3,3,3-trifluoro-propyl)-amide Show/Hide	C24H31F3N4O	1
1	Ki = 73 nM Bioactivity Info	TI LI LO TS
CP0508075 Compound Info	7-(2,4-Dichloro-6-methyl-phenyl)-2-ethyl-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-propyl-amide Show/Hide	C22H28Cl2N4O	1
1	Ki = 75 nM Bioactivity Info	TI LI LO TS
CP0423072 Compound Info	4-methoxy-2-(2-methoxy-4,6-dimethylphenyl)-N,N,6-tripropylpyrimidin-5-amine Show/Hide	C23H35N3O2	1
1	Ki = 76 nM Bioactivity Info	TI LI LO TS
CP0522499 Compound Info	5-[[ethyl(2-phenylethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C21H19Cl3F3N3S	1
1	Ki = 79 nM Bioactivity Info	TI LI LO TS
CP0535438 Compound Info	2-((1R,2S)-1-(3,6-diethyl-5-(4-methylpyridin-2-yloxy)pyrazin-2-ylamino)-2,3-dihydro-1H-inden-2-yloxy)ethanol Show/Hide	C25H30N4O3	1
1	Ki = 82 nM Bioactivity Info	TI LI LO TS
CP0408847 Compound Info	5-Dipropylamino-2-(2-methoxy-4,6-dimethyl-phenyl)-3,6-dimethyl-3H-pyrimidin-4-one Show/Hide	C21H31N3O2	1
1	Ki = 90 nM Bioactivity Info	TI LI LO TS
CP0505455 Compound Info	N-(cyclopropylmethyl)-N-[[4-methyl-7-(2,4,6-trimethylphenyl)-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]ethanamine Show/Hide	C25H31N5	1
1	Ki = 93 nM Bioactivity Info	TI LI LO TS
CP0436970 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-ethyl-amide Show/Hide	C23H32N4O	1
1	Ki = 94 nM Bioactivity Info	TI LI LO TS
CP0449372 Compound Info	7-(2-Chloro-4,6-dimethyl-phenyl)-2-ethyl-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-propyl-amide Show/Hide	C23H31ClN4O	1
1	Ki = 94 nM Bioactivity Info	TI LI LO TS
CP0486465 Compound Info	4-methoxy-2-(2-methoxy-4,6-dimethylphenyl)-6-methyl-N-(pentan-3-yl)pyrimidin-5-amine Show/Hide	C20H29N3O2	1
1	Ki = 94 nM Bioactivity Info	TI LI LO TS
CP0498577 Compound Info	5-[[propyl(pyridin-4-ylmethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C20H18Cl3F3N4S	1
1	Ki = 100 nM Bioactivity Info	TI LI LO TS
CP0501427 Compound Info	5-[[prop-2-enyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C17H17Cl3F3N3S	1
1	Ki = 100 nM Bioactivity Info	TI LI LO TS
CP0496898 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid dipropylamide Show/Hide	C23H34N4O	1
1	Ki = 100 nM Bioactivity Info	TI LI LO TS
CP0454073 Compound Info	1-(2,4-dichlorophenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C22H24Cl2N2	1
1	Ki = 103 nM Bioactivity Info	TI LI LO TS
CP0535071 Compound Info	3-(2,4-dichlorophenyl)-N-hexyl-2,5-dimethylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C19H23Cl2N5	1
1	Ki = 112 nM Bioactivity Info	TI LI LO TS
CP0490438 Compound Info	3-(2,4-dichlorophenyl)-2,5-dimethyl-N-propyl-N-(2-pyrrolidin-1-ylethyl)pyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C22H28Cl2N6	1
1	Ki = 115 nM Bioactivity Info	TI LI LO TS
CP0511630 Compound Info	5-N-(3,5-dichloropyridin-2-yl)-3,6-diethyl-2-N-pentan-3-ylpyrazine-2,5-diamine Show/Hide	C18H25Cl2N5	1
1	Ki = 115 nM Bioactivity Info	TI LI LO TS
CP0502545 Compound Info	5-[[benzyl(ethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C20H17Cl3F3N3S	1
1	Ki = 120 nM Bioactivity Info	TI LI LO TS
CP0454065 Compound Info	1-(2,4-dimethyl-6-(2-(piperidin-1-yl)ethoxy)phenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C31H43N3O	1
1	Ki = 120 nM Bioactivity Info	TI LI LO TS
CP0548856 Compound Info	7-(2-Bromo-4,6-dimethyl-phenyl)-2-ethyl-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-propyl-amide Show/Hide	C23H31BrN4O	1
1	Ki = 126 nM Bioactivity Info	TI LI LO TS
CP0482058 Compound Info	5-(2,4-dichlorophenyl)-3,6-diethyl-N,N-bis(2-methoxyethyl)pyrazin-2-amine Show/Hide	C20H27Cl2N3O2	1
1	Ki = 128 nM Bioactivity Info	TI LI LO TS
CP0497045 Compound Info	(5-{[Phenethyl-(3,3,3-trifluoro-propyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C22H18Cl3F6N3S	1
1	Ki = 130 nM Bioactivity Info	TI LI LO TS
CP0502541 Compound Info	5-[[propyl(thiophen-2-ylmethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C19H17Cl3F3N3S2	1
1	Ki = 130 nM Bioactivity Info	TI LI LO TS
CP0460378 Compound Info	5-Dipropylamino-3,6-dimethyl-2-(2,4,6-trimethyl-phenyl)-3H-pyrimidin-4-one Show/Hide	C21H31N3O	1
1	Ki = 135 nM Bioactivity Info	TI LI LO TS
CP0402525 Compound Info	N'-[3-(2,4-dichlorophenyl)-2,5-dimethylpyrazolo[4,3-d]pyrimidin-7-yl]-N,N-dimethyl-N'-propylethane-1,2-diamine Show/Hide	C20H26Cl2N6	1
1	Ki = 145 nM Bioactivity Info	TI LI LO TS
CP0394978 Compound Info	5-[[ethyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C16H17Cl3F3N3S	1
1	Ki = 150 nM Bioactivity Info	TI LI LO TS
CP0524566 Compound Info	5-(2,4-dichlorophenyl)-3-ethoxy-6-ethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C19H25Cl2N3O	1
1	Ki = 151 nM Bioactivity Info	TI LI LO TS
CP0431529 Compound Info	(5-Dipropylaminomethyl-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C17H19Cl3F3N3S	1
1	Ki = 160 nM Bioactivity Info	TI LI LO TS
CP0530410 Compound Info	1-(2-methoxy-4,6-dimethylphenyl)-3-methyl-N-propylisoquinolin-4-amine Show/Hide	C22H26N2O	1
1	Ki = 165 nM Bioactivity Info	TI LI LO TS
CP0424469 Compound Info	5-(2,4-dichlorophenyl)-6-ethyl-3-fluoro-N-pentan-3-ylpyrazin-2-amine Show/Hide	C17H20Cl2FN3	1
1	Ki = 167 nM Bioactivity Info	TI LI LO TS
CP0515972 Compound Info	1-(2,4-dimethyl-6-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C30H41N3O	1
1	Ki = 173 nM Bioactivity Info	TI LI LO TS
CP0501008 Compound Info	N-cyclohexyl-3-(2,4-dichlorophenyl)-2,5-dimethylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C19H21Cl2N5	1
1	Ki = 174 nM Bioactivity Info	TI LI LO TS
CP0478359 Compound Info	5-Dipropylamino-2-(2-methoxy-4,6-dimethyl-phenyl)-6-methyl-3-propyl-3H-pyrimidin-4-one Show/Hide	C23H35N3O2	1
1	Ki = 190 nM Bioactivity Info	TI LI LO TS
CP0503692 Compound Info	3-(2,4-dichlorophenyl)-N-ethyl-2,5-dimethylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C15H15Cl2N5	1
1	Ki = 192 nM Bioactivity Info	TI LI LO TS
CP0440857 Compound Info	N-[(1R,2S)-2-cyclopropyloxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C26H30N4O2	1
1	Ki = 214 nM Bioactivity Info	TI LI LO TS
CP0501737 Compound Info	1-(2-methoxy-4,6-dimethylphenyl)-3-methyl-N-propyl-N-(2-(pyrrolidin-1-yl)ethyl)isoquinolin-4-amine Show/Hide	C28H37N3O	1
1	Ki = 215 nM Bioactivity Info	TI LI LO TS
CP0405840 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid propyl-(3,3,3-trifluoro-propyl)-amide Show/Hide	C23H31F3N4O	1
1	Ki = 220 nM Bioactivity Info	TI LI LO TS
CP0502904 Compound Info	2-Methyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-propyl-amide Show/Hide	C23H32N4O	1
1	Ki = 220 nM Bioactivity Info	TI LI LO TS
CP0526009 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid phenethyl-propyl-amide Show/Hide	C28H36N4O	1
1	Ki = 220 nM Bioactivity Info	TI LI LO TS
CP0453921 Compound Info	3,6-diethyl-N-((1R,2S)-2-methoxy-2,3-dihydro-1H-inden-1-yl)-5-(4-methylpyridin-2-yloxy)pyrazin-2-amine Show/Hide	C24H28N4O2	1
1	Ki = 222 nM Bioactivity Info	TI LI LO TS
CP0528715 Compound Info	5-(2,4-dichlorophenyl)-N-(1,3-dimethoxypropan-2-yl)-3,6-diethylpyrazin-2-amine Show/Hide	C19H25Cl2N3O2	1
1	Ki = 224 nM Bioactivity Info	TI LI LO TS
CP0376183 Compound Info	5-[[2-methylpropyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C18H21Cl3F3N3S	1
1	Ki = 240 nM Bioactivity Info	TI LI LO TS
CP0390414 Compound Info	8-mesityl-3-(piperidin-1-ylmethyl)-2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine Show/Hide	C22H29F3N4	1
1	Ki = 245 nM Bioactivity Info	TI LI LO TS
CP0510695 Compound Info	3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-(1-phenylethyl)pyrazin-2-amine Show/Hide	C22H26N4O	1
1	Ki = 251 nM Bioactivity Info	TI LI LO TS
CP0402485 Compound Info	3-Cyclopropylmethyl-2-(2,4-dimethoxy-phenyl)-5-dipropylamino-6-methyl-3H-pyrimidin-4-one Show/Hide	C23H33N3O3	1
1	Ki = 260 nM Bioactivity Info	TI LI LO TS
CP0461226 Compound Info	1-(2-(2-(dimethylamino)ethoxy)-4,6-dimethylphenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C28H39N3O	1
1	Ki = 265 nM Bioactivity Info	TI LI LO TS
CP0535441 Compound Info	3,6-diethyl-N-((1R,2S)-2-(2-fluoroethoxy)-2,3-dihydro-1H-inden-1-yl)-5-(pyridin-2-yloxy)pyrazin-2-amine Show/Hide	C24H27FN4O2	1
1	Ki = 266 nM Bioactivity Info	TI LI LO TS
CP0486961 Compound Info	7-(2-Bromo-4-isopropyl-phenyl)-2-ethyl-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-(2,2,2-trifluoro-ethyl)-amide Show/Hide	C23H28BrF3N4O	1
1	Ki = 270 nM Bioactivity Info	TI LI LO TS
CP0490721 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid (4-chloro-benzyl)-(3,3,3-trifluoro-propyl)-amide Show/Hide	C27H30ClF3N4O	1
1	Ki = 270 nM Bioactivity Info	TI LI LO TS
CP0459479 Compound Info	2-(2,6-dimethoxyphenyl)-4-methoxy-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C20H29N3O3	1
1	Ki = 277 nM Bioactivity Info	TI LI LO TS
CP0485589 Compound Info	5-[[propyl(pyridin-3-ylmethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C20H18Cl3F3N4S	1
1	Ki = 290 nM Bioactivity Info	TI LI LO TS
CP0501426 Compound Info	5-[[butyl(ethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C17H19Cl3F3N3S	1
1	Ki = 290 nM Bioactivity Info	TI LI LO TS
CP0498022 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid butyl-ethyl-amide Show/Hide	C23H34N4O	1
1	Ki = 290 nM Bioactivity Info	TI LI LO TS
CP0510650 Compound Info	2-(2,6-Dimethoxy-phenyl)-5-dipropylamino-3-ethyl-6-methyl-3H-pyrimidin-4-one Show/Hide	C21H31N3O3	1
1	Ki = 310 nM Bioactivity Info	TI LI LO TS
CP0535443 Compound Info	3,6-diethyl-N-(2-isopropoxy-1-phenylethyl)-5-(4-methylpyridin-2-yloxy)pyrazin-2-amine Show/Hide	C25H32N4O2	1
1	Ki = 337 nM Bioactivity Info	TI LI LO TS
