Brief Information of the Compound and Protein
Compound Name
8-mesityl-3-((4-methyl-1,4-diazepan-1-yl)methyl)-2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine
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PubChem ID
CID: 46881399
Canonical SMILES
CN1CCCN(Cc2c(nc3N(CCCn23)c2c(C)cc(C)cc2C)C(F)(F)F)CC1
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Compound Formula C23H32F3N5
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  1
1
Ki > 5000 nM
   TI
   LI
   LO
   TS