Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-(4-(2-fluorophenyl)piperazine-1-carbonyl)-8-mesityl-2-methyl-5,6-dihydroimidazo[1,2-a]pyrimidin-7(8H)-one
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 PubChem ID
CID: 46881390
Canonical SMILES
Cc1nc2N(C(=O)CCn2c1C(=O)N1CCN(CC1)c1ccccc1F)c1c(C)cc(C)cc1C
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Compound Formula C27H30FN5O2
Compound Structure
Protein Name
 Protein Info 
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32
 Cell Line Info 
Homo sapiens (Human)  1
1
Ki > 5000 nM
   TI
   LI
   LO
   TS