CP0453240 Compound Info	2-mesityl-4-methoxy-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C21H31N3O	1
1	Ki = 354 nM Bioactivity Info	TI LI LO TS
CP0526591 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-ethylethanamine Show/Hide	C22H26ClN5	1
1	Ki = 360 nM Bioactivity Info	TI LI LO TS
CP0390415 Compound Info	3-((5,6-dihydropyridin-1(2H)-yl)methyl)-8-mesityl-2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine Show/Hide	C22H27F3N4	1
1	Ki = 364 nM Bioactivity Info	TI LI LO TS
CP0459834 Compound Info	N-(2-ethoxy-1-phenylethyl)-3,6-diethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C24H30N4O2	1
1	Ki = 384 nM Bioactivity Info	TI LI LO TS
CP0550909 Compound Info	(5-{[Benzyl-(2,2,2-trifluoro-ethyl)-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C20H14Cl3F6N3S	1
1	Ki = 390 nM Bioactivity Info	TI LI LO TS
CP0477963 Compound Info	3,6-dimethyl-5-(4-methylpyridin-2-yloxy)-N-(pentan-3-yl)pyrazin-2-amine Show/Hide	C17H24N4O	1
1	Ki = 401 nM Bioactivity Info	TI LI LO TS
CP0528713 Compound Info	2-butan-2-ylsulfanyl-5-(2,4-dichlorophenyl)-3,6-diethylpyrazine Show/Hide	C18H22Cl2N2S	1
1	Ki = 401 nM Bioactivity Info	TI LI LO TS
CP0448869 Compound Info	(5-{[(2-Cyclopropyl-ethyl)-propyl-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C19H21Cl3F3N3S	1
1	Ki = 420 nM Bioactivity Info	TI LI LO TS
CP0399586 Compound Info	N-[(1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(3-methylphenoxy)pyrazin-2-amine Show/Hide	C26H31N3O2	1
1	Ki = 436 nM Bioactivity Info	TI LI LO TS
CP0447404 Compound Info	4-((8-mesityl-2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-3-yl)methyl)thiomorpholine Show/Hide	C21H27F3N4S	1
1	Ki = 441 nM Bioactivity Info	TI LI LO TS
CP0490595 Compound Info	N-[(1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(5-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C25H30N4O2	1
1	Ki = 456 nM Bioactivity Info	TI LI LO TS
CP0395121 Compound Info	2-(2,4-Dimethoxy-phenyl)-5-dipropylamino-3,6-dimethyl-3H-pyrimidin-4-one Show/Hide	C20H29N3O3	1
1	Ki = 470 nM Bioactivity Info	TI LI LO TS
CP0399585 Compound Info	N-[(1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(6-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C25H30N4O2	1
1	Ki = 472 nM Bioactivity Info	TI LI LO TS
CP0524567 Compound Info	2-N-[5-(2,4-dichlorophenyl)-3,6-diethylpyrazin-2-yl]-1-N,1-N-dimethylpropane-1,2-diamine Show/Hide	C19H26Cl2N4	1
1	Ki = 489 nM Bioactivity Info	TI LI LO TS
CP0459480 Compound Info	2-(2,4-dimethoxyphenyl)-4-methoxy-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C20H29N3O3	1
1	Ki = 507 nM Bioactivity Info	TI LI LO TS
CP0506614 Compound Info	N-[(1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(3-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C25H30N4O2	1
1	Ki = 509 nM Bioactivity Info	TI LI LO TS
CP0501736 Compound Info	1-(2,4-dimethyl-6-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C31H44N4O	1
1	Ki = 524 nM Bioactivity Info	TI LI LO TS
CP0538719 Compound Info	3,6-diethyl-N-(2-methyl-1-phenylpropyl)-5-(4-methylpyridin-2-yloxy)pyrazin-2-amine Show/Hide	C24H30N4O	1
1	Ki = 530 nM Bioactivity Info	TI LI LO TS
CP0448012 Compound Info	2-(2,6-Dimethoxy-phenyl)-5-dipropylamino-3,6-dimethyl-3H-pyrimidin-4-one Show/Hide	C20H29N3O3	1
1	Ki = 530 nM Bioactivity Info	TI LI LO TS
CP0528741 Compound Info	5-(2,4-dichlorophenyl)-6-ethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C17H21Cl2N3	1
1	Ki = 545 nM Bioactivity Info	TI LI LO TS
CP0377338 Compound Info	5-[[methyl(2-phenylethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C20H17Cl3F3N3S	1
1	Ki = 560 nM Bioactivity Info	TI LI LO TS
CP0509175 Compound Info	5-Dipropylamino-6-ethyl-2-(2-methoxy-4,6-dimethyl-phenyl)-3H-pyrimidin-4-one Show/Hide	C21H31N3O2	1
1	Ki = 560 nM Bioactivity Info	TI LI LO TS
CP0505977 Compound Info	3-(2,4-dichlorophenyl)-2,5-dimethyl-N-(2-piperidin-1-ylethyl)-N-propylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C23H30Cl2N6	1
1	Ki = 561 nM Bioactivity Info	TI LI LO TS
CP0497736 Compound Info	2-(2-methoxy-4,6-dimethylphenyl)-4-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C20H29N3O	1
1	Ki = 561 nM Bioactivity Info	TI LI LO TS
CP0522325 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-methyl-2-pyridin-3-ylethanamine Show/Hide	C26H27ClN6	1
1	Ki = 570 nM Bioactivity Info	TI LI LO TS
CP0535078 Compound Info	8-(2-chloro-4,6-dimethyl-phenyl)-2-methyl-3-(2-phenyl-pyrrolidin-1-ylmethyl)-8H-1,3a,7,8-tetraaza-cyclopenta[a]indene Show/Hide	C28H28ClN5	1
1	Ki = 580 nM Bioactivity Info	TI LI LO TS
CP0453241 Compound Info	1-(5-(dipropylamino)-6-methoxy-2-(2-methoxy-4,6-dimethylphenyl)pyrimidin-4-yl)-2-methylpropan-2-ol Show/Hide	C24H37N3O3	1
1	Ki = 604 nM Bioactivity Info	TI LI LO TS
CP0430907 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid (2-cyclopropyl-ethyl)-ethyl-amide Show/Hide	C24H34N4O	1
1	Ki = 610 nM Bioactivity Info	TI LI LO TS
CP0392027 Compound Info	2-(2-Difluoromethoxy-6-methoxy-phenyl)-5-dipropylamino-3-ethyl-6-methyl-3H-pyrimidin-4-one Show/Hide	C21H29F2N3O3	1
1	Ki = 620 nM Bioactivity Info	TI LI LO TS
CP0496794 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid (2-cyclopropyl-ethyl)-(3,3,3-trifluoro-propyl)-amide Show/Hide	C25H33F3N4O	1
1	Ki = 650 nM Bioactivity Info	TI LI LO TS
CP0505499 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid benzyl-(3,3,3-trifluoro-propyl)-amide Show/Hide	C27H31F3N4O	1
1	Ki = 660 nM Bioactivity Info	TI LI LO TS
CP0522328 Compound Info	3-(3-benzyl-pyrrolidin-1-ylmethyl)-8-(2-chloro-4,6-dimethyl-phenyl)-2-methyl-8H-1,3a,7,8-tetraaza-cyclopenta[a]indene Show/Hide	C29H30ClN5	1
1	Ki = 700 nM Bioactivity Info	TI LI LO TS
CP0541073 Compound Info	8-(2-chloro-4,6-dimethyl-phenyl)-2-methyl-3-(3-phenethyl-pyrrolidin-1-ylmethyl)-8H-1,3a,7,8-tetraaza-cyclopenta[a]indene Show/Hide	C30H32ClN5	1
1	Ki = 700 nM Bioactivity Info	TI LI LO TS
CP0538720 Compound Info	3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N,N-dipropylpyrazin-2-amine Show/Hide	C20H30N4O	1
1	Ki = 711 nM Bioactivity Info	TI LI LO TS
CP0397686 Compound Info	2-(2,4-Dimethoxy-phenyl)-5-dipropylamino-6-methyl-3-propyl-3H-pyrimidin-4-one Show/Hide	C22H33N3O3	1
1	Ki = 720 nM Bioactivity Info	TI LI LO TS
CP0486418 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid allyl-propyl-amide Show/Hide	C23H32N4O	1
1	Ki = 740 nM Bioactivity Info	TI LI LO TS
CP0467344 Compound Info	3-(2-chlorophenyl)-2,5-dimethyl-N,N-dipropylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C19H24ClN5	1
1	Ki = 765 nM Bioactivity Info	TI LI LO TS
CP0498576 Compound Info	5-[[furan-2-ylmethyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C19H17Cl3F3N3OS	1
1	Ki = 770 nM Bioactivity Info	TI LI LO TS
CP0441918 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid (2-cyclopropyl-ethyl)-propyl-amide Show/Hide	C25H36N4O	1
1	Ki = 770 nM Bioactivity Info	TI LI LO TS
CP0397649 Compound Info	5-Dipropylamino-2-(2-methoxy-4,6-dimethyl-phenyl)-6-methyl-3H-pyrimidin-4-one Show/Hide	C20H29N3O2	1
1	Ki = 930 nM Bioactivity Info	TI LI LO TS
CP0552931 Compound Info	1-(4-chlorophenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C22H25ClN2	1
1	Ki = 962 nM Bioactivity Info	TI LI LO TS
CP0486738 Compound Info	N-(2-imidazol-1-ylethyl)-1-(2-methoxy-4,6-dimethylphenyl)-3-methyl-N-propylisoquinolin-4-amine Show/Hide	C27H32N4O	1
1	Ki = 1063 nM Bioactivity Info	TI LI LO TS
CP0372677 Compound Info	(5-Methylsulfanyl-[1,2,3]thiadiazol-4-yl)-[2-(2,4,6-trichloro-phenylamino)-4-trifluoromethyl-thiazol-5-ylmethyl]-amine Show/Hide	C14H9Cl3F3N5S3	1
1	Ki = 1100 nM Bioactivity Info	TI LI LO TS
CP0394980 Compound Info	(5-{[(2-Cyclopropyl-ethyl)-ethyl-amino]-methyl}-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C18H19Cl3F3N3S	1
1	Ki = 1100 nM Bioactivity Info	TI LI LO TS
CP0483777 Compound Info	1-(5-(dipropylamino)-6-methoxy-2-(2-methoxy-4,6-dimethylphenyl)pyrimidin-4-yl)propan-2-ol Show/Hide	C23H35N3O3	1
1	Ki = 1150 nM Bioactivity Info	TI LI LO TS
CP0502939 Compound Info	2-[3,6-diethyl-5-(pentan-3-ylamino)pyrazin-2-yl]-5-methoxyphenol Show/Hide	C20H29N3O2	1
1	Ki = 1181 nM Bioactivity Info	TI LI LO TS
CP0444901 Compound Info	3,6-dimethyl-5-(4-methylpyridin-2-yloxy)-N,N-dipropylpyrazin-2-amine Show/Hide	C18H26N4O	1
1	Ki = 1185 nM Bioactivity Info	TI LI LO TS
CP0535077 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-methyl-1-pyridin-4-ylmethanamine Show/Hide	C25H25ClN6	1
1	Ki = 1200 nM Bioactivity Info	TI LI LO TS
CP0527164 Compound Info	N-(cyclopropylmethyl)-N-propyl-2-(trifluoromethyl)-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C24H31F3N4O	1
1	Ki = 1200 nM Bioactivity Info	TI LI LO TS
CP0399588 Compound Info	N-(cyclopropylmethyl)-3,6-dimethyl-5-(4-methylpyridin-2-yl)oxy-N-propylpyrazin-2-amine Show/Hide	C19H26N4O	1
1	Ki = 1207 nM Bioactivity Info	TI LI LO TS
CP0538717 Compound Info	2-N-(3,5-dichloropyridin-2-yl)-3,6-diethyl-5-N-[(1R,2S)-2-(2-fluoroethoxy)-2,3-dihydro-1H-inden-1-yl]-2-N-methylpyrazine-2,5-diamine Show/Hide	C25H28Cl2FN5O	1
1	Ki = 1208 nM Bioactivity Info	TI LI LO TS
CP0511629 Compound Info	N-[(1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-dimethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C23H26N4O2	1
1	Ki = 1217 nM Bioactivity Info	TI LI LO TS
CP0528214 Compound Info	3,6-diethyl-N-((1R,2S)-2-methoxy-2,3-dihydro-1H-inden-1-yl)-N-methyl-5-(4-methylpyridin-2-yloxy)pyrazin-2-amine Show/Hide	C25H30N4O2	1
1	Ki = 1261 nM Bioactivity Info	TI LI LO TS
CP0522327 Compound Info	8-(2-chloro-4,6-dimethyl-phenyl)-2-methyl-3-(2-phenethyl-pyrrolidin-1-ylmethyl)-8H-1,3a,7,8-tetraaza-cyclopenta[a]indene Show/Hide	C30H32ClN5	1
1	Ki = 1300 nM Bioactivity Info	TI LI LO TS
CP0394191 Compound Info	5-[[propyl(pyridin-2-ylmethyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C20H18Cl3F3N4S	1
1	Ki = 1300 nM Bioactivity Info	TI LI LO TS
CP0510941 Compound Info	8-(2-chloro-4,6-dimethyl-phenyl)-2-methyl-3-morpholin-4-ylmethyl-8H-1,3a,7,8-tetraaza-cyclopenta[a]indene Show/Hide	C22H24ClN5O	1
1	Ki = 1400 nM Bioactivity Info	TI LI LO TS
CP0447403 Compound Info	4-((8-mesityl-2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidin-3-yl)methyl)morpholine Show/Hide	C21H27F3N4O	1
1	Ki = 1510 nM Bioactivity Info	TI LI LO TS
CP0424471 Compound Info	N'-[5-(2,4-dichlorophenyl)-3,6-diethylpyrazin-2-yl]-N,N-dimethyl-N'-propylethane-1,2-diamine Show/Hide	C21H30Cl2N4	1
1	Ki = 1538 nM Bioactivity Info	TI LI LO TS
CP0535444 Compound Info	3,6-diethyl-N2-(pentan-3-yl)-N5-(2,4,6-trichlorophenyl)pyrazine-2,5-diamine Show/Hide	C19H25Cl3N4	1
1	Ki = 1540 nM Bioactivity Info	TI LI LO TS
CP0445484 Compound Info	7-(2-Bromo-4-isopropyl-phenyl)-2-ethyl-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid cyclopropylmethyl-propyl-amide Show/Hide	C24H33BrN4O	1
1	Ki = 1559 nM Bioactivity Info	TI LI LO TS
CP0511938 Compound Info	2-(5-(dipropylamino)-2-(2-methoxy-4,6-dimethylphenyl)-6-methylpyrimidin-4-yloxy)ethanol Show/Hide	C22H33N3O3	1
1	Ki = 1610 nM Bioactivity Info	TI LI LO TS
CP0500474 Compound Info	5-Dipropylamino-2-(2-methoxy-4,6-dimethyl-phenyl)-6-methyl-3-(2,2,2-trifluoro-ethyl)-3H-pyrimidin-4-one Show/Hide	C22H30F3N3O2	1
1	Ki = 1630 nM Bioactivity Info	TI LI LO TS
CP0486744 Compound Info	1-(2-chlorophenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C22H25ClN2	1
1	Ki = 1685 nM Bioactivity Info	TI LI LO TS
CP0382896 Compound Info	8-mesityl-2-methyl-N-phenethyl-N-propyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C28H36N4O	1
1	Ki = 1700 nM Bioactivity Info	TI LI LO TS
CP0538718 Compound Info	5-N-(3,5-dichloropyridin-2-yl)-3,6-diethyl-2-N-[(1R,2S)-2-(2-fluoroethoxy)-2,3-dihydro-1H-inden-1-yl]pyrazine-2,5-diamine Show/Hide	C24H26Cl2FN5O	1
1	Ki = 1733 nM Bioactivity Info	TI LI LO TS
CP0548894 Compound Info	5-[(2-ethylimidazol-1-yl)methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C16H12Cl3F3N4S	1
1	Ki = 1800 nM Bioactivity Info	TI LI LO TS
CP0490596 Compound Info	(1R,2S)-1-(3,6-diethyl-5-(4-methylpyridin-2-yloxy)pyrazin-2-ylamino)-2,3-dihydro-1H-inden-2-yl acetate Show/Hide	C25H28N4O3	1
1	Ki = 2021 nM Bioactivity Info	TI LI LO TS
CP0528215 Compound Info	3,6-dimethyl-5-(4-methylpyridin-2-yloxy)-N-(1-phenylpropyl)pyrazin-2-amine Show/Hide	C21H24N4O	1
1	Ki = 2123 nM Bioactivity Info	TI LI LO TS
CP0471530 Compound Info	N-(cyclopropylmethyl)-2-ethyl-N-propyl-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C25H36N4O	1
1	Ki = 2300 nM Bioactivity Info	TI LI LO TS
CP0477974 Compound Info	3,6-dimethyl-N-(2-methyl-1-phenylpropyl)-5-(4-methylpyridin-2-yloxy)pyrazin-2-amine Show/Hide	C22H26N4O	1
1	Ki = 2376 nM Bioactivity Info	TI LI LO TS
CP0467793 Compound Info	3,6-diethyl-5-(3-methylpyridin-2-yloxy)-N-(1-phenylpropyl)pyrazin-2-amine Show/Hide	C23H28N4O	1
1	Ki = 2434 nM Bioactivity Info	TI LI LO TS
CP0409477 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-methyl-1-pyridin-3-ylmethanamine Show/Hide	C25H25ClN6	1
1	Ki = 2700 nM Bioactivity Info	TI LI LO TS
CP0442356 Compound Info	5-N-(4-chlorophenyl)-3,6-diethyl-2-N-pentan-3-ylpyrazine-2,5-diamine Show/Hide	C19H27ClN4	1
1	Ki = 2703 nM Bioactivity Info	TI LI LO TS
CP0510940 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-methyl-2-pyridin-2-ylethanamine Show/Hide	C26H27ClN6	1
1	Ki = 2800 nM Bioactivity Info	TI LI LO TS
CP0510939 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]pentan-2-amine Show/Hide	C23H28ClN5	1
1	Ki = 2900 nM Bioactivity Info	TI LI LO TS
CP0437109 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid (4-chloro-benzyl)-propyl-amide Show/Hide	C27H33ClN4O	1
1	Ki = 3000 nM Bioactivity Info	TI LI LO TS
CP0500809 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid diallylamide Show/Hide	C23H30N4O	1
1	Ki = 3000 nM Bioactivity Info	TI LI LO TS
CP0434486 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-methyl-2-pyridin-4-ylethanamine Show/Hide	C26H27ClN6	1
1	Ki = 3200 nM Bioactivity Info	TI LI LO TS
CP0504552 Compound Info	N-(cyclobutylmethyl)-2-methyl-N-propyl-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C25H36N4O	1
1	Ki = 3300 nM Bioactivity Info	TI LI LO TS
CP0464662 Compound Info	3,6-diethyl-N2-(6-methylpyridin-2-yl)-N5-(pentan-3-yl)pyrazine-2,5-diamine Show/Hide	C19H29N5	1
1	Ki = 3382 nM Bioactivity Info	TI LI LO TS
CP0382895 Compound Info	N,N-bis(cyclopropylmethyl)-2-methyl-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C25H34N4O	1
1	Ki = 3400 nM Bioactivity Info	TI LI LO TS
CP0503467 Compound Info	3-butyl-5-(2,4-dichlorophenyl)-6-ethyl-N-pentan-3-ylpyrazin-2-amine Show/Hide	C21H29Cl2N3	1
1	Ki = 3657 nM Bioactivity Info	TI LI LO TS
CP0459835 Compound Info	5-N-(3,5-dichloropyridin-2-yl)-3,6-dimethyl-2-N-pentan-3-ylpyrazine-2,5-diamine Show/Hide	C16H21Cl2N5	1
1	Ki = 3980 nM Bioactivity Info	TI LI LO TS
CP0529763 Compound Info	2-(2,4-Dimethoxy-phenyl)-5-dipropylamino-3-(2-methoxy-ethyl)-6-methyl-3H-pyrimidin-4-one Show/Hide	C22H33N3O4	1
1	Ki = 4000 nM Bioactivity Info	TI LI LO TS
CP0434485 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-2-methoxy-N-(2-methoxyethyl)ethanamine Show/Hide	C24H30ClN5O2	1
1	Ki = 4100 nM Bioactivity Info	TI LI LO TS
CP0445764 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid benzyl-propyl-amide Show/Hide	C27H34N4O	1
1	Ki = 4100 nM Bioactivity Info	TI LI LO TS
CP0511229 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid (3-fluoro-benzyl)-propyl-amide Show/Hide	C27H33FN4O	1
1	Ki = 4200 nM Bioactivity Info	TI LI LO TS
CP0467792 Compound Info	2-(3,6-diethyl-5-(4-methylpyridin-2-yloxy)pyrazin-2-ylamino)-2-phenylethanol Show/Hide	C22H26N4O2	1
1	Ki = 4688 nM Bioactivity Info	TI LI LO TS
CP0390941 Compound Info	5-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C17H17Cl3F3N3OS	1
1	Ki = 5100 nM Bioactivity Info	TI LI LO TS
CP0535440 Compound Info	N-[(1S,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C25H30N4O2	1
1	Ki = 5473 nM Bioactivity Info	TI LI LO TS
CP0525325 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-1,3-dimethoxypropan-2-amine Show/Hide	C23H28ClN5O2	1
1	Ki = 5600 nM Bioactivity Info	TI LI LO TS
CP0394979 Compound Info	5-[[cyclohexylmethyl(propyl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C21H25Cl3F3N3S	1
1	Ki = 6300 nM Bioactivity Info	TI LI LO TS
CP0497310 Compound Info	N-(cyclopropylmethyl)-N-[[6-methyl-1-(2,4,6-trimethylphenyl)-2,3-dihydroimidazo[1,2-a]imidazol-5-yl]methyl]propan-1-amine Show/Hide	C23H34N4	1
1	Ki = 6600 nM Bioactivity Info	TI LI LO TS
CP0523121 Compound Info	5-(2,5-dihydropyrrol-1-ylmethyl)-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C15H11Cl3F3N3S	1
1	Ki = 6700 nM Bioactivity Info	TI LI LO TS
CP0431530 Compound Info	5-[[di(propan-2-yl)amino]methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C17H19Cl3F3N3S	1
1	Ki = 9800 nM Bioactivity Info	TI LI LO TS
CP0522326 Compound Info	N-[[7-(2-chloro-4,6-dimethylphenyl)-4-methyl-2,5,7,9-tetrazatricyclo[6.4.0.02,6]dodeca-1(8),3,5,9,11-pentaen-3-yl]methyl]-N-methyl-1-pyridin-2-ylmethanamine Show/Hide	C25H25ClN6	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0448870 Compound Info	(5-Pyrrolidin-1-ylmethyl-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C15H13Cl3F3N3S	1
1	Ki = 10000 nM Bioactivity Info	TI LI LO TS
CP0486870 Compound Info	5-[(2-phenylethylamino)methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C19H15Cl3F3N3S	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0440854 Compound Info	3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-(pentan-3-yl)pyrazin-2-amine Show/Hide	C19H28N4O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0440855 Compound Info	2-N-(1,3-dimethoxypropan-2-yl)-3,6-diethyl-5-N-(4-methylpyridin-2-yl)pyrazine-2,5-diamine Show/Hide	C19H29N5O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0442351 Compound Info	3,6-diethyl-N2-(pentan-3-yl)-N5-(pyridin-2-yl)pyrazine-2,5-diamine Show/Hide	C18H27N5	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0444895 Compound Info	2-N-[(1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-N-(4-methylpyridin-2-yl)pyrazine-2,5-diamine Show/Hide	C25H31N5O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0444896 Compound Info	5-N-(3,5-dichloropyridin-2-yl)-3,6-diethyl-2-N-(1-phenylpropyl)pyrazine-2,5-diamine Show/Hide	C22H25Cl2N5	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0444897 Compound Info	3,6-diethyl-N2-(5-nitropyridin-2-yl)-N5-(pentan-3-yl)pyrazine-2,5-diamine Show/Hide	C18H26N6O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0444898 Compound Info	5-N-(2,4-dichlorophenyl)-3,6-diethyl-2-N-pentan-3-ylpyrazine-2,5-diamine Show/Hide	C19H26Cl2N4	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0444899 Compound Info	N-(1,3-dimethoxypropan-2-yl)-3,6-diethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C19H28N4O3	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0453920 Compound Info	5-N-(3,5-dichloropyridin-2-yl)-3,6-diethyl-2-N-(1-phenylethyl)pyrazine-2,5-diamine Show/Hide	C21H23Cl2N5	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0454376 Compound Info	3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-((1R,2S)-2-(tetrahydro-2H-pyran-4-yloxy)-2,3-dihydro-1H-inden-1-yl)pyrazin-2-amine Show/Hide	C28H34N4O3	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0457931 Compound Info	N-[(1R,2S)-2-(3,6-dimethylpyrazin-2-yl)oxy-2,3-dihydro-1H-inden-1-yl]-3,6-dimethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C27H28N6O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0467787 Compound Info	3,6-dimethyl-5-(4-methylpyridin-2-yl)oxy-N-[(1R,2S)-2-propan-2-yloxy-2,3-dihydro-1H-inden-1-yl]pyrazin-2-amine Show/Hide	C24H28N4O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0467788 Compound Info	(1S,2R)-1-(3,6-diethyl-5-(4-methylpyridin-2-yloxy)pyrazin-2-ylamino)-2,3-dihydro-1H-inden-2-ol Show/Hide	C23H26N4O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0467789 Compound Info	3,6-diethyl-N2-(3-nitropyridin-2-yl)-N5-(pentan-3-yl)pyrazine-2,5-diamine Show/Hide	C18H26N6O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0477973 Compound Info	5-N-(3,5-dichloropyridin-2-yl)-2-N-(1,3-dimethoxypropan-2-yl)-3,6-diethylpyrazine-2,5-diamine Show/Hide	C18H25Cl2N5O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0484071 Compound Info	3,6-diethyl-N-(2-methoxy-1-phenylethyl)-5-(4-methylpyridin-2-yloxy)pyrazin-2-amine Show/Hide	C23H28N4O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0510694 Compound Info	N-[(1R,2R)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C25H30N4O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0524375 Compound Info	2-N-(3,5-dichloropyridin-2-yl)-2-N,3,6-triethyl-5-N-[(1R,2S)-2-(2-fluoroethoxy)-2,3-dihydro-1H-inden-1-yl]pyrazine-2,5-diamine Show/Hide	C26H30Cl2FN5O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0560210 Compound Info	5-N-(5,7-dimethyl-2,1,3-benzothiadiazol-4-yl)-3,6-diethyl-2-N-pentan-3-ylpyrazine-2,5-diamine Show/Hide	C21H30N6S	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0560211 Compound Info	3,6-diethyl-N2-(4-methylpyridin-2-yl)-N5-(pentan-3-yl)pyrazine-2,5-diamine Show/Hide	C19H29N5	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0562542 Compound Info	N-[(1S,2R)-2-ethoxy-2,3-dihydro-1H-inden-1-yl]-3,6-diethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine Show/Hide	C25H30N4O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0399616 Compound Info	1-(3-chlorophenyl)-3-methyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C22H25ClN2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0501738 Compound Info	1-(2-methoxy-4,6-dimethylphenyl)-3-methyl-N-(2-(pyrrolidin-1-yl)ethyl)isoquinolin-4-amine Show/Hide	C25H31N3O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0530464 Compound Info	3-methyl-1-phenyl-N,N-dipropylisoquinolin-4-amine Show/Hide	C22H26N2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0496792 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid morpholin-4-ylamide Show/Hide	C21H29N5O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0500755 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid [4-(2-fluoro-phenyl)-piperazin-1-yl]-amide Show/Hide	C27H33FN6O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0524423 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid piperazin-1-ylamide Show/Hide	C21H30N6O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0524424 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid (4-acetyl-piperazin-1-yl)-amide Show/Hide	C23H32N6O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0524450 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid phenylamide Show/Hide	C23H26N4O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0525838 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid (2-dimethylamino-ethyl)-ethyl-amide Show/Hide	C23H35N5O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0526008 Compound Info	2-Ethyl-7-(2,4,6-trimethyl-phenyl)-6,7-dihydro-5H-imidazo[1,2-a]imidazole-3-carboxylic acid dibenzylamide Show/Hide	C31H34N4O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0453238 Compound Info	4-methoxy-2-(2-methoxy-4,6-dimethylphenyl)-6-methyl-N-neopentylpyrimidin-5-amine Show/Hide	C20H29N3O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0490265 Compound Info	2-(2,4-dichlorophenyl)-4-methoxy-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C18H23Cl2N3O	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0549510 Compound Info	4-methoxy-2-(2-methoxy-4,6-dimethylphenyl)-6-methyl-N-propylpyrimidin-5-amine Show/Hide	C18H25N3O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0497983 Compound Info	5-(3,6-dihydro-2H-pyridin-1-ylmethyl)-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C16H13Cl3F3N3S	1
1	Ki = 12000 nM Bioactivity Info	TI LI LO TS
CP0523119 Compound Info	N'-(cyclopropylmethyl)-N,N-dimethyl-N'-[[2-(2,4,6-trichloroanilino)-4-(trifluoromethyl)-1,3-thiazol-5-yl]methyl]ethane-1,2-diamine Show/Hide	C19H22Cl3F3N4S	1
1	Ki = 13000 nM Bioactivity Info	TI LI LO TS
CP0377342 Compound Info	(5-Imidazol-1-ylmethyl-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C14H8Cl3F3N4S	1
1	Ki = 18000 nM Bioactivity Info	TI LI LO TS
CP0501428 Compound Info	N'-ethyl-N,N-dimethyl-N'-[[2-(2,4,6-trichloroanilino)-4-(trifluoromethyl)-1,3-thiazol-5-yl]methyl]ethane-1,2-diamine Show/Hide	C17H20Cl3F3N4S	1
1	Ki = 19000 nM Bioactivity Info	TI LI LO TS
CP0392309 Compound Info	N-(cyclopropylmethyl)-N-[[6-ethyl-1-(2,4,6-trimethylphenyl)-2,3-dihydroimidazo[1,2-a]imidazol-5-yl]methyl]propan-1-amine Show/Hide	C24H36N4	1
1	Ki = 19000 nM Bioactivity Info	TI LI LO TS
CP0492023 Compound Info	5-[(cyclopropylmethylamino)methyl]-N-(2,4,6-trichlorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine Show/Hide	C15H13Cl3F3N3S	1
1	Ki = 29000 nM Bioactivity Info	TI LI LO TS
CP0390942 Compound Info	(5-Piperidin-1-ylmethyl-4-trifluoromethyl-thiazol-2-yl)-(2,4,6-trichloro-phenyl)-amine Show/Hide	C16H15Cl3F3N3S	1
1	Ki = 55000 nM Bioactivity Info	TI LI LO TS
CP0392319 Compound Info	3-(4-chlorophenyl)-2,5-dimethyl-N,N-dipropylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C19H24ClN5	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0439803 Compound Info	3-(3-chlorophenyl)-2,5-dimethyl-N,N-dipropylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C19H24ClN5	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0505986 Compound Info	3-(2,4-dichlorophenyl)-N,2,5-trimethylpyrazolo[4,3-d]pyrimidin-7-amine Show/Hide	C14H13Cl2N5	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0507027 Compound Info	(2,5-Dimethyl-3-phenyl-2H-pyrazolo[4,3-d]pyrimidin-7-yl)-dipropyl-amine Show/Hide	C19H25N5	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0373785 Compound Info	N-butyl-N,2-diethyl-7-oxo-8-(2,4,6-trimethylphenyl)-5,6-dihydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C24H34N4O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0373786 Compound Info	8-mesityl-3-((4-methyl-1,4-diazepan-1-yl)methyl)-2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine Show/Hide	C23H32F3N5	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0382897 Compound Info	N-benzyl-2-methyl-N-propyl-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C27H34N4O	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0382898 Compound Info	N-(cyclopropylmethyl)-2-ethyl-7-oxo-N-propyl-8-(2,4,6-trimethylphenyl)-5,6-dihydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C25H34N4O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0447408 Compound Info	8-mesityl-2-methyl-7-oxo-N,N-dipropyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C23H32N4O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0471531 Compound Info	2-methyl-7-oxo-N,N-bis(prop-2-enyl)-8-(2,4,6-trimethylphenyl)-5,6-dihydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C23H28N4O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0480009 Compound Info	2-ethyl-8-mesityl-7-oxo-N,N-dipropyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C24H34N4O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0485598 Compound Info	2-methyl-N-prop-2-enyl-N-propyl-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C23H32N4O	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0485599 Compound Info	2-ethyl-7-oxo-N,N-bis(prop-2-enyl)-8-(2,4,6-trimethylphenyl)-5,6-dihydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C24H30N4O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0520354 Compound Info	N-benzyl-N,2-diethyl-7-oxo-8-(2,4,6-trimethylphenyl)-5,6-dihydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C27H32N4O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0526344 Compound Info	3-(4-(2-fluorophenyl)piperazine-1-carbonyl)-8-mesityl-2-methyl-5,6-dihydroimidazo[1,2-a]pyrimidin-7(8H)-one Show/Hide	C27H30FN5O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0527163 Compound Info	N-(cyclopropylmethyl)-2-methyl-N-propyl-8-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-imidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C24H34N4O	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0527165 Compound Info	N-(cyclopropylmethyl)-2-methyl-7-oxo-N-propyl-8-(2,4,6-trimethylphenyl)-5,6-dihydroimidazo[1,2-a]pyrimidine-3-carboxamide Show/Hide	C24H32N4O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0527166 Compound Info	8-mesityl-2-methyl-3-(morpholine-4-carbonyl)-5,6-dihydroimidazo[1,2-a]pyrimidin-7(8H)-one Show/Hide	C21H26N4O3	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS
CP0486466 Compound Info	4-isopropoxy-2-(2-methoxy-4,6-dimethylphenyl)-6-methyl-N,N-dipropylpyrimidin-5-amine Show/Hide	C23H35N3O2	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS

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About MolBiC

Correspondence

Prof. Feng ZHU

Prof. Leo, Lianyi Han