8-(4-chlorophenyl)-1h-pyrrolo[2'',3'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

8-(4-methylphenyl)-1h-pyrrolo[2'',3'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

9-(4-chlorophenyl)-2,3-dihydro-3(R)-methyl-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

4-fluoro-N-methyl-N-(4-(6-(methylamino)pyrimidin-4-yl)thiazol-2-yl)benzamide

9-(4-chlorophenyl)-2,3-dihydro-3(S)-methyl-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

2,3-dihydro-9-(4-methylphenyl)-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

2,3-dihydro-9-(4-methoxyphenyl)-3(R)-methyl-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

N-[4-(6-aminopyrimidin-4-yl)-1,3-thiazol-2-yl]-4-fluoro-N-methylbenzamide

2,3-dihydro-9-(4-methoxyphenyl)-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

tert-butyl 4-[1-(3-fluoropyridin-2-yl)triazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

2-cyclopropyl-5-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)-2,3-dihydro-1H-inden-1-one

9-(4-chlorophenyl)-2,3-dihydro-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

2-ethyl-5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl)isoindolin-1-one

2-cyclopropyl-5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl)isoindolin-1-one

5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl)-2-propylisoindolin-1-one

N-[4-[6-(ethylamino)pyrimidin-4-yl]-1,3-thiazol-2-yl]-4-fluoro-N-methylbenzamide

4-O-[(2S)-3,3-dimethylbutan-2-yl] 2-O-propyl 3-methyl-1H-pyrrole-2,4-dicarboxylate

8-(4-methoxyphenyl)-1h-pyrrolo[2'',3'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

6-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)quinoline

4-fluoro-N-(4-(6-(isopropylamino)pyrimidin-4-yl)thiazol-2-yl)-N-methylbenzamide

2,3-dihydro-3(R)-methyl-9-(4-methylphenyl)-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl)-2-isopropylisoindolin-1-one

4-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl)-N-isopropyl-N-methyl-5,6-dihydropyridine-1(2H)-carboxamide

8-bromo-3-(4-chloro-phenyl)-9-methylamino-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one

8-(4-chlorophenyl)-1h-imidazo[4'',5'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

4-fluoro-N-methyl-N-(4-(pyridin-2-yl)thiazol-2-yl)benzamide

tert-butyl 4-[1-(2-fluorophenyl)triazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

tert-butyl 4-[1-(3-fluoropyridin-2-yl)-5-methyltriazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

propan-2-yl 4-[1-(2-fluoropyridin-3-yl)-5-methyltriazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

9-dimethylamino-3-(4-methoxy-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one

8-(4-chlorophenyl)-1-methyl-1H-imidazo[4'',5'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

tert-butyl 4-(1-phenyltriazol-4-yl)-3,6-dihydro-2H-pyridine-1-carboxylate

4-fluoro-N-methyl-N-(4-(pyrimidin-4-yl)thiazol-2-yl)benzamide

tert-butyl 4-[1-(2-methylphenyl)triazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

2,2-dimethyl-5-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)-2,3-dihydro-1H-inden-1-one

9-(4-chlorophenyl)-2,3-dihydro-2(S)-methyl-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

tert-butyl 4-[1-(4-fluorophenyl)triazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

8-(4-methylphenyl)-1H-pyrazolo[3'',4'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

tert-butyl 4-[1-(3-fluorophenyl)triazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

N-ethyl-4-fluoro-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide

4-O-(2-bicyclo[2.2.1]heptanyl) 2-O-ethyl 3-methyl-1H-pyrrole-2,4-dicarboxylate

cyclopropyl-[4-(5-methyl-1-pyridin-3-yltriazol-4-yl)phenyl]methanone

9-(4-chlorophenyl)-2,3-dihydro-2(R)-methyl-1H-pyrimido[4'',5'':4',5']thieno[3',2':5,6]pyrido[3,4-b][1,4]oxazin-8(9H)-one

2-[[4-(2,3-dihydro-1H-inden-2-ylamino)-5,6,7,8-tetrahydroquinazolin-2-yl]sulfanyl]ethanol

[(2S)-3,3-dimethylbutan-2-yl] 5-(2-methoxyethylcarbamoyl)-4-methyl-1H-pyrrole-3-carboxylate

propan-2-yl 4-(5-methyl-1-pyridin-3-yltriazol-4-yl)benzoate

8-(4-chlorophenyl)-1h-pyrazolo[3'',4'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

propan-2-yl 4-[1-(2-fluoropyridin-3-yl)triazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

tert-butyl 4-(1-pyridin-2-yltriazol-4-yl)-3,6-dihydro-2H-pyridine-1-carboxylate

4-fluoro-N-methyl-N-(4-(pyrazin-2-yl)thiazol-2-yl)benzamide

4-fluoro-N-methyl-N-(4-(pyridin-4-yl)thiazol-2-yl)benzamide

tert-butyl 4-(1-pyridin-3-yltriazol-4-yl)-3,6-dihydro-2H-pyridine-1-carboxylate

N-tert-butyl-4-[1-(2-fluorophenyl)triazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxamide

4-chloro-N-methyl-N-(4-(pyridin-4-yl)thiazol-2-yl)benzamide

5-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)-2,3-dihydro-1H-inden-1-one

4-fluoro-N-(4-(6-(isopropyl(methyl)amino)pyrimidin-4-yl)thiazol-2-yl)-N-methylbenzamide

N-methyl-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)benzamide

4-fluoro-N-propyl-N-(4-(pyridin-2-yl)thiazol-2-yl)benzamide

N,4-dimethyl-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)benzamide

4-O-(2-bicyclo[2.2.1]heptanyl) 2-O-ethyl 3,5-dimethyl-1H-pyrrole-2,4-dicarboxylate

3-fluoro-N-methyl-N-(4-(pyridin-4-yl)thiazol-2-yl)benzamide

1-(3,3-Dimethylbutanolyl)-4-[1-(2-fluorophenyl)-1H-1,2,3-triazol-4-yl]-1,2,3,6-tetrahydorohydropyridine

2-fluoro-N-methyl-N-(4-(pyridin-4-yl)thiazol-2-yl)benzamide

2-bicyclo[2.2.1]heptanyl 5-(2-methoxyethylcarbamoyl)-4-methyl-1H-pyrrole-3-carboxylate

1-(4-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)phenyl)propan-1-one

2-bicyclo[2.2.1]heptanyl 5-(4-acetamidobutylcarbamoyl)-4-methyl-1H-pyrrole-3-carboxylate

4-bromo-N-methyl-N-(4-(pyridin-4-yl)thiazol-2-yl)benzamide

4-(5-methyl-1-pyridin-3-yltriazol-4-yl)-N-propan-2-ylbenzamide

tert-butyl 4-(1-pyridin-4-yltriazol-4-yl)-3,6-dihydro-2H-pyridine-1-carboxylate

4-fluoro-N-methyl-N-(4-(pyridin-3-yl)thiazol-2-yl)benzamide

5-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)-1H-indole

3-(5-methyl-4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)pyridine

2-bicyclo[2.2.1]heptanyl 5-(2-methoxyethylcarbamoyl)-2,4-dimethyl-1H-pyrrole-3-carboxylate

8-(4-methylphenyl)thiazolo[4'',5'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidine-2,7(1H,8H)-dione

1-(4-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)phenyl)ethanone

1,2-dihydro-8-(4-methylphenyl)-2-thioxothiazolo[4'',5'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

tert-butyl 4-[1-(2-methoxyphenyl)triazol-4-yl]-3,6-dihydro-2H-pyridine-1-carboxylate

8-(4-methylphenyl)-2-(methylthio)thiazolo[4'',5'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one

N-methyl-4-(5-methyl-1-pyridin-3-yltriazol-4-yl)-N-propan-2-ylbenzamide

4-fluoro-N-(4-(pyridin-2-yl)thiazol-2-yl)benzamide

2-bicyclo[2.2.1]heptanyl 5-(4-acetamidobutylcarbamoyl)-2,4-dimethyl-1H-pyrrole-3-carboxylate

4-fluoro-N-methyl-N-(4-(pyrimidin-5-yl)thiazol-2-yl)benzamide

4-methoxy-N-methyl-N-(4-(pyridin-4-yl)thiazol-2-yl)benzamide

2-methyl-5-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)benzo[d]thiazole

(4-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)phenyl)(pyrrolidin-1-yl)methanone

4-fluoro-N-isopropyl-N-(4-(pyridin-2-yl)thiazol-2-yl)benzamide

propan-2-yl 3-(5-methyl-1-pyridin-3-yltriazol-4-yl)benzoate

(4-(5-methyl-1-(pyridin-3-yl)-1H-1,2,3-triazol-4-yl)phenyl)(phenyl)methanone

4-fluoro-N-methyl-N-(4-(pyrimidin-2-yl)thiazol-2-yl)benzamide

4-fluoro-N-methyl-N-(4-phenylthiazol-2-yl)benzamide

N-methyl-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)-4-(trifluoromethoxy)benzamide

5-(1-(2,4-difluorophenyl)-5-methyl-1H-1,2,3-triazol-4-yl)-2-isopropylisoindolin-1-one

N-(4-fluorophenyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-amine

2-(3-methylanilino)-7,8-dihydro-6H-quinazolin-5-one

N4-(bicyclo[2.2.1]heptan-2-yl)-N2-(2-methoxyethyl)-3-methyl-1H-pyrrole-2,4-dicarboxamide