Brief Information of the Compound and Protein
Compound Name
N-(1,3-dimethoxypropan-2-yl)-8-(4-methoxy-2-methylphenyl)-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-4-amine
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PubChem ID
CID: 42618174
SID: 81078833
Canonical SMILES
COCC(COC)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1C
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Compound Formula C20H27N5O3
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  1
1
Ki = 2 nM
   TI
   LI
   LO
   TS