Brief Information of the Cell Line and Protein
Cell Line ID: CL000026 , CHO-K1
Synonyms
CHO K1
CHOK1
CHO cell clone K1
GM15452
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0214
Protein ID: PT03308 , G-protein coupled receptor 35
Gene Name GPR35
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q9HC97
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000026  Protein ID: PT03308
 
Compound ID Compound Name Compound Formula
CP0419202
4,17-dioxo-3,18-dioxatetracyclo[12.4.0.02,7.08,13]octadeca-1(14),2(7),5,8,10,12,15-heptaene-5,16-dicarboxylic acid
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C18H8O8
 2
1
EC50 = 0.31 nM
   TI
   LI
   LO
   TS
2
IC50 = 0.47 nM
   TI
   LI
   LO
   TS
CP0419205
10-methyl-4,6-dioxo-1,9-dihydropyrido[3,2-g]quinoline-2,8-dicarboxylic acid
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C15H10N2O6
 2
1
EC50 = 1.08 nM
   TI
   LI
   LO
   TS
2
IC50 = 0.74 nM
   TI
   LI
   LO
   TS
CP0285587
2-[2-[4-[(4-chlorophenyl)-phenyl-methyl]piperazino]ethoxy]ethanol
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C23H16O6
 2
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
2
EC50 = 500 nM
   TI
   LI
   LO
   TS
CP0444735
4,6-dichloro-10-methylpyrido[3,2-g]quinoline-2,8-dicarboxylic acid
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C15H8Cl2N2O4
 2
1
EC50 = 5.08 nM
   TI
   LI
   LO
   TS
2
IC50 = 3.52 nM
   TI
   LI
   LO
   TS
CP0419207
6-(4-methoxyphenyl)-2,8-dioxopyrano[2,3-f]chromene-3,9-dicarboxylic acid
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C21H12O9
 2
1
EC50 = 6.93 nM
   TI
   LI
   LO
   TS
2
IC50 = 2.45 nM
   TI
   LI
   LO
   TS
CP0419201
4,6-dimethoxy-10-methylpyrido[3,2-g]quinoline-2,8-dicarboxylic acid
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C17H14N2O6
 2
1
EC50 = 8.13 nM
   TI
   LI
   LO
   TS
2
IC50 = 6.11 nM
   TI
   LI
   LO
   TS
CP0389119
6-bromo-8-[(4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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C18H12BrNO6
 1
1
EC50 = 12.1 nM
   TI
   LI
   LO
   TS
CP0520866
10-bromo-2,8-dioxopyrano[3,2-g]chromene-3,7-dicarboxylic acid
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C14H5BrO8
 2
1
EC50 = 12.72 nM
   TI
   LI
   LO
   TS
2
IC50 = 9.31 nM
   TI
   LI
   LO
   TS
CP0510397
4,10-dioxo-1,7-dihydro-1,7-phenanthroline-2,8-dicarboxylic acid
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C14H8N2O6
 1
1
EC50 = 13 nM
   TI
   LI
   LO
   TS
CP0517077
6-bromo-2,8-dioxo-3-(2H-tetrazol-5-yl)pyrano[2,3-f]chromene-9-carboxylic acid
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C14H5BrN4O6
 2
1
EC50 = 25.92 nM
   TI
   LI
   LO
   TS
2
IC50 = 15.9 nM
   TI
   LI
   LO
   TS
CP0382598
2-[3-cyano-5-(3,4-dichlorophenyl)-4,5-dimethylfuran-2-ylidene]propanedinitrile
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C16H9Cl2N3O
 2
1
EC50 = 32 nM
   TI
   LI
   LO
   TS
2
EC50 = 10200 nM
   TI
   LI
   LO
   TS
CP0082759
CROMOLYN
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C23H16O11
 2
1
EC50 = 52 nM
   TI
   LI
   LO
   TS
2
EC50 = 7000 nM
   TI
   LI
   LO
   TS
CP0037172
3-(2-propoxyphenyl)-2,4,7,8,9-pentazabicyclo[4.3.0]nona-1,3,6-trien-5-one
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C13H13N5O2
 4
1
EC50 = 62.83 nM
   TI
   LI
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   TS
2
EC50 = 160 nM
   TI
   LI
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3
EC50 = 4200 nM
   TI
   LI
   LO
   TS
4
IC50 = 48.15 nM
   TI
   LI
   LO
   TS
CP0419208
10-(4-methoxyphenyl)-2,8-dioxopyrano[3,2-g]chromene-3,7-dicarboxylic acid
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C21H12O9
 2
1
EC50 = 62.83 nM
   TI
   LI
   LO
   TS
2
IC50 = 48.15 nM
   TI
   LI
   LO
   TS
CP0070834
3,3''''-methylenebis(4-hydroxy-coumarin
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C19H12O6
 1
1
EC50 = 1300 nM
   TI
   LI
   LO
   TS
CP0192012
DOXANTRAZOLE
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C14H8N4O3S
 1
1
EC50 = 3400 nM
   TI
   LI
   LO
   TS
CP0322785
Aphthasol
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C16H14N2O4
 1
1
EC50 = 4000 nM
   TI
   LI
   LO
   TS
CP0533478
Lodoxamide
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C11H6ClN3O6
 1
1
EC50 = 4000 nM
   TI
   LI
   LO
   TS