Brief Information of the Compound and Protein
Compound Name
N-[(1R,2S)-2-(3,6-dimethylpyrazin-2-yl)oxy-2,3-dihydro-1H-inden-1-yl]-3,6-dimethyl-5-(4-methylpyridin-2-yl)oxypyrazin-2-amine
    Show/Hide
PubChem ID
CID: 44443637
Canonical SMILES
Cc1ccnc(Oc2nc(C)c(N[C@H]3[C@H](Cc4ccccc34)Oc3nc(C)cnc3C)nc2C)c1
    Show/Hide
Compound Formula C27H28N6O2
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
>
Corticotropin releasing factor receptor
>
Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS