Brief Information of the Compound and Protein
Compound Name
2-N-(3,5-dichloropyridin-2-yl)-2-N,3,6-triethyl-5-N-[(1R,2S)-2-(2-fluoroethoxy)-2,3-dihydro-1H-inden-1-yl]pyrazine-2,5-diamine
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PubChem ID
CID: 44443662
Canonical SMILES
CCN(c1ncc(Cl)cc1Cl)c1nc(CC)c(N[C@H]2[C@H](Cc3ccccc23)OCCF)nc1CC
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Compound Formula C26H30Cl2FN5O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS